Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
02/2004
02/18/2004EP1389461A1 Pyrimidones with antiviral properties
02/18/2004EP1389460A1 Cxcr4-antagonistic drugs comprising nitrogen-containing compound
02/18/2004EP1389202A1 2,6-substituted chroman derivatives useful as beta-3 adrenoreceptor agonists
02/18/2004EP1389201A1 N-oxide anthranylamide derivatives and their use as medicaments
02/18/2004EP1389194A2 Inhibitors of bace
02/18/2004EP1389110A2 Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
02/18/2004EP1389103A2 Synthesis and evaluation of novel phthalimide mimics as anti-angiogenic agents
02/18/2004EP1178958B1 N-cyanomethyl amides as protease inhibitors
02/18/2004EP1049691B1 Substituted 5-(2,2-difluoro-1,3-benzodioxol-5-yl) cyclopentenopyridine derivative
02/18/2004EP0716088B1 Process for producing 2-(tetrazol-5-yl)-4-oxo-4h-benzopyrans
02/18/2004CN1476442A Pyridine derivatives with IKB-kinase (IKK-beta) INhibiting activity
02/18/2004CN1476436A Novel compounds for use as HIV protease inhibitors
02/18/2004CN1476430A Delta 1-pyrrolines used as pesticides
02/18/2004CN1476429A EP4 receptor selective agonists in treatment of osteoporosis
02/18/2004CN1138774C Substituted 6,6-hetero-bicyclic derivatives
02/18/2004CN1138773C 4-alkenyl (and alkynyl) oxindoles as inhibitors of cell cycle protein dependent kinases, in particular CDK2
02/18/2004CN1138546C Certain 1,4,5-tri-substituted imidazole compounds useful as cytokine
02/17/2004US6693201 1,3-dimethyl-2-indolylmethlene(isopropylidene)succinic anhydrides
02/17/2004US6693200 2-(substituted-phenyl)amino-imidazoline derivatives
02/17/2004US6693194 By reacting 4,6-dichloro-2-(methylthio)pyrimidine in an inert organic solvent with an alkali metal methoxide, transferring to an aqueous acid medium and oxidation; using the product to prepare 7-((4,6-
02/17/2004US6693190 Tetraazacyclododecane macrocycle derivatives including metal complexes; magnetic resonance imaging agents
02/17/2004US6693123 (4-(3-pyridylaminomethylene)-2-phenylbenzoyl)-n -methylmethionine, methyl ester for example; restenosis, hyperplasia
02/17/2004US6693121 As inhibitors of serine proteases of the coagulation cascade and compounds, used for anticoagulant therapy forprophylaxis of a variety of thrombotic conditions including coronary artery and cerebrovascular diseases
02/17/2004US6693118 E.G., 1-(2-(6,7-METHYLENEDIOXYNAPHTH-2-YL)-ETHYL)-4-(3-TRIFLUOROMETHYLPHENYL)-1,2,3,6-TETRAHYDROPYRIDINE AND 1-2-(4-CYCLOHEXENYLPHENYL)-ETHYL)-4-(3-TRIFLUOROMETHYLPHENYL)-1,2,3,6 -TETRAHYDROPYRIDINE; apoptosis inhibition; treatment of graft rejection or of acute or chronic rheumatoid arthritis
02/17/2004US6693117 Compounds with analgesic effect
02/17/2004US6693101 Alkanoic acid derivative; integrin receptor antagonist
02/17/2004US6693099 Substituted piperazine compounds optionally containing a quinolyl moiety for treating multidrug resistance
02/17/2004US6693098 Carboxylic acid or tetrazole derivatives containing carbamate groups are useful for treating the conditions associated with the urinary tract, pain, inflammation, respiratory states, edema formation of hypotensive vascular diseases
02/17/2004US6692657 Alkenyl compound with 2,3-difluorophenyl group
02/17/2004CA2302965C Processes and intermediates for preparing anti-cancer compounds
02/17/2004CA2290918C Heteroaromatic bicyclic derivatives useful as anticancer agents
02/17/2004CA2280279C Indole, indazole and benzimidazole derivatives as antithrombotic agents
02/17/2004CA2124680C Piperazine derivatives as 5-ht1a antagonists
02/12/2004WO2004013135A1 2-phenylpyridin-4-yl derivatives as alk5 inhibitors
02/12/2004WO2004013129A1 4-trifluoromethylpyrazolyl substituted pyridines and pyrimidines
02/12/2004WO2004013125A1 Pyridinyl substituted (1,2,3,)triazoles as inhibitors of the tgf-beta signalling pathway
02/12/2004WO2004013120A1 Novel benzodioxoles
02/12/2004WO2004013104A1 Novel tetrahydroquinoline derivatives
02/12/2004WO2004013098A1 Novel gamma-lactams as beta-secretase inhibitors
02/12/2004WO2004012736A1 Biaryl compounds having anti-infective activity
02/12/2004WO2004012735A2 New effector conjugates, process for their production and their pharmaceutical use
02/12/2004WO2004012663A2 Hydantoin derivatives as inhibitors of matrix metalloproteinases and/or tnf-alpha converting enzyme
02/12/2004WO2004012656A2 Thiophene and furan derivatives as prostaglandin agonists and use thereof
02/12/2004WO2004012649A2 Novel compounds for stimulation of nerve growth, for the inhibition of scar tissue formation and/or reduction of secondary damage
02/12/2004WO2004012648A2 Substituted diaryl heterocycles, method for the production and use thereof as medicaments
02/12/2004WO2003103604A3 Gamma lactams as prostaglandin agonists and use thereof
02/12/2004WO2003049702A3 Vanilloid receptor ligands and their use in treatments
02/12/2004US20040030156 Substituted amino-furan-2-yl-acetic acid and amino-thien-2-yl-acetic acid derivatives and their use in the treatment of migraine and pain
02/12/2004US20040030138 Process for 8-carboxamido-2,6-methano-3-benzazocines
02/12/2004US20040029935 Heterocyclic aromatic compounds useful as growth hormone secretagogues
02/12/2004US20040029920 2-(biarylalkyl)amino-3-(heterocyclylcarbonylamino)-pyridine derivatives
02/12/2004US20040029919 Respiratory system disorders; bronchitis; irritable bowel disorders; incontinence
02/12/2004US20040029902 2,4-Pyrimidinediamine compounds and their uses
02/12/2004US20040029901 Obesity therapy; administering orlistat
02/12/2004US20040029898 Anticancer agents
02/12/2004US20040029897 Frangible compounds for pathogen inactivation
02/12/2004US20040029887 Cardiovascular disorders; antiinflammatory agents; central nervous system diosrders; psychological disorders
02/12/2004US20040029883 Beta-amino acid compounds as integrin antagonists
02/12/2004US20040029880 Anthranyl amides and their use as medicaments
02/12/2004US20040029875 Novel aminotriazolone compounds, method for preparing same and pharmaceutical compositions containing same
02/12/2004US20040029874 Anticoagulants; cardiovascular disorders
02/12/2004US20040029861 Using compound containing pyridine ring
02/12/2004US20040029857 Anticancer agents; central nervous system disorders; antiinflamamtory agents
02/12/2004DE10234975A1 New effector conjugates of epithilones useful to treat e.g. diseases associated with proliferative processes, neurodegenerative diseases, multiple sclerosis, Alzheimer's disease and rheumatoid arthritis
02/12/2004DE10233817A1 Substituierte Diarylheterocyclen, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel Substituted Diarylheterocyclen, processes for their preparation and their use as medicaments
02/12/2004DE10233366A1 In 6-Stellung substituierte Indolinonderivate, ihre Herstellung und ihre Verwendung als Arzneimittel In the 6-position substituted indolinone derivatives, their preparation and their use as medicaments
02/12/2004DE10136131B4 Polyaminosäure-katalysiertes Verfahren zur enantioselektiven Epoxidierung von α,β-ungesättigten Enonen und α,β-ungesättigten Sulfonen Polyamino acid-catalyzed process for the enantioselective epoxidation of α, β-unsaturated enones and α, β-unsaturated sulfones
02/12/2004CA2494139A1 Biaryl compounds having anti-infective activity
02/12/2004CA2493749A1 4-trifluoromethylpyrazolyl substituted pyridines and pyrimidines
02/12/2004CA2492437A1 New effector conjugates, process for their production and their pharmaceutical use
02/11/2004EP1388342A1 Acylated, heteroaryl-condensed cycloalkenylamines and their use as pharmaceuticals
02/11/2004EP1387841A1 Novel azole or triazole derivatives, method for preparing same and use thereof as fungicides
02/11/2004EP1387838A1 Cyanoanthranilamide derivatives and the use thereof as medicaments
02/11/2004EP1387836A1 Phthalazine derivatives with angiogenesis inhibiting activity
02/11/2004EP1387833A1 Protease-inhibitors
02/11/2004EP1387679A1 Sulfonamides
02/11/2004EP1387674A2 Hedgehog antagonists, methods and uses related thereto
02/11/2004EP1299356B1 Novel compounds
02/11/2004EP1183251B1 Indolylpiperidine derivatives as antihistaminic and antiallergic agents
02/11/2004EP1042300B1 Phthalazine derivatives useful as phosphodiesterase 4 inhibitors
02/11/2004EP1034169B1 Trisaryl-1,3,5-triazine ultraviolet light absorbers
02/11/2004EP1006110B1 Derivatives of acyl-piperazinil-pyrimidins, preparation thereof and application as medicaments
02/11/2004EP0936912B1 Inhibitors of cysteine protease
02/11/2004CN1474816A 4-amino-quinazolines
02/11/2004CN1474815A 4-amino-quinazolines
02/11/2004CN1474813A Substituted 2-phenylaminomidazoline phenyl ketone derivatives as IP antagonists
02/11/2004CN1474803A Novel amide derivatives and medicinal use thereof
02/11/2004CN1474703A Taxoid conjugates as antimitotic and antitumor agents
02/11/2004CN1474691A Novel uses of combined 5-HT 1A agonists and serotonin reuptake inhibitor
02/11/2004CN1474688A Novel uses of combined selective dopamine D2 receptor antagonists and 5-HT1A receptor agonists
02/11/2004CN1474652A Substituted 4,5-dihydro-1,2,4-triazin -6-ones, 1,2,4-triazin-6-ones, and their use as fungicides and insecticides
02/11/2004CN1473814A Intemediate for preparing alkyl-dihalogeno phenyl substituted keto-enol
02/11/2004CN1137886C Novel 2,3-dioxo-1,2,3,4-tetrahydro-quinoyxalinyl derivatives
02/11/2004CN1137884C Indazole compounds and pharmaceutical compositions for inhibiting protein kinases and methods for their use
02/10/2004US6689889 Using n-acryloxyphenylaniline neomenthylamide
02/10/2004US6689883 Substituted pyridines and pyridazines with angiogenesis inhibiting activity
02/10/2004US6689801 Certain heteroaryl substituted thiol inhibitors of endothelin-converting enzyme
02/10/2004US6689799 Non-nucleoside-derivative viricides
02/10/2004US6689798 Benzofuran derivatives
02/10/2004US6689797 Tetrahydropyridines, preparation method and pharmaceutical compositions containing same