Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
08/2000
08/17/2000WO2000012076A9 Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use
08/17/2000WO2000009109A3 Pipecolic acid derivatives for vision and memory disorders
08/17/2000DE19907480A1 New epothilone derivatives, useful for treating malignant tumors such as ovarian, stomach, colon, breast and lung carcinoma, acute lymphocytic and myelocytic leukemia and chronic inflammatory diseases such as psoriasis
08/17/2000CA2360952A1 Epothilon derivatives, method for the production and the use thereof as pharmaceuticals
08/17/2000CA2360305A1 Lactam inhibitors of fxa and method
08/17/2000CA2360164A1 5-ht1f agonists
08/16/2000EP1027359A2 Monocyclic l-nucleosides, analogs and uses thereof
08/16/2000EP1027349A1 Tetrahydrofuran phosphate- and hydroxy esters, as prodrugs for the corresponding antifungal agent
08/16/2000EP1027344A2 Pharmaceutical compounds isolated from aristolochia taliscana
08/16/2000EP1027336A1 Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors
08/16/2000EP1027335A1 Ortho-hydroxypyridinone derivatives as iron chelating and antioxidant agents
08/16/2000EP1027332A1 Novel lactam metalloprotease inhibitors
08/16/2000EP1027328A1 Substituted anilides
08/16/2000EP1027052A1 Novel combination
08/16/2000EP1026950A1 Treatment of schizophrenia with ampakines and neuroleptics
08/16/2000EP0842171B1 Herbicidal sulphonylamino(thio)carbonyl triazolinones with heterocyclyloxy substituents
08/16/2000EP0805802B1 Substituted phenyl compounds as endothelin antagonists
08/16/2000EP0707481B1 L-2',3'-dideoxy nucleoside analogs as anti-hepatitis b (hbv) and anti-hiv agents
08/16/2000CN1055477C Intermediate compound for synthesizing nucleoside derivative
08/16/2000CN1055470C Paroxetine and process for preparing medical salts thereof
08/16/2000CN1055467C Taxoids compound, their preparation and pharmaceutical compositions containing them
08/16/2000CN1055465C Optical active 2-imidazoline-5-thione derivatives and preparating method and use thereof
08/15/2000US6103936 Reacting aldehyde, sulfide, sulfone, or sulfoxide with formamide in presence of acid catalyst, and optionally a dehydrating agent
08/15/2000US6103910 D-proline derivatives
08/15/2000US6103905 Quinoline-indole antimicrobial agents, uses and compositions related thereto
08/15/2000US6103899 Bicyclic aminoimidazoles
08/15/2000US6103762 A biaromatic compounds in which the aromatic nuclei are connected by a propynylene or allenylene divalent radical, useful as human or veterinary medicine or used in cosmetics or keratinization disorders
08/15/2000US6103750 Pyrazole substituted tetrafluorodihydrobenzofuranyl or tetrafluorodihydroisobenzofuranyl compounds useful as pesticides, insecticides and miticides
08/15/2000US6103738 Quinoline and quinazoline compounds useful in therapy
08/15/2000US6103718 Selective cyclic nucleotide phosphodiesterase (pde) inhibitors (specifically of type 4) which are effective bronchial therapeutics; bronchodilators; respiratory system disorders
08/15/2000US6103715 Compounds that bind to the dopamine d4 receptor and their use as anxiolytic agents, treatment for schizophrenia, and drug screening; side effect reductioon
08/15/2000US6103700 Fluoro labelled anthracyclinone and anthracycline derivatives
08/15/2000US6103667 Phenylpyrazole herbicides
08/15/2000US6103665 Inhibition of glutathione transferase by haloenol lactones
08/15/2000CA2202280C Sugar modified nucleosides and their use for synthesis of oligonucleotides
08/15/2000CA2105385C Treatment of cognitive disorders
08/10/2000WO2000046221A1 Sulfamato hydroxamic acid metalloprotease inhibitor
08/10/2000WO2000046212A1 Method of producing substituted pyrimidine derivatives
08/10/2000WO2000046208A1 Substituted pyrazole carboxylic acids used to combat anaemias
08/10/2000WO2000046203A2 G-protein coupled heptahelical receptor binding compounds and methods of use thereof
08/10/2000WO2000046199A2 Indole derivatives as anti-inflammation agents
08/10/2000WO2000046198A1 Anti-inflammatory indole derivatives
08/10/2000DE19904406A1 Substituierte Pyrazolcarbonsäuren Substituted pyrazole
08/10/2000CA2362401A1 G-protein coupled heptahelical receptor binding compounds and methods of use thereof
08/10/2000CA2362230A1 Sulfamato hydroxamic acid metalloprotease inhibitor
08/10/2000CA2361816A1 Substituted pyrazole carboxylic acids used to combat anaemias
08/10/2000CA2357013A1 Anti-inflammatory indole derivatives
08/10/2000CA2355734A1 Indole derivatives as anti-inflammation agents
08/09/2000EP1026165A1 O-substituted Hydroxycoumaranone derivatives as antitumor and antimetastatic agents
08/09/2000EP1026151A1 Aryl and heteroarylcyclopropyl oxime ethers and their use as fungicides and insecticides
08/09/2000EP1025095A1 Substituted chroman derivatives
08/09/2000EP1025090A1 Vitronectin receptor antagonists
08/09/2000EP1024814A2 Use of antifungal agents for the topical treatment of fungus-induced mucositis
08/09/2000EP1024799A1 Method for treating disease-related or drug-induced dyskinesias
08/09/2000EP1024697A1 Method for treating alzheimer's disease
08/09/2000CN1262684A 2,4,4-trisubstituted-1,3-dioxolane antifungals
08/09/2000CN1262683A Soluble prodrugs of paclitaxel
08/09/2000CN1262682A Itraconazole with improved solubility, method of preparing same and pharmaceutical composition for oral administration comprising same
08/09/2000CN1262681A 4,5-dihydro-[1H]-benz [g] indazole-3-carboxylic acid derivatives
08/09/2000CN1262679A IL-5 inhibiting 6-azauracil derivatives
08/09/2000CN1262678A Triazole compounds and use thereof as dopamine-D3-ligands
08/09/2000CN1262676A 吡啶衍生物 Pyridine derivatives
08/09/2000CN1262675A (+)-Norcisapride useful for 5-HT3 and 5-HT4 mediated disorbers
08/09/2000CN1262674A Gatrokinetic monocyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidine derivatives
08/09/2000CN1262621A Gastrokinetic bicyclc benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidine derivatives
08/09/2000CN1262269A Aryl and heteroaryl cyclopropyl oximidoether and its application as bactericide and pesticide
08/08/2000US6100291 Pyrrolidine-indole compounds having 5-HT6 affinity
08/08/2000US6100284 Antiallergens
08/08/2000US6100268 Vasoconstrictive dihydrobenzopyran derivatives
08/08/2000US6100267 Enzyme inhibitor for treatment of neurodegenerative disorders, strokes, traumatic brain injury, cataracts
08/08/2000US6100257 2-haloalkyl,3-(haloalkyl, alkenyl, or alkynyl),5-(substituted phenyl or heterocycle),6-alkyl-pyrimidin-4-one compounds of given structure; use as herbicides
08/08/2000US6100253 Tricycle substituted with azaheterocyclic carboxylic acids
08/08/2000CA2185512C Treatment of tinnitus using neuroprotective agents
08/08/2000CA2072575C Anticholinergic agents
08/08/2000CA2018438C Imidazolyl-alkenoic acids
08/03/2000WO2000044737A1 Aminoalkylbenzofurans as serotonin (5-ht(2c)) agonists
08/03/2000WO2000044730A1 2,3,4,5-tetrahydro-1h-[1,4]benzodiazepine-3-hydroxamic acid as matrix metalloproteinase inhibitors
08/03/2000WO2000044728A1 Substituted bicyclic derivatives useful as anticancer agents
08/03/2000WO2000044726A1 2h-phthalazin-1-one derivatives and drugs comprising these derivatives as the active ingredient
08/03/2000WO2000044722A1 Chondrongenesis promotors and indolin-2-one derivatives
08/03/2000WO2000044379A2 Methods for restoring and/or enhancing accommodation in pseudo phakia
08/03/2000WO2000044376A1 Antidepressant heterocyclic compounds
08/03/2000WO2000044362A2 The use of 4-h-1-benzopyran-4-one derivatives as inhibitors of smooth muscle cell proliferation
08/03/2000WO2000005208A9 Amino-aldehyde solid support, linker therefor and methods of preparation and use thereof
08/03/2000CA2361516A1 Aminoalkylbenzofurans as serotonin (5-ht(2c)) agonists
08/03/2000CA2360683A1 Antidepressant heterocyclic compounds
08/03/2000CA2356313A1 Alkynyl containing hydroxamic acid derivatives, their preparation and their use as matrix metalloproteinase (mmp) inhibitors/tnf-alpha converting enzyme (tace) inhibitors
08/03/2000CA2356267A1 2,3,4,5-tetrahydro-1h-¬1,4|benzodiazepine-3-hydroxamic acid as matrix metalloproteinase inhibitors
08/02/2000EP1024134A1 Aminobutanoic acid derivatives
08/02/2000EP1023287A1 3-oxo-2(h)-1,2,4-triazine derivatives as ligands of 5ht1a receptors
08/02/2000EP1023281A1 Hiv integrase inhibitors
08/02/2000EP1023273A1 Cyclohexane derivatives difunctionalised in 1,4 as ligands of 5t h1a receptors
08/02/2000EP1023269A1 Beta3-adrenoreceptor agonists, agonist compositions and methods of using
08/02/2000EP1023268A1 Isoquinolines as urokinase inhibitors
08/02/2000EP1023267A1 Pyridyl compounds and pharmaceutical compositions containing them
08/02/2000EP1023265A1 Azetidinone derivatives for the treatment of hcmv infections
08/02/2000EP1023068A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
08/02/2000EP1023063A1 INDENO 1,2-c]-, NAPHTHO 1,2-c]- AND BENZO 6,7]CYCLOHEPTA 1,2-c]PYRAZOLE DERIVATIVES
08/02/2000EP0731796B1 1,3,5-trisubstituted pyrazole compounds for treatment of inflammation
08/02/2000EP0691953B1 1-amidinophenyl-pyrrolidones/ piperidinones as platelet aggregation inhibitors