Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
04/2004
04/29/2004CA2501547A1 Substituted indoles and their use as hcv inhibitors
04/29/2004CA2501539A1 Benzimidazole derivatives and their use as vanilloid receptor ligands
04/29/2004CA2501418A1 Novel compounds
04/29/2004CA2500320A1 Novel compounds with antibacterial activity
04/29/2004CA2500083A1 Tetrahydroquinoline derivatives as crth2 antagonists
04/28/2004EP1413580A1 Furanone derivatives as inhibitors of Cathepsin S
04/28/2004EP1413576A2 Substituted imidazole derivatives having agonist-like activity at alpha 2B or 2B/2C adrenergic receptors
04/28/2004EP1413306A1 Tetrahydroquinoline derivatives as CRTH2 antagonists
04/28/2004EP1412376A2 Compositions and methods for labeling oligonucleotides
04/28/2004EP1412364A1 Platelet adp receptor inhibitors
04/28/2004EP1412351A1 Reductive cleavage of the exocyclic ester of uk-2a or its derivatives and products formed therefrom
04/28/2004EP1412350A1 Paroxetine isethionate salt, process of preparation and use in the treatment of depression
04/28/2004EP1412349A2 Piperazine oxyquinoline (naphthaline) platelet adenosine diphosphate receptor antagonists
04/28/2004EP1412348A1 Compounds derived from diaminopyrazole substituted by a heteroaromatic radical and their use in oxidation dyeing of keratinous fibres
04/28/2004EP1412344A1 Iodobenzopyran-4-one derivatives having fungicidal activity
04/28/2004EP1412343A1 New compounds, which are potent inhibitors of na+/ca2+ exchange mechanism and are useful in the treatment of arrhythmias
04/28/2004EP1412327A2 Inhibitors of protein kinase for the treatment of disease
04/28/2004EP1411954A2 Modified nucleosides for treatment of viral infections and abnormal cellular proliferation
04/28/2004EP1411948A1 Tetrahydroquinoxalines acting as bradykinin antagonists
04/28/2004EP1411945A1 Substituted pyridin-4-ones and their use as gonadotropin-releasing hormone receptor antagonists
04/28/2004EP1411944A1 Sulfonamide derivatives as gamma secretase inhibitors
04/28/2004EP1411942A1 Substituted anilinic piperidines as mch selective antagonists
04/28/2004EP1411928A1 Viral polymerase inhibitors
04/28/2004EP1042313B1 Benzopyran and benzothiopyran derivatives having retinoid antagonist like activity
04/28/2004EP0513200B2 Method and compositions for the synthesis of bch-189 and related compounds
04/28/2004CN1492865A š�-lactam compounds, process for producing the same and serum cholesterol-lowering agents containing the same
04/28/2004CN1492860A 喹唑啉衍生物 Quinazoline derivatives
04/28/2004CN1492856A Pyridone derivative having affinity for cannabinoid 2-type receptor
04/28/2004CN1491949A Pyridazine-3-one derivatives, their use, and intermediate preparing them
04/28/2004CN1491947A C10 ester carbonate substituted taxadane
04/28/2004CN1491946A C 10 ester substituted taxadane
04/28/2004CN1491941A Heterobicyclic sulfonamide derivative and sulfonic ester derivative
04/28/2004CN1147504C New thrombin inhibitors, their preparation and use
04/28/2004CN1147486C 4-and 5-alkynyloxindoles and 4-and 5-alkenyloxindoles
04/28/2004CN1147476C Pyrazole derivatives as P-38 MAP kinase inhibitors
04/27/2004US6727364 Antiinflammatory agents
04/27/2004US6727275 Pyrrolidinone derivatives
04/27/2004US6727264 Substituted anilinic piperidines as MCH selective antagonists
04/27/2004US6727263 Serotonine reuptake inhibitor; antidepressants; side effect reduction
04/27/2004US6727257 Hypotensive agents for intraocular pressure; anticholesterol agents; relaxing urinary tract tissue; benign prostatic hyperplasia, impotency, and cardiovascular disorders; antiarrhythmia agents
04/27/2004US6727256 4-aminoquinazoline derivatives as anticarcinogenic agents
04/27/2004US6727251 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease
04/27/2004US6727250 Administering compounds such as trans-3-(naphth-2-yl)-but-2-enoic acid-n-(2-carboxy-phenyl)-amide or like for therapy of conditions associated with increased telomerase activity, e.g. tumour diseases
04/27/2004US6727248 Substituted quinolinecarboxamides as antiviral agents
04/27/2004US6727244 Mammalian metabolites of a tachykinin receptor antagonist
04/27/2004US6727239 Inhibitory activity on no- synthase enzymes producing nitrogen monoxide no and/or an activity which traps the reactive oxygen species (ros)
04/27/2004CA2299400C Method for treating disease-related or drug-induced dyskinesias
04/27/2004CA2136745C Heterocyclically disubstituted sulphonylamino(thio)carbonyl compounds
04/22/2004WO2004033632A2 Hydantoin derivatives as inhibitors of matrix metalloproteinases and/or tnf-alpha converting enzyme (tace)
04/22/2004WO2004033447A1 Imidazole derivatives and their use as peripherally-selective inhibitors of dopamine-beta-hydroxylase
04/22/2004WO2004033435A1 Quinazolinone derivatives useful as anti-hyperalgesic agents
04/22/2004WO2004033434A1 Pyrazole compounds for treatment of neurodegenerative disorders
04/22/2004WO2004033428A1 Substituted 1,4-di-piperidin-4-yl-piperazine derivatives and their use as neurokinin antagonists
04/22/2004WO2004033427A1 1,4-disubstituted piperidine derivatives and their use as 11-betahsd1 inhibitors
04/22/2004WO2004033422A2 Modulation of anxiety through blockade of anandamide hydrolysis
04/22/2004WO2004032908A2 Method of inhibiting angiogenesis
04/22/2004WO2004032871A2 Piperazine and piperazinone inhibitors of factor xa
04/22/2004WO2004032848A2 Pgd2 receptor antagonists for the treatment of inflammatory diseases
04/22/2004WO2004032846A2 Triazolone and triazolethione derivatives
04/22/2004WO2004032845A2 R-nsaid esters and their use
04/22/2004WO2004022544A8 Novel aminoindazole derivatives as medicines and pharmaceutical compositions containing same
04/22/2004WO2004020430A3 Derivatives of dioxane-2-alkyl carbamates, preparation method thereof and application of same in therapeutics
04/22/2004WO2004020410A3 Dihydropyridinone derivatives as hne inhibitors
04/22/2004WO2004016597A3 Protein kinase inhibitors and uses thereof
04/22/2004WO2004014300A3 Tyrosine kinase inhibitors
04/22/2004WO2004002986A3 Novel benzimidazole derivatives
04/22/2004WO2003082263A8 Sulfamic acids as inhibitors of human cytoplasmic protein tyrosine phosphatases
04/22/2004WO2003078403A3 Derives d’aminoindazoles comme inhibiteurs de proteine-kinase
04/22/2004WO2003072541A3 Chemical compounds
04/22/2004WO2003005999A8 Methods of treating cytokine mediated diseases
04/22/2004WO2002074767A8 Metalloproteinase inhibitors
04/22/2004WO2002074752A8 Metalloproteinase inhibitors
04/22/2004WO2002074748A8 Metalloproteinase inhibitors
04/22/2004US20040077877 Jun n-terminal kinase inhibitors
04/22/2004US20040077861 Asymmetric addition of organometallic compounds to chiral sulfinimine to give adducts in predominantly one diastereomer can subsequently be transferred into pure enantiomers of by cleavage of the chiral auxilliary
04/22/2004US20040077712 Resolution with acid; salt formation, cyclization
04/22/2004US20040077707 Pyrrole based inhibitors of glycogen synthase kinase 3
04/22/2004US20040077706 Piperidine and azepine derivatives; anxiolytic, analgesic, antidepressant, antiemetic, antiinflammatory, and hypotensive agents; sexual and psychological disorders; Alzheimer*s, Parkinson*s, Lesche-Nyhane, Wilson*s, and Tourette*s syndrome
04/22/2004US20040077702 Administering indazole derivative; or thienyl-, furyl-, or pyrrolyl- fused pyrazole derivative to treat Alzheimer*s, Parkinson*s, or Huntington*s disease
04/22/2004US20040077699 Substituted triazole diamine derivatives as kinase inhibitors
04/22/2004US20040077693 Integrin receptor inhibitors
04/22/2004US20040077684 Piperidinyl compounds that selectively bind integrins
04/22/2004US20040077671 Sorbitol dehydrogenase inhibitors
04/22/2004US20040077670 Novel sulfamides and their use as endothelin receptor antagonists
04/22/2004US20040077668 Compounds, compositins, and methods
04/22/2004US20040077667 Quinazolinone derivatives
04/22/2004US20040077656 Quinolines and nitrogenated derivatives thereof substituted in 4-position by a piperazine-containing moiety and their use as antibacterial agents
04/22/2004US20040077655 Piperazine derivatives for treatment of bacterial infections
04/22/2004US20040077654 Anticholesterol agents; cardiovascular disorders
04/22/2004US20040077650 Cannabinoid receptor ligands and uses thereof
04/22/2004US20040077648 Antiproliferative agents for smooth muscle cells; antiinflammatory agents for endothelial cells; restenosis, atherosclerosis
04/22/2004US20040077647 Fluorinated di-aryl urea compounds
04/22/2004US20040077646 Indole nitriles
04/22/2004US20040077644 Administering quinoline derivative as analgesic
04/22/2004US20040077643 3,4 Dihydroisoquinoline derivative compounds and drugs containing these compounds as the active ingredient
04/22/2004US20040077641 Insecticides for crops
04/22/2004US20040077635 Trypsin-like serine protease inhibitors; treating thromboembolic disorders; anticoagulants
04/22/2004CA2501611A1 1,4-disubstituted piperidine derivatives and their use as 11-betahsd1 inhibitors
04/22/2004CA2501529A1 Quinazolinone derivatives useful as anti-hyperalgesic agents
04/22/2004CA2501506A1 Modulation of anxiety through blockade of anandamide hydrolysis