Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
09/2000
09/21/2000CA2368148A1 Novel compounds and compositions as protease inhibitors
09/21/2000CA2368122A1 Novel compounds and compositions as protease inhibitors
09/21/2000CA2367895A1 Compounds and methods for modulation of estrogen receptors
09/21/2000CA2367461A1 Heterocyclic aromatic compounds useful as growth hormone secretagogues
09/21/2000CA2367352A1 Amine derivatives as protease inhibitors
09/20/2000EP1036073A1 (benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties
09/20/2000EP1036072A1 Thrombin receptor antagonists
09/20/2000EP1036065A1 Substituted imidazole derivatives having agonist-like activity at alpha 2b or 2b/2c adrenergic receptors
09/20/2000EP1036062A1 Hydroxamic acid derivatives as matrix metalloprotease (mmp) inhibitors
09/20/2000EP0705816B1 Benzene derivative useful for ischemic diseases
09/20/2000CN1267300A Benzo (5,6) cyclohepta (1,2-b) pyridine derivs useful for inhibition of farnesyl protein transferase
09/20/2000CN1267299A Aminooxyamide tricyclic inhibitors of farnesylprotein transferase
09/20/2000CN1267293A Benzo (5,6) cyclohepta (1,2-b) pyridine derivs. useful for inhibition of farnesyl-protein transferase
09/20/2000CN1267284A Carbostyril derivs. for inhibiting skin erythema and/or skin pigmentation
09/20/2000CN1266850A O-substd. hydroxy coumaranone derivs as antineoplastic and antitransfer agent
09/20/2000CN1056610C Piperidine or piperazine derivs, pharmaceutical compositions contg. them and their use
09/20/2000CN1056602C Esters and amides as PLAZ inhibitors
09/19/2000US6121451 Anticancer drugs
09/19/2000US6121448 Liquid crystalline compounds
09/19/2000US6121433 For diagnostic, research and therapeutic use; mimic or modulate proteins, enzymes, nucleic acids and lipids
09/19/2000US6121431 Nucleoside derivatives
09/19/2000US6121313 Pharmaceutical composition in a form of self-emulsifying formulation for lipophilic compounds
09/19/2000US6121310 By contacting plants or plant products with the antibiotic blasticidin a or salt thereof; inhibits production of aflatoxin, without inhibiting the growth of the aflatoxigenic organisms
09/19/2000US6121309 Fused-ring carboxylic acid derivatives
09/19/2000US6121308 Indole and benzimidazole antithrombotic compounds, such as 1-methyl-2-(n-(4-amidinophenyl)-aminomethyl)-5-(n-(hydroxycarbonylmethyl) -quinoline-8-sulphonylamino)-indole
09/19/2000US6121307 Side effect reduction; administering to treat depression
09/19/2000US6121283 N-substituted-6-(2-(4-trifluoromethylphenyl)phenylcarbonyl-amino) -1,2,3,4-tetrahydroisoquinolines; treating disorders including obesity, hyperlipidemia, and diabetes; microsomal triglyceride transfer protein (mtp); apolipoprotein b (apo-b)
09/19/2000US6121274 Phosphodiesterase inhibitor for treatment of respiratory system disorders
09/19/2000US6121270 N-(epoxyalkyl)xanthine derivatives which modulate cellular responses to noxious, pro-inflammatory stimuli
09/19/2000US6121267 Substituted piperazines and piperidines as central nervous system agents
09/19/2000US6121260 Appetite stimulation with dosage of neuropeptide y (npy) receptor agonist
09/19/2000US6121204 Selective control of monocotyledonous and dicotyledonous weeds in monocotyledonous and dicotyledonous crops, both pre-emergence and post-emergence
09/19/2000US6120696 Proton conductors in liquid form
09/14/2000WO2000053597A2 Benzofuran-2-ones as colorants for organic materials
09/14/2000WO2000053594A1 Aminomethylpyrrolidine derivatives having aromatic substituents
09/14/2000WO2000053583A1 Inhibitors of protein tyrosine phosphatase
09/14/2000WO2000053579A2 Solid phase synthesis of 4-aminoproline derivatives and/or combinatorial libraries thereof
09/14/2000WO2000053563A1 Novel ligands of nuclear receptors ppar's
09/14/2000WO2000053547A1 Method of preparing surface-active alcohols and surface-active alcoholic ethers, products obtained by said method and their use
09/14/2000WO2000044722A8 Chondrongenesis promotors and indolin-2-one derivatives
09/14/2000DE19910370A1 Verfahren zur Herstellung von Tensidalkoholen und Tensidalkoholethern, die hergestellten Produkte und ihre Verwendung A process for the preparation of surfactant alcohols and surfactant alcohol ethers, the manufactured products and their use
09/14/2000CA2366308A1 Inhibitors of protein tyrosine phosphatase
09/14/2000CA2366281A1 Novel ligands of nuclear receptors ppar's
09/13/2000EP1035113A2 Process for the preparation of 2-aryl-5-(perfluoroalkyl)pyrrole compounds from N-[1-chloro-1-(perfluoroalkyl)methyl]arylimidoyl chloride compounds
09/13/2000EP1034169A1 Trisaryl-1,3,5-triazine ultraviolet light absorbers
09/13/2000EP1034167A1 Alpha-alkylthio substituted pyrimidine ethers and thioethers as viral reverse transcriptase inhibitors
09/13/2000EP1034166A1 Substituted 2-phenyl-3(2h)-pyridazinones
09/13/2000EP1034165A1 Pyrazolylpyrazoles substituted by 1-methyl-5- alkylsulphonyl, 1-methyl-5- alkylsuphinyl and 1-methyl-5- alkylthio, methods for preparing them and use as herbicides
09/13/2000EP1034164A1 Substituted beta-alanine derivatives as cell adhesion inhibitors
09/13/2000EP0839146B1 Piperazine derivatives and their use as 5-ht1a antagonists
09/13/2000EP0764166B1 Corticotropin releasing factor antagonists
09/13/2000EP0607193B1 Triazole antifungal agents
09/13/2000EP0586570B1 Backbone modified oligonucleotide analogues
09/13/2000CN1266433A Benzpyrido cycloheptane compounds useful for inhibition of franesyl protein transferase
09/13/2000CN1266431A Aroyl-piperazine derivatives, their preparation and their use as tachykinin antagonists
09/13/2000CN1266427A New amidino derivatives and their use as thrombin inhibitors
09/13/2000CN1056369C Pyridazinone derivatives or their salts, processes of their production, and anti-shock agents containing them
09/12/2000US6117940 Solid phase synthesis of compounds such as the imidazoles, benzodiazepines, pyrazines, and steroid mimics.
09/12/2000US6117892 Crop protection products
09/12/2000CA2105384C Treatment of addiction to drugs and substances of abuse
09/12/2000CA1341098C Liquid crystal composition and use thereof
09/09/2000CA2300412A1 Process for the preparation of 2-aryl-5-(perfluoro-alkyl) pyrrole compounds from n-[1-chloro-1-(perfluoroalkyl) methyl] arylimidoyl chloride compounds
09/08/2000WO2000051991A1 4-AMINO-QUINAZOLINE AND QUINOLINE DERIVATIVES HAVING AN INHIBITORY EFFECT ON SIGNAL TRANsSDUCTION MEDIATED BY TYROSINE KINASES
09/08/2000WO2000051986A1 Cyclopentanone dihydropyridine compounds useful as potassium channel openers
09/08/2000WO2000051984A1 2-aryl indole derivatives as antagonists of tachykinins
09/08/2000WO2000051967A1 Oxyalkylene-substituted aminophenol intermediate
09/08/2000WO2000051614A1 Inhibitors of prenyl-protein transferases
09/08/2000WO2000051611A1 Inhibitors of prenyl-protein transferase
09/08/2000WO2000051610A1 Pyrrolidine modulators of chemokine receptor activity
09/08/2000WO2000051609A1 3-alkyl substituted pyrrolidine modulators of chemokine receptor activity
09/08/2000WO2000051608A1 3-thienyl and 3-furanyl pyrrolidine modulators of chemokine receptor activity
09/08/2000WO2000051607A1 3-cyclopropyl and 3-cyclobutyl pyrrolidine modulators of chemokine receptor activity
09/08/2000WO2000034260A3 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group
09/08/2000CA2362495A1 Inhibitors of prenyl-protein transferases
09/08/2000CA2362493A1 Inhibitors of prenyl-protein transferase
09/08/2000CA2330541A1 Cyclopentanone dihydropyridine compounds useful as potassium channel openers
09/07/2000DE19910403A1 Medicaments containing hydroxy-benzo-cyclopentabenzazepine-dione derivatives, useful as cellular hyperproliferation inhibitors, especially antitumor agents
09/06/2000EP1032571A1 Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance p antagonists
09/06/2000EP1032556A1 Pharmaceutically active compounds and methods of use
09/06/2000EP1032393A1 QUINOLINE-CONTAINING $g(a)-KETOAMIDE CYSTEINE AND SERINE PROTEASE INHIBITORS
09/06/2000CN1265665A Benzimidazole derivatives
09/06/2000CN1265658A 5-naphthalen-1-yl-1,3-dioxane derivatives, preparation and therapeutic application
09/06/2000CN1265656A O-substituted hydroxycumaranone derivatives as anttumor and antimetastatic agents
09/06/2000CN1265652A 2-acrylaminopropanamines as tachykinin receptor antagonists
09/06/2000CN1265645A Urokinase inhibitors
09/06/2000CN1265593A Novel process for manufacturing paroxetine solid dispersions
09/06/2000CN1265591A Coumpound
09/06/2000CN1265585A (Imidazol-5-yl) methyl-2-quinolinone derivatives as inhibitors of smooth muscle cell proliferation
09/06/2000CN1265394A Compound as intermediates for use in preparation of optically active 2-imidazoline-5-one or 2-imidazoline-5-thionone derivatives
09/06/2000CN1056144C New use of 6-heterocyclic-4-amino-3,4,5-tetrahydrobenz (CD) indoles compound
09/06/2000CN1056140C Biphenyl derivatives, their preparation and theirt use for treatment of hypertension and cardiac disease
09/05/2000US6114549 Process of making 3-phenyl-1-methylenedioxyphenyl-indane-2-carboxylic acid derivatives
09/05/2000US6114539 Reacting imidazole derivative with sulfur with a strong base in presence of diluent, and then hydrolyzing the product with water, or with sulfur in presence of diluent having high boiling point; controlling undesired microorganism in plants
09/05/2000US6114536 Indolin-2-one derivatives
09/05/2000US6114532 Anticoagulant
09/05/2000US6114493 Contacting a compound to be phosgenated with an excess of a phosgene source in the form of a solid phase reagent; supports in combinatorial synthesis for the creation of libraries of compounds for lead identification
09/05/2000US6114374 2-and 2,5-substituted phenylketoenols
09/05/2000US6114371 3-(cyclohexanoheteroarylidenyl)-2-indolinone protein tyrosine kinase inhibitors
09/05/2000US6114368 Triazolyl disulphides
09/05/2000US6114360 Pyrrole compounds