Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
01/2004
01/08/2004DE10224844A1 Nicht-peptidische BRS-3-Agonisten Non-peptidic BRS-3 agonist
01/08/2004CA2491089A1 Compounds useful for the inhibition of aldh
01/08/2004CA2490138A1 Novel tetrahydropyridine derivatives as renin inhibitors
01/08/2004CA2489560A1 Substituted quinoline ccr5 receptor antagonists
01/08/2004CA2489433A1 Inhibitors of hcv ns5b polymerase
01/07/2004EP1378508A1 Various forms of paroxetine hydrochloride anhydrate
01/07/2004EP1378246A1 Remedies for arteriosclerosis
01/07/2004EP1377976A2 Optical data carrier that contains a merocyanine dye as the light-absorbing compound in the information layer
01/07/2004EP1377975A2 Optical data medium containing, in the information layer, a dye as a lightabsorbing compound and having a protective covering layer of predetermined thickness
01/07/2004EP1377971A1 Optical data carrier that contains a cationic aminoheterocyclic dye as the light-absorbing compound in the information layer
01/07/2004EP1377970A1 Optical data carrier containing a cyclizable compound in the information layer
01/07/2004EP1377570A1 Substituted 2-carba-3,5-dicyano-4-aryl-6-aminopyridines and the use of the same as selective ligands of the adenosine receptor
01/07/2004EP1377569A1 Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines with adenosine receptor-binding activity and their use as cardiovascular preparations
01/07/2004EP1377565A1 Tetrahydropyran derivatives as neurokinin receptor antagonists
01/07/2004EP1377564A2 Transition-metal-catalyzed process for the preparation of sterically hindered n-substituted alkoxyamines
01/07/2004EP1377556A1 Pyrazole derivatives for treating hiv
01/07/2004EP1377555A1 Novel compounds
01/07/2004EP1377553A1 Tetrahydroquinoline derivatives as stat6-modulators, preparation and use thereof
01/07/2004EP1377549A1 Functionalized heterocycles as modulators of chemokine receptor function and methods of use therefor
01/07/2004EP1377293A1 Aryl and biaryl piperidines used as mch antagonists
01/07/2004EP1377290A2 Malonyl-coa decarboxylase inhibitors useful as metabolic modulators
01/07/2004EP1377283A2 Compounds of the formula r1-x-y-z-nr2r3 as abca-1 elevating agents against coronary artery disease or atherosclerosis
01/07/2004EP1056733B1 Histamine h3 receptor ligands
01/07/2004CN1466577A 3,4-dihydroisoquinoline derivative compounds and drugs containing these compounds as the active ingredient
01/07/2004CN1133634C Heterocyclic derivatives which inhibit factor Xa
01/07/2004CN1133372C Insecticidal N-(substituted arylmethyl)-4-[bis(substituted phenyl or pyridyl)methyl] piperidines
01/06/2004US6673941 Disubstituted imidazoles useful in the treatment of bacterial infections
01/06/2004US6673938 Substituted pyridine herbicides
01/06/2004US6673937 Analogs of deoxypreussomerin, palmarumycin cpi and related naphthoquinone spiroketals; inhibit thioredoxin-thioredoxin reductase system
01/06/2004US6673833 As antitumor agent
01/06/2004US6673829 Treatment of diseases of the central nervous system, the peripheral nervous system, the cardiovascular system, the pulmonary system, the gastrointestinal system and the endocrinological system.
01/06/2004US6673807 Administering compound possessing inhibitory activity on production of nitric oxide and tricyclic macrolide or salt, solvate or hydrate thereof to increase graft survival time in transplantation subject
01/06/2004US6673803 Quinazoline derivatives and pharmaceutical compositions containing them
01/06/2004US6673797 Cyclooxygenase-2 inhibitors; treating inflammatory disease induced by cyclooxygenase-2
01/06/2004US6673790 Indolin-2-one derivatives, preparation and their use as ocytocin receptor ligands
01/06/2004US6673789 2-pyridinylguanidine urokinase inhibitors
01/06/2004CA2285891C Triazole antifungal agents
01/02/2004EP1375503A1 Dioxino derivatives and their use as dopanine agonists
01/02/2004EP1375498A1 Optically active epoxy compound
01/02/2004EP1375494A1 Tetraether lipids with small headgroups, method of their synthesis and uses thereof
01/02/2004EP1375486A1 Nitrogen-containing heteroaryl compounds having hiv integrase inhibitory activity
01/02/2004EP1375483A1 6-chloro-3-pyridylmethylpropylamine derivatives, preparation process thereof and bactericides
01/02/2004EP1373271A1 Indole derivatives having an inhibitory effect on protein kinases
01/02/2004EP1373265A1 Substituted 2,6-diamino-3,5-dicyano-4-aryl-pyridines and their use as adenosine receptor-selective ligands
01/02/2004EP1373262A2 Azacycloalkyl substituted acetic acid derivatives for use as mmp inhibitors
01/02/2004EP1373261A2 Cyclopropaheterocycles as non-nucleoside reverse transcriptase inhibitors
01/02/2004EP1373259A1 Pyridazinone aldose reductase inhibitors
01/02/2004EP1373258A1 Ether derivatives useful as inhibitors of pde4 isozymes
01/02/2004EP1373257A1 Inhibitors of c-jun n-terminal kinases (jnk) and other protein kinases
01/02/2004EP1373252A1 Chemical derivatives and their use as anti-telomerase agent
01/02/2004EP1373251A2 Non-imidazole compounds as histamine h3 antagonists
01/02/2004EP1373244A2 Substituted benzopyranones as telomerase inhibitors
01/02/2004EP1373241A1 Method for producing optically active dihydropyrones
01/02/2004EP1373233A1 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
01/02/2004EP1373224A1 New spirotricyclic derivatives and their use as phosphodiesterase-7 inhibitors
01/02/2004EP1373223A1 Cyano-substituted dihydropyrimidine compounds and their use to treat diseases
01/02/2004EP1373221A2 Novel cyano-substituted dihydropyrimidine compounds and their use to treat diseases
01/02/2004EP1373219A1 Thiohydantoins and use thereof for treating diabetes
01/02/2004EP1373217A1 2-mercapto-4,5-diarylimidazole derivatives and the use thereof as cyclooxygenase inhibitors
01/02/2004EP1373210A1 Heterocyclic diamide invertebrate pest control agents
01/02/2004EP1373202A1 Preparation of non-crystalline atorvastatin calcium
01/02/2004EP1373199A2 Spiro-cyclic beta-amino acid derivatives as inhibitors of matrix metalloproteinases and tnf-alpha converting enzyme (tage)
01/02/2004EP1373196A2 Sulfoxides or sulfones grafted onto polymers
01/02/2004EP1373194A1 BENZAMIDE INHIBITORS OF FACTOR Xa
01/02/2004EP1214315B9 1,4-dihydropyridine-5-carboxylic acid ester derivatives and method for the preparation thereof
01/02/2004EP1036062B1 Hydroxamic acid derivatives as matrix metalloprotease (mmp) inhibitors
01/01/2004US20040002528 CBI analogs of CC-1065 and the duocarmycins
01/01/2004US20040002525 Obesity; osteoporosis
01/01/2004US20040002524 Cardiovascular disorders; osteoporosis; central nervous system disorders
01/01/2004US20040002515 Antihistamines; antiallergens; antiinflammatory agents; autoimmune diseases; rheumatic diseases
01/01/2004US20040002508 Antitumor agents; anticancer agents; sexual disorders; cardiovascular disorders
01/01/2004US20040002491 Melatonergic receptors
01/01/2004US20040002490 Melatonergic receptors
01/01/2004US20040002487 Bone disorders; osteoporosis; oral diseases; antiarthritic agents
01/01/2004US20040002461 Amelioration of the development of cataracts and other ophthalmic diseases
01/01/2004US20040002424 2-Amino-4-bicyclylamino-6H-1,3,5-triazines, processes for their preparation and their use as herbicides and plant growth regulators
12/2003
12/31/2003WO2004000835A1 Method for the production of 1,2,4-triazolylmethyl-oxiranes
12/31/2003WO2004000834A1 Novel 3-(4-oxo-4h-chromen-2-yl)-(1h)-quinoline-4-one derivatives, method for preparing same and pharmaceutical compositions containing same
12/31/2003WO2004000831A1 Indole derivatives useful as histamine h3 antagonists
12/31/2003WO2004000826A1 Processes for producing epoxytriazole derivative and intermediate therefor
12/31/2003WO2004000819A1 New use of pyrimidine - or triazine- 2-carbonitiles for treating diseases associated with cysteine protease activity and novel pyrimidine-2-carbonitile derivatives
12/31/2003WO2004000817A2 Benzimidazole compounds and their use as estrogen agonists/antagonists
12/31/2003WO2004000816A1 Androgen receptor agonist
12/31/2003WO2004000811A1 Arylsulfonylhydroxamic acid and amide derivatives and their use as protease inhibitors
12/31/2003WO2004000808A2 N-substituted piperidine derivatives as serotonin receptor agents
12/31/2003WO2004000807A1 Cannabinoid receptor agonists
12/31/2003WO2004000806A1 Amides of cyclic amino acids used as pde 4 inhibitors
12/31/2003WO2004000764A2 BENZO(b)FURAN DIMERS
12/31/2003WO2003078627A3 A building block capable of functional entity transfer to nucleophil
12/31/2003WO2003078446A3 A building block forming a c-c or a c-hetero atom bond upon reaction
12/31/2003WO2003074513A3 Indole amide derivatives and their use as glycogen phosphorylase inhibitors
12/31/2003WO2003060475A3 Melanin concentrating hormone receptor ligands: substituted 2-(4-benzyl-piperazin-1-ylmethyl)- and 2-(4-benzyl-diazepan-1-ylmethyl)-1h-benzoimidazole analogues
12/31/2003WO2003059269A3 Acridone inhibitors of impdh enzyme
12/31/2003WO2002060378A3 Substituted aryl compounds as cyclooxygenase-2 selective inhibitors, compositions and methods of use
12/31/2003WO2002040060A3 Conjugates of an antioxidants with metal chelating ligands
12/31/2003CN1132828C O-substd. hydroxy coumaranone derivs as antineoplastic and antitransfer agent
12/31/2003CN1132676C 用于降低血制品中小有机分子的方法和装置 For reducing blood products of small organic molecules method and apparatus
12/31/2003CA2490646A1 Arylsulfonylhydroxamic acid and amide derivatives and their use as protease inhibitors
12/31/2003CA2490397A1 N-substituted piperidine derivatives as serotonin receptor agents
12/31/2003CA2487346A1 Cannabinoid receptor agonists