| Patents for C07D 305 - Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms (5,442) |
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| 02/27/2003 | WO2003016543A2 Enzymatic resolution of t-butyl taxane derivatives |
| 02/27/2003 | US20030040508 Altering the conformational equilibrium of the A- ring of a 1 alpha -hydroxylated vitamin D compound to favor a chair conformation for A-ring that presents the 1 alpha-hydroxyl in an axial orientation |
| 02/26/2003 | EP1285920A1 C10 Ester sustituted taxanes as antitumor agents |
| 02/26/2003 | EP1285919A1 C10 Carbonate substituted taxanes as antitumor agents |
| 02/26/2003 | EP1285918A1 C7 Ester substituted taxanes as antitumor agents |
| 02/26/2003 | CN1398859A Process of preparing 10-deacetyl Bakatin III from taxad branch and leaf residue |
| 02/20/2003 | WO2003013503A1 C-2' methylated derivatives of paclitaxel for use as antitumour agents |
| 02/20/2003 | WO2002030882A9 Sulfoxide and bis-sulfoxide compounds and compositions for cholesterol management and related uses |
| 02/20/2003 | WO2002030860A9 Ketone compounds and compositions for cholesterol management and related uses |
| 02/20/2003 | US20030036661 For therapy of cancer |
| 02/20/2003 | CA2456523A1 C-2' methylated derivatives of paclitaxel for use as antitumour agents |
| 02/19/2003 | EP1032565B1 Method for preparing derivatives of the taxoid class |
| 02/19/2003 | EP0690867B1 Taxanes having furyl or thienyl substituted side-chain |
| 02/19/2003 | EP0687260B1 Process for the preparation of 9-desoxotaxanes |
| 02/18/2003 | US6521660 3′-alkyl substituted taxanes and pharmaceutical compositions containing them |
| 02/13/2003 | WO2002051388A3 Treatment of inoperable tumors by stereotactic injection of microspheres |
| 02/13/2003 | US20030032820 Extractions, separations, and purifications of plant material for pure paclitaxel and/or cephalomannine and/or 9-dihydro-13 -acetylbaccatin III and/or 10-deacetylbaccatin III |
| 02/12/2003 | CN1396947A Polymerizable liquid crystalline dioxetanes, their preparation and use |
| 02/12/2003 | CN1396919A Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-pyran-2-one |
| 02/12/2003 | CN1396917A Chromatographic separation method of paclitaxel and cephalomannin |
| 02/06/2003 | US20030028039 Starting from various bicyclo(5.3.1)undec-10-ene compounds of given formula having protected hydroxyl groups; use as antitumor agents |
| 02/06/2003 | US20030028038 Semi-synthetic taxanes with antitumor and antiangiogenetic activities |
| 02/06/2003 | US20030027855 Preparation of a derivative or analog of baccatin III or 10-desacetyl baccatin III having a C9 hydroxy substituent by selective reduction of the C9 keto compound |
| 02/05/2003 | EP1280786A1 Simple and efficient hydrazinolysis of c-10 and c-13 ester functionalities of taxanes to obtain 10-dab iii |
| 02/05/2003 | CN1395571A Semi-synthetic taxanes with antitumor and antiangiogenetic activities |
| 02/05/2003 | CN1394961A Method for mass production of taxinol by utilizing batch or semi-continuous culture |
| 02/05/2003 | CN1100771C Phosphononooxymethyl ethers for taxame derivatives |
| 02/05/2003 | CN1100770C Hydrolysis-promoitng taxane hydrophobic derivatives |
| 02/04/2003 | US6515152 Process for production of an oxetane |
| 02/04/2003 | US6515151 Method for the preparation of novel sidechain-bearing taxanes and intermediates thereof |
| 02/04/2003 | US6515016 Treating or preventing multiple sclerosis, by administering an antimicrotubule agent; treating various other inflammatory diseases |
| 02/04/2003 | US6514732 Acetylation of 10-deacetylbaccatin using acetyl transferase with acetyl coA; 10-hydroxytaxa-O-acetyltransferase; Used in preparation of taxol. |
| 01/31/2003 | CA2354486A1 C7 ester substituted taxanes |
| 01/31/2003 | CA2354478A1 C10 carbonate substituted taxanes |
| 01/31/2003 | CA2354471A1 C10 ester substituted taxanes |
| 01/30/2003 | US20030022865 Sulfoxide and bis-sulfoxide compounds and compositions for cholesterol management and related uses |
| 01/29/2003 | EP0983255B1 Substituted 2-benzoyl-cyclohexane-1,3-diones |
| 01/29/2003 | CN1393438A Taxane derivative and its preparing process and usage |
| 01/23/2003 | WO2003006430A1 Taxol enhancer compounds |
| 01/23/2003 | US20030018013 Cardiovascular disorders; antilipemic agents; Alzheimer's disease |
| 01/22/2003 | EP1157018B1 A process for the preparation of taxanes from 10-deacetylbaccatin iii |
| 01/22/2003 | CN1392145A Semi synthetic method for taxol |
| 01/21/2003 | US6509484 Trifluoroacetic acid amine salt taxane derivatives useful for taxol production |
| 01/16/2003 | WO2003004482A1 Efficient process for the production of 10-dab iii by selective hydrazinolysis of various taxanes |
| 01/16/2003 | WO2002072527A3 1-butyric acid derivatives such as carbomethoxypropionyl cyanide or leflunomide derivatives, and the therapeutic use thereof |
| 01/16/2003 | US20030013899 Production of taxol and taxanes |
| 01/16/2003 | US20030013889 Process for the preparation of taxane derivatives |
| 01/16/2003 | CA2452847A1 Efficient process for the production of 10-dab iii by selective hydrazinolysis of various taxanes |
| 01/15/2003 | EP1275389A1 Compositions containing C7 Taxanes |
| 01/15/2003 | EP1274698A1 Percyquinnin, a process for its production and its use as a pharmaceutical |
| 01/15/2003 | CN1098846C Water-soluble polyhydroxyl derivative of taxol and its preparing process |
| 01/14/2003 | US6506912 Method of locking 1α-OH of vitamin D compounds in axial orientation |
| 01/14/2003 | US6506411 Anti-angiogenic compositions and methods of use |
| 01/09/2003 | US20030009039 Reacting a beta -lactam with an alkoxide to form substituted isoserine ester compound |
| 01/08/2003 | EP1194423B1 Process for extraction and purification of paclitaxel from natural sources |
| 01/08/2003 | CN1389461A Chlorohydrination process of producing epoxypropane and its production equipment |
| 01/08/2003 | CN1098356C Method for monitoring high peak of cell growth and taxol synthesis in cultivation of rew cell |
| 01/07/2003 | US6504035 3-deoxy-desmycosin derivatives and process for their preparation |
| 01/07/2003 | US6503396 Solvent extraction, liquid-liquid separation and column chromatography of needles and other parts of yew trees |
| 01/07/2003 | CA2149055C Antitumoral compositions containing taxan derivatives |
| 01/07/2003 | CA2143208C Sulfonamide inhibitors of hiv-aspartyl protease |
| 01/02/2003 | US20030004210 Coupling to cell binding agent; killing cells |
| 01/02/2003 | US20030003094 Compound which disrupts microtubule function and polymeric carrier, with proviso that polymeric carrier is not a capsule |
| 01/02/2003 | EP1270564A1 Process for preparing 3-fluoroalkoxymethyl-3-alkyloxetanes |
| 01/02/2003 | EP1270563A1 Fluorinated oxetane derivatives and production process thereof |
| 01/02/2003 | EP1268458A1 Conversion of 9-dihydro-13-acetylbaccatin iii to baccatin iii and 10-deacetylbaccatin iii |
| 01/01/2003 | CN1388245A Method of raising taxol yield of south taxad |
| 01/01/2003 | CN1388106A Tubular reactor and reaction method for alcoholizing propenyl chloride |
| 01/01/2003 | CN1387948A Formula and prepn process for epoxidating propylene to prepare epoxy propane catalyst in oxy-hydrogen atmosphere |
| 01/01/2003 | CN1097586C Process for synthesizing paclitaxel |
| 12/31/2002 | US6500966 Process for the preparation of taxanes from 10-deacetylbaccatin III |
| 12/31/2002 | US6500859 Administering microtubule stabilizing chemotherapeutic agent for prophylaxis of arterial disease |
| 12/31/2002 | US6500858 For therapy of cancer |
| 12/26/2002 | US20020198141 Molecular conjugates for use in treatment of cancer |
| 12/26/2002 | US20020197245 Antitumour compositions containing taxane derivatives |
| 12/25/2002 | CN1097044C Taxane derivs. and drugs contg. same |
| 12/18/2002 | CN1096453C Method for acylating 10-deacatylbaccatin III selectively at the C-10 position |
| 12/17/2002 | US6495705 10-deacetyl baccatin iii (10-dab iii); containing a solvent reactive with hydrazine hydrate and a spectrum of taxanes, such as unwanted taxanes; precursor in the formation of paclitaxel |
| 12/17/2002 | US6495704 Process for the preparation of a derivative or analog of baccatin iii or 10-desacetyl baccatin iii having a c9 substituent other than keto in which the c9 keto substituent of taxol, a taxol analog, baccatin iii or 10-desacetyl |
| 12/17/2002 | US6495663 Method and composition for enhancing transport across biological membranes |
| 12/17/2002 | US6495636 A 3-(ethyleneoxyalkyloxyalkyl)oxetane and derivatives; copolymerized with a 1,1-difluoroethylene or derivative; very compatible and copolymerizable with unsaturated compounds; waterproofing; radiation transparent |
| 12/12/2002 | US20020187992 Prodrugs via acylation with cinnamate |
| 12/11/2002 | EP1263749A1 Taxane anticancer agents |
| 12/11/2002 | EP1263431A1 Condensation derivatives of thiocolchicine and baccatin as antitumor agents |
| 12/05/2002 | US20020183385 Administering a therapeutically effective amount of arsenic compounds to a mammal for treating solid tumor |
| 12/04/2002 | EP1261657A2 Poly(3-cyclopropyl-3-hydroxypropionate) and processes for its preparation and derivatives thereof |
| 12/04/2002 | EP1261596A1 Method and apparatus for preparing taxol using supercritical fluid from source materials |
| 12/04/2002 | EP1022277B1 New taxane derivatives |
| 12/04/2002 | EP0690856B1 Anti-tumor compounds, pharmaceutical compositions, methods for preparation thereof and for treatment |
| 12/04/2002 | CN1095464C Tech process of oxidizing propylene with hydrogen peroxide solution to produce epoxy propane continuously |
| 12/04/2002 | CN1095400C Catalyst for preparing gamma-butyrolactone from cis-aldehyde by ordinary-pressure gas-phase hydrogenation and its use |
| 11/28/2002 | US20020177609 Fatty alcohol drug conjugates |
| 11/27/2002 | EP1260507A1 Synthesis of taxol, analogs and intermediates with variable A-nng side chains |
| 11/27/2002 | EP1260223A1 Taxanes having furyl or thienyl substituted side-chain |
| 11/27/2002 | EP1260222A1 Butenyl-substituted taxanes and composition |
| 11/27/2002 | CN1094940C Taxol derivative with antineoplastic activity |
| 11/26/2002 | CA2148103C Process for preparing taxane derivatives |
| 11/26/2002 | CA2130333C Process for preparing .beta.-phenylisoserine and analogues thereof |
| 11/21/2002 | WO2002092600A1 Retinol derivatives potentiation of active substances by micellar preparation |
| 11/21/2002 | WO2002078690A3 Taxoid anti-tumor agents and pharmaceutical compositions thereof |