Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
08/1999
08/19/1999WO1999024024A3 Treatment of t-helper cell type 2 mediated immune diseases with retinoid antagonists
08/19/1999WO1999021832A3 Orally-active nipecotamide glycolamide esters for the treatment of thrombosis disorders
08/19/1999WO1999015894A3 Method of identification of leads or active compounds
08/19/1999WO1998052514A3 Treatment of hepatic cirrhosis
08/19/1999DE19806438A1 New pyrimidinyloxy-propionic acid derivatives useful as endothelin receptor antagonists in treatment of e.g. cardiac insufficiency, restenosis, hypertension, kidney failure, asthma and prostate cancer
08/19/1999CA2321146A1 Novel acetamide derivative and use thereof
08/19/1999CA2320378A1 Cyclic dipeptides and azetidinone compounds and their use in treating cns injury and neurodegenerative disorders
08/19/1999CA2320319A1 1,4-dihydropyridine derivatives
08/18/1999EP0936216A1 Novel acetamide derivatives and protease inhibitors
08/18/1999EP0935465A1 Novel substituted imidazole compounds
08/18/1999CN1226246A Noval tricyclic N-cyanoimines useful as inhibitors of farnesyl-protein transferase
08/18/1999CN1226245A Compounds with pharmacologically active, preparation method and use thereof
08/18/1999CN1226244A Carbanilides used as pesticides
08/18/1999CN1226238A Sulphonyl-mercapto-triazolyl derivative and their use as microbiocides
08/18/1999CN1226237A Thiocyano-triazolyl derivatives and their use as microbicides
08/18/1999CN1226231A Process for preparing 3-pyrroline-2-carboxylic acid derivative
08/18/1999CN1044707C Substituted aminoalkylaminopyridine, preparation method, its use and medicinal composition containing same compound
08/17/1999US5939587 N-protected/N-substituted-beta-amino hydroxy sulfonates
08/17/1999US5939559 Herbicides from pyrazole ketones
08/17/1999US5939557 Inhibitors of farnesyl-protein transferase
08/17/1999US5939462 NPY5 receptor antagonists and methods for using same
08/17/1999US5939449 Novel compounds having high affinity for the neurotensin receptors
08/17/1999US5939443 Selective β3 adrenergic agonists
08/17/1999US5939441 Substituted pyridylpyrazoles
08/17/1999US5939440 Fungicides and bactericides
08/17/1999US5939439 Enzyme inhibitors in carriers for ras proteins
08/17/1999US5939436 Pyrazole compounds with piperidine groups for treatment of schizophrenia and depression
08/17/1999US5939426 Also for motion sickness and vertigo
08/17/1999US5939416 Inhibit ras function, use for treating tumor cells expressing an activated ras oncogene in mammals
08/17/1999US5939413 Tachykinin mediated diseases in humans for respiratory system disorders like asthma, bronchitis, rhinitis or eye diseases or skin disorders
08/17/1999US5939268 Diels-alder reaction product of a diene and a dienophile; chemical intermediates for drugs, solid phase synthesis
08/17/1999CA2195622C Process for preparing trans-piperidine-2,5-dicarboxylates
08/17/1999CA1340706C Process for producing 1-substituted aryl-1,4-dihydro-4-oxonaphthyridine derivative, intermediates therefor and processes for producing the intermediates
08/12/1999WO1999040083A2 Bifunctional tryptase inhibitors
08/12/1999WO1999040082A2 2-(pyrazolyloxy)-pyridin-3-ylacetic acid derivatives, agents containing the same and use thereof against noxious fungi and animal parasites
08/12/1999WO1999040080A1 Hydroxamic and carboxylic acid derivatives
08/12/1999WO1999040075A1 Sulfonamide derivatives, process for producing the same and utilization thereof
08/12/1999WO1999040073A2 Tryptase inhibitors
08/12/1999WO1999040072A1 Five-membered, benzo-condensed heterocycles used as antithrombotic agents
08/12/1999WO1999040071A1 Urocanic acid derivatives
08/12/1999WO1999040068A2 2-aminoquinoline derivatives having d4-agonistic activity
08/12/1999WO1999040064A1 Biphenylsulfonyl cyanamides, method for the production thereof and their utilization as a medicament
08/12/1999WO1999026940A3 Method for producing 8-methoxy-quinoline carboxylic acids
08/12/1999WO1999006032A3 Oral pharmaceutical preparation comprising an antiulcer activity compound, and process for its production
08/12/1999DE19851299A1 Tryptase-Inhibitoren Tryptase inhibitors
08/12/1999DE19804486A1 2-(Pyrazolyloxy)-pyridin-3-ylessigsäure- Derivate, sie enthaltende Mittel und ihr 2- (pyrazolyloxy) pyridine-3-ylessigsäure- derivatives, compositions containing them and their
08/12/1999CA2319555A1 Biphenylsulfonyl cyanamides, method for the production thereof and their utilization as a medicament
08/12/1999CA2319494A1 5-membered heterocyclic condensed benzoderivatives, the preparation thereof and their use as pharmaceuticals
08/12/1999CA2319060A1 Urocanic acid derivatives
08/12/1999CA2317476A1 Hydroxamic and carboxylic acid derivatives
08/12/1999CA2317017A1 Sulfonamide derivatives, their production and use
08/11/1999EP0934934A2 Methods of preparing substituted 3-phenyl- and 3-pyridyl-4(3H)-quinazolinones and atropisomers thereof
08/11/1999EP0934931A2 3-Benzylidene-2-indolinones and their analogues as tyrosine kinase activity modulators
08/11/1999EP0934316A1 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
08/11/1999EP0934313A1 N-substituted azaheterocyclic compounds
08/11/1999EP0934312A1 1,4-disubstituted piperazines
08/11/1999EP0934311A2 New heterocyclylmethyl-substituted pyrazol derivates
08/11/1999EP0934310A1 THIO ACID DERIVED MONOCYCLIC $i(N)-HETEROCYCLICS AS ANTICOAGULANTS
08/11/1999EP0934309A1 New pyridyl alkane acid amides as cytostatics and immunosuppressives
08/11/1999EP0934308A1 3-pyridyloxymethyl heterocyclic ether compounds useful in controlling chemical synaptic transmission
08/11/1999EP0934307A1 Substituted azabicylic compounds and their use as inhibitors of the production of tnf and cyclic amp phosphodiesterase
08/11/1999EP0934306A1 N-substituted azaheterocyclic compounds
08/11/1999EP0934304A1 2-pyrimidineamine derivatives and processes for their preparation
08/11/1999EP0934303A2 Compounds useful for inhibition of farnesyl protein transferase
08/11/1999EP0934293A1 Novel compounds and compositions for treating diseases associated with tryptase activity
08/11/1999EP0934291A1 Protease inhibitors
08/11/1999EP0934285A1 Substituting 2-amino-4-alkylamino-1,3,5-triazine as herbicide
08/11/1999EP0934284A1 Substituted 2-amino-4-alkylamino-1,3,5-triazines as herbicides
08/11/1999EP0934283A2 Arthropodicidal and fungicidal cyclic amides
08/11/1999EP0934282A1 1,4-benzodiazepinones and their uses as cck antagonists
08/11/1999EP0934281A1 1-phenyl-benzimidazole compounds and their use as baga- a? receptor modulators
08/11/1999EP0934276A1 Anthranilic acid derivatives as multi drug resistance modulators
08/11/1999EP0934274A1 Substituted pyridines and biphenyls as anti-hypercholesterinemic, anti-hyperlipoproteinemic and anti-hyperglycemic agents
08/11/1999EP0934273A1 New derivates from piperidine-keto acid, their preparation and use
08/11/1999EP0934270A1 A method of treating cancer
08/11/1999EP0934265A1 Amidinophenyl-pyrrolidines, -pyrrolines, and -isoxazolidines and derivatives thereof
08/11/1999EP0934264A1 Pyrrolidinyl and pyrrolinyl ethylamine compounds as kappa agonists
08/11/1999EP0934263A1 Heterocyclic thioesters and ketones
08/11/1999EP0934080A2 1,3-bis-(n-lactamyl) propane and the pharmaceutical and cosmetic use thereof
08/11/1999EP0934068A1 Compounds and methods
08/11/1999EP0934058A2 Stable drug form for oral administration with benzimidazole derivatives as active ingredient and process for the preparation thereof
08/11/1999EP0584223B1 Novel immunosuppressive compounds
08/11/1999CN1225629A Novel pyrrole derivatives
08/10/1999US5936123 Compounds such as 3-isopropyl-4-hydrazinobenzoic acid and its salts
08/10/1999US5936098 Process for producing indoline compounds and intermediates for the production of the same
08/10/1999US5936089 Dipeptides which promote release of growth hormone
08/10/1999US5935989 N-linked ureas and carbamates of heterocyclic thioesters
08/10/1999US5935986 Pesticides, fungicides; etherification
08/10/1999US5935985 Phenoxyacetic acid derivatives
08/10/1999US5935982 Methods of treating retroviral infection and compounds useful therefor
08/10/1999US5935981 α-unsaturated amines, their production and use
08/10/1999US5935977 Substituted vinyl pyridine derivative and drugs containing the same
08/10/1999US5935976 Viricides, hiv
08/10/1999US5935974 Diphenylmethylene piperidine derivatives
08/10/1999US5935966 Compounds that block the activation of transcription factors through inhibition of a family of specific kinases, decreasing proinflammatory proteins to treat autoimmune diseases and as general antiinflammatory agents
08/10/1999US5935961 Compounds such as n-methyl 2-(2-(6'-(3?,4?-dichlorophenyl)-pyridazin-3'-on-2'yl)-methylphenyl)-2 -methoxyiminoacetamide useful against powdery mildew, blight in cucumbers, tomatoes, and wheat for example
08/10/1999US5935957 Compounds, compositions and methods for treating influenza
08/10/1999US5935955 Substituted 3,6-dibenzylidene-2,5-piperazinediones, modulators of multidrug resistance
08/10/1999US5935954 Compounds with improved multi-drug resistance activity
08/10/1999US5935952 Quinolone- or naphthylidone-carboxylic acid derivates or their salts