| Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979) |
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| 01/06/2000 | WO2000000479A1 1,3-benzodiazepin-2-ones and 1,3-benzoxazepin-2-ones useful as hiv reverse transcriptase inhibitors |
| 01/06/2000 | WO2000000478A1 Substituted quinoxalin-2(1h)-ones useful as hiv reverse transcriptase inhibitors |
| 01/06/2000 | WO2000000477A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases |
| 01/06/2000 | WO2000000473A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them |
| 01/06/2000 | WO2000000472A1 5-ht7 receptor antagonists |
| 01/06/2000 | WO2000000198A1 Piperidine derivatives having effects on serotonin related systems |
| 01/06/2000 | WO2000000197A1 4-benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective nmda receptor antagonists |
| 01/06/2000 | WO1999043661A3 Substituted cycloalkyl-4-oxonicotinic carboxamides; gaba brain receptor ligands |
| 01/06/2000 | CA2336625A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases |
| 01/06/2000 | CA2336254A1 5-ht1f agonists |
| 01/06/2000 | CA2336117A1 Piperidine derivatives having effects on serotonin related systems |
| 01/06/2000 | CA2335921A1 Carboxylic and hydroxamic acid compounds inhibiting metalloproteases, method for preparing same and pharmaceutical compositions containing them |
| 01/06/2000 | CA2335595A1 Bifunctional antagonists of cytokine-sensitive protein kinase activation cascades and methods for use as anti-inflammatory agents |
| 01/06/2000 | CA2334332A1 Substituted quinoxalin-2(1h)-ones useful as hiv reverse transcriptase inhibitors |
| 01/06/2000 | CA2330110A1 1,3-benzodiazepin-2-ones and 1,3-benzoxazepin-2-ones useful as hiv reverse transcriptase inhibitors |
| 01/06/2000 | CA2327888A1 4-benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective nmda receptor antagonists |
| 01/05/2000 | EP0969071A1 Alkenyl compound having a negative delta epsilon value, liquid crystal composition and liquid crystal display device |
| 01/05/2000 | EP0969003A2 Process for the preparation of benzo[f]quinolinone derivatives and intermediates |
| 01/05/2000 | EP0968715A1 Loratadine for use as an antiarrhymthmic |
| 01/05/2000 | EP0968208A1 Quinoline and quinazoline compounds useful in therapy, particularly in the treatment of benign prostatic hyperplasia |
| 01/05/2000 | EP0968206A1 N-heterocyclic derivatives as nos inhibitors |
| 01/05/2000 | EP0968205A1 Process for the preparation of 2- (2-pyridinyl)methyl]sulfinyl]-1h-benzimidazoles and novel compounds of use for such purpose |
| 01/05/2000 | EP0968204A1 Process for the preparation of 2- (2-pyridinyl)methyl]sulfinyl]-1h-benzimidazoles and novel compounds of use for such purpose |
| 01/05/2000 | EP0968194A1 Atropisomers of 3-aryl-4(3h)-quinazolinones and their use as ampa-receptor antagonists |
| 01/05/2000 | EP0968193A1 Phenylsulphonyl ureas, processes for their preparation and their use as herbicides and plant-growth regulators |
| 01/05/2000 | EP0968191A1 Phenylbenzimidazole derivatives as ligands for gaba receptors |
| 01/05/2000 | EP0968190A1 Substituted isoquinoline derivatives and their use as anticonvulsants |
| 01/05/2000 | EP0968188A1 Substituted 2-benz(o)ylpyridines, their preparation and their use as herbicides |
| 01/05/2000 | EP0666856B1 4-arylmethyloxymethyl piperidines as tachykinin antagonists |
| 01/05/2000 | EP0664792B1 Fibrinogen receptor antagonists |
| 01/05/2000 | EP0539420B1 substituted thiazolyl and substituted pyridinyl derivatives |
| 01/05/2000 | EP0427765B1 Alkoxy-4(1h)-pyridone derivatives, processes for preparing them and their use as drugs |
| 01/05/2000 | DE19829964A1 New benzimidazolyl amidine or nitrile compounds, used as thrombin inhibitors, antithrombotic agents or intermediates |
| 01/05/2000 | CN1240443A Novel carboxy substituted cyclic carboxamide derivatives |
| 01/05/2000 | CN1240442A Heterocyclyl uracils |
| 01/05/2000 | CN1240441A Heterocyclyluracil |
| 01/05/2000 | CN1240428A Diphenyl alkyl-tetrahydropyridines, process for their preparation, and pharmaceutical compositions containing them |
| 01/05/2000 | CN1240427A 1-phenylalkyl-1,2,3,6-tetrahydropyridines for treating alzheimer's disease |
| 01/05/2000 | CN1240426A Novel tetrahydrobenzindolone derivatives |
| 01/04/2000 | US6011158 Aromatic heterocyclic derivatives as enzyme inhibitors |
| 01/04/2000 | US6011155 N-(substituted glycyl)-2-cyanopyrrolidines, pharmaceutical compositions containing them and their use in inhibiting dipeptidyl peptidase-IV |
| 01/04/2000 | US6011154 Substituted heterocyclic compounds, method of preparing them and pharmaceutical compositions in which they are present |
| 01/04/2000 | US6011150 Synthetic intermediate of a 1 beta-methylcarbapenem derivative |
| 01/04/2000 | US6011039 Aminopyridine derivatives |
| 01/04/2000 | US6011038 Pyrazinone thrombin inhibitors |
| 01/04/2000 | US6011035 Libraries of these compounds can also be used to identify antagonists for other targets. compounds containing benzhydril and 6-membered heterocyclic moieties |
| 01/04/2000 | US6011033 Phenylene derivatives |
| 01/04/2000 | US6011029 Benzodiazepine compounds |
| 01/04/2000 | US6011028 Cyclic amidino agents useful as nitric oxide synthase inhibitors |
| 12/29/1999 | WO1999067238A2 Tetrahydroquinoline-indole derivatives antimicrobial agents, their uses and compositions containing them |
| 12/29/1999 | WO1999067237A1 4,5,6 and 7-indole and indoline derivatives, their preparation and use |
| 12/29/1999 | WO1999067235A1 Five-membered ring compounds |
| 12/29/1999 | WO1999067230A1 INHIBITORS OF α4β1 MEDIATED CELL ADHESION |
| 12/29/1999 | WO1999067221A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/29/1999 | WO1999067220A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/29/1999 | WO1999067219A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/29/1999 | WO1999067215A1 Amidino and guanidino azetidinone tryptase inhibitors |
| 12/29/1999 | WO1999066944A1 Methods for identifying novel multimeric agents that modulate receptors |
| 12/29/1999 | WO1999066934A1 CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING β-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS |
| 12/29/1999 | WO1999054326A8 Dihydropyrimidines |
| 12/29/1999 | WO1999054315A3 Triazolones with a neuroprotective action |
| 12/29/1999 | EP0967212A1 Pyrazoline compounds and use as plant disease control agent |
| 12/29/1999 | EP0967207A1 Nitrone derivatives, process for their preparation and pharmaceutical compositions containing them |
| 12/29/1999 | EP0967205A1 Labeling reactants and their use |
| 12/29/1999 | EP0966473A1 Thiazolobenzoheterocycles, preparation and medicines containing same |
| 12/29/1999 | EP0966464A1 Substituted 2,4-diaminopyrimidines |
| 12/29/1999 | EP0966462A1 Heterocyclic compounds useful as oxido-squalene cyclase inhibitors |
| 12/29/1999 | EP0966461A1 Pyrazole derivatives as herbicides |
| 12/29/1999 | EP0966460A1 Heterocyclic compounds useful as oxido-squalene cyclase inhibitors |
| 12/29/1999 | EP0966454A1 Disubstituted bicyclic heterocycles, their production and use as medicaments |
| 12/29/1999 | EP0966447A1 Small molecules useful in the treatment of inflammatory disease |
| 12/29/1999 | EP0966446A1 Bicyclic inhibitors of protein farnesyl transferase |
| 12/29/1999 | EP0966445A1 Processes for preparing pesticidal intermediates |
| 12/29/1999 | EP0966444A1 Process for preparing pyrazole derivatives |
| 12/29/1999 | EP0966443A1 Heteroaryl-hexanoic acid amide derivatives, their preparation and their use as selective inhibitors of mip-1-alpha binding to its ccr1 receptor |
| 12/29/1999 | EP0966442A1 Quinoline and quinazoline derivatives having corticotropin releasing factor (crf) antagonist activity |
| 12/29/1999 | EP0966436A1 Aryl sulfonamides and analogues thereof and their use in the treatment of neurodegenerative diseases |
| 12/29/1999 | EP0966285A1 Use of (+)mefloquine for the treatment of malaria |
| 12/29/1999 | EP0966282A1 Use of angiotensin ii antagonists to treat symptomatic heart failure |
| 12/29/1999 | EP0612314B1 2-pyrazinylethylamine derivatives and their use as pharmaceuticals |
| 12/29/1999 | CN1239959A Subsitutted 2(2,6-dioxopiperidin-3-yl) phthalimides and -1-xoisoindolines and method of reducing TNF-alpha levels |
| 12/29/1999 | CN1239957A Substituting 2-amino-4-alkylamino-1,3,5-triazine as herbicide |
| 12/29/1999 | CN1239956A Substituted 2-amino-4-alkylamino-1,3,5-triazines as herbicides |
| 12/29/1999 | CN1239955A Substituted 2,4-diamino-1,3,5-triazine as herbicide |
| 12/29/1999 | CN1239952A 6-phenylpyridyl-2-amine derivatives useful as NOS inhibitors |
| 12/29/1999 | CN1239950A New derivates from piperidine-keto acid, their preparation and use |
| 12/29/1999 | CN1239949A Novel heterocyclically substituted benzamides and their use in fighting diseases |
| 12/29/1999 | CN1239895A Radiopharmaceuticals for imaging infection and inflammation |
| 12/29/1999 | CN1047777C Pyridyltetrazolinone derivatives, its preparation, composition and use |
| 12/29/1999 | CN1047776C Pharmacologically active pyridine derivatives and process for the preparation thereof |
| 12/29/1999 | CN1047775C N-piperidino 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl pyrazole-3-formyl amide, its preparation and drug composition |
| 12/29/1999 | CA2342778A1 Inhibitors of .alpha.4.beta.1 mediated cell adhesion |
| 12/29/1999 | CA2336003A1 Amidino and guanidino azetidinone tryptase inhibitors |
| 12/29/1999 | CA2335711A1 4,5,6 and 7-indole and indoline derivatives, their preparation and use |
| 12/29/1999 | CA2325389A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/29/1999 | CA2325388A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/29/1999 | CA2324475A1 Cyclic amino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds |
| 12/29/1999 | CA2324474A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/29/1999 | CA2319650A1 Methods for identifying novel multimeric agents that modulate receptors |
| 12/28/1999 | US6008370 Fungicidal imidazolinone and imidazolinethione compounds for use in plant protection |