Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
11/2000
11/08/2000EP1049671A1 Azetidinecarboxamide derivatives for the treatment of cns disorders
11/08/2000EP1049472A1 Antagonists of gonadotropin releasing hormone
11/08/2000EP0769006B1 Small molecule inhibitors of rotamase enzyme activity
11/08/2000CN1272842A 2-acylaminopropanamines as tachykinin receptor antagonists
11/08/2000CN1272841A Novel lactam metalloprotease inhibitors
11/08/2000CN1272493A Novel amino-triazole compound, its preparation method and drug composition containing them
11/08/2000CN1058262C Novel 1-phenylalkanone 5-HT4 receptor ligands
11/07/2000US6143909 Epoxidation; producing cryptophycin compounds having an epoxide functionality
11/07/2000US6143907 3-phenyl-1-methylenedioxyphenyl-indane-2-carboxylic acid derivatives
11/07/2000US6143892 Process for making 5-substituted pyrazoles
11/07/2000US6143780 Compounds for treatment of aids containing furan or thiophene groups
11/07/2000US6143779 Benzofuranone derivatives and a method for producing them
11/07/2000US6143774 Imidazole n-benzyldioxol derivatives, method for preparing same, resulting intermediates, pharmaceutical compositions and use of said derivatives as endothelin antagonists
11/07/2000US6143766 Benzopyranone and quinolone inhibitors of ras farnesyl transferase
11/07/2000US6143764 Quinoline and quinazoline derivatives inhibiting platelet-derived growth factor receptor autophosphorylation and pharmaceutical compositions containing the same
11/07/2000US6143762 Tetrahydroisoquinoline derivatives and their pharmaceutical use
11/07/2000US6143751 Pyridine derivatives and pharmaceutical compositions containing them
11/07/2000US6143747 Bis-sulfonamide hydroxyethylamino retroviral protease inhibitors
11/07/2000US6143696 Substituted 4-(3-alkenylbenzoyl)pyrazoles
11/07/2000CA2179306C Dopamine receptor ligands
11/07/2000CA2156455C Glycinamide derivatives, processes for their preparation and medicines containing them
11/07/2000CA2083913C Piperazinyl-and piperidinyl-cyclohexanols
11/02/2000WO2000064891A1 Farnesyl transferase inhibitors having a pyrrole structure and process for preparation thereof
11/02/2000WO2000064888A1 Di-aryl acid derivatives as ppar receptor ligands
11/02/2000WO2000064885A1 Heteroaryl diazacycloalkanes, their preparation and use
11/02/2000WO2000064876A1 Tri-aryl acid derivatives as ppar receptor ligands
11/02/2000WO2000064874A2 Heterosubstituted pyridine derivatives as pde 4 inhibitors
11/02/2000WO2000064872A1 INHIBITORS OF c-JUN N-TERMINAL KINASES (JNK)
11/02/2000WO2000064445A1 Bicyclic acyl guanidine sodium/proton exchange inhibitors and method
11/02/2000WO2000038730A3 Use of a cyclooxygenase-2 inhibitor and one or more antineoplastic agents for combination therapy in neoplasia
11/02/2000WO2000037464A3 4-(aminoalkoxy)benzofurans as n-myristoyltransferase inhibitors
11/02/2000EP1048658A1 Alicyclic acylated heterocyclic derivatives
11/02/2000EP1048640A1 Apoptosis inhibitors
11/02/2000EP1047979A2 Compound, composition and use
11/02/2000EP1047694A1 Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors
11/02/2000EP1047684A1 Substituted alpha,beta-anellated butyrolactones
11/02/2000EP1047678A1 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
11/02/2000EP1047675A1 Chemokine receptor antagonists and methods of use therefor
11/02/2000EP1047415A1 Pig appeasing pheromones to decrease stress, anxiety and aggressiveness
11/02/2000EP0808312B1 Indole derivatives as 5-ht receptor antagonist
11/02/2000DE19921086A1 New stable 6-alkenyl- or 6-alkynyl-epothilone derivatives, are cell division regulators useful for treating malignant tumors, angiogenesis or chronic inflammatory disease
11/02/2000CA2371308A1 Tri-aryl acid derivatives as ppar receptor ligands
11/02/2000CA2370607A1 Bicyclic acyl guanidine sodium/proton exchange inhibitors and method
11/02/2000CA2369092A1 Heterosubstituted pyridine derivatives as pde 4 inhibitors
11/02/2000CA2367695A1 Heteroaryl diazacycloalkanes, their preparation and use
11/01/2000CN1058010C Novel quinoline carboxylic acid derivatives having 7-(4-aminomethyl-3-oxime) pyrrolidine substituent and process for preparing thereof
11/01/2000CN1058008C Phenyl heterocycles as cyclooxygenase-2 inhibitors
10/2000
10/31/2000US6140513 Color forming dye precursor, composition containing the same and color forming heat-sensitive recording material
10/31/2000US6140361 For inhibiting binding of human immunodeficiency virus rev protein to rev responsive elements (rre)
10/31/2000US6140358 Substituted phenyl keto enols as pesticides and herbicides
10/31/2000US6140357 Small molecule inhibitors of rotamase enzyme activity
10/31/2000US6140352 Carbazolyl-substituted ethanolamines as selective β-3 agonists
10/31/2000US6140349 Cyclic amine modulators of chemokine receptor activity
10/31/2000US6140345 For treating psychoses and pain
10/31/2000US6140344 For treating pathological conditions such as asthma, rhinitis, eczema and parasitic infections featuring tissue eosinophilia
10/31/2000US6140340 Derivatives of 2-[3-phenyl-2-propenyl]-1,2,3,4-tetrahydro isoquinoline, their process and their use as fungicides
10/31/2000US6140338 For treating acute inflammatory diseases, chronic inflammatory diseases, acquired immune deficiency syndrome, cancer, ischemic reflow disorder and/or arteriosclerosis
10/31/2000US6140334 For treating high blood pressure, benign prostate hyperplasia
10/31/2000US6140331 For treating anxiety disorders, depression, psychosis, impulse control disorders, alcohol abuse, ischaemic diseases, cardiovascular disorders, side effects induced by conventional antipsychotic agents and senile dementia
10/31/2000US6140273 Herbicides; made by reacting a cyclohexane-1,3-dione with an activated benzoic acid or benzoic acid compound, to give an acylation product, and subsequent rearrangement
10/31/2000US6140272 Substituted 4-benzoyl-pyrazoles
10/31/2000US6140271 1-alkyl-4-benzoyl-5-hydroxypyrazole compounds and their use as herbicides
10/26/2000WO2000063207A1 Pesticidal indazole or benzotriazole derivatives
10/26/2000WO2000063204A2 Substituted azoles
10/26/2000WO2000063198A1 2,2-disubstituted cyclic ether derivatives and hair tonics containing the same
10/26/2000WO2000063171A1 Tricyclic compounds
10/26/2000WO2000063165A1 Mmp inhibitor
10/26/2000WO2000062765A2 ESTROGEN RECEPTOR-β LIGANDS
10/26/2000WO2000039120A3 Compounds and methods for modulation of estrogen receptors
10/26/2000WO2000035886A3 (hetero)aryl-bicyclic heteroaryl derivatives, their preparation and their use as protease inhibitors
10/26/2000CA2370417A1 Substituted azoles
10/26/2000CA2370265A1 Pesticidal indazole or benzotriazole derivatives
10/26/2000CA2370126A1 Estrogen receptor-.beta. ligands
10/25/2000EP1045846A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof
10/25/2000EP1045842A2 Methods of use and compositions for benzylidene- and cinnamylidene-anabaseines
10/25/2000EP1045839A2 Novel amines as pharmaceutical agents
10/25/2000EP1045836A1 Pyridones as src family sh2 domain inhibitors
10/25/2000EP1045834A1 4(3)substituted-4(3)-aminomethyl-(thio)pyran or -piperidine derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
10/25/2000EP1045833A1 2,3-substituted indole compounds as cox-2 inhibitors
10/25/2000CN1271357A bisethers of 1-oxa, aza and thianaphthalen-2-ones as phospholamban inhibitors
10/25/2000CN1271356A Tetrahydrofuran phosphate- and hydroxy esters, as prodrugs for corresponding antifungal agent
10/25/2000CN1271352A Process for making 3-aryloxy, 4-arylfuran-2-ones useful as inhibitors of cox-2
10/25/2000CN1271349A Substituted quinazoline derivatives and their use as tyrosine kinase inhibitors
10/25/2000CN1271346A Method for producing substituted 2-nitroguanidine derivative
10/25/2000CN1271345A Method for producing substituted 2-nitroguanideine derivatives
10/24/2000US6137002 Glycoprotein IIb/IIIa antagonists
10/24/2000US6136977 Processes for producing phenoxy propionic acid derivatives
10/24/2000US6136969 Azepanes
10/24/2000US6136848 Antiallergens; asthma therapy
10/24/2000US6136844 5-aroylpyrrol-2-ylmethylarene derivatives
10/24/2000US6136843 Indole derivatives useful as endothelin receptor antagonists
10/24/2000US6136842 Sulphur derivatives comprising an amide bond, method for preparing same, use thereof as drugs, and pharmaceutical compositions containing such derivatives
10/24/2000US6136832 Racemic mixtures and enantiomorphs
10/24/2000US6136826 Aminopiperidine compounds substituted with alkanoyl
10/24/2000US6136825 Sulfonamide compounds having 5-HT receptor activity
10/24/2000US6136824 1-piperidinyl-propan-2-derivatives and their use as therapeutic agents
10/24/2000US6136822 Quinolinone derivative, method for preparing the same, and anti-allergic agent
10/24/2000US6136812 Methods of administering AMPA receptor antagonists to treat dyskinesias associated with dopamine agonist therapy
10/24/2000US6136808 Antitumor agents from plants
10/19/2000WO2000061579A1 New endothelin converting enzyme inhibitors, their production and their use