Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
03/2004
03/11/2004US20040048844 Acylsemicarbazides as cyclin dependent kinase inhibitors useful as anti-cancer and anti-proliferative agents
03/11/2004US20040048843 And aza- and diaza-derivatives thereof; especially treating allergy or nasal congestion
03/11/2004US20040048797 Regulation of TNF-alpha
03/11/2004DE10236910A1 Substituierte 1,2,3,4-Tetrahydrochinolinderivate Substituted 1,2,3,4-tetrahydroquinoline
03/11/2004CA2496887A1 Oxytocin inhibitors
03/11/2004CA2495853A1 2,5-dioxoimidazolidin-4-yl acetamides and analogues as inhibitors of metalloproteinase mmp12
03/11/2004CA2495248A1 Anabaseine derivatives useful in the treatment of neurodegenerative diseases
03/11/2004CA2488739A1 Nitrogen-containing aromatic derivatives
03/10/2004EP1396490A1 3-quinoline-2-(1h)-ylideneindolin-2-one derivatives
03/10/2004EP1396489A1 Heteroaromatic bicyclic derivatives useful as anticancer agents
03/10/2004EP1396487A1 Phenylpyridine carbonyl piperazine derivative
03/10/2004EP1395606A1 Pyrrolidin-2-one derivatives as inhibitors of factor xa
03/10/2004EP1395578A1 Carbazole derivatives and their use for the preparation of pharmaceutical compositions for the treatment of npy related diseases
03/10/2004EP1395576A1 4-(phenyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395575A1 4-(penyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395574A1 4-(phenyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395571A1 Compounds and methods for the treatment or prevention of flavivirus infections
03/10/2004EP1395568A1 4-aminopyrimidine derivatives
03/10/2004EP1395565A1 Herbicidal substituted benzoylpyrazoles
03/10/2004EP1395564A1 Quinoline derivatives as ligands for the neuropeptide y receptor
03/10/2004EP1395561A1 Carbamate and oxamide compounds as inhibitors of cytokine production
03/10/2004EP1395559A1 4-(phenyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain anxiety or gastrointestinal disorders
03/10/2004EP1395558A1 4-(phenyl-(piperidin-4-yl)-amino)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395557A1 4-(phenyl-(piperidin-4-yl)-amino)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395556A1 4-(phenyl-(piperidin-4-yl)-amino)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395555A1 4-(phenyl-(piperidin-4-yl)-amino)-benzamide derativatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395256A2 Prodrugs via acylation with cinnamate
03/10/2004EP1136477B1 Benzofuran derivatives, process for the preparation of the same and uses thereof
03/10/2004EP1081132B1 Hydroxamic acid derivatives and medicinal utilization thereof
03/10/2004EP0804435B1 Novel imidazole derivatives, method for preparing same, novel intermediates thus obtained, medicinal applications of same and pharmaceutical compositions containing same
03/10/2004CN1481380A Novel benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists
03/10/2004CN1481377A Cyclic Beta-amino acid derivatives as inhibitors of matrix metalloproteases and TNF alhpa
03/10/2004CN1481376A Oxybenzamides derivatives as factor xa inhibitors
03/10/2004CN1481370A Quinazoline derivatives, medicaments contg. said compounds, their utilization and method for prodn. thereof
03/10/2004CN1481368A Gyrase imhibitors and uses thereof
03/10/2004CN1481363A N-alkoxy-4, 4-dioxy-polyalkyl-piperidines as polymerisation in hibitors
03/10/2004CN1481361A Piperidine MCH antagonists and their use in treatment of obesity
03/10/2004CN1481360A 蕈毒碱拮抗剂 Muscarinic antagonist
03/10/2004CN1481358A Carboxylic acid amide derivatives and their use in treatment of thromboembolic diseases and tumours
03/10/2004CN1480451A Photoactive compound used as intermediate for preparing photoactive 2-imidazoline-5-ketone or 2-imdazoline-5-thio-ketone derivative
03/10/2004CN1141298C Carbostyril derivs. for inhibiting skin erythema and/or skin pigmentation
03/10/2004CN1141295C Indoline derivatives as progesterohe antagonists
03/09/2004USRE38460 Huperzine A derivatives, their preparation and their use
03/09/2004US6703525 Antiinflammatory agents; coupling sulfonyl halide with aromatic amine compound
03/09/2004US6703510 More stable and durable; automotive coatings, candle wax
03/09/2004US6703509 Reduction of 5-arylnicotinic acids by catalytic hydrogenation in the presence of carboxylic anhydrides in which the catalyst used is a palladium/ligand complex to produce aryinicotinaldehydes
03/09/2004US6703506 Amino acid ester containing azole antifungals
03/09/2004US6703503 Pyridazin-3-one derivatives, their use, and intermediates for their production
03/09/2004US6703408 N-formyl derivatives of paroxetine
03/09/2004US6703397 Pyrimidinyl methyl indole derivatives with antibacterial activity
03/09/2004US6703396 Cis-4-amino-5-fluoro-1-(2-hydroxymethyl-1,3-oxathiolane-5-yl) -(1h)-pyrimidin-2-one
03/09/2004US6703387 Inhibitors of HPV E1 helicase enzyme
03/04/2004WO2004018486A1 Azole derivatives as antifungal agents
03/04/2004WO2004018485A1 Azole derivatives as antifungal agents
03/04/2004WO2004018461A2 Antibacterial benzoic acid derivatives
03/04/2004WO2004018460A1 Amino methyl imidazoles as c5a receptor modulators
03/04/2004WO2004018458A1 2-thio-substituted imidazole derivatives and their use in pharmaceutics
03/04/2004WO2004018457A1 Pyrrolidinedione substituted piperidine-phthalazones as pde4 inhibitors
03/04/2004WO2004018455A1 Pyrrole based inhibitors of glycogen synthase kinase 3
03/04/2004WO2004018452A1 Pyrimidine derivatives as selective cox-2 inhibitors
03/04/2004WO2004018451A1 Pyridazinone-derivatives as pde4 inhibitors
03/04/2004WO2004018450A1 Piperidine-n-oxide-derivatives
03/04/2004WO2004018438A2 Microbiocidal (e.g. fungicidal) 1,2,3-triazole derivatives
03/04/2004WO2004018433A1 Pyrimidine derivatives and their use as cb2 modulators
03/04/2004WO2004018429A2 Substituted hihydroquinolines as glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
03/04/2004WO2004018428A1 Antibacterial benzoic acid derivatives
03/04/2004WO2004018420A1 Indolylalkylamino-methylidenecarbamate derivatives useful as gnrh antagonists
03/04/2004WO2004018419A2 Benzimidazole quinolinones and uses thereof
03/04/2004WO2004018414A2 Antibacterial agents
03/04/2004WO2004017974A1 Piperidine-pyridazones and phthalazones as pde4 inhibitors
03/04/2004WO2004017961A2 Derivatives of 3-hydroxy-4-(cyclyl-alkylaminoalkyl)-5-phenyl-1h-pyrazole as antagonists of the gonadotropin releasing hormone (gnrh) for use in the treatment of sex hormone related conditions, such as prostatic of uterine cancer
03/04/2004WO2004017911A2 Protease inhibitors
03/04/2004WO2004005264A3 Imidazole compounds for the treatment of hepatitis c virus infections
03/04/2004WO2003094845A3 Pyridine-based thyroid receptor ligands
03/04/2004WO2003088917A3 Regulation of tnf-alpha
03/04/2004WO2003082350A3 Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands
03/04/2004WO2003024928A3 Novel aminoazetidine, -pyrrolidine and -piperidine derivatives
03/04/2004WO2003004464A8 Heterocyclic amide derivatives and the use thereof as pesticides
03/04/2004WO2002098856A3 Piperazine oxyquinoline (naphthaline) platelet adenosine diphosphate receptor antagonists
03/04/2004WO2002096867A3 Inhibitors of protein kinase for the treatment of disease
03/04/2004US20040044211 Substituted 4-phenyltetrahydroisoquinolinium, process for their preparation, their use as a medicament, and medicament containing them
03/04/2004US20040044204 Glycoprotein antagonist; anticholesterol agents; cardiovascular disorders; strokes; antiischemic agents
03/04/2004US20040044203 Anticancer agents
03/04/2004US20040044201 Bone disorders; osteoporosis; oral diseases; antiarthritic agents
03/04/2004US20040044075 Alpha acyloxyacetamides for kallikrein and urokinase inhibition
03/04/2004US20040044057 5- substituted tetralones as inhibitors of ras farnesyl trransferase
03/04/2004US20040044051 Cannabinoid receptor agonists
03/04/2004US20040044047 Alpha and beta-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
03/04/2004US20040044037 Sleep disorders; antidepressants; analgesics; central nervous system disorders
03/04/2004US20040044031 Controlling appetite; dietetics; sleep disorders
03/04/2004US20040044015 Quinazoline derivatives
03/04/2004US20040044014 Controlling signal transduction; tyrosine kinase inhibitors; benign prostatic hyperplasmia; respiratory system disorders; antitumor agents
03/04/2004US20040044003 Therapeutic agents useful for treating pain
03/04/2004US20040044000 Cardiovascular disorders; antiarthritic agents; inflammatory bowel disorders; vision defects; respiratory system disorders
03/04/2004US20040043999 Phthalazine derivatives as phosphodiesterase 4-inhibitors
03/04/2004US20040043989 Therapy for drug resistant bacteria; topoisomerase inhibitor
03/04/2004US20040043988 Cycloalkyl alkanoic acids as intergrin receptor antagonists
03/04/2004US20040043986 Cardiovascular disorders; inflammatory bowel disorders; antiarthritic agents; skin disorders; vision defects; osteoporosis
03/04/2004US20040043984 3,4-Dihydroquinolin-2-one, 5,6-fused oxazin-3-one, and 5,6-fused thiazin-3-one derivatives as matrix metalloproteinase inhibitors
03/04/2004US20040043983 Cardiovascular disorders; antiarthritic agents; inflammatory bowel disorders; vision defects; respiratory system disorders