Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
09/2004
09/30/2004CA2519372A1 Substituted cyclohexyl and piperidinyl derivates as melanocortin-4 receptor modulators
09/30/2004CA2519220A1 Amino cyclobutylamide modulators of chemokine receptor activity
09/30/2004CA2519026A1 Therapeutic and/or preventive agent for chronic skin disease
09/30/2004CA2518973A1 Methods for isolating crystalline form i of 5-azacytidine
09/30/2004CA2517446A1 6-sulfonamide quinoline and chromene derivative as androgen receptor antagonists
09/29/2004EP1461334A2 Pyrazole derived kinase inhibitors
09/29/2004EP1461330A1 3h-naphtho 2,1-b]-pyrane derivatives and the use of the same
09/29/2004EP1461321A1 3,4-di-substituted pyridazinediones as cxc chemokine receptor antagonists
09/29/2004EP1461320A2 Enantioselective transformation of alfa,beta-unsaturated ketones using chiral organic catalysts
09/29/2004EP1389202B1 2,6-substituted chroman derivatives useful as beta-3 adrenoreceptor agonists
09/29/2004EP1189881B1 Propanoic acid derivatives that inhibit the binding of integrins to their receptors
09/29/2004EP1181278B1 Cyclic amine derivatives and their uses
09/29/2004EP1165557B1 ARYL AND HETEROARYL FUSED AMINOALKYL-IMIDAZOLE DERIVATIVES: SELECTIVE MODULATORS OF GABAa RECEPTORS
09/29/2004EP1051397A4 Method for preparing an n- (aliphatic or aromatic)carbonyl]-2-aminoacetamide compound and a cyclyzed compound
09/29/2004EP1012140B1 New amidino derivatives and their use as thrombin inhibitors
09/29/2004EP0901487B9 2,3,6 trisubstituted-4(3h)-quinazolinones
09/29/2004CN1533382A 哌嗪衍生物 Piperazine derivatives
09/29/2004CN1532635A Organic light sensitive body with epoxy charge transfer compound
09/29/2004CN1168722C Diresorinyl-alkoxy-and-aryloxy-s-triazines
09/29/2004CN1168720C Aryl alkanoylpyridazines compounds
09/29/2004CN1168719C 6-phenylpyridyl-2-amine derivatives and pharmaceutical composition and use
09/29/2004CN1168704C Aryl and heteroaryl cyclopropyl oximidoether and its application as bactericide and pesticide
09/28/2004US6797820 Succinate compounds, compositions and methods of use and preparation
09/28/2004US6797714 Hypoglycemic agents; antidiabetic agents; side effect reduction
09/28/2004US6797713 1,4 substituted piperazines, 1,4 substituted piperidines, and 1-substituted,4-alkylidenyl piperidine compounds; dual acting molecules having both leukotriene inhibition properties
09/28/2004US6797712 Substituted amino-furan-2-yl-acetic acid and amino-thien-2-yl-acetic acid derivatives and their use in the treatment of migraine and pain
09/28/2004US6797710 Cardiovascular disorders; serine protease inhibitor; administering by mouth; bioavailability
09/28/2004US6797708 Enzyme inhibitors such as 4-(2-(1-benzhydryl-2-(2-((benzyl-sulfonyl)amino)ethyl)-5-chloro-1h-indol-3 -yl)ethoxy) benzoic acid, used as analgesics or antiinflammatory agents
09/23/2004WO2004081005A1 Melanin-concentrating hormone receptor antagonists and compositions and methods related thereto
09/23/2004WO2004081004A1 Substituted azetidinone compounds, formulations and uses thereof for the treatment of hypercholesterolemia
09/23/2004WO2004081003A1 Substituted azetidinone compounds, formulations and uses thereof for the treatment of hypercholeterolemia
09/23/2004WO2004080999A1 Pyrazole compounds useful in the treatment of inflammation
09/23/2004WO2004080990A1 C-glycoside derivatives and salts thereof
09/23/2004WO2004080982A1 Pyrazine compounds as transforming growth factor (tgf) inhibitors
09/23/2004WO2004080981A1 Pyrimidin-2-one compounds and their use as dopamine d3 receptor ligands
09/23/2004WO2004080980A1 2, 4- di (phenylamino) pyrimidines useful in the treatment of neoplastic diseases, inflammatory and immune system disorders
09/23/2004WO2004080977A1 4-substituted-5-cyano-1h-pyrimidin-6-(thi)ones as gsk-3 inhibitors
09/23/2004WO2004080976A1 Phthalazinone derivatives
09/23/2004WO2004080973A1 Fused tri and tetra-cyclic pyrazole kinase inhibitors
09/23/2004WO2004080972A1 Pirazole modulators of atp-binding cassette transporters
09/23/2004WO2004080969A1 Quinolinone / benzoxazinone derivatives and uses thereof
09/23/2004WO2004080968A1 6-substituted nicotinamide derivatives as opioid receptor antagonists
09/23/2004WO2004080480A1 Pharmaceutical preparations comprising acid-stabilised insulin
09/23/2004WO2004080463A1 Heterocyclic kinase inhibitors: methods of use and synthesis
09/23/2004WO2004080411A2 Melanin-concentrating hormone receptor antagonists and compositions and methods related thereto
09/23/2004WO2004050613A3 2-substituted-3-propenamide derivatives and methods of using the same
09/23/2004WO2004043884A3 Novel acylating reagents
09/23/2004WO2004041258A3 Cyclic nucleotide phosphodiesterase inhibitors, preparation and uses
09/23/2004WO2004005472A3 Inhibitors of ftsz and uses thereof
09/23/2004WO2003072552A8 Method for preparing benzisoxazole methane sulfonyl chloride and its amidation to form zonisamide
09/23/2004WO2003011219A3 Mediators of hedgehog signaling pathways, compositions and uses related thereto
09/23/2004US20040186296 Process to produce derivatives from uk-2a derivatives
09/23/2004US20040186295 G protein-coupled receptors activators such as 2-[2-(3-chlorophenyl)-2H-tetrazol-5-yl]pyridine, used as analgesics, anxiolytic, antidepressants, and for prophylaxis of psychological disorders
09/23/2004US20040186287 heterocyclic imines such as 2-(2,6-difluorophenyl)-5-phenyl-3,4-dihydro-2H-pyrrole, formed by cyclocondensation, for use as insecticides or miticides
09/23/2004US20040186284 Methods for isolating crystalline form I of 5-azacytidine
09/23/2004US20040186170 Benzofuran derivatives, pharmaceutical composition containing the same, and a process for the preparation of the active ingredient
09/23/2004US20040186168 Such as spiroadamantane on one side and 4-substituted spiro-cyclohexyl on other side; structurally simple, nontoxic, easy synthesis, potent parasiticides
09/23/2004US20040186159 used to treat glaucomatous optic neuropathy and/or lower and control intraocular pressure (IOP) associated with normal-tension glaucoma, ocular hypertension, and/or glaucoma in warm blooded animals, including man
09/23/2004US20040186156 useful for solid tumors and leukemia; auto-immune diseases such as psoriasis, alopecia and multiple sclerosis; cardiovascular diseases such as stenoses, arterioscleroses and restenoses; infectious diseases caused by unicellular parasites; nephrological diseases, neurodegenerative diseases
09/23/2004US20040186153 Pharmaceutical use of N-carbamoylazole derivatives
09/23/2004US20040186151 E.g., 2-[3-(4'-Methoxyphenyl)-propionylamino]-2-(4'-n-butoxy-3'-carboxyphenyl)-2-ethyl[4-(4'-nitrophenyl)]imidazole; inhibitors of protein tyrosine phosphatases; antidiabetic, -carcinogenic, -inflammation agents; antiallergens; infections; modulation of growth hormones/factors; Alzeimer's; obesity
09/23/2004US20040186148 E.g., 1-(pyrid-2-yl-so2-),2-((4-(isopropylphenyl)-so2-),5-(isopropoxy)benzene; antiinflammatory agents; immunomodulatory activity rheumatoid arthritis, asthma, allergy, psoriasis, Crohn's disease, systemic lupus erythematosus, multiple sclerosis, diabetes, cancer, glaucoma, osteoporosis, renal ischemia
09/23/2004US20040186140 Cyclic derivatives as modulators of chemokine receptor activity
09/23/2004US20040186134 Inhibitors of Factor Xa are useful as anticoagulants in the treatment of cardiovascular disorders associated with thromboses; e.g., 1,1-dimethylethyl 1-[1-(-2-(-3-[2-(5-Chloro-thiophen-2-yl)-ethenesulfonylamino]-2-oxo-piperidin-1-yl)-acetyl)-pyrrolidin-2- yl-methyl]-pyrrolidin-3-yl}-methyl-carbamate
09/23/2004US20040186133 preferably antagonists used in the therapeutic and/or preventive treatment of disfunctions of the heart, kidney, respiratory system, central nervous system
09/23/2004US20040186125 E.g , 3-cyclohexyl-2-furan-3-yl-1Hindole-5-carboxylic acid; hepatitis C viricides that target RNA dependent RNA polymerases (Ns5B) in mammals, an enzyme essential to viral replication; used in conjunction with an mmunomodulatory agent, such as beta -, delta - gamma -, and omega -interferon
09/23/2004US20040186119 glycogen synthase kinase (GSK-3) inhibitors; for treatment of diabetes and alzheimer's disease
09/23/2004US20040186118 Chk-, Pdk- and Akt-inhibitory pyrimidines, their production and use as pharmaceutical agents
09/23/2004US20040186116 such as 2-(7-acetylamino-1-furano-2-ylmethyl-2,4-dioxo-1,4-dihydro-2H-quinazolin-3-yl)-succinic acid; for treatment of autoimmune diseases, proliferative diseases, angiogenic disorders, and/or cancers; catheters, prosthetics
09/23/2004US20040186113 Heterocyclic amines for the treatment of conditions associated with gsk-3
09/23/2004US20040186099 Novel heterocyclic compounds, their preparation, pharmaceutical compositions containing them and their use in medicine
09/23/2004US20040186098 Method for preventing and treating hearing loss using sensorineurotrophic compounds
09/23/2004US20040186097 such as N-phenyl-3-[[4-(phenylmethyl)-1-piperidinyl]methyl]-1-piperidinecarboxamide for prevention of asthma and allergies
09/23/2004US20040186092 Tertiary carbocyclic amides such as 1-(3-Piperazin-1-yl-benzyl)-3,4-dihydro-1H-quinolin-2-one, used as serotonin receptor antagonists for prophylaxis of nervous system disorders and gastrointestinal disorders
09/23/2004US20040186090 New amidino derivatives and their use as thrombin inhibitors
09/23/2004US20040185553 Apparatus comprised of highly absorbent particles immobilized to inert matrix for removal of substances from blood products; dialysis
09/23/2004US20040185544 Batch devices for the reduction of compounds from biological compositions containing cells and methods of use
09/23/2004US20040185255 Indeno-fused photochromic naphthopyrans, naphthols and photochromic articles
09/23/2004DE10311065A1 New 1-(cyclic amino-alkyl)-pyrimidin-2(1H)-one derivatives, are selective dopamine D3 receptor ligands useful for treating CNS disorders, especially schizophrenia or depression
09/23/2004CA2518403A1 Quinolinone/benzoxazinone derivatives and uses thereof
09/23/2004CA2518398A1 Heterocyclic kinase inhibitors: methods of use and synthesis
09/23/2004CA2518194A1 6-substituted nicotinamide derivatives as opioid receptor antagonists
09/23/2004CA2517885A1 Fused tri and tetra-cyclic pyrazole kinase inhibitors
09/23/2004CA2517720A1 Pyrazine compounds as transforming growth factor (tgf) inhibitors
09/22/2004EP1460073A1 Substituted piperidine and piperazine derivatives as melanocortin-4 receptor modulators
09/22/2004EP1460072A1 Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors
09/22/2004EP1460070A1 Substituted piperidine and piperazine derivatives as melanocortin-4 receptor modulators
09/22/2004EP1460069A1 Substituted cyclohexyl and piperidinyl derivatives as melanocortin-4 receptor modulators
09/22/2004EP1460062A1 Nitrogenous cyclic ketone derivative, process for producing the same, and use
09/22/2004EP1458714A1 3,4-dihydro-1h-isoquinoloin-2-yl-derivatives
09/22/2004EP1458712A2 Novel compounds
09/22/2004EP1458703A1 Isochroman compounds for treatment of cns disorders
09/22/2004EP1458700A2 Substituted 2-phenyl benzofurans as estrogenic agents
09/22/2004EP1458691A2 Benzodiazepine derivatives, preparation thereof and use thereof
09/22/2004EP1458687A2 Pyrimidine compounds
09/22/2004EP1458686A1 Benzocyclodecane derivatives with antitumor activity
09/22/2004EP1458685A2 Substituted phenyl derivatives
09/22/2004EP1458684A2 Therapeutic heterocycles
09/22/2004EP1458679A2 Pyrrolidine derivatives as prostaglandin modulators
09/22/2004EP1458394A1 Use of oxindole derivatives in the treatment of dementia related diseases, alzheimer s disease and conditions associated with glycogen synthase kinase-3