Patents
Patents for C07D 305 - Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms (5,442)
12/2001
12/13/2001WO2001094328A1 Stable isotope labeling of paclitaxel
12/13/2001US20010051736 Methods of treating cell lines expressing multidrug resistance P-glycoprotein
12/13/2001US20010051640 C7 carbamoyloxy substituted taxanes
12/13/2001US20010051639 Exceptional utility as antitumor agents; bioavailability and nontoxic; oral administration; e.g., 10-propionyl-10-deacetyl Baccatin III; anticarcinogenic agents
12/13/2001CA2409944A1 Stable isotope labeling of paclitaxel
12/11/2001US6329193 Taxol production by a microbe
12/06/2001WO2001092245A1 Novel paclitaxel derivatives for the treatment of cancer
12/05/2001EP1160252A1 Avermectin derivatives
12/05/2001EP1159975A2 Anti-angiogenic compositions and methods of use
12/05/2001EP1159974A1 Anti-angiogenic compositions and methods of use
12/05/2001EP0956284A4 Process for selective derivatization of taxanes
11/2001
11/28/2001EP1157018A1 A process for the preparation of taxanes from 10-deacetylbaccatin iii
11/28/2001EP0832080B1 Paclitaxel synthesis from precursor compounds and methods of producing the same
11/28/2001EP0690712B1 Taxanes having a pyridyl substituted side-chain
11/27/2001US6323347 Used for dehydrocyclization reaction of a diol under a gas phase to form lactone; activity, long lifetime and high selectivity of products
11/22/2001US20010044549 Process for the preparation of a paclitaxel C-4 methyl carbonate analog
11/21/2001EP1155691A2 Anti-angiogenic compositions and methods of use
11/21/2001EP1155690A2 Anti-angiogenic compositions and method of use
11/21/2001EP1155689A2 Anti-angiogenic compositions and methods of use
11/21/2001EP1155008A1 C-7 metal alkoxides of baccatin iii
11/21/2001EP0802911B1 Hydrophobic taxane derivatives
11/21/2001EP0708642B1 Taxol derivatives
11/21/2001CN1075066C Taxanes having an alkyl substituted side-chain and pharmaceutical compositions containing them
11/15/2001US20010041803 Blocking with polymer
11/15/2001US20010041796 Taxol derivative; antitumor agents
11/08/2001WO2001083560A1 An antibody selective for a tumor necrosis factor-related apoptosis-inducing ligand receptor and uses thereof
11/08/2001WO2001082859A2 Method for producing r-teatrol analogs having an antineoplastic activity
11/08/2001CA2407965A1 An antibody selective for a tumor necrosis factor-related apoptosis-inducing ligand receptor and uses thereof
11/07/2001EP0923565B1 Process for preparing paclitaxel
11/07/2001EP0912535B1 Conjugates of cis-docosahexaenoic acid and paclitaxel
11/07/2001EP0837846B1 C-2' hydroxyl-benzyl protected, n-carbamate protected (2r,3s)-3-phenylisoserine and production process therefor
11/07/2001EP0776322B1 Method for the preparation of taxol and its derivatives
11/07/2001CN1320598A Process for preparing perfluoroepoxide
11/01/2001US20010037020 Method for preparation of taxol
11/01/2001CA2523096A1 Improved process for the preparation of 3,4-dihydroxybutanoic acid
10/2001
10/31/2001CN1319596A Synthesis of 3,6-dialkyl 5,6-dihydro-4-hydroxide-2H-pyran-2-ketone
10/30/2001US6310201 (3r-cis)-1-benzoyl-3-(1-methoxy-1-methylethoxy)-4-phenyl-2-aze tidinone.
10/24/2001EP1148055A1 C9 taxane derivatives and pharmaceutical compositions containing them
10/24/2001EP1060172A4 Synthesis of paclitaxel baccatin iii by protecting the 7-hydroxyl using a strong base and an electrophile
10/23/2001US6307088 Synthesis of taxol, taxol analogs and their intermediates with variable A-ring side chain structures and compositions thereof
10/23/2001US6307071 Synthesis of paclitaxel from baccatin III by protection of the 7-hydroxyl of baccatin III using a strong base and an electrophile
10/23/2001US6307064 Process to prepare taxol
10/23/2001US6306993 Method and composition for enhancing transport across biological membranes
10/23/2001US6306894 Seals on containers for piclitaxel and sealed containers and drugs
10/18/2001WO2001077094A1 Percyquinnin, a process for its production and its use as a pharmaceutical
10/18/2001CA2405066A1 Percyquinnin, a process for its production and its use as a pharmaceutical
10/17/2001EP1146043A1 Taxanes having an alkyl substituted side-chain and pharmaceutical compositions containing them
10/17/2001EP1144377A1 Oxetanone derivatives
10/17/2001EP1143933A2 Novel hydrogel isolated cochleate formulations, process of preparation and their use for the delivery of biologically relevant molecules
10/17/2001CN1073108C Texane derivatives having pyridil substituted C13 side chain, their prepn. and their use as anti-tumor agents
10/17/2001CN1073106C Taxoids compound, preparation thereof, and pharmaceutical compsns. contg. same
10/17/2001CN1073105C Semi-synthetic taxanes with anti-tumoural activity
10/16/2001CA2035967C Oxetanones
10/11/2001WO2001074800A1 Process for preparing 3-fluoroalkoxymethyl-3-alkyloxetanes
10/11/2001WO2001074799A1 Fluorinated oxetane derivatives and production process thereof
10/10/2001EP1142886A1 Percyquinnin, a process for its production and its use as a pharmaceutical
10/10/2001EP1140885A1 Method for high yield extraction of paclitaxel from paclitaxel-containing material
10/10/2001EP1140884A1 Process for production of an oxetane
10/10/2001EP0923566A4 High molecular weight polymer-based prodrugs
10/10/2001CN1072665C Preparation of unsaturated cyclic ethers
10/09/2001CA2195844C Semi-synthetic taxanes with anti-tumoural activity
10/09/2001CA2029787C Method for preparation of taxol using an oxazinone
10/04/2001EP1137690A2 Peg-based macromonomers, chemically inert polymers prepared therefrom and the use of these polymers for organic synthesis and enzyme reactions
10/02/2001US6297329 Coating composition comprising a bicyclo- or spiro-orthoester functional compound
10/02/2001CA2156908C C9 taxane derivatives and pharmaceutical compositions containing them
09/2001
09/27/2001WO2001070718A1 Taxane anticancer agents
09/27/2001WO2001070717A1 Conversion of 9-dihydro-13-acetylbaccatin iii to baccatin iii and 10-deacetylbaccatin iii
09/27/2001US20010025036 Modifying the structure of a 1alpha-hydroxylated vitamin D compound to increase its in vivo activity by altering the conformational equilibrium of the A-ring to favor a chair conformation that presents 1alphahydroxy in axial orientation
09/27/2001CA2403429A1 Conversion of 9-dihydro-13-acetylbaccatin iii to baccatin iii and 10-deacetylbaccatin iii
09/27/2001CA2400645A1 Taxane anticancer agents
09/26/2001EP0839141B1 Method for extracting and isolating 10-deacetylbaccatin iii
09/25/2001CA2214051C Beta-lactams useful in preparation of taxols
09/20/2001WO2001068624A1 Simple and efficient hydrazinolysis of c-10 and c-13 ester functionalities of taxanes to obtain 10-dab iii
09/20/2001WO2001068089A1 Condensation derivatives of thiocolchicine and baccatin as antitumor agents
09/20/2001WO2001015675A3 Use of docetaxel for treating hepatocellular carcinoma
09/20/2001US20010023255 Phosphonooxymethyl ethers of taxane derivatives
09/20/2001CA2403227A1 Simple and efficient hydrazinolysis of c-10 and c-13 ester functionalities of taxanes to obtain 10-dab iii
09/19/2001EP0600062B1 Polymer-bound paclitaxel derivatives
09/19/2001CN1313764A New use of taxoid derivatives
09/18/2001US6291692 Water solubility; as chemical intermediate in synthesis of taxanes
09/18/2001US6291691 Process for selective derivatization of taxanes
09/18/2001US6291690 Hydrophobic taxane derivatives
09/13/2001WO2001066535A1 Process for manufacturing paclitaxel and 13-acetyl-9-dihydrobaccatin iii
09/13/2001US20010021783 New taxoids, their preparation and pharmaceutical compositions containing them
09/12/2001CN1312714A Pharmaceutical composition containing lipase inhibitors and chitosan
09/05/2001EP1070057A4 7-hexanoyltaxol and methods for preparing the same
09/05/2001EP0826688B1 Pentacyclic compounds
08/2001
08/30/2001WO2001062753A1 Method and apparatus for preparing taxol using supercritical fluid from source materials
08/30/2001US20010018531 Therapy for mammary or colon tumors
08/29/2001EP1127886A1 Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-2H-pyran-2one
08/28/2001US6281368 Simple and efficient hydrazinolysis of C-10 and C-13 ester functionalities of taxanes to obtain 10-DAB III
08/28/2001US6281365 (Gem-heterocyclodimethanamine-n,n′)platinum complexes
08/28/2001CA2017252C Retroviral protease inhibiting compounds
08/22/2001EP0876361B1 4,10beta-diacetoxy-2alpha-benzoyloxy-5beta,20-epoxy-1-hydroxy-9-oxo-19-nor-cyclopropa(g]tax-11-ene-13alpha-yl (2r,3s)-tert-butoxycarbonylamino-2-hydroxy-3-phenylpropionate dihydrate, and method for preparing same
08/21/2001US6278026 Intermediates for tricyclic or tetracyclic taxanes
08/16/2001US20010014746 Preparation of substituted isoserine esters using metal alkoxides and beta-lactams
08/16/2001EP0885208B1 Taxoids, their preparation and pharmaceutical compositions containing them
08/16/2001EP0874838B1 Novel taxoids, preparation thereof and pharmaceutical compositions containing same
08/15/2001CN1308609A Method of locking 1 & alpha, -OH of vitamin d compounds in axial orientation
08/15/2001CN1308073A Partially synthetic seco-taxinane with antineoplastic activity
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