Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
04/2005
04/14/2005WO2005033056A2 Triphenylethylene compounds as selective estrogen receptor modulators
04/14/2005WO2005032471A2 Benzylether and benzylamino beta-secretase inhibitors for the treatment of alzheimer's disease
04/14/2005WO2004113391A3 Improved pharmaceutical drug candidates and methods for preparation thereof
04/14/2005WO2003090678A3 Antileishmanial dinitroaniline sulfonamides with activity against parasite tubulin
04/14/2005US20050080271 Peptidomimetic ligands for cellular receptors and ion channels
04/14/2005US20050080141 Amino diols useful in the treatment of alzheimer's disease
04/14/2005US20050080119 Diaminopropionic acid derivatives
04/14/2005US20050080099 Methods and kits for treating depression or preventing deterioration of cognitive function
04/14/2005US20050080090 Such as 7-(Imidazolo[4,5-b]pyridin-1-yl)-1-(1-methylpyrrolidin-3-yl)naphthalene; for treating depression, anxiety, eating disorders, drug abuse, cluster headache, migraine, pain, and other disorders arising from deficient serotonergic neurotransmission
04/14/2005US20050080088 Novel compounds
04/14/2005US20050080077 Serotonin receptor antagonists such as cis-4,N-dimethyl-N-(3-(4-methylpiperidin-1-yl)cyclopentyl)-benzenesulfonamide for treatment of neurological conditions (depression and sleep disorders)
04/14/2005US20050080073 Sulfonylaminocarboxiylic acid N-arylamides as guanylate cyclase activators
04/14/2005US20050080072 Such as 11-[4-[2-(2-hydroxyethoxy)ethyl]-1-pinerazinyl]dibenzo[b,f][1,4]thiazepine (quetiapine) via reduction, cyclization, and deprotection
04/14/2005US20050080067 Omega aminoalkylamides of R-2 aryl propionic acids as inhibitors of the chemotaxis of polymorphonucleate and mononucleate cells
04/14/2005CA2540826A1 Melanin concentrating hormone antagonists
04/14/2005CA2540638A1 Quinoxaline compounds
04/14/2005CA2540452A1 Benzylether and benzylamino beta-secretase inhibitors for the treatment of alzheimer's disease
04/13/2005EP1521748A1 Novel anthracene derivatives and the use thereof as a medicament
04/13/2005EP1521740A2 Probucol derivatives
04/13/2005EP1521733A1 Modulators of the glucocorticoid receptor
04/13/2005EP1077962B1 Isocyanate derivatizing agent and methods of production and use
04/13/2005CN1606548A Aryloxyphenyl and arylsulfanylphenyl piperazine derivatives
04/13/2005CN1606543A Alpha-cyanoacrylates
04/13/2005CN1196680C Modulators of dopamine neurotransmission
04/13/2005CN1196673C (-)-Verbenzone derivs.
04/12/2005US6878736 Histamine H3 receptor ligands
04/12/2005US6878732 5,7-diazaspiro(3.4)octane and -octene derivatives; treating diseases including emesis, depression, anxiety and cough
04/12/2005US6878724 Polyarylcarboxamides useful as lipid lowering agents
04/12/2005US6878712 E.g., (R)-((2S,5R)-2-methyl-5-methyl-4-(4-carboxyphenyl-sulphonyl)-1-(3,3,3 -trifluoro-2-hydroxy-2-methylpropionyl)-piperazine); antidiabetic agents
04/12/2005US6878707 Carboxamides useful as inhibitors of microsomal triglyceride transfer protein and of apolipoprotein b secretion
04/12/2005US6878706 N-(morpholinocarbonylmethyl)-N-isobutyl(benzylcarbonyl-N -cyanoamino)acetamide; treating rheumatoid arthritis, autoimmune diseases, osteoporosis, asthma, Alzheimer's disease, atherosclerosis and endometriosis.
04/12/2005US6878700 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
04/12/2005CA2203936C Boronic ester and acid compounds, synthesis and uses
04/12/2005CA2122571C Adhesion receptor antagonists
04/07/2005WO2005030188A2 Phenyl-piperazine derivatives as modulators of muscarinic receptors
04/07/2005WO2005030135A2 Nitrosated glutamic acid compounds, compositions and methods of use
04/07/2005WO2005019147A3 Pesticidally active phenol derivatives
04/07/2005WO2005014533A3 Aryl and heteroaryl compounds, compositions, and methods of use
04/07/2005WO2005007076A3 Colchicine derivatives
04/07/2005WO2005000845A3 Bicyclic derivatives as nk-1 and nk-2 antagonists
04/07/2005WO2004110364A9 Thiotungstate analogues and uses thereof
04/07/2005WO2003028728A8 4-(4-substituted piperazinyl-1yl)-butylcarboxamides as d3 dopamine subtype selective ligands
04/07/2005US20050075392 cyclopentyl substituted glutaramide derivatives; inhibitors of neutral endopeptidase which may be used to treat cardiovascular disorders, especially hypertension
04/07/2005US20050075381 a [4-(5-phenyl)oxazolyl]-N-acetyl pyrrolidine or a [1-amino-2-hydroxy-2-phenylethyl]-N-acetyl pyrrolidine; enzyme inhibitors; anticarcinogenic, antitumor agents
04/07/2005US20050075374 Sulfonyl aryl or heteroaryl hydroxamic acid compounds
04/07/2005US20050075368 Solvent extracting natural E2,E4-decadienal and undecadienal from ground, dried fruit of piper species; oxidation, esterification and transamidation; taste and aroma enhancers; bactercidel, fungicide and insecticidide activity
04/07/2005US20050075367 Ester compound and medicinal use thereof
04/07/2005US20050075344 Melanocortin receptor agonists
04/07/2005US20050075324 Melanin concentrating hormone antagonists
04/07/2005US20050074533 Conjugated dienamides, methods of production thereof, compositions containing same and uses thereof
04/07/2005CA2540186A1 Phenyl-piperazine derivatives as modulators of muscarinic receptors
04/07/2005CA2539973A1 Nitrosated glutamic acid compounds, compositions and methods of use
04/06/2005EP1520850A2 Conjugated dienamides, methods of production thereof, compositions containing same and uses thereof
04/06/2005EP1519932A1 Bisarylsulfonamide compounds and their use in cancer therapy
04/06/2005EP1519915A2 Tricyclic steroid hormone nuclear receptor modulators
04/06/2005CN1604890A 取代的环己烷衍生物 Substituted cyclohexane derivatives
04/06/2005CN1603291A Novel intermediates useful for the preparation of antihistaminic piperidine derivatives
04/06/2005CN1195738C 2'-substd. 1, 1'-biphenyl-2-carbonamides, method for production thereof, use thereof as medicament and pharmaceutical preparation contg. said compounds
04/06/2005CN1195737C HIV proteinase inhibitor
04/06/2005CN1195735C Sulfonylamino derivatives which inhibit matrix-degrading metallopr teinases
04/05/2005US6875831 Mono and multifunctional alkoxyamines for the preparation of functionalized macromers
04/05/2005US6875780 Compounds that modulate PPAR activity and methods for their preparation
04/05/2005US6875775 Triphenylalkene derivatives and their use as selective estrogen receptor modulators
04/05/2005US6875765 Inhibitors of interleukin-1 beta converting enzyme and other cysteine proteases in the ICE family
04/05/2005US6875764 Urea and thiourea compounds useful for treatment of coccidiosis
04/05/2005US6875760 Glucagon antagonists/inverse agonists
04/05/2005US6875759 Anticancer agents; analgesics
04/05/2005CA2245686C In situ block copolymer formation during polymerization of a vinyl aromatic monomer
03/2005
03/31/2005WO2005028459A1 Preparation method for quetiapine
03/31/2005WO2005028458A1 Preparation of quetiapine
03/31/2005WO2005028457A1 Preparation of quetiapine
03/31/2005WO2005028427A1 Aminoalkylamide substituted cyclohexyl derivatives
03/31/2005WO2005028426A1 Novel 4-phenylamino-benzaldoxime derivative and use thereof as mek inhibitor
03/31/2005WO2005028409A1 Alpha-hydroxy-benzeneacetic acid derivatives, and compounds having two 5-membered lactone rings fused to central cyclohexa-1,4-diene nucleus based upon the same, and uses of the compounds
03/31/2005WO2005019193A3 Phenylurea derivatives useful in the treatment of conditions mediated by polo-like kinases (plk)
03/31/2005WO2005005394A3 Thiophenylaminoimidazolines as prostaglandin i2 antagonists
03/31/2005WO2004113270A3 Propionic acid derivatives useful in the treatment of lipid disorders
03/31/2005WO2004098591A3 Inhibitors of glutaminyl cyclase and their use in the treatment of neurological diseases
03/31/2005US20050070719 Central nervous system disorders; antidiabetic agents; antiinflammatory agents; antiarthritic agents;obesity; osteoporosis ; anticancer agents
03/31/2005US20050070582 For example,1-{[2-(3,5-dimethylphenoxy)-5-nitrophenyl]sulfonyl}-4-ethylpiperazine or 1-{[2-(3,5-dichlorophenoxy)-5-nitrophenyl]sulfonyl}piperazine; for the treatment of asthma, atopic dermatitis, allergic rhinitis and other inflammatory/immunological disorders
03/31/2005US20050070559 Use of oxindole derivatives in the treatment of dementia related diseases, alzheimer's disease and conditions associated with glycogen synthase kinase-3
03/31/2005US20050070539 Such as 1-(4-{4-[2-(cyclopropylmethyl-amino)-5-nitro-benzoyl]-piperazin-1-yl}-3-fluoro- phenyl)-ethanone for treatment of psychoses, pain, neurodegenerative disfunction in memory and learning, schizophrenia, dementia, attention deficit disorders, or Alzheimer's disease
03/31/2005US20050070527 For leukocyte recruitment inhibition, treating or preventing inflammation and H4 receptor-mediated conditions
03/31/2005US20050070485 Phenylalanine derivatives
03/31/2005US20050069555 Vaccine adjuvants; hepatitis c virus; modulation immunology response
03/31/2005US20050066451 Para-phenylenediamine derivatives comprising a cyclic diaza group substituted with a cationic radical, and use of these derivatives for dyeing keratin fibers
03/31/2005CA2539159A1 Aminoalkylamide substituted cyclohexyl derivatives
03/31/2005CA2538866A1 Preparation of quetiapine
03/31/2005CA2538745A1 Preparation of quetiapine
03/30/2005EP1518553A2 Use of nitrate ester compounds for treating pain or providing analgesia
03/30/2005EP1517900A1 Process for the production of n-(2,6-dimethyl-phenyl)-2-piperazin-1-yl-acetamide
03/30/2005EP1517898A1 Arylcarbonylpiperazines and heteroarylcarbonylpiperazines and the use thereof for treating benign and malignant tumour diseases
03/30/2005EP1517882A1 Amide linker peroxisome proliferator activated receptor modulators
03/30/2005EP1517879A1 Aminoalkylphenols, methods of using and making the same
03/30/2005EP1360184B1 Piperidine derivatives as neurokinin 1 antagonists
03/30/2005EP1235831B1 New oxabispidine compounds useful in the treatment of cardiac arrhythmias
03/30/2005EP1192127B1 Substituted benzamide inhibitors of rhinovirus 3c protease
03/30/2005CN1602292A Unsaturated 1-amino-alkylcyclohexane NMDA, 5HT3 and neuronal nicotinic receptor antagonists
03/30/2005CN1602191A Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
03/29/2005US6872851 Melatonergic receptors; antiinflammatory agents; anticancer agents