| Patents for C07D 305 - Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms (5,442) |
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| 04/11/2001 | EP1090637A2 Compositions and methods for treating or preventing inflammatory diseases |
| 04/11/2001 | EP1068192A4 Novel crystalline complexes of baccatin iii with imidazole, 2-methylimidazole or isopropanol |
| 04/11/2001 | EP1056736A4 Alternate method for acylating 10-deacetylbaccatin iii selectively at the c-10 position |
| 04/11/2001 | EP1047682A4 Recovery of taxanes from plant material |
| 04/10/2001 | US6215000 Crystalline complexes of baccatin III with imidazole, 2-methylimidazole or isopropanol |
| 04/10/2001 | US6214863 Synergistic therapy for breast cancer consisting of taxol or taxotere and derivatives, with alkylating agent such as cyclophosphamide and anthracycline antibiotic (daunorubicin or doxorubicin); avoiding/ delaying multi-drug resistance |
| 04/10/2001 | CA2222299C Novel taxoids |
| 04/05/2001 | WO2000009120A8 New use of taxoid derivatives |
| 04/04/2001 | EP1087955A1 The semi-synthesis of baccatin iii |
| 04/04/2001 | EP1087926A2 Analytic substrates and antioxidative agents |
| 04/04/2001 | CN1290305A Method for producing baccatin |
| 04/04/2001 | CN1290304A Process for extracting taxol from taxus cuspidata |
| 04/03/2001 | US6211363 Taxane compounds; antitumor agents |
| 03/28/2001 | CN1288890A Water soluble taxad alcohol derivative |
| 03/22/2001 | WO2001019810A1 Water-soluble cephalomannine esters with poly-amino-acid or the salts thereof, pharmaceutical compositions containing them and their use in medicine |
| 03/21/2001 | EP1085018A1 Taxoid compound and method for producing the same |
| 03/21/2001 | CN1288463A Alternate method for acylating 10-deactetylbaccatin III selectively at the C-10 position |
| 03/21/2001 | CN1288010A Water soluble cephalotaxin phosphorus poly aminoacid ester or its salt, pharmaceutical compositions contg. same, and pharmaceutical use thereof |
| 03/14/2001 | EP1082316A1 Methods and useful intermediates for paclitaxel synthesis from c-7, c-10 di-cbz baccatin iii |
| 03/14/2001 | CN1287120A Taxad alcohol purifying method from its mixture with target spot microtulule protein |
| 03/13/2001 | US6201140 7-0-ethers of taxane derivatives |
| 03/08/2001 | WO2001015675A2 Use of docetaxel for treating hepatocellular carcinoma |
| 03/07/2001 | EP1019347A4 Method for the synthesis of taxanes |
| 03/07/2001 | CN1286686A Taxane derivs |
| 03/06/2001 | US6197981 Oxidation; blocking, deprotecting; anticarcinogenic, antitumor agents |
| 03/06/2001 | US6197980 4-Acetoxy-2α-benzoyloxy-5β,20-epoxy-1β,7β,10β-trihydroxy-9-oxo-11-taxen-13α-yl(2R,3S)-3-t-butoxycarbonylamino-3-phenyl-2-hydroxypropionate trihydrate |
| 02/28/2001 | EP1077937A1 METHOD OF LOCKING 1$g(a)-OH OF VITAMIN D COMPOUNDS IN AXIAL ORIENTATION |
| 02/28/2001 | CN1285412A Method for monitoring high peak of cell growth and taxol synthesis in cultivation of rew cell |
| 02/28/2001 | CN1285351A Taxane with alkyl subtituted lateral chain and medicinal composition containing said compound |
| 02/28/2001 | CN1062561C 7-halo-and 7beta, 8 beta-methano-taxols, antineoplastic use and pharmaceutical compositions containing them |
| 02/27/2001 | US6194582 Multi-drug resistance |
| 02/27/2001 | US6194451 Prevent release tumor necrosis factor; antiinflammatory agents |
| 02/21/2001 | CN1284502A Method of initially separating taxad alcohol from yew plant cell culturing liquid |
| 02/21/2001 | CN1284501A Compound for synthetic taxol, taxol analog and intermediate |
| 02/20/2001 | US6191287 Treating the taxane with a silyamide or a bissilylamide to form c10 silylated taxane |
| 02/15/2001 | WO2001010856A1 Process for the preparation of a paclitaxel c-4 methyl carbonate analog |
| 02/15/2001 | CA2381401A1 Process for the preparation of a paclitaxel c-4 methyl carbonate analog |
| 02/14/2001 | CN1283619A Water-soluble polyhydroxyl derivative of taxusol and its preparing process |
| 02/13/2001 | US6187916 Process for the preparation of taxane derivatives and β-lactam intermediates therefor |
| 02/06/2001 | US6184395 Reaction conditions for the cleavage of silyl ethers in the preparation of paclitaxel(taxol®) and paclitaxel analogues |
| 01/31/2001 | CN1282218A Compositions and method for treatment of primary and metastatic neoplastic diseases using arsenic compounds |
| 01/31/2001 | CN1061339C Novel sulfonamide inhibitors of aspartyl protease |
| 01/30/2001 | US6180802 Method for selective protection of baccatin derivatives and its application to taxane synthesis |
| 01/25/2001 | WO2001005871A1 Amorphous polyether glycols based on bis-substituted oxetane monomers |
| 01/25/2001 | CA2379371A1 Amorphous polyether glycols based on bis-substituted oxetane monomers |
| 01/24/2001 | EP1070502A2 Compositions and methods for treating or preventing inflammatory diseases |
| 01/24/2001 | EP1070057A1 7-hexanoyltaxol and methods for preparing the same |
| 01/23/2001 | US6177573 Process to prepare taxol |
| 01/23/2001 | US6177456 Monohalocephalomannines having anticancer and antileukemic activity and method of preparation therefor |
| 01/23/2001 | US6177033 Pressurization |
| 01/17/2001 | EP1069120A1 Naphthalene derivative, binaphthalene derivative and biphenyl derivative and cationically curable compound |
| 01/17/2001 | EP1068192A1 Novel crystalline complexes of baccatin iii with imidazole, 2-methylimidazole or isopropanol |
| 01/17/2001 | EP1067923A1 2-aroyl-4-acyl paclitaxel (taxol) analogs |
| 01/16/2001 | US6175023 Synthesis of water soluble 9-dihydro-paclitaxel derivatives from 9-dihydro-13-acetylbaccatin III |
| 01/16/2001 | US6175022 Making a nucleophilic group-terminated 2-oxetanone multimer of given formula by reacting a compound having nucleophilic group with a molar excess of a dicarboxylic acid chloride in the presence of basic catalyst and removing salt by-product |
| 01/11/2001 | WO2001002407A2 Taxane derivatives and processes for the preparation thereof |
| 01/10/2001 | EP0898557A4 Water soluble tri-substituted 1,2-dioxetane compounds having increased storage stability, synthetic processes and intermediates |
| 01/10/2001 | CN1279677A Intermediates and methods useful in the semisynthesis of paclitaxel and analogs |
| 01/10/2001 | CN1060476C Preparation process of taxad alcohol |
| 01/03/2001 | EP1064285A1 Novel cephalotaxane derivatives and process for their preparation |
| 12/28/2000 | WO2000078741A2 Process for extraction and purification of paclitaxel from natural sources |
| 12/28/2000 | WO2000078707A1 C-2 hydroxyl protected-n-acyl(2r,3s)-3-phenylisoserine activated esters and methods for production thereof |
| 12/28/2000 | CA2375343A1 C-2 hydroxyl protected-n-acyl(2r,3s)-3-phenylisoserine activated esters and methods for production thereof |
| 12/27/2000 | EP1063234A2 Hydrophobic taxane derivates |
| 12/26/2000 | US6166234 Tripodal cyclopentadiene derivatives and their use |
| 12/26/2000 | US6166228 Reacting a trimethylolalkane with a dialkyl carbonate usinga basic catalyst; first stage stirring and refluxing for 6 hours; second stage distilling off the alcohol formed; and third stage, raising the temperature to decarboxylate |
| 12/22/2000 | CA2275980A1 Process for recovering pacitaxeline from natural sources |
| 12/20/2000 | EP1060172A1 Synthesis of paclitaxel baccatin iii by protecting the 7-hydroxyl using a strong base and an electrophile |
| 12/19/2000 | US6162920 Taxane derivatives having a pyridyl substituted C13 side chain, their preparation and their use as anti-tumor agents |
| 12/12/2000 | US6160135 Taxoids, preparation thereof and pharmaceutical compositions containing same |
| 12/07/2000 | WO2000073293A1 Semi-synthesis of paclitaxel using dialkyldichlorosilanes |
| 12/07/2000 | CA2375253A1 Semi-synthesis of paclitaxel using dialkyldichlorosilanes |
| 12/06/2000 | EP1056736A1 Alternate method for acylating 10-deacetylbaccatin iii selectively at the c-10 position |
| 12/05/2000 | US6156911 Purification of lipstatin |
| 11/30/2000 | WO2000042989A3 Novel hydrogel isolated cochleate formulations, process of preparation and their use for the delivery of biologically relevant molecules |
| 11/29/2000 | CN1275120A Method for synthesis of taxanes |
| 11/28/2000 | US6153756 Salt formation by dissolving paclitaxel and a 2-halo-1-onium tosylate salt in a dry organic solvent, adding a quaternary compound forming agent to the mixture, purification by high performance liquid chromatography |
| 11/28/2000 | US6153217 Nanocochleate formulations, process of preparation and method of delivery of pharmaceutical agents |
| 11/23/2000 | WO2000069840A1 Novel reaction conditions for the cleavage of silyl ethers in the preparation of paclitaxel (taxol®) and paclitaxel analogues |
| 11/23/2000 | CA2373819A1 Novel reaction conditions for the cleavage of silyl ethers in the preparation of paclitaxel (taxol) and paclitaxel analogues |
| 11/22/2000 | EP1053345A1 Method for producing baccatin |
| 11/22/2000 | CN1058714C Method of preparing metal alkoxides |
| 11/21/2000 | US6150541 Anticancer agent; antileukemia agent |
| 11/21/2000 | US6150537 Methods for the esterification of alcohols and compounds useful therefor as potential anticancer agents |
| 11/16/2000 | WO2000068290A2 Poly(3-cyclopropyl-3-hydroxypropionate) and processes for its preparation and derivatives thereof |
| 11/15/2000 | EP1051505A1 Process of extracting taxol from taxus cuspidata |
| 11/15/2000 | CN1058497C Process for preparing 7-trialklsilki baccatin III |
| 11/14/2000 | US6147234 C9 taxane derivatives |
| 11/09/2000 | WO2000066602A1 3-deoxy-desmycosin derivatives and process for their preparation |
| 11/09/2000 | CA2368249A1 3-deoxy-desmycosin derivatives and process for their preparation |
| 11/09/2000 | CA2365776A1 Method for treating abnormal cell proliferation in the brain |
| 11/08/2000 | EP1049686A1 Intermediates and methods useful in the semisynthesis of paclitaxel and analogs |
| 11/08/2000 | EP1049667A1 Novel naphthyl substituted and heterocyclic substituted sulfonamides |
| 11/08/2000 | EP1049666A1 Novel naphthyl-substituted and anilide-substituted sulfonamides |
| 11/07/2000 | US6143902 Semi-synthesis of paclitaxel using a protected c-2 hydroxyl protected-n-acyl (2r,3s)-3-phenylisoserine activated esters |
| 11/07/2000 | US6143900 Stereoselective synthesis of oxazoline derivative |
| 11/02/2000 | EP1047682A1 Recovery of taxanes from plant material |
| 11/01/2000 | CN1271729A New beta-caprolactam, process for preparing taxane, and taxanes with side chain |
| 10/31/2000 | US6140359 Injectable composition |
| 10/31/2000 | US6140273 Herbicides; made by reacting a cyclohexane-1,3-dione with an activated benzoic acid or benzoic acid compound, to give an acylation product, and subsequent rearrangement |