Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
09/2004
09/30/2004US20040192681 N-acylsulfonamide apoptosis promoters
09/30/2004US20040192680 Novel amides that activate soluble guanylate cyclase
09/30/2004US20040192676 Ligands of melanocortin receptors and compositions and methods related thereto
09/30/2004US20040192657 9-Aminoacyl tetracycline compounds and methods of use thereof
09/30/2004CA2519582A1 Substituted p-diaminobenzene derivatives
09/30/2004CA2519440A1 Substituted piperidine and piperazine derivatives as melanocortin-4 receptor modulators
09/30/2004CA2519220A1 Amino cyclobutylamide modulators of chemokine receptor activity
09/29/2004EP1462445A1 Paraphenyldiamine derivatives concisting of a cyclic diaza group substituted by a cationic radical and use of these derivatives for dyeing keratin fibres
09/29/2004EP1462091A1 Composition for dyeing of keratinic fibers comprising a cationic derivative of p-phenylenediamine substituted by a diazacyclohexane or a diazacyloheptane
09/29/2004EP1461313A1 Human adam-10 inhibitors
09/29/2004EP1461311A2 Urea derivatives as vr1-antagonists
09/29/2004EP1461310A1 Bacterial enzyme inhibitors
09/29/2004EP1461306A1 Quaternary ammonium compounds and their use as antimuscarinic agents
09/29/2004EP1461038A1 Arylsulfonamide derivatives for use as ccr3 antagonists in the treatment of inflammatory and immunological disorders
09/29/2004EP1299350B1 Substituted benzamides for immune enhancement and for the treatment of cancer, infection and manic-depressive illness
09/29/2004EP1198462B1 Process for preparing a 10,11-methanodibenzosuberane derivative
09/29/2004EP1192189B1 Catalysts containing n-pyrrolyl substituted nitrogen donors
09/29/2004EP1169302B1 N-(2-phenyl-4-amino-butyl)-1-naphthamides as neurokinin-1 receptor antagonists
09/29/2004EP1100483B1 Glucocorticoid-selective anti-inflammatory agents
09/29/2004EP1051397A4 Method for preparing an n- (aliphatic or aromatic)carbonyl]-2-aminoacetamide compound and a cyclyzed compound
09/29/2004EP0993439B1 4-bromo or 4-iodo phenylamino benzhydroxamic acid derivatives and their use as mek inhibitors
09/29/2004CN1533382A 哌嗪衍生物 Piperazine derivatives
09/29/2004CN1533292A Medicament inhititing sodium/calcium exchange system
09/29/2004CN1168717C Novel intermediates for prepn. of antihisatminic piperidine derivatives
09/29/2004CN1168700C Cyclic amine substd. phenylalkanone and preparing method thereof
09/28/2004US6797820 Succinate compounds, compositions and methods of use and preparation
09/28/2004US6797713 1,4 substituted piperazines, 1,4 substituted piperidines, and 1-substituted,4-alkylidenyl piperidine compounds; dual acting molecules having both leukotriene inhibition properties
09/28/2004CA2299013C Neuropeptide y antagonists
09/28/2004CA2224125C Pharmaceutical composition comprising a proteinase inhibitor and a monoglyceride
09/23/2004WO2004081643A1 Lenslet array with polarization conversion
09/23/2004WO2004080986A1 Phenyl sulfone derivatives and their use in the treatment of cns disorders
09/23/2004WO2004080974A1 A purification method of ionic liquids to obtain their high purity
09/23/2004WO2004080947A1 Imino ether derivative compounds and drugs containing the compounds as the active ingredient
09/23/2004WO2004080391A2 Novel antibacterial agents
09/23/2004WO2004050613A3 2-substituted-3-propenamide derivatives and methods of using the same
09/23/2004WO2003082268A3 Hemiasterlin derivatives and uses thereof in the treatment of cancer
09/23/2004US20040186294 Method for producing biperiden iv
09/23/2004US20040186148 E.g., 1-(pyrid-2-yl-so2-),2-((4-(isopropylphenyl)-so2-),5-(isopropoxy)benzene; antiinflammatory agents; immunomodulatory activity rheumatoid arthritis, asthma, allergy, psoriasis, Crohn's disease, systemic lupus erythematosus, multiple sclerosis, diabetes, cancer, glaucoma, osteoporosis, renal ischemia
09/23/2004US20040186146 E.g., R-N-2-[4-(pyrrolidin-1'-yl)methylphenyl]propionyl-methanesulfonamide; inhibition of chemotaxis of neutrophils induced by interleukin-8; antiinflammatory agents; psoriasis, ulcerative cholitis, glomerular nephritis, acute respiratory insufficiency, idiopathic fibrosis, and rheumatoid arthritis
09/23/2004US20040186145 Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them
09/23/2004US20040186136 E.g., mono-, poly- or perdeuteriated tolperisone and eperisone; appreciably better pharmacokinetic and/or pharmacodynamic properties than the undeuterated compounds; muscular disorders; muscle relaxants (skeletal); antispasmodic agents; vasodilation
09/23/2004US20040186112 Polymorphic forms of dihydrochloride salts of cetirizine and processes for preparation thereof
09/23/2004US20040186104 Novel pyridinone and related heterocyclic derivatives
09/23/2004US20040186080 Beta 2-adrenergic receptor agonists
09/23/2004US20040186061 Novel derivatives of 3,3-diphenylpropylamines
09/23/2004CA2801100A1 Novel antibacterial agents
09/23/2004CA2518986A1 Imino ether derivative compounds and drugs containing the compounds as the active ingredient
09/22/2004EP1458689A1 Aryloxyphenyl and arylsulfanylphenyl derivatives
09/22/2004EP1458684A2 Therapeutic heterocycles
09/22/2004EP1458676A2 Compounds for the treatment of inflammatory disorders
09/22/2004EP1458675A1 Alpha-cyanoacrylates
09/22/2004EP1458394A1 Use of oxindole derivatives in the treatment of dementia related diseases, alzheimer s disease and conditions associated with glycogen synthase kinase-3
09/22/2004EP1458375A2 Compositions for decreasing activity of hormone-sensitive lipase
09/22/2004EP1458374A2 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
09/22/2004EP1100503B1 Non-imidazole alkylamines as histamine h 3?-receptor ligands and their therapeutic applications
09/22/2004EP0706524B1 Processes and intermediates for the preparation of 5- 2-(4-(benzoisothiazol-3-yl)-piperazin-1-yl)ethyl]-6-chloro-1,3-dihydro-indol-2-one
09/22/2004CN1531531A Novel arylsusfonamide compounds for treatment of obesity, type II diabetes and CNS-disorders
09/22/2004CN1531520A Self-reducing anthraquinone compounds
09/22/2004CN1531459A Method for hydrogenating organic compounds by means of RU/SIO2 catalysts
09/22/2004CN1531425A Urea derivatives as integrin alpha 4 antagonists
09/22/2004CN1167701C Method for preparing oxazolidone amine
09/22/2004CN1167694C 1-phenyl-4-(1-[2-aryl]cyclopropyl) methylpiperazines: dopamine receptor ligands
09/22/2004CN1167673C Fluorovinyloxyacetamides, process for preparing the same and herbicidal composition comprising the same
09/21/2004US6794545 Conformationally restricted polyamine analogs as disease therapies
09/21/2004US6794511 An enzyme inhibitors of metalloprotease; treating connective tissue degradation caused by inflammation or tumor
09/21/2004US6794507 Compounds that inhibit factor Xa activity
09/21/2004US6794400 4-substituted-1-(arylmethylidene)thiosemicarbazide, 4-substituted-1-(arylcarbonyl)thiosemicarbazide and analogs as activators of caspases and inducers of apoptosis and the use thereof
09/21/2004US6794392 Cell differentiation inducer
09/21/2004US6794372 Nitrate salts of antimicrobial agents
09/16/2004WO2004071445A3 2-(aminomethyl)arylamide analgesics
09/16/2004WO2004069782A3 2-aryl-acetic acids, their derivatives and pharmaceutical compositions containing them
09/16/2004WO2003096989A3 Anti tubercular drug: compositions and methods
09/16/2004US20040181057 Aminothiol compound
09/16/2004US20040180964 anti-obestic activity; Neuropeptide Y antagonist
09/16/2004US20040180944 Pyrazolopyrimidinones which inhibit type 5 cyclic guanosine 3',5'-monophosphate phosphodiesterase (cGMP-PDE5) for the treatment of sexual dysfunction
09/16/2004US20040180906 Anti-inflammatory medicaments
09/16/2004US20040180894 Benzamide inhibitors of the P2X7 receptor
09/16/2004US20040180892 control of cardiovascular homeostasis is achieved through a combination of both direct neuronal control and systemic neurohormonal activation
09/16/2004US20040180876 Selective beta 2-adrenoreceptor agonists; rapid onset of action, long duration; such as 3-(4-{[6-{(-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)benzenesulfonamide; synthesis
09/16/2004US20040180871 Anti-inflammatory compositions and methods
09/16/2004US20040180863 Novel, nitric oxide-releasing amidine- and enamine-derived diazeniumdiolates, compositions and uses thereof and method of making same
09/15/2004EP1456171A1 Substituted cyclohexane derivatives
09/15/2004EP1456151A1 Method for forming a carbon-carbon or carbon-heteroatom linkage
09/15/2004EP1455777A1 Glyt1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders
09/15/2004EP1077925B1 Compounds having reversible inhibiting activity of carnitine palmitoyl-transferase
09/15/2004EP0986384A4 Inhibitors of protein isoprenyl transferases
09/15/2004EP0775689B9 Novel amine derivative, process for producing the same, and use thereof as antiarrhythmic
09/15/2004CN1529699A Novel sulfonic acid derivatives
09/15/2004CN1529691A N-Benzyl-M-Phenylenedimine derivatives and dyes containing said compounds
09/15/2004CN1529599A Acylic piperazine and piperidine derivatives which are used for treating neuronal damage
09/15/2004CN1528742A Compound for treating asthma, irritability an a inflammation and its intermediate
09/15/2004CN1166654C Benzoylguanidine derivatives wit advantageous properties, method for producing them and their use in production of medicaments
09/15/2004CN1166653C Process for producing benzylamine compound
09/15/2004CN1166652C Preparation method of carbonyl aplpha-substitution nitrogenous compound
09/15/2004CN1166646C Process for synthesis of azacyclic compounds
09/15/2004CN1166643C 4-phenyl-pyrimidine derivatives
09/15/2004CN1166633C New alpha-amino acid sulfuryl compounds, its preparing method and medicinal composition containing them
09/15/2004CN1166629C Benzene sulfonamide compounds, its preparing method and medicinal compsns. contg. same
09/15/2004CN1166610C Diglycol material for preparing morpholine
09/14/2004US6790996 Hydrogenating nitriles in the presence of a supported cobalt containing catalyst to form primary amines