Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
06/2001
06/07/2001WO2001040211A1 A PROCESS FOR THE PREPARATION OF {2-[4-(α-PHENYL-p-CHLOROBENZYL)PIPERAZIN-1-YL]ETHOXY}ACETIC ACID AND NOVEL INTERMEDIATES THEREFOR
06/07/2001WO2001040188A1 Curcumin analogues for treating cancer
06/07/2001WO2001040147A1 Catalysis using phosphine oxide compounds
06/07/2001WO2001039769A1 Hypoglycemics comprising organic zinc (ii) complexes
06/07/2001WO2001030749B1 Novel compounds
06/07/2001US20010003121 Adamantane derivatives such as 2,4-dichloro-N-(tricyclo(3.3.1.13,7)dec-1-methyl)-benzamide; administering to treat rheumatoid arthritis; immunosuppressant
06/07/2001DE19958496A1 Verfahren zur Herstellung von 5-(1-Piperazinyl)-benzofuran-2-carboxamid durch Übergangsmetallkatalysierte Aminierung A process for the preparation of 5- (1-piperazinyl) benzofuran-2-carboxamide by transition metal amination
06/07/2001CA2393440A1 Curcumin analogs with anti-tumor and anti-angiogenic properties
06/06/2001EP1104413A2 Piperidine and piperazine derivatives, process for their preparation and pharmaceutical compounds containing them
06/06/2001EP0873329B1 Novel n-aminoalkylfluorenecarboxamides; a new class of dopamine receptor subtype specific ligands
06/06/2001CN1298399A Substituted alxoxycarbonyl compounds
06/06/2001CN1298299A Antibacterial agents
06/05/2001US6242644 N-(4-carbamimidoyl-phenyl)-glycine derivatives
06/05/2001US6242606 Reacting a a,a-dimethylphenylacetic acid amide with a w-halo compound produces w'-halo-a-keto-a,a-dimethylphenylacetic acid amide and reacting it with a piperidine compound; 2-(4-(4-chloro-butyryl)-phenyl)-2-methy-propionic acid
06/05/2001US6242605 Aryloxy-alkyl-dialkylamines
06/05/2001US6242596 Preparation of betamethyl carbapenem intermediates
06/05/2001US6242495 Compounds and compositions for delivering active agents
06/05/2001US6242494 Angiogenesis inhibitors, antitumor agents, diabetic retinopathy, and antiinflammatory agents
06/05/2001US6242470 Rheumatic diseases; antiarthritic agents, antiallergens; irritable bowel syndrome; amidation
06/05/2001CA2039073C Method of removing water from a dilute solution of n-methylmorpholine-n-oxide, n-methylmorpholine, or morpholine
05/2001
05/31/2001WO2001038561A1 Methods of use of peptide deformylase inhibitors as novel antibacterial agents
05/31/2001WO2001038309A1 β-AMINO ACID-, ASPARTIC ACID- AND DIAMINOPROPIONIC-BASED INHIBITORS OF FACTOR Xa
05/31/2001WO2001037826A1 Npyy5 antagonists
05/31/2001WO1999064041A9 Multibinding agents that modulate nmda receptors
05/31/2001DE19957672A1 Purification and drying of crude pyrrolidine, used as intermediate e.g. in synthesis of plant protection agents and pharmaceuticals, involves continuous distillation in distillation and concentration column at reduced pressure
05/31/2001CA2392576A1 .beta.-amino acid-, aspartic acid- and diaminopropionic-based inhibitors of factor xa
05/30/2001EP1103552A1 Benzothiepin derivatives, process for the preparation of the same and uses thereof
05/30/2001EP1103536A1 Process for the preparation of chiral amines by asymmetric hydrogenation of enamines
05/30/2001EP1102743A1 Amide derivatives which are useful as cytokine inhibitors
05/30/2001EP1102739A1 Glucocorticoid and thyroid hormone receptor ligands for the treatment of metabolic disorders
05/30/2001EP1102597A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht 4 receptors
05/30/2001EP1102538A1 Plant growth regulator compositions
05/30/2001CN1297441A Heterocyclically substd. amides used as calpain inhibitors
05/30/2001CN1066444C Nitrogenous derivs. for elemene and their use as anticancer drugs
05/30/2001CN1066438C Preparation of beta-methyl carbapenem intermediates
05/29/2001US6239313 From an inclusion complex of epoxide with cyclodextrin and nucleophilic compound
05/29/2001US6239277 Alkylation of amine group in piperazine ring
05/29/2001US6239179 N-aminoalkyl-2-anthracenecarboxamides; new dopamine receptor subtype specific ligands
05/29/2001US6239175 Carbamoyloxy derivatives of mutiline and their use as antibacterials
05/29/2001US6239154 Arylacetamides, agonists at kappa opioid receptors.
05/29/2001US6239151 Compounds as inhibitor of tumor necrosis factor alpha release
05/29/2001US6239135 Arylpiperazines having activity at the serotonin 1A receptor
05/25/2001WO2001036403A1 Urea derivatives as anti-inflammatory agents
05/25/2001WO2001036386A1 Diabetic remedy containing dipiperazine derivative
05/25/2001WO2001036376A1 Novel phenylalanine derivatives
05/25/2001WO2001036375A1 Aminoalcohol derivatives useful for the treatment of gastrointestinal disorders
05/25/2001WO2001036374A2 Bis-basic compounds for use as tryptase inhibitors, method for producing the same and their use as medicaments
05/25/2001WO2001036360A1 Triphenylalkene derivatives and their use as selective estrogen receptor modulators
05/25/2001WO2000077027A3 Serine protease inhibitors
05/25/2001WO2000039081A3 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
05/24/2001US20010001799 Anticoagulant
05/23/2001EP1101755A1 Anthranilic acid derivatives
05/23/2001EP1100794A1 COMPOUNDS SPECIFIC FOR THE HUMAN $g(a) 1d? ADRENERGIC RECEPTOR AND USES THEREOF
05/23/2001EP1100790A1 Antidiabetic piperazine derivatives, processes for their preparation and compositions containing them
05/23/2001EP1100763A1 Diketoacid-derivatives as inhibitors of polymerases
05/23/2001EP1100519A1 Multibinding agents that modulate nmda receptors
05/23/2001EP1100503A2 Non-imidazole alkylamines as histamine h 3?-receptor ligands and their therapeutic applications
05/23/2001EP1100495A1 Propenamides as ccr5 modulators
05/23/2001EP1100485A1 Substituted anilide compounds and methods
05/23/2001EP1100483A2 Glucocorticoid-selective anti-inflammatory agents
05/23/2001EP0689536B1 Naphthalene derivatives
05/23/2001DE19955476A1 Bis-basische Verbindungen als Tryptase-Inhibitoren, Verfahren zu deren Herstellung sowie deren Verwendung als Arzneimittel Bis-basic compounds as tryptase inhibitors, to processes for their preparation and their use as medicaments
05/23/2001CN1296478A Histamine H3 receptor ligands
05/23/2001CN1296477A Piperazine derivatives and process for the preparation thereof
05/23/2001CN1296411A Remedies for cardiac dilastolit disorders
05/23/2001CN1296382A Plant growth regulator compositions
05/22/2001US6235938 Transition metal-catalyzed process for preparing N-aryl amine compounds
05/22/2001US6235929 Tripeptide α-ketoamides
05/22/2001US6235927 Process for the separation of a mixture of enantiomers
05/22/2001US6235875 Human and animal anthelmintic
05/22/2001US6235791 Using cis n-cyclohexyl-n-ethyl(3-(3-chloro-cyclohexylphenyl)allyl)amine
05/22/2001US6235787 Antiinflammatory agents; rheumatic diseases; bone disorders; skin disorders; multiple sclerosis
05/22/2001US6235778 Anticoagulants
05/22/2001US6235736 3-anilino-2-cycloalkenone derivatives
05/22/2001US6235732 Neurokinin antagonists
05/22/2001US6235218 Reacting heterocyclic amine with monoaldehyde or dialdehyde and hydrogen cyanide or alkali metal cyanide in aqueous medium, quaternizing amine with alkylating agent at ph controlled to prevent formation of protonated intermediate
05/17/2001WO2001034591A2 Substituted 4h-chromene and analogs as activators of caspases and inducers of apoptosis and the use thereof
05/17/2001WO2001034588A1 Process for producing benzylamine compound
05/17/2001WO2001034587A2 Process for preparing n-(4-hydroxy-phenyl)-n'-(4'-aminophenyl)-piperazine
05/17/2001WO2001034586A2 Branched adamantyl and noradamantyl aryl- and aralkylpiperazines with serotonin 5-ht1a activity
05/17/2001WO2001034578A1 Compounds with anti-helicobacter pylori activity
05/17/2001WO2001034569A1 Pancreatitis remedies
05/17/2001WO2001034561A1 Processes for the preparation of sumatriptan and related compounds
05/17/2001WO2001034135A2 Oncolytic combinations for the treatment of cancer
05/17/2001CA2390789A1 Oncolytic combinations for the treatment of cancer
05/17/2001CA2390524A1 Branched adamantyl and noradamantyl aryl- and aralkylpiperazines with serotonin 5-ht1a activity
05/17/2001CA2389514A1 Processes for the preparation of sumatriptan and related compounds
05/16/2001EP1099692A1 N,n-substituted cyclic amine derivatives
05/16/2001EP1098892A1 Biphenyl derivatives
05/16/2001EP1098870A2 Nitric esters and nitrate salts of specific drugs
05/16/2001EP1098864A1 Method for hydrogenating unsaturated heterocyclic compounds
05/16/2001EP1098651A2 Novel urokinase inhibitors
05/16/2001EP1098642A1 Methods for treating conditions modulated by lactosylceramide
05/16/2001CN1295479A Beta 2-adrenergic receptor agonist
05/16/2001CN1295475A Medicine for improving optic disc circulation
05/15/2001US6232476 Intermediates in a process for cis-1-{2-[4-(6-methoxy-2-phenyl-1,2,3,4-tetrahydronaphthalen-1-yl)phenoxy]ethyl}pyrrolidine
05/15/2001US6232467 Biosynthesis of an amine with ketone and boron compound; compoundlibraries
05/15/2001US6232342 Protease inhibitors
05/15/2001US6232336 Nitric oxide-releasing amidine- and enamine-derived diazeniumdiolates, compositions and uses thereof and method of making same
05/15/2001US6232314 Arylalkylpiperazine compounds as antioxidants