Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
06/2004
06/17/2004WO2004050630A1 The use of aryl- and heteroaryl-substituted tetrahydroisoquinolines in the treatment of chronic and neuropathic pain, migraine headaches, and urge, stress and mixed urinary incontinence
06/17/2004WO2004050624A1 Substituted 1h-pyridine-2-one derivatives
06/17/2004WO2004050621A2 Indol derivatives and their use as kinase inhibitors
06/17/2004WO2004050619A1 Hydroxyethylamine derivatives for the treatment of alzheimer's disease
06/17/2004WO2004050613A2 2-substituted-3-propenamide derivatives and methods of using the same
06/17/2004WO2004050609A1 Substituted ureas and carbamates
06/17/2004WO2004050087A1 3-(2-hydroxy-phenyl)-1h-pyrazole-4-carboxylic acid amide derivatives as hsp90 inhibitors for the treatment of cancer
06/17/2004WO2004050082A1 The novel coumarin-amide derivatives and its preparation, said drug composition and its use
06/17/2004WO2004050035A2 Benzimidazoles and analogs thereof as antivirals
06/17/2004WO2004050024A2 3-aminopyrrolidine derivatives as modulators of chemokine receptors
06/17/2004WO2004050018A2 Dicationic 2,5-diarylfuran aza-analogs as anti-protozoan agents
06/17/2004WO2004049797A2 Pesticidal sulphonylaminopyrazoles
06/17/2004WO2004018414A3 Antibacterial agents
06/17/2004WO2004014869A3 5,6-fused 3,4-dihydropyrimidine-2-one derivatives as matrix metalloproteinase inhibitors
06/17/2004WO2003105781A3 Ophthalmic compositions for treating ocular hypertension
06/17/2004US20040116710 N3 alkylated benzimidazole derivatives as MEK inhibitors
06/17/2004US20040116706 Therapeutic ureas
06/17/2004US20040116695 2-Mercapto-4,5-diarylimidazole derivatives and the use thereof as cyclooxygenase inhibitors
06/17/2004US20040116694 Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors
06/17/2004US20040116507 2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
06/17/2004US20040116499 treatment of inflammatory or proliferative diseases of the skin and other organ systems; from yeast of the genus Malassezia; for example, 2,3-dihydro-4,5-bis(indol-3-yl)furan-2,3-dione; against multiresistent staphylococci
06/17/2004US20040116497 Chromane derivatives, process for their preparation and their use as antitumor agents
06/17/2004US20040116491 Therapy for infections; autoimmune diseases; vision defects; asthma:eating disorders; cardiovascular disorders; liver disorders; antiallergens; antiinflammatory agents; antiulcer agnets
06/17/2004US20040116486 Metalloproteinase inhibitors
06/17/2004US20040116480 Oxime ether compound and agricultural or horticultural bactericide
06/17/2004US20040116476 Imidazolidinone compounds
06/17/2004US20040116474 Novel pyrazole compounds as transforming growth factor (TGF) inhibitors
06/17/2004US20040116472 inhibit angiogenesis, tumor metastasis and growth, osteoporosis, Paget's disease, hypercalcemia of malignancy, retinopathy, macular degeneration, arthritis, periodontal disease, smooth muscle cell migration and viral diseases
06/17/2004US20040116471 Indolylpiperidine derivatives as antihistaminic aand antiallergic agents
06/17/2004US20040116465 Novel compounds
06/17/2004US20040116455 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
06/17/2004US20040116454 Pyrazole compounds useful as protein kinase inhibitors
06/17/2004US20040116443 Dopamine D4 ligands for the treatment of novelty-seeking disorders
06/17/2004US20040116440 Useful for diagnosis, treatment of male or female sexual dysfunction
06/17/2004US20040116431 Substituted aryl compounds as novel cyclooxygenase-2 selective inhibitors, compositions and methods of use
06/17/2004US20040116424 Aryl imidazoles and related compounds as C5a receptor modulators
06/17/2004US20040116423 5-Aryltetrazole compounds, compositions thereof, and uses therefor
06/17/2004US20040116422 Drugs as enzyme inhibitors for tyrosine kinases and for treatment of psoriasis
06/17/2004US20040116420 Remedial agent for viral infectious disease
06/17/2004US20040116417 Thiohydantoins and use thereof for treating diabetes
06/17/2004US20040116399 for preventing or treating coagulation disorders
06/17/2004US20040116388 triazine compoound inhibitors of enzymes that catalyze phosphoryl transfer and/or that bind ATP/GTP nucleotides
06/17/2004US20040116353 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
06/17/2004DE19742593B4 Neuer farbbildender Farbstoffvorläufer, Zusammensetzung, die denselben enthält und farbbildendes wärmeempfindliches Aufzeichnungsmaterial New color-forming dye precursor composition comprising the same and color-forming heat-sensitive recording material
06/17/2004DE10256405A1 New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
06/17/2004DE10247233A1 New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
06/17/2004CA2508574A1 3-(2-hydroxy-phenyl)-1h-pyrazole-4-carboxylic acid amide derivatives as hsp90 inhibitors for the treatment of cancer
06/17/2004CA2508329A1 Substituted dihydrophenanthridinesul fonamides
06/17/2004CA2508325A1 Hydroxyethylamine derivatives for the treatment of alzheimer's disease
06/17/2004CA2507780A1 Indol derivatives and their use as kinase inhibitors
06/17/2004CA2507484A1 Substituted ureas and carbamates
06/17/2004CA2505893A1 Oxime ester photoinitiators with heteroaromatic groups
06/17/2004CA2504742A1 Process for synthesis bis-aryl diamidoxime compounds
06/17/2004CA2504740A1 Dicationic 2,5-diarylfuran aza-analogs as anti-protozoan agents
06/16/2004EP1428822A2 1-phenylpiperazine derivative as modulators of dopamine neurotransmission
06/16/2004EP1427724A1 Novel use of substituted aminomethyl chromans
06/16/2004EP1427723A1 Tetrahydropyran derivatives and their use as therapeutic agents
06/16/2004EP1427722A2 Pyrrole-type compounds, compositions, and methods for treating cancer, treating viral diseases and causing immunosuppression
06/16/2004EP1427708A1 Amino-phthalazinone derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions containing them
06/16/2004EP1427707A1 Substituted indazole compounds for the treatment of inflammation
06/16/2004EP1427421A1 2,4-disubstituted pyrimidinyl derivatives for use as anticancer agents
06/16/2004EP1427417A1 3-substituted 6,7-dihydroxytetrahydroisoquinoline derivatives for use as antibacterial agents
06/16/2004EP1427416A2 3-glyoxlylamideindoles for treating cancer
06/16/2004EP1427408A2 CYCLIC HYDROXAMIC ACIDS AS INHIBITORS OF MATRIX METALLOPROTEINASES AND/OR TNF-$g(a) CONVERTING ENZYME (TACE)
06/16/2004EP1427407A2 Fatty amine drug conjugates
06/16/2004EP1351958B1 Imidazolo-5-yl-2-anilino-pyrimidines as agents for the inhibition of the cell proliferation
06/16/2004EP1341763B1 N-alkoxy-4,4-dioxy-polyalkyl-piperidine compounds, with glycidyl or alkylcarbonyl groups as functional initiators for controlled radical polymerization
06/16/2004EP1339406B1 Piperazine derivatives, their preparation and their use for treating central nervous system (cns) disorders
06/16/2004EP1282616B1 Hydroxyphenyl-piperidin-4-ylidene-methyl-benzamide derivatives for the treatement of pain
06/16/2004EP1263751B1 2-phenylpyran-4-one derivatives
06/16/2004EP1255751B1 1,3-dihydro-2h-indol-2-one derivatives and their use as ligands for v1b or v1b and v1a arginine-vasopressin receptors
06/16/2004EP1219173B1 Insecticides and acaricides
06/16/2004EP1214074B1 Dioxolane nucleoside analogs for the treatment or prevention of viral infection
06/16/2004EP1194411B1 Benzoylpyridazines
06/16/2004EP1147083B1 Arylpiperazinyl-cyclohexyl indole derivatives for the treatment of depression
06/16/2004EP0983243B1 Novel quinoline- and naphthalenecarboxamides, pharmaceutical compositions and methods of inhibiting calpain
06/16/2004EP0979079B1 Use of tetrahydropyridine derivatives to prepare medicines for treating diseases causing demyelination
06/16/2004EP0960104B1 N-(amidinophenyl)-n'-(subst.)-3h-2,4-benzodiazepin-3-one derivatives as factor xa inhibitors
06/16/2004EP0823423B1 1,4-disubstituted piperidine derivatives
06/16/2004CN1505628A Triazole compounds useful in treating diseases associated with unwanted cytokine activity
06/16/2004CN1505625A Triazole compounds useful in treating diseases associated with unwanted cytokine activity
06/16/2004CN1505624A Piperazino-derivatives and their use as pde4 inhibitor
06/16/2004CN1505617A Peptides as met-ap2 inhibitors
06/16/2004CN1505613A Substituted indoles, pharmaceutical compositions containing such indoles and their use as ppar-gamma binding agents
06/16/2004CN1505514A Combinations of aldose reductase inhibitors and cyclooxygenase-2 inhibitors
06/16/2004CN1504462A Pyrimidinyl derivatives as interleukin inhibitors
06/16/2004CN1153770C Substitued nitrogen heterocyclic ring as inhibitors of P38 protein kinase
06/16/2004CN1153766C Nitroketone compound, its preparing process and pharmaceutical composition containing same
06/16/2004CN1153764C Substituted benzylaminopiperidine compounds
06/15/2004US6750357 Rhodamine-based fluorophores useful as labeling reagents
06/15/2004US6750353 Preparation of pharmaceutically acceptable atorvastatin salts in non-crystalline form
06/15/2004US6750349 Superior gastrokinetic properties
06/15/2004US6750348 Protective effects against infection by hiv through binding to chemokine receptors, including cxcr4 and ccr5;n-(2-pyridinylmethyl)-n'-(2-(phenylureido)ethyl)-n'-(5,6,7,8-tetrahydro-8-quinolinyl)-1,4-benzenedimethanamine
06/15/2004US6750346 Chromenes as terminal end groups
06/15/2004US6750338 Process for making 5-substituted pyrazoles
06/15/2004US6750254 Nitric oxide-releasing amidine—and enamine-derived diazeniumdiolates, compositions and uses thereof and method of making same
06/15/2004US6750245 C7 carbamate substituted taxanes
06/15/2004US6750243 COMPETITIVE INHIBITORS OF TRYPSIN-LIKE SERINE PROTEASES, ESPECIALLY THROMBIN; chemical synthesis; anticoagulants; treatment of thrombosis
06/15/2004US6750242 Positive modulators of nicotinic receptor agonists
06/15/2004US6750241 Two or more ligand moieties covalently linked together by one or more linking groups enabling binding to multiple binding sites; increased efficacy, selectivity and duration; anti-proliferative and anticarcinogenic