Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
09/2001
09/20/2001WO2001068591A1 Carboxylic acid derivatives as ip antagonists
09/20/2001WO2001068585A1 Novel amide compounds
09/20/2001WO2001068063A2 Novel use of (r)-(-)-2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]-chromane and its physiologically acceptable salts
09/20/2001WO2001034591A3 Substituted 4h-chromene and analogs as activators of caspases and inducers of apoptosis and the use thereof
09/20/2001WO2001014369A3 Process for the preparation of paroxetin.hcl
09/20/2001US20010023292 3-((3,5-difluoro-6-(3-(1-methylimidazolin-2-yl)phenoxy)-4 -(2,3 -dihydroxypropoxy)pyridin-2-yl)oxy)-4-hydroxybenzamidine, for example
09/20/2001US20010023291 Polyhydroxylated monocyclic N-heterocyclic derivatives as anti-coagulants
09/20/2001US20010023253 Novel compound
09/20/2001US20010023250 Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p56lck tyrosine kinases
09/20/2001DE10013126A1 New 6-aminoalkyl-dihydropyrimidine-5-carboxylate ester derivatives, useful as antiviral agents having strong activity against hepatitis B virus and low cytotoxicity
09/20/2001CA2403149A1 2-phenylpyran-4-one derivatives
09/20/2001CA2402402A1 Use of (r)-(-)-2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]-chromane for treating adverse effects of anti-parkinsonian drugs
09/20/2001CA2373411A1 5-substituted arylpyrimidines
09/19/2001EP1134214A1 Picolinamide derivatives and pest controllers containing the same as the active ingredient
09/19/2001EP1133492A1 Process for the preparation of paroxetine hydrochloride
09/19/2001EP1133491A1 Novel benzofurane derivatives, preparation method, use as medicines and pharmaceutical compositions containing same
09/19/2001EP1133489A1 Isonipecotamides for the treatment of integrin-mediated disorders
09/19/2001EP1133488A1 Propanoic acid derivatives as integrin inhibitors
09/19/2001EP1133484A2 Heterocyclic derivatives and their use as integrin inhibitors
09/19/2001EP1133483A1 Il-5 inhibiting 6-azauracil derivatives
09/19/2001EP1133481A1 Quinoline and quinoxaline compounds as pdgf-r and/or lck tyrosine kinase inhibitors
09/19/2001EP1133480A1 Quinoline and quinoxaline compounds as pdgf-receptor and/or lck tyrosine kinase inhibitors
09/19/2001EP1133479A1 Quinoline and quinoxaline compounds
09/19/2001EP1133475A1 Substituted benzo de]isoquinoline-1,3-diones
09/19/2001EP0869952B1 5-naphthalen-1-yl-1,3-dioxane derivatives, preparation and therapeutical use thereof
09/19/2001EP0839144B1 Piperazine derivatives as therapeutic agents
09/19/2001EP0800516B1 FIBRINOGEN RECEPTOR ANTAGONISTS HAVING SUBSTITUTED (b)-AMINO ACID RESIDUES AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME
09/19/2001EP0612244B1 Endothelin receptor antagonists
09/19/2001CN1313855A Inhibitors of alpha4Betal mediated cell adhesion alpha Beta
09/19/2001CN1313854A Antiviral pyrimidinedione derivatives and process for the preparation thereof
09/19/2001CN1313853A Oxindole derivatives as growth hormone releasers
09/19/2001CN1313284A N-(3-benzofuryl) urea derivative
09/19/2001CN1313280A Benzheterocyclic derivatives
09/19/2001CN1071332C Enterokinetic benzamide
09/19/2001CN1071331C Anti-helicobacter acyl derivatives of azolones
09/18/2001US6291687 Used aspartyl protease inhibitors of human immunodeficiency virus (hiv)
09/18/2001US6291683 N-arloxyethyl-alkylamines for the treatment of depression
09/18/2001US6291679 Process for preparing benzoperhydroisoindole compounds
09/18/2001US6291672 Human NK3 receptor-selective antagonist compounds, method for obtaining them and pharmaceutical compositions containing them
09/18/2001US6291510 Small molecule inhibitors of rotamase enzyme activity
09/18/2001US6291508 Potent ability to bind to retinoic acid receptors thus useful in treating psoriasis and rheumatoid arthritis.
09/18/2001US6291500 Administering an antifungal agent
09/18/2001US6291499 2-cyclohexyl benzimidazole NMDA/NR2B antagonists
09/18/2001US6291489 Process for substituted pyridines
09/18/2001US6291485 Treatment of post-ptca restenosis
09/18/2001US6291482 N-hydroxyurea derivative and pharmaceutical composition containing the same
09/18/2001US6291481 Conditions related to a hampered or impaired gastric emptying and more generally to treat conditions related to a hampered or impaired gastrointestinal transit.
09/18/2001US6291480 Diaryl piperidyl pyrrole derivatives as antiprotozoal agents
09/18/2001US6291476 Pyrazole carboxamides useful for the treatment of obesity and other disorders
09/18/2001US6291456 Compounds and methods for modulation of estrogen receptors
09/18/2001US6291451 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
09/18/2001US6289745 High temperature insertion type flow element and mounting extension
09/18/2001CA2236814C Quinoline and quinazoline compounds useful in therapy
09/13/2001WO2001066539A1 Imidazol derivatives as raf kinase inhibitors
09/13/2001WO2001066534A2 Cyclic and bicyclic diamino histamine-3 receptor antagonists
09/13/2001WO2001066523A1 6-chloro-3-pyridylmethylpropylamine derivatives, preparation process thereof and bactericides
09/13/2001WO2001066521A1 Azacyclic compounds for use in the treatment of serotonin related diseases
09/13/2001WO2001066520A1 Indole derivatives, process for preparation of the same and use thereof
09/13/2001WO2001066114A1 Novel methods using cholinesterase inhibitors
09/13/2001WO2001009138A3 Chemokine receptor antagonists and methods of use therefor
09/13/2001US20010021776 Spray drying
09/13/2001US20010021719 2-phenyl-1- [4- (2-aminoethoxy) - benzyl] - indoles as estrogenic agents
09/13/2001US20010021715 Gastrointestinal disorders
09/13/2001US20010021709 Integrin inhibitors used to treat circulatory disorders, for thrombosis, myocardial infarct, coronary heart disease, arteriosclerosis, osteoporosis, pathological processes maintained or propagated by angiogenesis and tumor therapy
09/13/2001US20010021708 Acylurea compound containing imidazolidine ring
09/13/2001DE19954228A1 New epothilone derivatives used for treating e.g. malignant melanoma, breast carcinoma, psoriasis, multiple sclerosis and arthritis
09/13/2001CA2402174A1 Indole derivatives, process for preparation of the same and use thereof
09/12/2001EP1132379A1 Novel thiol derivatives, process for producing the same and utilization thereof
09/12/2001EP1131318A1 Process for making 5-substituted pyrazoles using dithietanes
09/12/2001EP1131315A1 Polyhydroxylated heterocyclic derivatives as anti-coagulants
09/12/2001EP1131291A1 4-aroyl-piperidin-ccr-3 receptor antagonists iii
09/12/2001EP1131288A1 Pyrrolidine derivatives-ccr-3 receptor antagonists
09/12/2001EP1044200A4 Preparation of terazosin hydrochloride dihydrate
09/12/2001EP0891354B1 N-aminoalkyldibenzofurancarboxamides as dopamine receptor subtype specific ligands
09/12/2001EP0888317B1 Substituted 4-hydroxy-phenylalcanoic acid derivatives with agonist activity to ppar-gamma
09/12/2001EP0863141B1 Substituted heteroaromatic derivatives
09/12/2001EP0832066B1 Substituted n-(indole-2-carbonyl-) amides and derivatives as glycogen phosphorylase inhibitors
09/12/2001EP0794945B1 Iminooxybenzylcrotonic acid esters, process for their preparation and use thereof
09/12/2001CN1312807A Inhibitors of glycogen synthase kinase 3
09/12/2001CN1312803A Novel benzopykan or thiobenzopyran derivatives
09/12/2001CN1312799A Bispiperidines as antithrombotic agents
09/12/2001CN1312733A Reactor comprising a contact tube bundle
09/12/2001CN1070701C Pyrimidine ortriazine carboxylic acid derivatives to be used as medicaments
09/11/2001US6288247 Catalytic multistage process forming a racemic mixture of compounds
09/11/2001US6288234 Fluorinated heterocyclic amido amine compounds as drugs
09/11/2001US6288230 2-(2, 3-dihydrobenzofuran-5-yl)-4-aminomethylimidazoles: dopamine receptor subtype specific ligands
09/11/2001US6288228 Triazine angiogenesis inhibitors
09/11/2001US6288102 Substituted phenylketoenols and their use as pesticides and herbicides
09/11/2001US6288092 Triaryl compounds
09/11/2001US6288085 Piperidine derivatives for treating psychoses
09/11/2001US6288084 Administering comounds such as 4-(4-chlorophenyl)-1-(4-(3-methoxyphenyl)-4-(3-pyridinyl)-3 -butenyl)piperidin-4-ol to treat diseases associated with aberrant leukocyte recruitment and/or activation
09/11/2001US6288083 Chemokine receptor antagonists and methods of use therefor
09/11/2001US6288068 Administering 1,4-disubstited piperidine derivative; alzheimer*s disease, cognition activators; anticholinergic agents
09/11/2001US6288066 Antidiabetic agents; oxidation, hydrolysis
09/11/2001US6288059 Acylated hetero-alicyclic derivatives
09/11/2001US6288058 Treating muscular, nervous system, psychological and gastrointestinal disorders
09/11/2001CA2217171C New process for preparing (-)-trans-n-p-fluorobenzoylmethyl-4-(p-fluorophenyl)-3-¢¢3,4-(methylenedioxy)phenoxy!methyl!-piperidine
09/11/2001CA2200742C Quinoxaline derivatives useful in therapy
09/11/2001CA2115426C Novel cyclic ureas useful as antiarrhythmic and antifibrillatory agents
09/07/2001WO2001064676A2 INHIBITORS OF p38-α KINASE