Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
09/1999
09/29/1999EP0945440A1 Aminopyrazole derivatives
09/29/1999EP0945439A1 Novel aminopyrazole derivatives
09/29/1999EP0945438A1 Pyrazole derivatives
09/29/1999EP0945437A1 Pyrazolyl acrylic acid- and pyrazolyl oximino-acetic acid derivatives, their preparation and their use as fungicides
09/29/1999EP0945435A1 Novel pyridonecarboxylic acid derivatives or salts thereof and drugs containing the same as the active ingredient
09/29/1999EP0944673A1 Trifluormethylpyridone based indolenine methine dyes
09/29/1999EP0944672A1 Helium-neon excitable reticulocyte dyes derivable from halolepidines
09/29/1999EP0944619A1 Novel integrin receptor antagonists
09/29/1999EP0944618A1 Novel n-benzenesulphonyl-l-proline derivatives, method for preparing and therapeutic use
09/29/1999EP0944617A1 Crystals of benzimidazole derivatives and their production
09/29/1999EP0944616A1 Bicyclic aryl carboxamides and their therapeutic use
09/29/1999EP0944606A1 4,5-diaminopyrimidine derivatives and a method for the preparation thereof
09/29/1999EP0944603A1 Process for making 2-amino-2-imidazoline, guanidine, and 2-amino-3,4,5,6-tetrahydropyrimidine derivatives
09/29/1999EP0944602A1 Apo b-secretion/mtp inhibitory amides
09/29/1999EP0944597A1 Metalloproteinase inhibitors
09/29/1999EP0944595A1 5-cyclo indole compounds as 5-ht1d receptor ligands
09/29/1999EP0944594A1 Inhibitors of the enzymatic activity of psa
09/29/1999EP0944582A1 Ketobenzamides as calpain inhibitors
09/29/1999EP0944388A2 Inhibitors of farnesyl-protein transferase
09/29/1999EP0944386A1 Sulfonic acid or sulfonylamino n-(heteroaralkyl)-azaheterocyclylamide compounds
09/29/1999EP0944322A1 Quarternary ammonium salts and their use in agricultural formulations
09/29/1999EP0944314A1 Methyl substituted fungicides and arthropodicides
09/29/1999EP0553107B1 Protein kinase c modulators with anti-inflammatory and antiviral activity
09/29/1999CN1230196A Modified aminoacids, pharmaceuticals containing these compounds and method for their prodn.
09/29/1999CN1230187A Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors
09/29/1999CN1230180A D4 receptor selectivity piperazine derivatives
09/29/1999CN1230110A Cell adhesion inhibitors
09/29/1999CN1045294C Method for prepn. of indole derivatives
09/29/1999CN1045293C Substituted pyrazoles compounds and medicinal compositions containing same
09/28/1999US5959123 Reacating substituted amino acid with 3-amino-4-substituted-azetidine-2-one compound to form 3, 4-disubstituted-azetidine-2-one compound; useful for treating muscular dystrophy, arthritis, viral and parasitic infections
09/28/1999US5959121 Process for preparing 3-substituted indazoles
09/28/1999US5959113 Reacting a diketone derivative with an aldehyde derivative; administering to treat atherosclerosis, psoriasis, alopecia and tumors
09/28/1999US5959109 Compounds and methods for increasing endogenous levels of corticotropin-releasing factor
09/28/1999US5959107 Inhibitory activity on neuronal cell death (apoptotic cell death-type) caused by excessive apoptosis in a nervous system and they are useful for prevention or treatment of neurodegenerative disorders
09/28/1999US5958955 Method for the synthesis of a benzimidazole compound
09/28/1999US5958954 2,2-dialkyl-4-aryl-substituted benzopyran and benzothiopyran derivatives
09/28/1999US5958953 Substituted indazole derivatives
09/28/1999US5958952 Substituted phenylamindines, medicaments containing these compounds and process for producing them
09/28/1999US5958949 N-linked ureas and carbamates of piperidyl thioesters
09/28/1999US5958948 Corticotropin releasing factor; therapy for stress
09/28/1999US5958947 DNA-affinic hypoxia selective cytotoxins
09/28/1999US5958944 Treatment of circulatory diseases in coronary, cerebral, renal and peripheral arteries, as a therapeutic agent for hypertension, angina pectoris, and renal and peripheral circulation disorder, antiasthmatic agent
09/28/1999US5958940 Antitumor agent inhibiting growth of cells expressing an activated ras oncogene in mammals
09/28/1999US5958939 Tricyclic compounds useful for inhibition of a g-protein function and for treatment of proliferative diseases
09/28/1999US5958935 Substituted 2-anilinopyrimidines useful as protein kinase inhibitors
09/28/1999US5958927 Psychological and nervous system disorders
09/28/1999US5958926 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
09/28/1999US5958925 Pyridazinones and their use as fungicides
09/28/1999US5958924 Hypotensive agents, cardiovascular disorders, antiischemic agents, restenosis, anticoalugants, respiratory system disorders
09/28/1999US5958918 Substituted (sulfinic acid, sulfonic acid, sulfonylamino or sulfinylamino) N- (aminominomethyl)phenylalkyl!-azaheterocyclylamide compounds
09/28/1999US5958890 Antitumor
09/28/1999US5958838 Controlling weeds in crops.
09/28/1999US5958837 2-(phenylmethoxy or carbonyloxy-(1,4-phenylene)-),3-halo,5-haloalkylpyridines; herbicides effecting desiccation and defoliation of plants; good activity and better tailored control of weeds
09/28/1999CA2014457C Pyrimidine derivatives
09/28/1999CA2012539C Process for the preparation of o-carboxypyridyl-and 0-carboxyquinolylimidazolines
09/23/1999WO1999047545A2 Inhibitors of caspases
09/23/1999WO1999047517A1 Novel heterocyclic compounds
09/23/1999WO1999047515A1 Arylpiperidine derivatives and use thereof
09/23/1999WO1999047514A1 Chemical process for the production of sulphinyl derivatives by oxidation of the corresponding co-derivatives with perborates
09/23/1999WO1999047513A1 Heteroaromatic derivatives
09/23/1999WO1999047512A1 2-(2,6-dioxopiperidin-3-yl)isoindoline derivatives, their preparation and their use as inhibitors of inflammatory cytokines
09/23/1999WO1999047511A1 Indole derivatives as 5-ht2a receptor antagonists
09/23/1999WO1999047503A1 Aminoisoquinoline derivatives
09/23/1999DE19812331A1 New benzo-heterocyclic substituted piperidine derivatives useful as excitatory aminoacid receptor antagonists, used e.g. for treating neurodegenerative diseases
09/23/1999CA2324550A1 Arylpiperidine derivatives and use thereof
09/23/1999CA2324268A1 Aromaheterocyclic derivatives
09/23/1999CA2324153A1 Aminoisoquinoline derivatives
09/23/1999CA2323422A1 Chemical process for the production of sulphinyl derivatives by oxidation of the corresponding co-derivatives with perborates
09/22/1999EP0943616A1 Substituted imidazole derivatives and their use as cytokine inhibitors
09/22/1999EP0943615A1 1,4-dihydropyridine derivatives
09/22/1999EP0943008A1 Metal mediated serine protease inhibitors
09/22/1999EP0942906A2 Compounds useful for inhibition of farnesyl protein transferase
09/22/1999EP0942902A2 Novel immunotherapeutic imides/amides
09/22/1999EP0942735A1 Use of nk-1 receptor antagonists for treating schizophrenic disorders
09/22/1999CN1229412A Inhibitors of interleukin-1'beta' converting emzyme
09/22/1999CN1229408A Dihydroindole derivatives useful as 5-HT-2C receptor antagonists
09/22/1999CN1229405A Novel acetamide derivatives and protease inhibitors
09/22/1999CN1229082A Amine compound and its acid addition salt
09/22/1999CN1229081A Process for preparation of aqueous nicotinaldehyde
09/22/1999CN1045206C Method for preparing cyclic amide derivative
09/22/1999CN1045204C 10,11-methanodibenzosuberane derivatives, preparation method and composition
09/21/1999US5955501 Derived from phorboids of the diterpene- and benzolactam-classes.
09/21/1999US5955487 Treating high blood pressure, cardiac insufficiency, glaucoma
09/21/1999US5955482 Use of 1,4-dihydropyridine-3,5-dicarboxylic acid esters as medicaments
09/21/1999US5955480 Glucagon receptor antagonists, cytokine inhibitors
09/21/1999US5955476 Substituted 2-(2,6-dioxo-3-fluoropiperidin-3-yl)-isoindolines and method of reducing inflammatory cytokine levels
09/21/1999US5955473 Fungicidal quinolines
09/21/1999US5955464 4-anilinoquinazoline derivatives bearing a heteroaryl substituted at the 6-position and possessing anti-cell-proliferation properties
09/21/1999US5955463 Antitumor, antiinflammatory, and antiarthritic agents
09/21/1999US5955461 Quinoxalinedione derivatives, their production and use in pharmaceutical agents
09/21/1999US5955365 Introducing polynucleotides into cells
09/21/1999CA2192975C Benzimidazolone derivatives
09/21/1999CA2005235C Tetramethyl piperidyl terminated triazine oligomeric esters and amides
09/21/1999CA2005234C Triazine-based light stabilizers for plastics
09/16/1999WO1999046264A1 New compounds
09/16/1999WO1999046260A1 New compounds
09/16/1999WO1999046259A1 5-heteroaryl substituted indoles
09/16/1999WO1999046258A1 SUBSTITUTED 2-(2,6-DIOXO-3-FLUOROPIPERIDIN-3-YL)-ISOINDOLINES AND THEIR USE TO REDUCE TNFα LEVELS
09/16/1999WO1999046248A1 1,2-diazepane derivatives as interleukin-1beta converting enzyme inhibitors
09/16/1999WO1999046247A1 Pyrazole compounds and agricultural chemicals containing the same as active ingredient