Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
07/1999
07/01/1999DE19756236A1 Neue piperazinylsubstituierte Pyridylalkan-, alken- und -alkincarbonsäureamide New piperazinyl substituted pyridylalkane, alkene and -alkincarbonsäureamide
07/01/1999DE19756235A1 Neue piperidinylsubstituierte Pyridylalkan- alken- und -alkincarbonsäureamide New piperidinylsubstituierte pyridylalkane alkene and -alkincarbonsäureamide
07/01/1999DE19756212A1 Neue, mit einem cyclischen Imid substituierte Pyridylalkan-, alken- und -alkincarbonsäureamide Novel substituted with a cyclic imide pyridylalkane, alkene and -alkincarbonsäureamide
07/01/1999CA2315941A1 Novel substituted pyridine compounds useful as modulators of acetylcholine receptors
07/01/1999CA2315910A1 Novel dihydropyridine derivative
07/01/1999CA2315720A1 Inhibition of p38 kinase activity using substituted heterocyclic ureas
07/01/1999CA2315226A1 Hypoglycemic imidazoline compounds
07/01/1999CA2315070A1 Ortho-anthranilamide derivatives as anti-coagulants
07/01/1999CA2314980A1 Compounds of heteroaryl substituted imidazole, their pharmaceutical compositions and uses
07/01/1999CA2314869A1 Catalyst and method for amide formation
07/01/1999CA2314401A1 Nitrogen containing heteroaromatics with ortho-substituted p1's as factor xa inhibitors
07/01/1999CA2309882A1 4-hydroxyquinoline-3-carboxamides and hydrazides as antiviral agents
07/01/1999CA2309661A1 Catalytic composition based on chiral ligands with molybdenum, tungsten or chromium and method for asymmetric alkylation of allylic substrates
06/1999
06/30/1999EP0926137A1 Picolin acid derivatives useful in the treatment of IL-1 and TNF mediated diseases
06/30/1999EP0925302A1 Palladium catalyzed indolization
06/30/1999EP0925300A1 Pharmaceutically active compounds and methods of use
06/30/1999EP0925296A1 New pharmaceutically active compounds
06/30/1999EP0925295A1 N-benzenesulphonyl-l-proline derivatives as bradykinin b2 agonists
06/30/1999EP0925294A1 Substituted 2(2,6-dioxopiperidin-3-yl)phthalimides and -1-oxoisoindolines and method of reducing tnf-alpha levels
06/30/1999EP0925287A1 Heterocyclic metalloprotease inhibitors
06/30/1999EP0925286A1 Substituted pyrimidine derivatives and their pharmaceutical use
06/30/1999EP0925282A1 4-substituted quinoline derivatives having fungicidal activity
06/30/1999EP0756602B1 Cck or gastrin modulating 5-heterocyclic-1,5-benzodiazepines
06/30/1999CN1221422A Novel chiral bisphosphines
06/30/1999CN1221417A Thiazolidinedione compounds having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions thereof
06/30/1999CN1221407A Aminoisoquinolines and aminothienopyridine derivatives and their use as anti-inflammatory agents
06/30/1999CN1221405A Substituted amidinobenzene derivatives and medicinal compositions thereof
06/30/1999CN1043888C Fungicidal and herbicidal triazoles
06/30/1999CN1043886C Substituted pyrimidine, there process of preparation and use as sectivide and fungicide thereof
06/30/1999CN1043885C Herbicidal pyrimidine derivatives, process for preparation thereof and their use as herbicide
06/30/1999CN1043884C New substituted azacylobutanone, preparation method and medicinal use thereof
06/29/1999US5917048 Substituted aryl or heteroarylamides having retinoid-like biological activity
06/29/1999US5917046 Method for producing 2-naphthamide derivative, and compounds for producing 2-naphthamide derivative
06/29/1999US5917043 Intermediates
06/29/1999US5916908 Pharmaceutical pyrazole compositions useful as inhibitors of protein kinases
06/29/1999US5916900 7-(2-imidazolinylamino)quinoline compounds useful as alpha-2 adrenoceptor agonists
06/29/1999US5916891 Cytokine mediated diseases
06/29/1999US5916889 1,4-disubstituted piperazines
06/29/1999US5916847 Displays low phytotoxicity; plant growth regulator
06/29/1999CA2131722C N,n'-disubstituted amide derivative
06/24/1999WO1999031099A1 Integrin receptor antagonists
06/24/1999WO1999031089A1 1-(1h-imidazol-2-yl)pyrrolidine and 1-(1h-imidazol-2-ylpiperidine) derivatives, preparation and therapeutic application
06/24/1999WO1999031088A1 Triazine angiogenesis inhibitors
06/24/1999WO1999031087A1 Cyclic imide-substituted pyridylalkane, alkene and alkine carboxamides useful as cytostatic and immunosuppressive agents
06/24/1999WO1999031086A1 Quinolinepiperazine and quinolinepiperidine derivatives, their preparation and their use as combined 5-ht1a, 5-ht1b and 5-ht1d receptor antagonists
06/24/1999WO1999031085A1 3-piperidyl-4-oxoquinazoline derivatives and medicincal compositions containing the same
06/24/1999WO1999031077A1 Arylpiperazines having activity at the serotonin 1a receptor
06/24/1999WO1999031075A1 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
06/24/1999WO1999031074A2 ((cyclo)alkyl substituted)-.gamma.-aminobutyric acid derivatives (=gaba analogues), their preparation and their use in the treatment of neurological disorders
06/24/1999WO1999031073A1 Novel pyrimidine-5-carboxamide derivatives
06/24/1999WO1999031070A1 Substituted phenylpyrazolones, method and intermediate products for the production thereof, and their utilization for combating parasitic fungi and animal parasites
06/24/1999WO1999031068A1 Substituted isoquinoline derivatives and their use as anticonvulsants
06/24/1999WO1999031066A1 Pyridones as src family sh2 domain inhibitors
06/24/1999WO1999031064A1 Aryl-substituted pyridylalkane, alkene, and alkine carboxamides useful as cytostatic and immunosuppressive agents
06/24/1999WO1999031063A1 New piperazinyl-substituted pyridylalkane, alkene and alkine carboxamides
06/24/1999WO1999031061A1 Integrin receptor antagonists
06/24/1999WO1999031060A2 Piperidinyl-substituted pyridylalkane, alkene and alkine carboxamides as cytostatics and immunesuppressants
06/24/1999WO1999031058A1 Novel heterocyclic compounds
06/24/1999WO1999031057A1 4(3)substituted-4(3)-aminomethyl-(thio)pyran or -piperidine derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
06/24/1999WO1999030713A1 Integrin receptor antagonists
06/24/1999WO1999030709A1 Integrin receptor antagonists
06/24/1999WO1999030696A1 A method for the prevention and treatment of stunned myocardium
06/24/1999WO1999019305A3 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system
06/24/1999DE19756388A1 New 2-aryl-4-amino-6,7-di:methoxy-quinazoline derivatives useful as guanylate cyclase activators for treating cardiovascular diseases, etc.
06/24/1999DE19756115A1 Substituierte Phenylpyrazolone, Verfahren und Zwischenprodukte zu ihrer Herstellung und ihre Verwendung zur Bekämpfung von Schadpilzen und tierischen Schädlingen Substituted phenylpyrazolones, processes and intermediates for their preparation and their use for controlling harmful fungi and animal pests
06/24/1999DE19756036A1 New indole amide derivatives
06/24/1999CA2506802A1 Arylpiperazines having activity at the serotonin 1a receptor
06/24/1999CA2315370A1 Integrin receptor antagonists
06/24/1999CA2315232A1 Integrin receptor antagonists
06/24/1999CA2315079A1 Substituted isoquinoline derivatives and their use as anticonvulsants
06/24/1999CA2313776A1 Triazine angiogenesis inhibitors
06/24/1999CA2313125A1 Quinolinepiperazine and quinolinepiperidine derivatives, their preparation and their use as combined 5-ht1a, 5-ht1b and 5-ht1d receptor antagonists
06/24/1999CA2311932A1 A method for the prevention and treatment of stunned myocardium
06/24/1999CA2280705A1 3-piperidyl-4-oxoquinazoline derivatives and pharmaceutical compositionscomprising the same
06/23/1999EP0924209A1 Hypoglycemic imidazoline compounds
06/23/1999EP0924205A1 Arylpiperazines having activity at the serotonin 1a receptor
06/23/1999EP0924201A1 Tricyclic-substituted pyrazolyl benzenesulfonamides and their use as cyclooxygenase II inhibitors
06/23/1999EP0923933A1 Substituted pyrazolyl benzenesulfonamides for use in the treatment of inflammation
06/23/1999EP0923580A1 Thiazolidinedione compounds having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions thereof
06/23/1999EP0923573A1 Preparation of aminomethyl-phenylimidazoles
06/23/1999EP0923571A2 Trisubstituted pyridine compounds for herbicidal use
06/23/1999EP0923570A1 Pyridyl alkene- and pyridyl alkine- acid amides as cytostatics and immunosuppressives
06/23/1999EP0923563A1 1,4-heterocyclic metallprotease inhibitors
06/23/1999EP0923556A1 An asymmetric conjugate addition reaction
06/23/1999EP0923555A1 Carboxamide derivatives of pyrrolidine, piperidine and hexahydroazepine for the treatment of thrombosis disorders
06/23/1999EP0923551A1 4-aminoethoxy indolone derivatives
06/23/1999EP0923547A1 Bidentate metalloprotease inhibitors
06/23/1999EP0923545A1 3-mercaptopyrrolidines as farnesyl protein transferase inhibitors
06/23/1999EP0923542A1 Aryl substituted cyclic amines as selective dopamine d3 ligands
06/23/1999CN1220604A Anti-HIV composition containing imidazole derivative
06/23/1999CN1220265A New piperazine and piperidine compounds
06/23/1999CN1043762C Compound used for excitary amino acid receptor antagonists and its drug composition
06/23/1999CN1043759C Process for preparation of 2-(4-hydroxypiperidino)-1-alkanol derivatives as antiischemic agents
06/22/1999US5914406 Azepanes and their ring homologues having protein kinase inhibiting activity
06/22/1999US5914405 Treating indazole compound with adamantane ring-containing piperidine compound
06/22/1999US5914335 Pesticidal 1-arylpyrazole-5-sulfinilimine derivatives
06/22/1999US5914332 Retroviral protease inhibiting compounds
06/22/1999US5914328 Control dopamine release, activate cholinergic channels
06/22/1999CA2151674C Methods of administering crf antagonists
06/22/1999CA1340608C Alkoxy-4(1h)-pyridone derivatives, processes for the preparation thereof and pharmaceutical compositions containing them