Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
05/2004
05/27/2004WO2004012735A3 New effector conjugates, process for their production and their pharmaceutical use
05/27/2004WO2003099812A8 Phenyl-furan or phenyl-thiophene derivatives, their preparation and their use as medicine
05/27/2004WO2003088908A3 Heterocyclo inhibitors of potassium channel function
05/27/2004WO2003031436A8 Heterocyclic compounds for use in the treatment of disorders of the urinary tract
05/27/2004WO2003016276A3 3-substituted oxindole beta-3 agonists
05/27/2004US20040102630 For therapy of cancer, auto-immune diseases, cardiovascular diseases, infectious diseases, nephrological diseases, neurodegenerative diseases and viral infections
05/27/2004US20040102626 Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines with adenosine receptor-binding activity and their use cardiovascular preparations
05/27/2004US20040102516 Crop protection agents
05/27/2004US20040102509 Kinase inhibitors for the treatment of disease
05/27/2004US20040102508 Naphathalene derivatives which bind to the ep4 receptor
05/27/2004US20040102507 Use of GALR3 receptor antagonists for the treatment of depression and/or anxiety and compounds useful in such methods
05/27/2004US20040102506 Pyrazole compositions useful as inhibitors of ERK
05/27/2004US20040102500 Peroxisome proliferator activated receptor alpha agonists
05/27/2004US20040102488 Antiinflamamtory agents; autoimmune diseases; antiarthritic agents; anticancer agents; Alzheimer's disease
05/27/2004US20040102483 Chemical compounds
05/27/2004US20040102479 Novel benzopyran or thiobenzopyran derivatives
05/27/2004US20040102466 Analgesics; antipyretics; antiinflammatory agents
05/27/2004US20040102461 Synergistic mixture with anticancer drugs
05/27/2004US20040102455 Autoimmune diseases; antiinflammatory agents; antiallergens; viricides; anticancer agents
05/27/2004US20040102450 Substituted oxoazaheterocyclyl compounds
05/27/2004US20040102449 Pyridinyl, pyrimidinyl and pyrazinyl amides as potassium channel openers
05/27/2004US20040102448 Substituted polycyclic aryl and heteroaryl pyrazinones useful for selective inhibition of the coagulation cascade
05/27/2004US20040102442 Central nervous system disorders; brain disorders
05/27/2004US20040102441 Ortho-substituted anthranilic acid amides and their use as medicaments
05/27/2004US20040102437 Prevention cytokine migration; hypotensive agents; asthma therapy
05/27/2004US20040102432 Asthma, rhinitis therapy
05/27/2004US20040102431 Protease inhibitors
05/27/2004US20040102423 Spironolactone and angiotensin II antagonist combination therapy for treatment of congestive heart failure
05/27/2004US20040101535 Administering nucleoside, or prodrug thereof; viricides
05/27/2004DE10252969A1 New 3-aminomethylene-indoline-2-(thi)one derivatives, are kinase inhibitors useful for treating proliferative diseases e.g. tumors, rheumatoid arthritis, neovascular glaucoma and arteriosclerosis
05/27/2004CA2765093A1 Bicyclic-substituted amines as histamine-3 receptor ligands
05/27/2004CA2505819A1 Indolyl pyrazinone derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis
05/27/2004CA2505557A1 Mucin synthesis inhibitors
05/27/2004CA2505361A1 Phenyl or heteroaryl amino alkane derivatives as ip receptor antagonist
05/27/2004CA2504737A1 Aromatic sulfone hydroxamic acids and their use as protease inhibitors
05/27/2004CA2501932A1 Use of benzimidazole quinolinones for treating cancer
05/26/2004EP1422219A1 Cyclic amine compound
05/26/2004EP1422218A1 Antiviral agent
05/26/2004EP1421082A1 New piperidinyl-morpholinyl derivatives as modulators of chemokine receptor activity
05/26/2004EP1421078A1 Beta-3 adrenergic agonists
05/26/2004EP1421071A2 Substituted piperazine and diazepane derivaives as histamine h3 receptor modulators
05/26/2004EP1421063A1 Disulfide and thiosulfonate ligands and libraries comprising these ligands
05/26/2004EP1420796A1 Androgen receptor modulators and methods of use thereof
05/26/2004EP1420784A1 Compounds effecting glucokinase
05/26/2004EP1420780A2 Cyclopropyl and cyclobutyl epothilone analogs
05/26/2004EP1206474B1 Sulfonylphenylpyrazole compounds useful as cox-2 inhibitors
05/26/2004EP1137645B1 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group
05/26/2004EP1117642B1 Substituted 1,3-diaryl-2-pyridine-2-yl-3-(pyridine-2-ylamino)-propanol derivatives, methods for their production, pharmaceutical compositions containing the same and their use
05/26/2004EP1027332B1 Novel lactam metalloprotease inhibitors
05/26/2004EP0968194B1 Atropisomers of 3-aryl-4(3h)-quinazolinones and their use as ampa-receptor antagonists
05/26/2004CN1500087A 哒嗪酮醛糖还原酶抑制剂 Pyridazinone aldose reductase inhibitors
05/26/2004CN1500086A Aminopiperidine derivatives
05/26/2004CN1500085A Lipid lowering biphenylcarboxamides
05/26/2004CN1500082A Cyano-5ubstituted dihydropyrimidine compounds and their use to treat diseases
05/26/2004CN1500081A Thiohydantonins and use thereof for treating diabetes
05/26/2004CN1500080A 稠合杂环化合物 Fused heterocyclic compounds
05/26/2004CN1500076A Sulfoxider or sulfones gralted onto polymers
05/26/2004CN1499970A Use of GAL3 receptor antagonists for treatment of. depression and/or anxiety and compounds useful in such methods
05/26/2004CN1151161C Medicine nitrate salts
05/26/2004CN1151148C Farnesy transferase inhibitors having pyrrole structure and process for preparation thereof
05/26/2004CN1151147C Indole derivatives as 5-HT receptor antagonist
05/26/2004CN1151136C Fused pyridazine compound
05/26/2004CN1151133C Anthranilic acid amides and use thereof as medicaments
05/26/2004CN1151131C Piperidine derivatives useful as CCR5 antagonists
05/26/2004CN1151130C Neuroprotective 3-(piperidinyl-1)-chroman-4,7-diol and 1-(4-hydrophenyl)-2-(piperidinyl-1)-alkane alcohol
05/26/2004CN1151127C Indole derivatives and their use in the treatment of malignant and other diseases caused by pathological cell proliferation
05/25/2004US6740760 Such as 1-((s)-3-mercapto-2-methyl-propionyl)-(r)-pyrrol-idine-2-carboxylic acid for treating diseases associated with amyloidosis (alzheimer's disease, diabetes, and familial amyloid polyneuropathy)
05/25/2004US6740682 Treatment of thrombotic diseases, asthma, emphysema, cirrhosis, arthritis, carcinoma, melanoma, restenois, atheroma, trauma, shock and reperfusion injury.
05/25/2004US6740655 3',5'-cyclic nucleotide phosphodiesterase 4-specific inhibitors reduce eosinophil influx to the lungs; side effect reduction; antiinflammatory agent; antiallergens; respiratory system disorders, especially asthma
05/25/2004US6740649 Cyclic hydroxamic acids as inhibitors of matrix metalloproteinases and/or TNF- α converting enzyme (TACE)
05/25/2004CA2302058C A process for preparing 5-methoxy-4-methyl-2,4-dihydro-3h-1,2,4-triazol-3-one
05/25/2004CA2115170C Imidazolyl-alkenoic acids
05/21/2004WO2004041811A1 3-cyano-quinoline derivatives
05/21/2004WO2004041810A1 Compounds useful as inhibitors of jak and other protein kinases
05/21/2004WO2004041807A1 Novel compounds
05/21/2004WO2004041791A1 N-aryl acetyl cyclic amine derivatives as orexin antagonists
05/21/2004WO2004041789A1 Compositions useful as inhibitors of jak and other protein kinases
05/21/2004WO2004041788A1 Novel pyrimidine-4,6-dicarboxamides for the selective inhibition of collagenases
05/21/2004WO2004041787A1 Process for producing quinolinecarbaldehyde
05/21/2004WO2004041784A1 Phenyl-piperidin-4-ylidene-methyl-benzamide derivatives for the treatment of pain or gastrointestinal disorders
05/21/2004WO2004041782A1 Indoles useful in the treatment of androgen-receptor related diseases
05/21/2004WO2004041755A2 Quinazolinone compounds as calcilytics
05/21/2004WO2004041274A1 Benzotriazoles and methods of prophylaxis or treatment of metabolic-related disorders thereof
05/21/2004WO2004041258A2 Cyclic nucleotide phosphodiesterase inhibitors, preparation and uses
05/21/2004WO2004041211A2 INHIBITORS OF β-SECRETASE, AND THEIR USE FOR THE PREVENTION OR TREATMENT OF ALZHEIMER’S DISEASE OR MILD COGNITIVE IMPAIRMENT
05/21/2004WO2004041209A2 Transcription factor modulating compounds and methods of use thereof
05/21/2004WO2004041201A2 Benzofuran compounds, compositions and methods for treatment and prophylaxis of hepatitis c viral infections and associated diseases
05/21/2004WO2004041161A2 Tetrahydropyranyl cyclopentyl benzylamide modulators of chemokine receptor activity
05/21/2004WO2004014860A3 Fused heterocyclic compounds as peptidase inhibitors
05/21/2004WO2004004629A3 3,6-disubstituted azabicyclo [3.1.0]hexane derivatives useful as muscarinic receptor antagonists
05/21/2004WO2004000817A3 Benzimidazole compounds and their use as estrogen agonists/antagonists
05/21/2004WO2003086605A3 Functionalized ionic liquids, and methods of use thereof
05/21/2004CA2507406A1 Compounds useful as inhibitors of jak and other protein kinases
05/21/2004CA2506772A1 Compositions useful as inhibitors of jak and other protein kinases
05/21/2004CA2505239A1 Process for producing quinolinecarbaldehyde
05/21/2004CA2504344A1 Benzofuran compounds, compositions and methods for treatment and prophylaxis of hepatitis c viral infections and associated diseases
05/21/2004CA2503716A1 Cyclic nucleotide phosphodiesterase inhibitors, preparation and uses
05/21/2004CA2502302A1 Quinazolinone compounds as calcilytics
05/21/2004CA2502174A1 Tetrahydropyranyl cyclopentyl benzylamide modulators of chemokine receptor activity
05/20/2004US20040097734 Aryl- and heteroarylcarbonylpiperazines and their use for the treatment of benign and malignant oncoses