Patents
Patents for C07D 403 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group (62,587)
06/2004
06/03/2004WO2004046120A2 Diaminotriazoles useful as inhibitors of protein kinases
06/03/2004WO2004046117A1 Pyridazinone derivatives as gsk-3beta inhibitors
06/03/2004WO2004046116A1 Novel process for the preparation of imidazolyl compounds
06/03/2004WO2004046107A1 Indole derivatives as somatostatin agonists or antagonists
06/03/2004WO2004046101A2 Cyanoguanidines and cyanoamidines as erbb2 and egfr inhibitors
06/03/2004WO2004026236A3 Cyclopentyl indole derivatives
06/03/2004WO2004022060A8 (1h-benzoimidazol-2-yl)-(piperazinyl)-methanone derivatives and related compounds as histamine h4-receptor antagonists for the treatment of inflammatory and allergic disorders
06/03/2004WO2004014868A3 Pyrimidine-2,4-dione derivatives as matrix metalloproteinase inhibitors
06/03/2004WO2003086371A3 Use of ep4 receptor ligands in the treatment of il-6 involved diseases
06/03/2004WO2003051842A3 Compositions decreasing activity of hormone-sensitive lipase
06/03/2004US20040106833 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
06/03/2004US20040106802 Novel compounds and therapeutic uses thereof
06/03/2004US20040106800 cannabinoid (cb1); treating disorders involving cannabinoid neurotransmission
06/03/2004US20040106792 Biphenyl compound
06/03/2004US20040106790 Novel compounds and method for preparing 3-methylcephams
06/03/2004US20040106669 inhibitor against type-X sPLA2 (secretary PLA2) as an active ingredient
06/03/2004US20040106667 novel specific indazoles exhibiting anticancer activity via the modulation of the activity of proteins, in particular of kinases
06/03/2004US20040106664 11-Beta-hydroxysteroid dehydrogenase 1 inhibitors useful for the treatment of diabetes, obesity and dyslipidemia
06/03/2004US20040106659 hydantoin, oxazoledione and thiazoledione (or dithiione) derivatives; e.g., 5-[1-(Biphenyl-4-yloxy)-ethyl]-5-methyl-imidazolidine-2,4-dione
06/03/2004US20040106655 pyrrolo-2yl-carbonyl-amino compounds; dipeptidyl peptidase inhibitor
06/03/2004US20040106652 such as (2S)-3,3-dimethyl-1-[2-(5-phenylpentanoyl) pyrrolidinyl]pentane-1,2-dione which has affinity for immunophilin; for treatment of neurological disorders/neurodegenerative diseases; nerve growth factors; FK binding proteins
06/03/2004US20040106645 Antagonists of melanin concentrating hormone receptor
06/03/2004US20040106634 Methods for treating or preventing an inflammatory or metabolic condition or inhibiting JNK
06/03/2004US20040106626 amidine containing compounds which inhibit serine proteases
06/03/2004US20040106620 5-Substituted-2-arylpyrazines
06/03/2004US20040106616 To treat one or more conditions responsive to capsaicin receptor modulation, such as pain, itch, urinary incontinence, cough, hiccup, and/or obesity
06/03/2004US20040106615 For treating or lessening the severity of a variety of disorders, including stroke, inflammatory disorders, autoimmune diseases such as SLE lupus and psoriasis, proliferative disorders such as cancer, and conditions associated with organ transplant
06/03/2004US20040106612 Selective inhibitor of cyclooxygenase-2 used as an antipyretic, an analgesic, and an antiinflammatory agent, with reduced side effects.
06/03/2004US20040106599 an aromatic or heteroaromatic amide compound useful as antiproliferative agent
06/03/2004US20040106598 Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting Beta-amyloid peptide release and/or its synthesis by use of such compounds
06/03/2004US20040106559 for inhibiting proteases
06/03/2004US20040106521 Pyrrolecarboxamides and pyrrolethioamides as fungicides
06/03/2004US20040106520 A pplying to plants; controlling weeds
06/03/2004DE10254092A1 New pyrimidine-4,6-dicarboxamide derivatives, are selective collagenase inhibitors useful e.g. for treating degenerative joint diseases, connective tissue disorders or cancer
06/03/2004CA2518917A1 Pyridazinone derivatives as cdk2-inhibitors
06/03/2004CA2506735A1 Indole derivatives as somatostatin agonists or antagonists
06/03/2004CA2506503A1 Cyanoguanidines and cyanoamidines as erbb2 and egfr inhibitors
06/03/2004CA2506025A1 Amino-heterocycles as vr-1 antagonists for treating pain
06/03/2004CA2506022A1 Pyridazinone derivatives as gsk-3beta inhibitors
06/03/2004CA2505789A1 Diaminotriazoles useful as inhibitors of protein kinases
06/03/2004CA2499133A1 Pyrazine compounds as crf modulators
06/02/2004EP1424063A1 Cosmetic sunscreen compositions comprising 3-(2-azacycloalkylidene)-1,3-dihydro-indol-2-one derivatives and uses thereof
06/02/2004EP1424062A1 Screening composition containing at least one dibenzoylmethane derivative and at least one 3-(2-azacycloalkylidene)-1,3-dihydro-indol-2-one; photostabilisation process
06/02/2004EP1423390A2 Purine inhibitors of phosphodiesterase (pde) 7
06/02/2004EP1423382A2 Pyrazole-derived kinase inhibitors and uses thereof
06/02/2004EP1423380A1 Pyrazole-derived kinase inhibitors and uses thereof
06/02/2004EP1423376A1 Bicyclic compound, production and use thereof
06/02/2004EP1423363A1 Oral antidiabetic agents
06/02/2004EP1423362A1 New mandelic acid derivatives and their use as thrombin inhibitors
06/02/2004EP1423122A2 Compositions and methods relating to novel benzodiazepine compounds and targets thereof
06/02/2004EP1423121A1 Cysteine protease inhibitors with 2-cyano-4-amino-pyrimidine structure and cathepsin k inhibitory activity for the treatment of inflammations and other diseases
06/02/2004EP1423120A1 2h-phthalazin-1-ones and methods for use thereof
06/02/2004EP1423110A2 Cbi analogues of cc-1065 and the duocarmycins
06/02/2004EP1423107A2 Fatty alcohol drug conjugates
06/02/2004EP1423006A1 Agonists and antagonists of 5h 3?-like receptors of invertebrate s as pesticides
06/02/2004CN1501917A Compounds useful as insecticides, compounds useful as acaricides, and processes to use and make same
06/02/2004CN1501796A Treatment of type 2 diabetes mellitus using inhibitors of dipeptidyl peptidase IV
06/02/2004CN1152030C Novel heterocyclic compounds
06/02/2004CN1151789C Use of aryl (or heteroaryl) pyrrolyl methanol derivatives
06/01/2004US6743919 2-aroylimidazole compounds for treating cancer
06/01/2004US6743810 Indol-3-yl derivatives
06/01/2004US6743795 Inhibitors for hepatitis b and acquired immune deficiency syndrome (aids) because they interfere with removal of rna strand from rna-dna hybrid formed during the reverse transcription of viral rna to dna
06/01/2004US6743793 Dp receptor antagonist; prostaglandin d
06/01/2004US6743792 Antiinflammatory agents
06/01/2004US6743791 Heterocyclic inhibitors of ERK2 and uses thereof
05/2004
05/29/2004WO2004035566A1 Cannabinoid receptor ligands and uses thereof
05/29/2004CA2502511A1 Cannabinoid receptor ligands and uses thereof
05/27/2004WO2004043950A1 Indolyl pyrazinone derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis
05/27/2004WO2004043949A1 4-substituted 1-aminocyclohexane derivatives for utilization as orl1-receptor and mu-opiate receptor ligands
05/27/2004WO2004043940A1 Phenylalanine derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
05/27/2004WO2004043926A1 Phenyl or heteroaryl amino alkane derivatives as ip receptor antagonist
05/27/2004WO2004043458A1 Bicyclic-substituted amines as histamine-3 receptor ligands
05/27/2004WO2004043369A2 Sulfonamides
05/27/2004WO2004043366A2 Sulfonamides
05/27/2004WO2004043354A2 Ophthalmic compositions for treating ocular hypertension
05/27/2004WO2004043337A2 Indole, azaindole and related heterocyclic 4-alkenyl piperidine amides
05/27/2004WO2004007482A3 Novel synthesis of irbesartan
05/27/2004WO2003088908A3 Heterocyclo inhibitors of potassium channel function
05/27/2004WO2003039549A3 Selective antibacterial agents
05/27/2004WO2003016276A3 3-substituted oxindole beta-3 agonists
05/27/2004US20040102635 Herbicides for combating weeds, preparation by mixing with extenders, surfactants; a tetrazolinone benzoyl with cyclohexyl-, isoxazole-, pyrazole-, or oxomethylene-derivatives
05/27/2004US20040102630 For therapy of cancer, auto-immune diseases, cardiovascular diseases, infectious diseases, nephrological diseases, neurodegenerative diseases and viral infections
05/27/2004US20040102510 Cancer; the compounds interact with the amino acids in the catalytic region of PKs and bind in the general space normally occupied by the adenine ring of ATP
05/27/2004US20040102509 Kinase inhibitors for the treatment of disease
05/27/2004US20040102508 Naphathalene derivatives which bind to the ep4 receptor
05/27/2004US20040102507 Use of GALR3 receptor antagonists for the treatment of depression and/or anxiety and compounds useful in such methods
05/27/2004US20040102506 Pyrazole compositions useful as inhibitors of ERK
05/27/2004US20040102502 Preventing/remedies for portal hypertension
05/27/2004US20040102500 Peroxisome proliferator activated receptor alpha agonists
05/27/2004US20040102492 Inflammation such as chronic inflammatory disease. Also disclosed are processes for preparing these compounds and pharmaceutical compositions comprising these compounds. Ar1 is carbocycle optionally substituted with one R1, and wherein Ar1
05/27/2004US20040102488 Antiinflamamtory agents; autoimmune diseases; antiarthritic agents; anticancer agents; Alzheimer's disease
05/27/2004US20040102483 Chemical compounds
05/27/2004US20040102467 Antiinflammatory agents; central nervous system disorders; antiproliferative agents
05/27/2004US20040102465 Pesticides; insecticides; fungicides
05/27/2004US20040102464 Hypotensive agents; cardiovascular disorders; anticancer agents; headaches; antihistamines; antiinflamamtory agents
05/27/2004US20040102457 Central nervous system disorders; anxiolytic agents; antidepressants; attention deficit disorders; Alzheimer's diseases
05/27/2004US20040102454 Anticancer agents; fungicides
05/27/2004US20040102450 Substituted oxoazaheterocyclyl compounds
05/27/2004US20040102448 Substituted polycyclic aryl and heteroaryl pyrazinones useful for selective inhibition of the coagulation cascade
05/27/2004US20040102437 Prevention cytokine migration; hypotensive agents; asthma therapy