Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
04/2001
04/17/2001US6218392 For therapy and prophylaxis of ischemic heart diseases such as angina pectoris, myocardial infarct and chronic and acute cardiac failure, pulmonary hypertension, arteriosclerosis and bronchial asthma
04/17/2001US6218391 Triazinones and derivatives thereof
04/17/2001US6218385 1,2,4,5-Tetrahydro-benzo[D]azepin derivatives
04/17/2001US6217856 Sunscreen agents
04/17/2001CA2179396C Tetrahydrofuran antifungals
04/17/2001CA2027765C Mevinic acid derivatives
04/12/2001WO2001025233A1 Piperidine derivatives
04/12/2001WO2001025232A1 Process for the preparation of paroxetine hydrochloride acetone solvate
04/12/2001WO2001025231A1 Process for the preparation of paroxetine hydrochloride acetone solvate
04/12/2001WO2001025230A1 Process for the preparation of paroxetine hydrochloride acetone solvate
04/12/2001WO2001025220A1 Triazine kinase inhibitors
04/12/2001WO2001025217A1 New pyrimidine-2,4,6-trione derivatives, processes for their production and pharmaceutical agents containing these compounds
04/12/2001WO2001025210A2 Substituted 2-thio-3,5-dicyano-4-aryl-6-aminopyridines and the use thereof as adenosine receptor ligands
04/12/2001WO2001025208A1 Pyridinium derivatives for the management of aging-related and diabetic vascular complications, process for their preparation and therapeutic uses thereof
04/12/2001WO2001025207A1 Novel nicotinonitrile compounds
04/12/2001WO2001025200A1 Cyclic amine compounds as ccr5 antagonists
04/12/2001WO2001025190A1 Novel diarylamide derivatives and use thereof as medicines
04/12/2001WO2001024828A2 MODULATORS OF CYTOKINE MEDIATED SIGNALLING PATHWAYS AND INTEGRIN αVβ3 RECEPTOR ANTAGONISTS FOR COMBINATION THERAPY
04/12/2001WO2001024827A2 INHIBITORS OF THE ENDOTHELIN SIGNALLING PATHWAY AND αVβ3 INTEGRIN RECEPTOR ANTAGONISTS FOR COMBINATION THERAPY
04/12/2001WO2001024796A1 1,2,4-triazole derivatives, composition, process of making and methods of use
04/12/2001WO1999063939A9 Multibinding inhibitors of cyclooxygenase-2
04/12/2001WO1999057117A3 Indole derivatives and their use in the treatment of malignant and other diseases caused by pathological cell proliferation
04/12/2001CA2608807A1 Cyclic amine compounds as ccr5 antagonists
04/12/2001CA2386457A1 Inhibitors of the endothelin signalling pathway and .alpha.v.beta.3 integrin receptor antagonists for combination therapy
04/12/2001CA2386218A1 Triazine kinase inhibitors
04/12/2001CA2386147A1 Substituted 2-thio-3,5-dicyano-4-aryl-6-aminopyridines and the use thereof
04/12/2001CA2385972A1 Novel diarylamide derivatives and use thereof as medicines
04/12/2001CA2385244A1 Novel nicotinonitrile compounds
04/11/2001EP1090918A1 Amorphous paroxetine hydrochloride and method of producing it
04/11/2001EP1089998A2 Epothilone derivatives and their synthesis and use
04/11/2001EP1089997A1 4,5,6 and 7-indole and indoline derivatives, their preparation and use
04/11/2001EP1089996A1 Paroxetine methanesulfonate
04/11/2001EP1089995A1 Paroxetine ascorbate
04/11/2001EP1089993A1 5-ht 1f? agonists
04/11/2001EP1089989A1 Inhibitors of alpha4beta1 mediated cell adhesion
04/11/2001EP1089980A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
04/11/2001EP1089979A1 Substituted quinoxalin-2(1h)-ones useful as hiv reverse transcriptase inhibitors
04/11/2001EP1089977A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
04/11/2001EP1089964A1 Hydrazine derivatives
04/11/2001EP1089735A1 4-benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective nmda receptor antagonists
04/11/2001EP0984963B1 Novel compounds
04/11/2001CN1291192A 5,6,7-trino-4,8-inter-m-phenylene PGI2 derivative and drugs containing the same
04/11/2001CN1291190A 5-substituted pyrimidine-2-yloxy carboxylic acid derivatives, the production of the same and their utilization as endothelin antagonist
04/11/2001CN1291093A Pig appeasing pheromones to decrease stress, anxiety and aggressiveness
04/11/2001CN1290698A Quinoline-4-base deviative I
04/11/2001CN1064356C New piperazine, piperidine and 1,2,5,6-tetrahydropyridine compounds process for preparation thereof, and pharmaceutical composition containing them
04/11/2001CN1064354C Trilcyclic benzazepine vasopressin antagnonists
04/10/2001US6215016 Hematopoietic agents; preventing cytopenia
04/10/2001US6214870 Antiarthritic agents; anticancer agents
04/10/2001US6214858 Caspases and apoptosis
04/10/2001US6214845 Insecticidal N-(substituted arylmethyl)-4[bis(substituted phenyl or pyridyl)methyl] piperidines
04/10/2001US6214822 Substituted aza and diazacycloheptane and cyclooctane compounds and their use
04/10/2001US6214813 Azopyrazoles
04/10/2001US6214551 Oligonucleoside linkages containing adjacent nitrogen atoms
04/10/2001CA2086974C R(+)-terazosin
04/10/2001CA2077252C Methods of making ureas and guanidines, and intermediates therefor
04/05/2001WO2001023381A1 Piperidine derivatives as reuptake inhibitors
04/05/2001WO2001023380A1 Piperidine derivatives as serotonine reuptake inhibitors
04/05/2001WO2001023378A1 Pharmaceutically active sulfonamide derivatives
04/05/2001WO2001023376A1 Isonipecotamides for the treatment of integrin-mediated disorders
04/05/2001WO2001023375A2 Substituted pyridines and pyridazines with angiogenesis inhibiting activity
04/05/2001WO2001023364A1 Quinazolinones
04/05/2001WO2001023362A2 Rate-controlled particles
04/05/2001WO2001023361A1 Pyrimidine derivatives, process for preparing the derivatives and drugs containing the same as the active ingredient
04/05/2001WO2001023360A1 Aryl sulfonamide-substituted benzimidazol derivatives thereof as tryptase inhibitors
04/05/2001WO2001023357A2 Fused cycloheptane and fused azacycloheptane compounds and their use as integrin receptor antagonists
04/05/2001WO2001023353A2 Method for producing indole derivatives on a solid phase
04/05/2001WO2001022966A1 Caspases and apoptosis
04/05/2001WO2001022950A2 Diosolane nucleoside analogs for the treatment or prevention of viral infection
04/05/2001WO2000073284A3 1,4-benzodiazepin-2-ones useful as hiv reverse transcriptase inhibitors
04/05/2001WO2000068198A3 Heterosubstituted pyridine derivatives as pde 4 inhibitors
04/05/2001WO2000066580A3 Antifungal ethers
04/05/2001WO2000044362A3 The use of 4-h-1-benzopyran-4-one derivatives as inhibitors of smooth muscle cell proliferation
04/05/2001DE19955087A1 Solid phase synthesis of indole derivatives comprises bonding of the indole nitrogen to a solid phase having vicinal diol groups by trans-acetalization of dialkoxymethyl protected indoles.
04/05/2001DE19947440A1 1-Aziridino-1-hydroxyiminomethyl-Derivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel 1-Aziridino-1-hydroxyiminomethyl derivatives, processes for their preparation and medicaments containing these compounds
04/05/2001CA2386092A1 Piperidine derivatives
04/05/2001CA2386085A1 Piperidine derivatives
04/05/2001CA2386074A1 Method for producing indole derivatives on a solid phase
04/05/2001CA2385918A1 Quinazolinones
04/05/2001CA2385349A1 Method for the treatment or prevention of viral infection using nucleoside analogues
04/05/2001CA2385292A1 Pyrimidine compounds, processes for the preparation thereof and pharmaceutical compositions comprising the compounds as active ingredient
04/05/2001CA2352957A1 Isonipecotamides for the treatment of integrin-mediated disorders
04/04/2001EP1088821A1 Pharmaceutically active sulfonamide derivatives
04/04/2001EP1088819A2 6-azauracil derivatives as thyroid receptor ligands
04/04/2001EP1088818A1 Quinolin-4-yl derivatives
04/04/2001EP1087964A1 N-benzodioxanylmethyl-1-piperidyl-methylamine compounds having affinity for 5-ht receptors
04/04/2001EP1087963A1 Inhibitors of glycogen synthase kinase 3
04/04/2001EP1087961A1 Phenoxylpropanolamines, method for the production thereof and pharmaceutical compositions containing the same
04/04/2001EP1087959A1 Novel benzopyran or thiobenzopyran derivatives
04/04/2001EP1087948A1 2,4-diamino-1,3,5-triazine, method for the production and use of the same as herbicides and plant growth regulators
04/04/2001EP1087946A1 Aryl alkanoylpyridazines
04/04/2001EP1087938A1 Inhibitors of neuraminidases
04/04/2001EP1087937A1 Cyclic hydroxamic acids as metalloproteinase inhibitors
04/04/2001EP1087766A1 Method of treatment
04/04/2001EP1087662A1 Composition for keeping away vermin
04/04/2001EP0636127B1 Disubstituted acetylenes bearing heterobicyclic groups and heteroaromatic or phenyl groups having retinoid like activity
04/04/2001CN1290266A Benzofuran-4-carboxamides and their therapeutical use
04/04/2001CN1290265A Thrombin receptor antagonists
04/04/2001CN1290264A Triazine angiogenesis inhibitors
04/04/2001CN1290263A Arylpiperidine derivatives and use thereof