Patents
Patents for C07D 305 - Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms (5,442)
05/1997
05/02/1997EP0770070A1 Method for preparing 4-acetoxy-2alpha-benzoyloxy-5alpha,20-epoxy-1,7beta,10beta-trihydroxy-9-oxo-tax-11-en-13alpha-yl(2r,3s)-3-tert-butoxycarbonylamino-2-hydroxy-3-phenylpropionate trihydrate
05/01/1997WO1997015562A1 Intermediary compounds for the hemisynthesis of taxanes and preparation processes therefor
05/01/1997CA2576943A1 Intermediates for the hemisynthesis of taxanes and processes for their preparation
04/1997
04/24/1997WO1997014954A1 Improved chemiluminescent 1,2-dioxetanes
04/24/1997CA2231191A1 Improved chemiluminescent 1,2-dioxetanes
04/23/1997EP0769064A1 A method for mass production of taxol by semi-continuous culture
04/23/1997EP0755388A4 Preparation of 10-deacetylbaccatin iii and 7-protected-10-deacetylbaccatin iii derivatives from 10-deacetyl taxol a, 10-deacetyl taxol b, and 10-deacetyl taxol c
04/22/1997US5622986 Water soluble antitumor agents
04/16/1997EP0767786A1 7-ether-taxol analogs, antineoplastic use and pharmaceutical compositions containing them
04/16/1997EP0767775A1 A method for the preparation of a novel a-ring precursor for taxoids and novel intermediates
04/16/1997EP0687259B1 Novel taxoids, preparation thereof and pharmaceutical compositions containing same
04/15/1997US5621121 Process for the preparation of taxane derivatives
04/15/1997US5620875 Transfer of taxol from yew tree cuttings into a culture medium over time
04/08/1997US5618952 Chemical intermediates; hydroxylation; reduction; recyclization
04/08/1997US5618538 Separating clippings form plants, drying, extracting with solvent, evaporating to form residue and partitioning between water and organic layer, removing aqueous layer, evaporating
04/02/1997CN1146722A Taxane class derivative based pharmaceutical compositions
04/01/1997US5616740 Process for making 9-deoxotaxane compounds
04/01/1997US5616739 Method of preparing taxane derivatives
04/01/1997US5616608 Method of treating atherosclerosis or restenosis using microtubule stabilizing agent
03/1997
03/26/1997EP0764643A1 Deacetoxytaxol derivative
03/26/1997EP0764156A1 New taxoids, preparation thereof and pharmaceutical compositions containing them
03/26/1997EP0764155A1 Taxoids, preparation and pharmaceutical compositions containing them
03/26/1997EP0764154A1 New taxoids, preparation thereof and pharmaceutical compositions containing them
03/26/1997EP0696279B1 Oxidation products of cephalomannine
03/25/1997US5614645 Methods for making 2-debenzoyl and -2-acyl taxol derivatives
03/25/1997US5614549 High molecular weight polymer-based prodrugs
03/20/1997WO1997010234A1 Hydrolysis-promoting taxane hydrophobic derivatives
03/20/1997WO1997010233A1 Biocatalytic methods for synthesizing and identifying biologically active compounds
03/20/1997WO1997009979A1 Radiosensitizing taxanes and their pharmaceutical preparations
03/20/1997CA2240468A1 Biocatalytic methods for synthesizing and identifying biologically active compounds
03/20/1997CA2231837A1 Radiosensitizing taxanes and their pharmaceutical preparations
03/19/1997EP0663901B1 Method for the stereoselective preparation of a derivative of beta-phenylisoserine and its use in the preparation of taxane derivatives
03/19/1997CN1145429A 2-oxetanone sizing agents and their preparation and use
03/12/1997EP0761662A1 Method for preparing unsaturated cyclic ethers
03/12/1997CN1145073A Process for preparing 7-trialkylsilkl baccatin III
03/12/1997CN1145070A Process for the preparation of 7-hydroxy taxanes
03/12/1997CN1144805A Prodrugs of paclitaxel derivatives
03/04/1997US5608102 Process for the preparation of β-phenylisoserine and its analogues
03/04/1997US5608087 Water soluble taxol derivatives
03/04/1997US5608073 Baccatin derivatives and processes for preparing the same
03/04/1997CA2051484C Decarboxylation processes using mixed metal oxide catalysts
02/1997
02/27/1997WO1997007110A1 Process for producing taxol derivatives and intermediates therefor
02/26/1997EP0690852B1 Method for purifying taxoids
02/26/1997CN1143641A Novel methods for preparation of taxanes using oxazolidine intermediates
02/26/1997CN1143640A Tetrahydrofuran derivative, its synthesizing process and use
02/25/1997US5606083 Process for the preparation of taxane derivatives, new derivatives thus obtained and the compositions which contain them
02/25/1997US5606068 Chemical intermediate for taxane
02/19/1997EP0758231A1 Taxane class derivative based pharmaceutical compositions
02/12/1997EP0663910B1 Method of obtaining 10-deacetylbaccatine iii
02/12/1997EP0663908B1 Method of preparing taxane derivatives
02/04/1997US5599978 Esterification, acylation
02/04/1997US5599942 Taxoid intermediates
02/04/1997US5599820 Anti-tumor compounds, pharmaceutical compositions, methods for preparation thereof and for treatment
01/1997
01/30/1997WO1997003105A1 Preparation of cyclic oligomers of substituted cyclic ethers
01/30/1997WO1997003061A1 Method for extracting and isolating 10-deacetylbaccatin iii
01/29/1997EP0755388A1 Preparation of 10-deacetylbaccatin iii and 7-protected-10-deacetylbaccatin iii derivatives from 10-deacetyl taxol a, 10-deacetyl taxol b, and 10-deacetyl taxol c
01/29/1997EP0755387A1 Oxidative purification of biomass extracts containing taxol and cephalomannine using ozone and girard reagents
01/28/1997US5597931 Total synthesis of taxol and analogues thereof
01/28/1997US5597779 Sulfonylureas
01/22/1997EP0754185A1 Process for preparing 7-trialkylsilyl baccatin iii
01/22/1997EP0754181A1 Process for the preparation of 7-hydroxy taxanes
01/22/1997EP0669916B1 Novel method for preparing taxane derivatives, novel derivatives thus obtained and compositions containing them
01/15/1997EP0663907B1 Method of preparing taxane derivatives
01/15/1997EP0663905B1 Novel method of esterification of baccatine iii an 10-deacetylbaccatine iii
01/15/1997CN1140170A Preparative liquid chromatography for extracting and purifying taxol and other taxanes derivs
01/14/1997US5594157 Process for making taxol derivatives
01/09/1997WO1997000870A1 Method for the preparation of taxol and its derivatives
01/08/1997EP0751963A1 Copolymers based on diketens, ethylenically unsaturated bicarboxylic acids or their derivatives and ethylenically unsaturated hydrocarbons
01/08/1997EP0663909B1 Method of obtaining 10-deacetylbaccatine iii
01/08/1997CN1139925A 'Delta' 12,13-iso-taxol analogs, antineoplastic use and pharmaceutical compositions containing them
01/02/1997EP0751136A1 Process for the preparation of 3-hydroxyoxetanes
12/1996
12/31/1996US5589502 Antitumor
12/27/1996EP0749432A1 9-deoxotaxane compounds
12/24/1996US5587493 Process for preparing taxoids
12/24/1996US5587489 Taxane and baccatin III analogs bearing new C2 and C4 functional groups
12/19/1996WO1996040667A1 Paclitaxel synthesis from precursor compounds and methods of producing the same
12/19/1996WO1996040666A1 Paclitaxel synthesis from precursor compounds and methods of producing the same
12/19/1996WO1996040624A1 C-2' hydroxyl-benzyl protected, n-carbamate protected (2r,3s)-3-phenylisoserine and production process therefor
12/19/1996WO1996040091A1 Dual functional cytotoxic/radiosensitizer compounds and methods for the preparation thereof
12/19/1996CA2222989A1 Paclitaxel synthesis from precursor compounds and methods of producing the same
12/19/1996CA2222919A1 Paclitaxel synthesis from precursor compounds and methods of producing the same
12/18/1996EP0748318A1 Process for preparing polyfluorooxetanes
12/18/1996EP0625146B1 Novel acid anhydrides and preparation and use thereof
12/17/1996US5585397 Viricides
12/11/1996EP0747385A1 Prodrugs of paclitaxel derivatives
12/11/1996EP0747372A1 Taxane derivatives from 14-beta-hydroxy-10 deacetybaccatin III
12/11/1996EP0663906B1 Method of preparing taxane derivatives
12/11/1996CN1137789A Synthesis of taxol and its derivatives
12/07/1996CA2176191A1 Prodrugs of paclitaxel derivatives
12/05/1996WO1996038138A1 Novel taxoids
12/03/1996US5580998 Process for preparing taxoids
12/03/1996US5580997 Baccatin III derivatives
12/03/1996US5580899 Stably associate with lipid carrier for improved delivery
11/1996
11/26/1996US5578739 Process for the preparation of Baccatin III and 10-deacetylbaccatin III derivatives
11/21/1996WO1996036622A1 10-deacetyl-14beta-hydroxybaccatine iii derivatives, a process for the preparation thereof and formulations containing them
11/19/1996US5576450 Process for preparing taxoids
11/19/1996US5576345 Method and means for inhibiting posterior capsule opacification
11/13/1996EP0742315A1 2-Oxetanone sizing agents and their preparation and use
11/13/1996EP0741716A1 Delta 12,13 -iso-taxol analogs, antineoplastic use and pharmaceutical compositions containing them
11/12/1996US5574156 N-carbonyl azetidin-2-ones
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