Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
06/1999
06/22/1999CA1340603C Tri-aza macrocycles and metal complexes thereof
06/17/1999WO1999029693A1 Imidazonaphthyridines and their use in inducing cytokine biosynthesis
06/17/1999WO1999029686A1 Novel compounds
06/17/1999WO1999029684A1 Morpholino end-capped, hindered amine substituted aminotriazine and their use as light stabilizers
06/17/1999WO1999029674A1 Retinoic acid mimetic anilides
06/17/1999WO1999029673A1 SELECTIVE β3 ADRENERGIC AGONISTS
06/17/1999WO1999029670A2 Aminocarbonyltetralin and dihydronaphtalene derivates as thrombin inhibitors
06/17/1999WO1999029667A1 Hydroxamic acid derivatives as matrix metalloprotease (mmp) inhibitors
06/17/1999WO1999029320A1 Novel administration form comprising an acid-labile active compound
06/17/1999WO1999029318A1 Antiviral compounds
06/17/1999WO1999029311A1 Hiv/fiv protease inhibitors having a small p3 residue
06/17/1999WO1999029299A1 Novel suppository form comprising an acid-labile active compound
06/17/1999WO1999007695A3 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONIST
06/17/1999CA2314408A1 Antiviral compounds
06/17/1999CA2312999A1 Morpholino end-capped, hindered amine substituted aminotriazine and their use as light stabilizers
06/17/1999CA2312987A1 Selective .beta.3 adrenergic agonists
06/17/1999CA2312720A1 Retinoic acid mimetic anilides
06/17/1999CA2312357A1 Novel compounds
06/16/1999EP0922697A1 Substituted Pyrazolyl benzenesulfonamides and their use as cyclooxygenase II inhibitors
06/16/1999EP0922042A1 Novel piperazine containing compounds
06/16/1999EP0922036A1 Arylalkanoyl pyridazines
06/16/1999EP0922035A1 Tetrahydroisoquinoline derivatives and their pharmaceutical use
06/16/1999EP0922032A1 Herbicidal pyridinyl and pyrazolylphenyl ketones
06/16/1999EP0922028A1 Inhibitors of phospholipase enzymes
06/16/1999EP0921801A1 Inhibitors of farnesyl-protein transferase
06/16/1999EP0753003B1 Aziridine derivatives, their production and use
06/16/1999EP0752424B1 Nicotinic acid derivative and herbicide
06/16/1999EP0553218B1 Indole derivatives
06/16/1999CN1219932A Aromatic amidine derivatives useful as selective thrombin inhibitors
06/16/1999CN1043639C New piperidine compounds, process for their preparation and pharmaceutical compositions which contain them
06/15/1999US5912350 Certain aminomethyl biphenyl, aminomethyl phenyl pyridine and aminomethyl phenyl pyrimidine derivatives; novel dopamine receptor subtype selective ligands
06/15/1999US5912342 Synthesis of combinatorial libraries by computer controlled robot
06/15/1999US5912260 Gastrin and CCK antagonists
06/15/1999US5912256 0-(4-indolyloxy)-3-(4-hydroxy-4-naphthylpiperidin-1-yl)propane s
06/15/1999US5911913 1-fluoroisoquinoline derivatives and the use thereof in liquid crystalline mixtures
06/15/1999CA2155664C Oxindole 1-[n-(alkoxycarbonyl)]carboxamides and 1-(n-carboxamido)carboxamides as antiinflammatory agents
06/15/1999CA2087032C Diphenylmethyl piperazine derivatives
06/10/1999WO1999028359A1 Preparation for prevention and healing of inflammation affections
06/10/1999WO1999028315A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof
06/10/1999WO1999028314A1 Inhibitors of farnesyl-protein transferase
06/10/1999WO1999028313A1 Inhibitors of farnesyl-protein transferase
06/10/1999WO1999028303A1 Process of preparing substituted pyrimidinones
06/10/1999WO1999028302A1 Substituted phenyl uracils
06/10/1999WO1999028301A1 Substituted pyrimidine and pyridine herbicides
06/10/1999WO1999028300A1 Substituted imidazole derivatives having agonist-like activity at alpha 2b or 2b/2c adrenergic receptors
06/10/1999WO1999028299A1 1,2-dihydro-2-oxoquinoline derivatives
06/10/1999WO1999028297A1 Substituted indoles, having a thrombin inhibiting effect
06/10/1999WO1999027933A1 Inhibitors of farnesyl-protein transferase
06/10/1999DE19754490A1 Durch einen Aminocarbonylrest substituierte Bicyclen, ihre Herstellung und ihre Verwendung als Arzneimittel By an aminocarbonyl radical substituted bicyclic compounds, their preparation and their use as medicaments
06/10/1999DE19753522A1 Substituierte Indole, ihre Herstellung und ihre Verwendung als Arzneimittel Substituted indoles, their preparation and their use as medicaments
06/10/1999CA2313055A1 1,2-dihydro-2-oxoquinoline derivatives
06/10/1999CA2312366A1 Inhibitors of farnesyl-protein transferase
06/10/1999CA2312361A1 Inhibitors of farnesyl-protein transferase
06/10/1999CA2312338A1 Process of preparing substituted pyrimidinones
06/10/1999CA2312334A1 Substituted imidazole derivatives having agonist-like activity at alpha 2b or 2b/2c adrenergic receptors
06/10/1999CA2311928A1 Inhibitors of farnesyl-protein transferase
06/10/1999CA2311557A1 Substituted phenyl uracils
06/10/1999CA2310629A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof
06/09/1999EP0921120A1 Selective beta 3 adrenergic agonists
06/09/1999EP0921119A1 Pyrrole derivatives, process for their preparation and pharmaceutical compositions containing them
06/09/1999EP0920865A1 Pharmaceutical compositions containing Norastemizole
06/09/1999EP0920428A1 Non-symmetrical bis-heteroarylmethoxyphenylalkyl carboxylates as inhibitors of leukotriene biosynthesis
06/09/1999EP0920426A1 New thiazole derivatives with phosphodiesterase-inhibiting effect
06/09/1999EP0920425A1 Substituted 4-(1h-benzimidazol-2-yl-amino)piperidines useful for the treatment of allergic diseases
06/09/1999EP0920424A1 Non-peptide bombesin receptor antagonists
06/09/1999EP0920419A1 Compounds, compositions and methods for treating influenza
06/09/1999EP0920416A1 Naphtholactams and lactones as bone morphogenetic protein active agents
06/09/1999EP0920318A1 Aryloxy- and arylthiosubstituted pyrimidines and triazines and derivatives thereof
06/09/1999EP0799223B1 Piperidineacetic acid derivatives useful as fibrinogen antagonist agent
06/09/1999CN1219172A Novel benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists
06/09/1999CN1219168A Quinoline carboxamides as TNF inhibitors and as PDC-IV inhibitors
06/09/1999CN1219131A Quinoline carboxamides as TNF inhibitors and as PDC-IV inhibitors
06/09/1999CN1219125A Intracoronary stents fixing mould containing quinazolinone derivatives
06/09/1999CN1218801A Tri-substituted imidazoles, and process of their preparation and using the same and having their pharmic composition
06/08/1999US5910593 Highly selective process for the preparation of enantiomerically pure phenylsubstituted 1,4-dihydropyridine-3,5-dicarboxylic acid derivatives
06/08/1999US5910586 Tricyclic aminoalkylcarboxamides; dopamine D3 receptor subtype specific ligands
06/08/1999US5910506 Imidazole derivatives as anti-HIV agents
06/08/1999US5910498 Pyridonecarboxylic acid derivatives or salts thereof and antibacterial agents comprising the same as active ingredient
06/08/1999CA2089972C Sulfonamidocarboxamides
06/08/1999CA1340588C Amino acid derivatives
06/03/1999WO1999026944A1 New compounds which are p2-purinoceptor 7-transmembrane (tm) g-protein coupled receptor antagonists
06/03/1999WO1999026943A1 Thrombin receptor antagonists
06/03/1999WO1999026941A1 Substituted amidinoaryl derivatives and their use as anticoagulants
06/03/1999WO1999026940A2 Method for producing 8-methoxy-quinoline carboxylic acids
06/03/1999WO1999026933A1 Substituted amidinoaryl derivatives and their use as anticoagulants
06/03/1999WO1999026930A2 Benzylidene pyrazolones and use as herbicide
06/03/1999WO1999026926A1 Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitors
06/03/1999WO1999026924A1 Substituted oximes as neurokinin antagonists
06/03/1999WO1999026921A1 SUBSTITUTED β-ALANINE DERIVATIVES AS CELL ADHESION INHIBITORS
06/03/1999WO1999026909A2 Alpha-hydroxy, -amino and -fluoro derivatives of beta-sulphonyl hydroxamic acids as matrix metalloproteinases inhibitors
06/03/1999WO1999026659A1 Combination of an aldose reductase inhibitor and a glycogen phosphorylase inhibitor
06/03/1999WO1999010312B1 N-alkanoylphenylalanine derivatives
06/03/1999WO1999002502A3 Sulphonamide derivatives being 5-ht6 receptor antagonists and process for their preparation
06/03/1999CA2311969A1 Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitors
06/03/1999CA2310401A1 Alpha-hydroxy, -amino and -halo derivatives of beta-sulfone hydroxamates as matrix metalloproteinase inhibitors
06/03/1999CA2310087A1 Benzylidene pyrazolones and use as herbicide
06/03/1999CA2310069A1 Combination of an aldose reductase inhibitor and a glycogen phosphorylase inhibitor
06/03/1999CA2309341A1 Substituted .beta.-alanine derivatives as cell adhesion inhibitors
06/02/1999EP0919553A1 cis-SUBSTITUTED AMINOCYCLOPROPANE DERIVATIVES
06/02/1999EP0919233A1 Therapeutic agent for kidney diseases