Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
06/2005
06/15/2005EP1539677A2 Succinic acid semi-amides as anti-corrosives agents
06/15/2005EP1539676A1 Monomer compound comprising several cationic groups, process for making the same, and polymers comprising units deriving therefrom
06/15/2005EP1539662A1 Cannabinoid receptor ligands
06/15/2005EP1539134A2 Nitrosated and/or nitrosylated cyclooxygenase-2 selective inhibitors, compositions and methods of use
06/15/2005EP1278740B1 Hydroxyphenyl-piperazinyl-methyl-benzamide derivatives for the treatment of pain
06/15/2005EP1256576B1 Fused imidazolium derivatives
06/15/2005EP1064252B1 Oxidation dyeing compositions containing a cationic coupling agent, novel cationic coupling agents
06/15/2005EP0956031B1 Inhibition of 26 s and 20 s proteasome by indanones
06/15/2005CN1628109A Novel aryl- and heteroarylpiperazines
06/15/2005CN1628107A Heteroaryl alkyl piperazine derivatives as fatty acid oxidation inhibitors
06/15/2005CN1627946A Carboximide derivatives as useful uro-selective alpha-1A adrenoceptor blockers
06/15/2005CN1626516A Novel intermediate for prepn. of pyrazolopyrimidinones
06/15/2005CN1206213C N-arylsulfonyl amino acid omega amides
06/14/2005US6906203 Anticancer agents; such as 2-Amino-3-cyano-4-(2-bromo-4,5-dimethoxyphenyl)-4H-indolo(4,5-b)pyran
06/14/2005US6906202 Purified racemic lasofoxifene and purified lasofoxifene D-tartrate and a method for effective purification of racemic lasofoxifene
06/14/2005US6906094 1,2,4-tribsubstituted benzenes as inhibitors of 15-lipoxygenase
06/14/2005US6906073 Piperazine CCR-3 receptor antagonists
06/14/2005US6906072 Central nervous system disorders
06/14/2005CA2155952C Novel process for trans-6-[2-(substituted-pyrrol-1-yl)alkyl]pyran-2-one inhibitors of cholesterol synthesis
06/09/2005WO2005051933A1 An improved process for the synthesis of 4-(4-benzyloxy-carbonylamino-2-fluorophenyl)-piperazine-1-carboxylic acid tert-butyl ester, a key intermediate for oxazolidinone antimicrobials and compounds prepared thereby
06/09/2005WO2005051914A1 Benzylether and benzylamino beta-secretase inhibitors for the treatment of alzheimer's disease
06/09/2005WO2005051895A1 Organic compounds
06/09/2005WO2005051892A1 Novel phenoxyacetamide derivatives and use thereof for the preparation of diphenylamines
06/09/2005WO2005051890A1 Aminophenylcyclopropyl carboxylic acids and derivatives as agonists to gpr40
06/09/2005WO2005051373A1 Receptor function regulating agent
06/09/2005WO2005040142A9 Novel keto-oxadiazole derivatives as cathepsin inhibitors
06/09/2005WO2004052845A8 Tetrahydro-naphthalene derivatives as vanilloid receptor antagonists
06/09/2005US20050124682 Such as N-{2-[5-(methylthio)-1H-indol-3-yl]ethyl}acetamide for treatment of disorders of the melatoninergic system; hormone replacement therapy
06/09/2005US20050124679 Alpha, beta-unsaturated hydroxamic acid derivatives and their use as histone deacetylase inhibitors
06/09/2005US20050124654 Compounds and methods of use
06/09/2005US20050124632 Use of aminobenzenesulfonic acid derivative or a salt, hydrate, or solvate thereof; treatment of heart failure or arrhythmia in diabetic ischemic heart disease
06/09/2005US20050124001 Method of producing highly functionalized 1,3-diamino-propan-2-ols from solid support
06/09/2005DE10353910A1 Verfahren zur Synthese optisch aktiver Piperidine Process for the synthesis of optically active piperidines
06/09/2005CA2547430A1 Receptor function regulating agent
06/09/2005CA2547281A1 Novel phenoxyacetamide derivatives and use thereof for the preparation of diphenylamines
06/09/2005CA2546142A1 Benzylether and benzylamino beta-secretase inhibitors for the treatment of alzheimer's disease
06/08/2005EP1538150A1 Novel pleuromutilin derivatives
06/08/2005EP1537075A2 Diarylurea derivatives and their use as chloride channel blockers
06/08/2005EP1537074A1 Cathepsin cysteine protease inhibitors
06/08/2005EP1370528B1 Mch antagonists and their use in the treatment of obesity
06/08/2005EP1252133B1 Pharmaceutical compounds
06/08/2005EP1042305B1 INHIBITION OF p38 KINASE USING SYMMETRICAL AND UNSYMMETRICAL DIPHENYL UREAS
06/08/2005EP0849256B1 Amide compounds and use of the same
06/08/2005CN1625553A Treatment of male sexual dysfunction
06/08/2005CN1625548A Purified LASOFOXIFENE and a method for purification of racemic LASOFOXIFENE by recrystallization
06/08/2005CN1623988A Biaryl sulfonamides and methods for using same
06/08/2005CN1205185C Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
06/08/2005CN1205180C 3-(2,5-diaminophenyl)-acrylamide derivatives and colouring agents containing said compounds
06/08/2005CN1205179C (P-amino-hydroxyphenyl)-acrylamide derivatives and dyes containing said compounds
06/08/2005CN1205177C Process for producing depsipeptide derivs, and noval intermidiates therefor
06/07/2005US6903120 Modulators of dopamine neurotransmission
06/07/2005US6903115 Bipiperidine compounds
06/07/2005US6903114 Carbocyclic alcohols such as 1,6-dinitronaphthalene-2,3-diol, used as catechol-O-methyltransferase inhibitors, for prophylaxis of Parkinson's disease
06/07/2005US6903102 17β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
06/07/2005US6903092 Naphthamide neurokinin antagonists for use as medicaments
06/07/2005US6903088 Compounds which inhibit leukocyte adhesion mediated by VLA-4
06/02/2005WO2005049604A2 Antithrombotic aromatic ethers
06/02/2005WO2005049594A1 N-acylsulfonamide apoptosis promoters
06/02/2005WO2005049593A2 N-acylsulfonamide apoptosis promoters
06/02/2005WO2005049589A2 Heterocyclic compounds for the treatment of hyperlipidemia, diabetes, obesity and similar diseases
06/02/2005WO2005049570A1 Method for synthesising optically active piperidines by the hydrogenation of optically active pyridines
06/02/2005WO2005049561A2 Processes for preparing novel methylene blue derivative
06/02/2005WO2005049023A1 Glyt1 transporter inhibitors
06/02/2005WO2005049009A1 Methods and agents for inhibiting dynamin-dependent endocytosis
06/02/2005WO2005048810A2 Sigma-2 receptor radiotracers for imaging the proliferative status of solid tumors
06/02/2005WO2004063150A3 Diagnostic and therapeutic alkyl piperidine/piperazine compounds and process
06/02/2005US20050119502 (Dialkylamino, morpholino, or imidazolyl)-alkoxyphenolic derivatives as drug delivery agents; improved bioavailability for oral administration
06/02/2005US20050119315 Cardiovascular disorders; antiarrhythmia agents; sodium channel moderators; potassium channel moderators; prevention fibrillation
06/02/2005US20050119306 Blocking transcription factor; culture product of transgenic fungi
06/02/2005US20050119275 Antiinflammatory agents; autoimmune disease; Alzheimer's disease; anticancer agents; antiarthritic agents; antidiabetic agents; lupus; interinflammatory agents
06/02/2005US20050119252 Ligands of melanocortin receptors and compositions and methods related thereto
06/02/2005US20050119250 Amino-derivatives as novel inhibitors of histone deacetylase
06/02/2005US20050119245 Alpha -, beta -, and gamma -amino acid derivatives, e.g., S)-2-{N'-[4-(4-Fluoro-phenoxy)-phenyl]-N''-cyano-guanidino}-3-phenyl-N-(3-pyrrolidin-1-yl-propyl)-propionamide for the treatment of central nervous system conditions such as muscle spasticity, tinnitus, epilepsy and neuropathic pain.
06/02/2005US20050119225 Phosphodiesterase 4 inhibitors, including N-substituted aniline and diphenylamine analogs
06/02/2005CA2556801A1 Methods and agents for inhibiting dynamin-dependent endocytosis
06/01/2005EP1534693A2 1, 3-diamino-2-hydroxypropane prodrug derivatives
06/01/2005EP1534689A1 Novel carboxamide compounds having an mch-antagonistic effect, medicaments containing said compounds, and methods for the production thereof
06/01/2005EP1534283A1 Formulation of liposomal derivatives of phenylalanine
06/01/2005EP1440118B1 Blends of waxes and polymer additives
06/01/2005EP1351959B1 Novel pleuromutilin derivatives
06/01/2005EP1115695B1 (r)-chiral halogenated 1-substitutedamino-(n+1)-alkanols useful for inhibiting cholesteryl ester transfer protein activity
06/01/2005EP1095015B1 Sulfonylamino carboxylic acid n-arylamides as guanylate cyclase activators
06/01/2005EP1049679B1 Sulphonamide derivatives for treatment of cns disorders
06/01/2005EP0994862B1 Sulphonamide derivatives being 5-ht6 receptor antagonists and process for their preparation
06/01/2005EP0993441B1 INHIBITORS OF p38
06/01/2005CN1622942A HIV protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
06/01/2005CN1622941A Glutaminyl based DPIV inhibitors
06/01/2005CN1204135C 1, 3-dioxolanes with antitussive activity
06/01/2005CN1204121C 1, 4-substituted cyclic amine derivatives or dihydro indole derivatives and medicines containing same
06/01/2005CN1203898C Perfluoroalkyl-containing metal complexes, its preparing method and use in NMR diagnostics
05/2005
05/31/2005US6900350 In aqueous solution; from secondary amine, dihaloalkane and alkali metal sulfite
05/31/2005US6900345 Antibiotics; mutilin 14-[N-(2-carbamoyloxyethoxycarbonyl)]carbamate; therapy for bacteria infections; chemical synthesis
05/31/2005US6900329 MCH antagonists and their use in the treatment of obesity
05/31/2005US6900244 Controlling lipid, cholesterol metabolism; anticholesterol agents
05/31/2005US6900237 Sulfonamide compounds as protease inhibitors
05/31/2005US6900218 Reducing oxidation stresses; central nervous system disorders; antiinflammatory agents
05/31/2005US6899830 Method for producing Grignard compounds
05/26/2005WO2005047899A2 Use of the lipoxin receptor, fprl1, as a tool for identifying compounds effective in the treatment of pain and inflammation
05/26/2005WO2005047249A1 Benzylether amine compounds useful as ccr-5 antagonists
05/26/2005WO2005047230A1 Bis-cationic compounds and use thereof