Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
10/1999
10/21/1999WO1999043643A3 Metal-catalyzed arylations and vinylations of hydrazines, hydrazones, hydroxylamines and oximes
10/21/1999WO1999040082A3 2-(pyrazolyloxy)-pyridin-3-ylacetic acid derivatives, agents containing the same and use thereof against noxious fungi and animal parasites
10/21/1999DE19817459A1 New heterocyclic amide derivatives useful as cysteine protease inhibitors for treating neurodegenerative diseases, neuronal damage, stroke, cranial trauma, Alzheimer's disease, etc.
10/21/1999DE19817265A1 Treating hepatitis B using new or known dihydropyrimidine derivative antiviral agents
10/21/1999DE19817264A1 New dihydropyrimidine derivatives and their corresponding mesomers useful as antiviral agents
10/21/1999DE19816983A1 New bicyclic heteroaromatic amidine or nitrile compounds, used as thrombin inhibitors, antithrombotic agents or intermediates
10/21/1999DE19816882A1 Use of known and new triazolone derivatives as medicaments, especially for treatment of neurodegenerative disorders and cerebral ischemia
10/21/1999DE19816624A1 Neue substituierte Indolinone, ihre Herstellung und ihre Verwendung als Arzneimittel New substituted indolinones, their preparation and their use as medicaments
10/21/1999CA2328211A1 Substituted pyrrolidine hydroxamate metalloprotease inhibitors
10/21/1999CA2327695A1 Amine compounds, their production and their use as somatostatin receptor antagonists or agonists
10/21/1999CA2327488A1 Amidine compounds
10/21/1999CA2326665A1 Heterocyclic glycyl beta-alanine derivatives as vitronectin antagonists
10/21/1999CA2325559A1 Non-endogenous, constitutively activated human serotonin receptors and small molecule modulators thereof
10/20/1999EP0950657A2 Substituted carbazoles, process for their preparation and their use as sPLA2 inhibitors
10/20/1999EP0950057A1 3-pyridyl enantiomers and their use as analgesics
10/20/1999EP0950056A2 N-(pyridinylamino)isoindolines and related compounds
10/20/1999EP0950049A1 Diphenyl alkyl-tetrahydropyridines, process for their preparation, and pharmaceutical compositions containing them
10/20/1999EP0950048A1 1-phenylalkyl-1,2,3,6-tetrahydropyridines for treating alzheimer's disease
10/20/1999EP0950047A1 Indolin-2-one derivatives, method for preparing them and pharmaceutical compositions containing them
10/20/1999EP0950046A1 3,4-disubstituted azetidin-2-one derivatives useful as cysteine proteinase regulators
10/20/1999EP0949865A1 The use of cd4-binding small molecules to inhibit immune responses
10/20/1999CN1232462A Muscarinic antagonists
10/20/1999CN1232457A 1,4-heterocyclic metalloprotease inhibitors
10/20/1999CN1232451A Substd. cyclic amine metalloprotease inhibitors
10/20/1999CN1232450A 2- and 2,5-substd. phenylketoenols
10/20/1999CN1232399A Inhibitors of cysteine protease
10/20/1999CN1232397A Use of H+, K+-ATPase inhibitor in treatment of nasal polyps
10/20/1999CN1232032A Substd. 1,2,3,4-tetrahydro-5-nitro-pyrimidines
10/20/1999CN1045775C Substd. nitropyrimidines, their preparing method and use in insecticides
10/20/1999CN1045774C Substd. arylthioalkylthiopyridines, their preparing method and pharmaceutical use
10/20/1999CN1045773C Preparation method of pyridine deriv.
10/20/1999CN1045772C Polyazacycloalkanes as dichelants
10/20/1999CN1045770C Method for preparation of 1-biphenylmethyl imidazole derivs.
10/20/1999CN1045769C Process for preparing sulfurous derivs. of imidazole
10/20/1999CN1045768C Angiotension II antagonists compounds, preparing method and use thereof
10/19/1999US5969184 Amide compounds
10/19/1999US5969141 Intermediates for 7-amino-1-cyclopropyl-6,8-dihalogeno-1,4-dihydro-4-oxo-3-quinolinecarbox ylic acid antibacterial agents
10/19/1999US5969140 Aminopyridine derivatives of naphthalene for treatment of asthma and bronchoconstrictor inhibitors
10/19/1999US5969139 Inhibitors of herpes simplex virus thymidine kinase
10/19/1999US5968977 Ketonitrile derivatives and antibacterial agent and drugs containing the same
10/19/1999US5968967 Pyrazolones derivatives
10/19/1999US5968959 Administering phospholamban inhibitor
10/19/1999US5968956 Substituted piperidine derivative and medicine comprising the same
10/19/1999US5968953 For side effect reduction
10/19/1999US5968952 Farnesyl transferase inhibiting 2-quinolone derivatives
10/19/1999US5968951 Benzenesulfonamide derivatives as bradykinin antagonists
10/19/1999US5968944 Substituted pyrazoles as corticotropin-releasing factor (CRF) antagonists
10/19/1999US5968929 Piperazino derivatives as neurokinin antagonists
10/19/1999US5968924 Benzo-fused lactams promote release of growth hormone
10/19/1999US5968923 (Azetidin-1-ylalkyl) lactams as tachykinin antagonists
10/19/1999CA2197298C Novel pyrimidine derivatives and processes for the preparation thereof
10/19/1999CA1340793C Process for producing 1-substituted aryl-1-4-dihydro-4-oxonaphthyridine derivative, intermediates therefor and processes for producing the intermediates
10/17/1999CA2269262A1 Substituted tricyclics
10/14/1999WO1999051590A1 Substituted indolinones as kinase inhibitors
10/14/1999WO1999051589A1 Substituted piperidines, method for their preparation and their use as pesticides and fungicides
10/14/1999WO1999051588A1 Quinolonecarboxylic acid derivatives or salts thereof
10/14/1999WO1999051582A1 Nitrogenous heterocyclic compounds
10/14/1999WO1999051580A1 Pyrazole inhibitors of cytokine production
10/14/1999WO1999051578A1 Biocidal benzylbiphenyl derivatives
10/14/1999WO1999051575A1 N-aryloxyethyl-indoly-alkylamines for the treatment of depression (5-ht1a receptor active agents)
10/14/1999WO1999051572A1 Sulfonamide derivatives
10/14/1999WO1999051564A1 Propanolamine derivatives
10/14/1999WO1999051224A1 Indolyl-3-glyoxylic acid derivatives with antitumoral activity
10/14/1999WO1999051215A2 Immunosuppressive imidazole derivatives and their combination preparations with tacrolimus or cyclosporins
10/14/1999WO1999045011A8 Glycine transport inhibitors
10/14/1999DE19909541A1 New pyrimidine derivatives useful as herbicides, especially for selective weed control
10/14/1999DE19814838A1 Indolyl-3-glyoxylsäure-Derivate mit Antitumorwirkung Indolyl-3-glyoxylic acid derivatives having anti-tumor activity
10/14/1999CA2327359A1 N-aryloxyethyl-indoly-alkylamines for the treatment of depression (5-ht1a receptor active agents)
10/14/1999CA2327290A1 Sulfonamide derivatives
10/14/1999CA2327185A1 Pyrazole inhibitors of cytokine production
10/14/1999CA2326159A1 Biocidal benzylbiphenyl derivatives
10/13/1999EP0949261A1 Substituted piperidinedione derivatives and herbicides
10/13/1999EP0949260A1 Acid-addition salts of optically active piperidine compound and process for producing the same
10/13/1999EP0949259A1 N-hydroxyurea derivatives and medicinal compositions containing the same
10/13/1999EP0949249A1 Process for producing imidazole derivatives
10/13/1999EP0948497A2 Substituted pyrimidine compounds and their use
10/13/1999EP0948496A2 Substituted pyrimidinone and pyridone compounds and methods of use
10/13/1999EP0948495A1 Aryl and heteroaryl substituted fused pyrrole antiinflammatory agents
10/13/1999EP0948487A1 Pesticidal 1-aryl and pyridylpyrazole derivatives
10/13/1999EP0948486A1 Pesticidal 1-arylpyrazoles
10/13/1999EP0948485A1 Pesticidal 1-arylpyrazoles
10/13/1999EP0948483A1 Farnesyl transferase inhibitors
10/13/1999EP0948257A1 Triaryl substituted imidazoles, compositions containing such compounds and methods of use
10/13/1999EP0936912A4 Inhibitors of cysteine protease
10/13/1999EP0579618B1 Pyridine- and imidazole-derived agents for cardiovascular diseases
10/13/1999CN1231665A Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
10/13/1999CN1231663A Arthropodicidal and fungicidal cyclic amides
10/13/1999CN1231662A Quinazoline derivatives and pharmaceutical compositions containing them
10/13/1999CN1231287A Benzosulfone derivatives
10/13/1999CN1231286A 1,2-Di-substituted piperidine derivative, hair growth promoter and external composition for skin using the same
10/13/1999CN1045597C Alkylenediamine derivatives having heterocyclic group and medicinal composition thereof
10/13/1999CN1045595C Process for the preparation of the intermediates used in the synthesis of 3-aminopiperidine derivatives
10/12/1999US5965745 Asthma; antiarthritic,-shock agents; bronchitis; respiratory system diseases, e.g. chronic obstructive airways diseases; psoriasis; allergic rhinitis; atopic dermatitis
10/12/1999US5965730 Selective phosphodiestearase iv inhibitor having bronchodialation and anti-inflammatory activity; prophylaxis and treatment of asthma
10/12/1999US5965600 Preventive and therapeutic method for treating arteriosclerosis and articular rheumatism; providing minimal liver toxicity
10/12/1999US5965592 Acyl compounds
10/12/1999US5965583 Substituted imidazoles useful in the treatment of inflammatory disease
10/12/1999US5965582 Antihistamines
10/12/1999US5965579 Antagonists of the neurotensin receptors; increasing affinity for human neurotensin receptors
10/12/1999US5965578 An enzyme inhibitor for farnesylation of the oncogene ras protein, a chemotherapeutic composition prevention of thiol-dependent chemical reactions, such as rapid autoxidation and disulfide formation with endogenous thiols