Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
02/1999
02/11/1999WO1999006361A2 N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases
02/11/1999WO1999006049A1 Integrin receptor antagonists
02/11/1999WO1999006042A1 Caspases and apoptosis
02/11/1999WO1999006032A2 Oral pharmaceutical preparation comprising an antiulcer activity compound, and process for its production
02/11/1999CA2298668A1 Caspases and apoptosis
02/11/1999CA2298544A1 Integrin receptor antagonists
02/11/1999CA2297757A1 Caspases and apoptosis
02/11/1999CA2296282A1 Substituted 2-(benzoaryl)pyridines
02/11/1999CA2295945A1 Heterocyclic derivatives which inhibit factor xa
02/10/1999EP0895475A1 Vitronectin receptor antagonists
02/10/1999CN1207738A Substd. aminocycloalkylpyrrolidine derivs.
02/10/1999CN1207735A Triazine derivs.
02/10/1999CN1207734A Metalloproteinase inhibitors, pharmaceutical compositions contg. them and their pharmaceutical uses, and methods and intermediates useful for their preparation
02/10/1999CN1207729A Quinoline-4-carboxamide derivs., their preparation and their use as neurokinin 3 (NK-3)- and neurokinin 2 (NK-2) receptor antagonists
02/10/1999CN1207727A Substd. aryl or heteroarylamides having retinoid-like biological activity
02/10/1999CN1207291A Use of substituted 2,4-imidazolidinedione compounds as analgesics
02/09/1999US5869685 Serotonin reuptake inhibitors
02/09/1999US5869680 Reacting a oxazolidine derivative with protected hydroxy-taxol; decyclization and amination
02/09/1999US5869675 Lactacystin derivatives
02/09/1999US5869674 Arylpyrazoles as leukotriene inhibitors
02/09/1999US5869670 7-(4-aminomethyl-3-methyloxyiminopyrrolidin-1-yl)-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid and the process for the preparation thereof
02/09/1999US5869663 Intermediates for neurokinin receptor antagonists
02/09/1999US5869660 From aromatic s(o)x substitituted isonitriles and heterocyclic-substituted imines
02/09/1999US5869655 Diamine compounds, methods of making same, method of use of same and intermediates
02/09/1999US5869517 2- (dihydro)pyrazol-3'-yloxymethylene!anilides, their preparation and their use
02/09/1999US5869516 4-(arylaminomethylene)-2,4-dihydro-3-pyrazolones
02/09/1999US5869504 Pesticidal tetrazole derivatives
02/09/1999US5869502 Treating depression, obsessive compulsive disorder, stuttering, trichotillomania
02/09/1999US5869501 Amidinonaphthyl derivative or salt thereof
02/09/1999US5869491 Pesticides
02/09/1999US5869490 Adminstering to treat brain dopamine dysregulation; schizophrenia
02/09/1999US5869489 Trypthophan ureas as neurokinnin antagonists
02/09/1999US5869488 Piperazino derivatives as neurokinin antagonists
02/09/1999US5869483 Tricyclic benzazepine vasopressin antagonists
02/09/1999US5869481 Treating epileptic disorders
02/09/1999CA2163274C Intermediates for producing neuroleptic perhydro-1h-pyrido¬1,2-a| pyrazines
02/04/1999WO1999005139A1 2-[pyrazolyl and triazolyl-3'-oxymethylene]-phenyl-isoxazolones, triazolones and tetrazolones as pesticides and fungicides
02/04/1999WO1999005138A1 Heterocyclic compounds and antitumor agent containing the same as active ingredient
02/04/1999WO1999005121A1 Derivatives of acyl-piperazinil-pyrimidins, preparation thereof and application as medicaments
02/04/1999WO1999005117A1 Hydantoin derivatives having an inhibitory activity for farnesyl transferase
02/04/1999WO1999005116A1 Nitrophenyl-sulfonyl-imidazoles and use thereof for controlling vegetable and animal pests
02/04/1999WO1999005113A1 Substituted 6-phenylphenanthridines
02/04/1999WO1999005111A1 Novel tetrazole derivatives
02/04/1999WO1999005104A1 Indole compounds as cox-2 inhibitors
02/04/1999WO1999004794A1 Cyclic amine modulators of chemokine receptor activity
02/04/1999WO1999004775A2 Method of treating dopaminergic and gaba-nergic disorders
02/04/1999DE19732846A1 Bisiminosubstituierte Phenylverbindungen Bisiminosubstituierte phenyl compounds
02/04/1999CA2297923A1 Novel tetrazole-substituted 6-phenyl-pheanathridines as pde inhibitors
02/04/1999CA2297410A1 Method of treating dopaminergic and gaba-nergic disorders
02/04/1999CA2296729A1 2-[pyrazolyl and triazolyl-3'-oxymethylene]-phenyl-isoxazolones, triazolones and tetrazolones as pesticides and fungicides
02/04/1999CA2296314A1 Cyclic amine modulators of chemokine receptor activity
02/03/1999EP0894796A1 Imidazolines substituted with a heterocyclic ring as alpha-2 antagonists
02/03/1999EP0894795A1 Benzimidazole, benzoxazole and benzothiazole derivatives, their preparation and pharmaceutical compositions containing them
02/03/1999EP0894792A1 Heterocycle-substituted benzene derivatives and herbicides
02/03/1999EP0894497A1 Use of substituted imidazolidin-2,4-diones as analgesics
02/03/1999EP0894088A1 Substituted sulfonic acid n- (aminoiminomethyl)phenylalkyl]-azaheterocyclamide compounds
02/03/1999EP0894085A1 Benzyl(idene)-lactam derivatives, their preparation and their use as selective (ant)agonists of 5-ht1a- and/or 5-ht1d receptors
02/03/1999EP0894084A1 Cinnamic acid derivatives and their use as integrin antagonists
02/03/1999CN1207097A Novel substituted 4-(1H-benzimidazol-2-YL) [1,4] diazepanes useful for the treatment of allergic diseases
02/03/1999CN1207096A 3-azetidinylalkylpiperidines or-pyrrolidines as tachykinin antagonists
02/03/1999CN1206712A Heterocyclic compound, preparation process thereof and medicinal composition containing same
02/03/1999CN1206589A Process for preparing medicine composition
02/03/1999CN1041923C Piperzine derivatives and preparation process and usage thereof
02/03/1999CN1041921C Bicyclic fibrinogen antagonists
02/03/1999CN1041920C Glycerin derivative and its pharmacological use
02/03/1999CN1041919C N-(3-piperidinylcarbonyl)-beta-alanine derivatives as PAF antagonists
02/02/1999US5866598 4h-carbazol-4-ones
02/02/1999US5866589 Alkyl substituted piperadinyl and piperazinyl anti-AIDS compounds
02/02/1999US5866583 Substituted 2,4-diaminopyrimidines
02/02/1999US5866579 Imidazole and imidazoline derivatives and uses thereof
02/02/1999US5866577 Aromatic amidine derivatives and salts thereof
02/02/1999US5866573 Pyrazinone thrombin inhibitors
02/02/1999US5866572 Receptor tyrosine kinase inhibitory properties, treatment of proliferative diseases such as cancer.
02/02/1999US5866568 Heterocyclic compounds
02/02/1999US5866567 Diazepinones, their production and use
02/02/1999US5866562 Ring-bridged bis-quinolines
02/02/1999US5866335 Preparation of derivatized 10,10'-substituted-9,9'-biacridine luminescent molecules and signal solutions
02/02/1999US5866293 Containing diazo compound and pyrazolone coupler; storage stability
01/1999
01/31/1999CA2244200A1 Use of substituted 2,4-imidazolidinedione compounds as analgesics
01/30/1999CA2244438A1 New benzimidazole, benzoxazole and benzothiazole derivatives, their preparation process and the pharmaceutical compositions containing them
01/30/1999CA2244435A1 New heterocyclic compounds, their preparation process and the pharmaceutical compounds containing them
01/28/1999WO1999003854A1 Crystal modification of a n-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use
01/28/1999WO1999003837A1 2-substituted imidazoles useful in the treatment of inflammatory diseases
01/28/1999WO1999003498A1 USE OF FVIIa OR FVIIai FOR THE TREATMENT OF ADVERSE CONDITIONS RELATED TO THE FVIIa MEDIATED INTRACELLULAR SIGNALLING PATHWAY
01/28/1999WO1999003472A1 Peripherally acting anti-pruritic opiates
01/28/1999WO1999003468A1 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith
01/28/1999WO1998049138A3 Vitamin d3 analogs with bis c-20 side chains
01/28/1999WO1998046589A3 Indazole amide compounds as serotoninergic agents
01/28/1999DE19731153A1 2-(Pyrazolyl- und Triazolyl-3'-oxymethylen)-phenyl-isoxazolone und -triazolone, Verfahren zu ihrer Herstellung und ihre Verwendung 2- (pyrazolyl and triazolyl-3'-oxymethylene) phenyl-isoxazolones and -triazolone, processes for their preparation and their use
01/28/1999CA2295021A1 2-substituted imidazoles useful in the treatment of inflammatory diseases
01/28/1999CA2289055A1 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith
01/28/1999CA2288833A1 Peripherally acting anti-pruritic opiates
01/27/1999EP0893446A1 Cephem compounds and drugs containing the compounds
01/27/1999EP0893442A1 Lymph-absorbable imidazole derivatives
01/27/1999EP0892797A1 Inhibitors of farnesyl protein transferase
01/27/1999EP0892796A1 Isatin derivatives as acetylcholinesterase inhibitors and analgesics
01/27/1999EP0892795A1 Piperidinylpyramidine derivatives
01/27/1999EP0892794A1 Acylated n-hydroxy methyl thalidomide prodrugs with immunomodulator action
01/27/1999EP0892791A1 Substituted benzenesulfonamide derivatives as prodrugs of cox-2 inhibitors
01/27/1999EP0892790A1 New quinazoline-4-amino-2-(piperidine-1-yl-4-substituted) derivatives having anti-hypertensive activity, a method for their preparation and their pharmaceutical use