Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
02/2004
02/26/2004CA2495383A1 Fused benzene derivative and use
02/25/2004EP1391952A2 Salts of pentacyclic or tetrapentaline derived anions, and their uses as ionic conductive materials
02/25/2004EP1391456A1 2-iminoimidazole derivative (2)
02/25/2004EP1391451A1 2-iminopyrrolidine derivates
02/25/2004EP1391450A1 N-(heterocycle-methyl)alkylamine derivative, process for producing the same, and bactericide
02/25/2004EP1390362A1 Substituted benzofurans and benzothiophenes, methods of making and methods of use as integrin antagonists
02/25/2004EP1390353A1 Triazole-derived kinase inhibitors and uses thereof
02/25/2004EP1390352A1 Pyrimidine derivatives
02/25/2004EP1390350A1 Novel compounds
02/25/2004EP1390349A1 Aminoquinoline and aminopyridine derivatives and their use as adenosine a3 ligands
02/25/2004EP1390340A1 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
02/25/2004EP1390034A1 N-substituted nonaryl-heterocyclo amidyl nmda/nr2b antagonists
02/25/2004EP1301503B1 Coumarin derivatives with comt inhibiting activity
02/25/2004EP1263756B1 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha
02/25/2004EP1230232B1 Substituted 4h-chromene and analogs as activators of caspases and inducers of apoptosis and the use thereof
02/25/2004EP1222171B1 Pyridinium derivatives for the management of aging-related and diabetic vascular complications, process for their preparation and therapeutic uses thereof
02/25/2004EP1211246B1 Pyrimidine derivatives and herbicides containing the same
02/25/2004EP1178986B1 Furanone derivatives as inhibitors of cathepsin s
02/25/2004EP1042296B1 Substituted isoquinoline derivatives and their use as anticonvulsants
02/25/2004CN1478136A Novel red fluorescent material and organic electroluminescent device containing same
02/25/2004CN1478094A Process and ester derivatives for preparing cephalosporins
02/25/2004CN1478089A Substituted derivatives of aminofuran-2-Y1-acetic acid and aminothien-2-Y1-acetic acid and use thereof for treating migraines and pain
02/25/2004CN1478085A ABCA-1 elevating compounds against coronary artery disease or atherosclerosis
02/25/2004CN1478079A Diaminopyrazole derivatives and their use for oxidation dyeing of keratinous fibres
02/25/2004CN1478078A Nitrogenous aromatic ring compounds
02/25/2004CN1478076A MCH antagonists and their use in treatment of obesity
02/25/2004CN1477961A Piperazine derivatives, their preparation and their use for treating central nervous system (CNS) disorders
02/25/2004CN1139588C Novel fluorinated imidazoline benzodioxane, preparation and therapeutic use thereof
02/24/2004US6696470 Pyridylthiophene compounds
02/24/2004US6696469 For treatment of diseases or pathological conditions in which endothelial dysfunction is known; atherosclerosis, dyslipidaemia, diabetes
02/24/2004US6696468 (s)-4-amino-5-chloro-2-methoxy-n-[1-[1-(2-tetrahydrofuryl-carbonyl)-4-piperidinylmethyl]-4-piperidinyl]benzamide, process for the preparation thereof, pharmaceutical composition containing the same, and intermediate therefor
02/24/2004US6696467 Quinoline derivatives
02/24/2004US6696456 Carbocyclic acids and salts such as (2s,3r)-3-ethylsulfanyl-2-(4'-fluoro-biphenyl-4-sulfonylamino)-3- phenylpropionic acid, used as metalloenzyme antagonists for the prophylaxis of degenerative joint disease and as wound healing agents
02/24/2004US6696452 Glycogen synthase kinase-3 and aurora-2 a serine/threonine protein kinase inhibitors; antidiabetic and anticancer agents and alzheimer's disease treatments
02/24/2004US6696449 Control degradation of conencting tissue; cardiovascular disorders
02/24/2004US6696447 Hydroxyphenyl-piperazinyl-methyl-benzamide derivatives for the treatment of pain
02/24/2004US6696446 Benzoylpyridazines, their preparation and use
02/24/2004US6696437 Polymerase inhibitors comprising heterocyclic amides such as 2-pyridin-2-ylbenzimidazole-4-carboxamide, used for prophylaxis of neurodegenerative disorders, damage to hearts or brains, and as anticarcinogenic agents
02/24/2004US6696434 Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p56lck tyrosine kinases
02/24/2004US6695969 Displacement chromatography and involves using a displacer for displacing the hmg-coa reductase inhibitor
02/24/2004CA2208141C Fungicidal mixture
02/24/2004CA2150944C New taxoids; process for preparing the same and pharmaceutical compositions containing them
02/24/2004CA2114542C Benzimidazolone derivatives as 5-ht1a and 5-ht2 antagonists
02/19/2004WO2004014919A1 Epothilone derivatives
02/19/2004WO2004014900A1 Benzimidazoles and benzothiazoles as inhibitors of map kinase
02/19/2004WO2004014898A1 Benzopyran derivatives substituted with secondary amines including imidazole, their preparation and pharmaceutical compositions containing them
02/19/2004WO2004014897A1 N-aryl-2-oxazolidinones and their derivatives
02/19/2004WO2004014896A1 Process for preparing 5-(4-fluorophenyl)-1-[2-((2r,4r)-4-hydroxy -6-oxo-tetrahydro-pyran-2-yl)ethyl]-2-isopropyl-4-phenyl-1h-pyrrole-3-carboxylic acid phenylamide
02/19/2004WO2004014878A1 1,2,4-triazole derivative, method for preparing the same, and pharmaceutical composition containing the same
02/19/2004WO2004014877A1 Process for preparing rizatriptan
02/19/2004WO2004014871A1 Vanilloid receptor ligands and their use in treatments
02/19/2004WO2004014870A1 Fluorinated phenyl-naphthalenyl-urea compounds as inhibitors of cytokines involved in inflammatory processes
02/19/2004WO2004014869A2 5,6-fused 3,4-dihydropyrimidine-2-one derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014868A2 Pyrimidine-2,4-dione derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014864A1 1h-indazole-3-carboxamide compounds as cyclin dependent kinases (cdk) inhibitors
02/19/2004WO2004014860A2 Fused heterocyclic compounds as peptidase inhibitors
02/19/2004WO2004014851A2 Tyrosine kinase inhibitors
02/19/2004WO2004014430A1 Compositions of a cyclooxygenase-2 selective inhibitor and a carbonic anhydrase inhibitor for the treatment of neoplasia
02/19/2004WO2004014389A1 3,4-dihydroquinolin-2-one, 5,6-fused oxazin-3-one, and 5,6-fused thiazin-3-one derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014379A1 Isoquinoline derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014377A1 4-hydroxyquinoline derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014372A1 Acylated, heteroaryl-condensed cycloalkenylamines and their use as pharmaceuticals
02/19/2004WO2004014366A1 Hetero biaryl derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014365A1 Phthalimide derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014352A2 Methods for treating carbonic anhydrase mediated disorders
02/19/2004WO2004014300A2 Tyrosine kinase inhibitors
02/19/2004WO2004007481A3 Substituted amine derivatives and methods of use in the treatment of angiogenesis relates disorders
02/19/2004WO2003065989A3 (oxime)carbamoyl fatty acid amide hydrolase inhibitors
02/19/2004WO2003049593A3 Prevention of flap necrosis in plastic surgery
02/19/2004WO2002032920A3 Modified nucleosides for treatment of viral infections and abnormal cellular proliferation
02/19/2004US20040034239 Inhibitors of nadh:ubiquinone oxidoreductase
02/19/2004US20040034230 Taxanes having a carbamoyloxy substituent at C(10), a hydroxy substituent at C(7), and a range of C(2), C(9), C(14), and side chain substitutions; anticarcinogenic agent
02/19/2004US20040034229 3,4-Di-substituted maleimide compounds as CXC chemokine receptor antagonists
02/19/2004US20040034222 Phenyloxyalkylamino substituted triazine compound, useful for applying to the parts of the plants, to plant seed or to the area under cultivation as plant growth regulator
02/19/2004US20040034217 An indole derivatives as intermediate for the synthesis of vindoline, is formed from a substituted aniline; synthetic efficiency, nontoxic reagents
02/19/2004US20040034205 Chiral (1pyrrolino) fullerene derivatives
02/19/2004US20040034084 Side effect reduction; for treatment of AIDS, cancer and arthritis
02/19/2004US20040034063 Antiallergens for treating and prevention of asthma
02/19/2004US20040034049 A benzofuran derivatives for treating neurodegenerative disease, such as Alzheimer's disease, Parkinson's disease, amyotropic lateral sclerosis and Huntington's disease
02/19/2004US20040034047 E.g. 5-(6,7-dimethoxy-2-(4-methoxybenzyl)benzofuran-4-yl-methyl-)pyrimidine-2,4 -diamine; bactericides for infections of grampositive and gramnegative pathogens; more potent than Trimethoprim, especially against respiratory tract pathogens
02/19/2004US20040034046 Quinazoline derivatives
02/19/2004US20040034034 Novel piperazine derivatives
02/19/2004US20040034032 Quinoline and quinazoline compounds useful in therapy
02/19/2004US20040034031 3,4-Disubstituted, 3,5-disubstituted and 3,4,5-substituted piperidines
02/19/2004US20040034025 Having a high residual activity, greater activity at lower application rates, curative activity, and a broader spectrum of efficacy; heterocyclic aromatic amides having a hydroxy group adjacent to the amide functionality
02/19/2004US20040034019 Piperazine and piperidine derivatives
02/19/2004US20040034018 2-amino-trihydroindole or tetrahydronapthalene-2-yl derivatives, useful for disease state associated with smooth muscle disorders, such as gastrointestinal and urogenital disorders
02/19/2004US20040033514 Detection of disease related genes
02/19/2004DE10236340A1 New heteroar(alkan)oyl-substituted phenyl-beta-alaninamide derivatives, useful as broad-spectrum antibacterial agents in human or veterinary medicine
02/19/2004DE10234697A1 Neue Verbindungen zur Stimulation des Nervenwachstums, zur Inhibition der Narbengewebsbildung und/oder Reduktion eines Sekundärschadens Novel compounds for stimulation of nerve growth, to inhibition of scar tissue formation and / or reduction of secondary damage
02/19/2004CA2497656A1 Pyrimidine-2,4-dione derivatives as matrix metalloproteinase inhibitors
02/19/2004CA2495516A1 Compositions of a cyclooxygenase-2 selective inhibitor and a carbonic anhydrase inhibitor for the treatment of neoplasia
02/19/2004CA2495502A1 Methods for treating carbonic anhydrase mediated disorders
02/19/2004CA2494824A1 Fluorinated phenyl-naphthalenyl-urea compounds as inhibitors of cytokines involved in inflammatory processes
02/19/2004CA2494269A1 Process for preparing 5-(4-fluorophenyl)-1-[2-((2r,4r)-4-hydroxy -6-oxo-tetrahydro-pyran-2-yl)ethyl]-2-isopropyl-4-phenyl-1h-pyrrole-3-carboxylic acid phenylamide
02/19/2004CA2494259A1 Epothilone derivatives
02/19/2004CA2494048A1 4-hydroxyquinoline derivatives as matrix metalloproteinase inhibitors
02/19/2004CA2493575A1 Tyrosine kinase inhibitors
02/19/2004CA2492019A1 Isoquinoline derivatives as matrix metalloproteinase inhibitors
02/19/2004CA2491287A1 N-aryl-2-oxazolidinones and their derivatives