Patents for C07D 305 - Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms (5,442) |
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12/13/2001 | WO2001094328A1 Stable isotope labeling of paclitaxel |
12/13/2001 | US20010051736 Methods of treating cell lines expressing multidrug resistance P-glycoprotein |
12/13/2001 | US20010051640 C7 carbamoyloxy substituted taxanes |
12/13/2001 | US20010051639 Exceptional utility as antitumor agents; bioavailability and nontoxic; oral administration; e.g., 10-propionyl-10-deacetyl Baccatin III; anticarcinogenic agents |
12/13/2001 | CA2409944A1 Stable isotope labeling of paclitaxel |
12/11/2001 | US6329193 Taxol production by a microbe |
12/06/2001 | WO2001092245A1 Novel paclitaxel derivatives for the treatment of cancer |
12/05/2001 | EP1160252A1 Avermectin derivatives |
12/05/2001 | EP1159975A2 Anti-angiogenic compositions and methods of use |
12/05/2001 | EP1159974A1 Anti-angiogenic compositions and methods of use |
12/05/2001 | EP0956284A4 Process for selective derivatization of taxanes |
11/28/2001 | EP1157018A1 A process for the preparation of taxanes from 10-deacetylbaccatin iii |
11/28/2001 | EP0832080B1 Paclitaxel synthesis from precursor compounds and methods of producing the same |
11/28/2001 | EP0690712B1 Taxanes having a pyridyl substituted side-chain |
11/27/2001 | US6323347 Used for dehydrocyclization reaction of a diol under a gas phase to form lactone; activity, long lifetime and high selectivity of products |
11/22/2001 | US20010044549 Process for the preparation of a paclitaxel C-4 methyl carbonate analog |
11/21/2001 | EP1155691A2 Anti-angiogenic compositions and methods of use |
11/21/2001 | EP1155690A2 Anti-angiogenic compositions and method of use |
11/21/2001 | EP1155689A2 Anti-angiogenic compositions and methods of use |
11/21/2001 | EP1155008A1 C-7 metal alkoxides of baccatin iii |
11/21/2001 | EP0802911B1 Hydrophobic taxane derivatives |
11/21/2001 | EP0708642B1 Taxol derivatives |
11/21/2001 | CN1075066C Taxanes having an alkyl substituted side-chain and pharmaceutical compositions containing them |
11/15/2001 | US20010041803 Blocking with polymer |
11/15/2001 | US20010041796 Taxol derivative; antitumor agents |
11/08/2001 | WO2001083560A1 An antibody selective for a tumor necrosis factor-related apoptosis-inducing ligand receptor and uses thereof |
11/08/2001 | WO2001082859A2 Method for producing r-teatrol analogs having an antineoplastic activity |
11/08/2001 | CA2407965A1 An antibody selective for a tumor necrosis factor-related apoptosis-inducing ligand receptor and uses thereof |
11/07/2001 | EP0923565B1 Process for preparing paclitaxel |
11/07/2001 | EP0912535B1 Conjugates of cis-docosahexaenoic acid and paclitaxel |
11/07/2001 | EP0837846B1 C-2' hydroxyl-benzyl protected, n-carbamate protected (2r,3s)-3-phenylisoserine and production process therefor |
11/07/2001 | EP0776322B1 Method for the preparation of taxol and its derivatives |
11/07/2001 | CN1320598A Process for preparing perfluoroepoxide |
11/01/2001 | US20010037020 Method for preparation of taxol |
11/01/2001 | CA2523096A1 Improved process for the preparation of 3,4-dihydroxybutanoic acid |
10/31/2001 | CN1319596A Synthesis of 3,6-dialkyl 5,6-dihydro-4-hydroxide-2H-pyran-2-ketone |
10/30/2001 | US6310201 (3r-cis)-1-benzoyl-3-(1-methoxy-1-methylethoxy)-4-phenyl-2-aze tidinone. |
10/24/2001 | EP1148055A1 C9 taxane derivatives and pharmaceutical compositions containing them |
10/24/2001 | EP1060172A4 Synthesis of paclitaxel baccatin iii by protecting the 7-hydroxyl using a strong base and an electrophile |
10/23/2001 | US6307088 Synthesis of taxol, taxol analogs and their intermediates with variable A-ring side chain structures and compositions thereof |
10/23/2001 | US6307071 Synthesis of paclitaxel from baccatin III by protection of the 7-hydroxyl of baccatin III using a strong base and an electrophile |
10/23/2001 | US6307064 Process to prepare taxol |
10/23/2001 | US6306993 Method and composition for enhancing transport across biological membranes |
10/23/2001 | US6306894 Seals on containers for piclitaxel and sealed containers and drugs |
10/18/2001 | WO2001077094A1 Percyquinnin, a process for its production and its use as a pharmaceutical |
10/18/2001 | CA2405066A1 Percyquinnin, a process for its production and its use as a pharmaceutical |
10/17/2001 | EP1146043A1 Taxanes having an alkyl substituted side-chain and pharmaceutical compositions containing them |
10/17/2001 | EP1144377A1 Oxetanone derivatives |
10/17/2001 | EP1143933A2 Novel hydrogel isolated cochleate formulations, process of preparation and their use for the delivery of biologically relevant molecules |
10/17/2001 | CN1073108C Texane derivatives having pyridil substituted C13 side chain, their prepn. and their use as anti-tumor agents |
10/17/2001 | CN1073106C Taxoids compound, preparation thereof, and pharmaceutical compsns. contg. same |
10/17/2001 | CN1073105C Semi-synthetic taxanes with anti-tumoural activity |
10/16/2001 | CA2035967C Oxetanones |
10/11/2001 | WO2001074800A1 Process for preparing 3-fluoroalkoxymethyl-3-alkyloxetanes |
10/11/2001 | WO2001074799A1 Fluorinated oxetane derivatives and production process thereof |
10/10/2001 | EP1142886A1 Percyquinnin, a process for its production and its use as a pharmaceutical |
10/10/2001 | EP1140885A1 Method for high yield extraction of paclitaxel from paclitaxel-containing material |
10/10/2001 | EP1140884A1 Process for production of an oxetane |
10/10/2001 | EP0923566A4 High molecular weight polymer-based prodrugs |
10/10/2001 | CN1072665C Preparation of unsaturated cyclic ethers |
10/09/2001 | CA2195844C Semi-synthetic taxanes with anti-tumoural activity |
10/09/2001 | CA2029787C Method for preparation of taxol using an oxazinone |
10/04/2001 | EP1137690A2 Peg-based macromonomers, chemically inert polymers prepared therefrom and the use of these polymers for organic synthesis and enzyme reactions |
10/02/2001 | US6297329 Coating composition comprising a bicyclo- or spiro-orthoester functional compound |
10/02/2001 | CA2156908C C9 taxane derivatives and pharmaceutical compositions containing them |
09/27/2001 | WO2001070718A1 Taxane anticancer agents |
09/27/2001 | WO2001070717A1 Conversion of 9-dihydro-13-acetylbaccatin iii to baccatin iii and 10-deacetylbaccatin iii |
09/27/2001 | US20010025036 Modifying the structure of a 1alpha-hydroxylated vitamin D compound to increase its in vivo activity by altering the conformational equilibrium of the A-ring to favor a chair conformation that presents 1alphahydroxy in axial orientation |
09/27/2001 | CA2403429A1 Conversion of 9-dihydro-13-acetylbaccatin iii to baccatin iii and 10-deacetylbaccatin iii |
09/27/2001 | CA2400645A1 Taxane anticancer agents |
09/26/2001 | EP0839141B1 Method for extracting and isolating 10-deacetylbaccatin iii |
09/25/2001 | CA2214051C Beta-lactams useful in preparation of taxols |
09/20/2001 | WO2001068624A1 Simple and efficient hydrazinolysis of c-10 and c-13 ester functionalities of taxanes to obtain 10-dab iii |
09/20/2001 | WO2001068089A1 Condensation derivatives of thiocolchicine and baccatin as antitumor agents |
09/20/2001 | WO2001015675A3 Use of docetaxel for treating hepatocellular carcinoma |
09/20/2001 | US20010023255 Phosphonooxymethyl ethers of taxane derivatives |
09/20/2001 | CA2403227A1 Simple and efficient hydrazinolysis of c-10 and c-13 ester functionalities of taxanes to obtain 10-dab iii |
09/19/2001 | EP0600062B1 Polymer-bound paclitaxel derivatives |
09/19/2001 | CN1313764A New use of taxoid derivatives |
09/18/2001 | US6291692 Water solubility; as chemical intermediate in synthesis of taxanes |
09/18/2001 | US6291691 Process for selective derivatization of taxanes |
09/18/2001 | US6291690 Hydrophobic taxane derivatives |
09/13/2001 | WO2001066535A1 Process for manufacturing paclitaxel and 13-acetyl-9-dihydrobaccatin iii |
09/13/2001 | US20010021783 New taxoids, their preparation and pharmaceutical compositions containing them |
09/12/2001 | CN1312714A Pharmaceutical composition containing lipase inhibitors and chitosan |
09/05/2001 | EP1070057A4 7-hexanoyltaxol and methods for preparing the same |
09/05/2001 | EP0826688B1 Pentacyclic compounds |
08/30/2001 | WO2001062753A1 Method and apparatus for preparing taxol using supercritical fluid from source materials |
08/30/2001 | US20010018531 Therapy for mammary or colon tumors |
08/29/2001 | EP1127886A1 Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-2H-pyran-2one |
08/28/2001 | US6281368 Simple and efficient hydrazinolysis of C-10 and C-13 ester functionalities of taxanes to obtain 10-DAB III |
08/28/2001 | US6281365 (Gem-heterocyclodimethanamine-n,n′)platinum complexes |
08/28/2001 | CA2017252C Retroviral protease inhibiting compounds |
08/22/2001 | EP0876361B1 4,10beta-diacetoxy-2alpha-benzoyloxy-5beta,20-epoxy-1-hydroxy-9-oxo-19-nor-cyclopropa(g]tax-11-ene-13alpha-yl (2r,3s)-tert-butoxycarbonylamino-2-hydroxy-3-phenylpropionate dihydrate, and method for preparing same |
08/21/2001 | US6278026 Intermediates for tricyclic or tetracyclic taxanes |
08/16/2001 | US20010014746 Preparation of substituted isoserine esters using metal alkoxides and beta-lactams |
08/16/2001 | EP0885208B1 Taxoids, their preparation and pharmaceutical compositions containing them |
08/16/2001 | EP0874838B1 Novel taxoids, preparation thereof and pharmaceutical compositions containing same |
08/15/2001 | CN1308609A Method of locking 1 & alpha, -OH of vitamin d compounds in axial orientation |
08/15/2001 | CN1308073A Partially synthetic seco-taxinane with antineoplastic activity |