Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
08/2005
08/25/2005US20050187198 Methods of preparing substituted tetracyclines with transition metal-based chemistries
08/25/2005US20050186176 Compounds and compositions for delivering active agents
08/25/2005CA2555884A1 Amino-substituted tricyclic derivatives and methods of use
08/24/2005EP1565422A1 Vitamin d receptor modulators
08/24/2005EP1565192A2 Method and compositions for temporarily incapaciting subjets
08/24/2005EP1565190A2 Arylcyclopropylcarboxylic amides as potassium channel openers
08/24/2005EP1565185A2 Neuroprotective iron chelators and pharmaceutical compositions comprising them
08/24/2005EP1565178A2 Method and compositions for treating persistent pulmonary hypertension using aralkyl ester soft drugs
08/24/2005EP1334085B1 Sulfamides as gamma-secretase inhibitors
08/24/2005EP1299349B1 Compounds to treat alzheimer's disease
08/24/2005EP1284722B1 Compositions containing a benzamide disulfide derivative for treating allergic diseases
08/24/2005EP1218341B1 Sulfonyl carboxamide derivatives, method for their production and their use as medicaments
08/24/2005EP1019075B1 Beta 2-adrenergic receptor agonists
08/24/2005CN1659157A Terphenyl derivatives, preparation thereof, compositions containing same
08/24/2005CN1659156A Novel guanidinobenzamides
08/24/2005CN1659155A 1-phenylalkyl-piperazines
08/24/2005CN1659134A Monomer compound comprising several cationic groups, process for making the same, and polymers comprising units deriving therefrom
08/24/2005CN1659131A (2-((2-alkoxy) -phenyl) -cyclopent-1-enyl) aromatic carbo and heterocyclic acid and derivatives
08/24/2005CN1658879A Neurotrophic factor production accelerator
08/24/2005CN1658872A Antiallergic
08/24/2005CN1658855A O-substituted hydroxyaryl derivatives
08/24/2005CN1216056C Sulfamato hydroxamic acid metalloprotease inhibitor
08/24/2005CN1216053C 2,2-disubstituted 1,3-dioxolanes as antitussive atents
08/24/2005CN1215834C Emulsion of perfluororganic compounds for medical purposes, method for producing said emulsion and methods for curing and preventing diseases with the aid of the emulsion
08/23/2005US6933393 Reacting methyl cyanoacetate with morphiline to form 3-morpholin-4-yl-3-oxo- propionitrile; forming salt; reacting with phenylacetic acid and 2-(2-(4-fluorophenyl)-2-oxo-1-phenyl-ethyl)-4-
08/23/2005US6933390 Process for the arylation of aza-heterocycles with activated aromatics in presence of caesium carbonate
08/23/2005US6933321 For therapy of androgen-dependent diseases such as prostate cancer, benign prostatic hyperplasia, precicious puberty, polycystic ovarian syndrome, acne, hirsutism, seborrhea, androgenic alopecia and premature male baldness
08/23/2005US6933319 Resorcinol derivatives
08/23/2005CA2469592C Hiv integrase inhibitors
08/23/2005CA2266884C Inhibition of 26s and 20s proteasome by indanones
08/23/2005CA2089442C Amino-substituted benzoylguanidines, process for their preparation, their use as a medicament and medicament containing them
08/18/2005WO2005075410A1 New compounds, methods for their preparation and use thereof
08/18/2005WO2005074919A1 Diurea derivatives
08/18/2005WO2004110387A3 Sigma ligands for neuronal regeneration and functional recovery
08/18/2005WO2003101931A3 Preparation of 4-(n, n-disubstitutedamino) butyraldehyde acetals
08/18/2005US20050182070 Method for the treatment of allergic conditions
08/18/2005US20050182069 For treatment of asthma, allergies, inflammation and anxiety; antihistamines; sedatives; tranquilizing agents; 2[2-[4-[(4-chlorophenyl)phenylmethyl]-1-piperazinyl]ethoxy]acetamide
08/18/2005US20050182068 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
08/18/2005US20050182057 Aryl N-cyanoguanidines and methods related thereto
08/18/2005US20050182040 Benzamide derivatives
08/18/2005US20050181034 3-Amidino- or 3-guanidino phenylalanine derivative which is effective as urokinase inhibitor; antitumor, anticarcinogenic, and antimetastasis agents
08/18/2005CA2552942A1 New compounds, methods for their preparation and use thereof
08/18/2005CA2551566A1 Diurea derivatives
08/17/2005EP1562925A1 Phenylalanine derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
08/17/2005EP1562924A1 4(phenyl-piperazinyl-methyl) benzamide derivatives and their use for the treatment of pain or gastrointestinal disorders
08/17/2005EP1562923A1 4(phenyl-piperazinyl-methyl) benzamide derivatives and their use for the treatment of pain or gastrointestinal disorders
08/17/2005EP1562922A1 4(phenyl-piperazinyl-methyl) benzamide derivatives and their use for the treatment of pain or gastrointestinal disorders
08/17/2005EP1562895A1 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication
08/17/2005EP1140841B1 3-phenyl-2,6-dioxopiperidin-3-yl propionamide derivatives and method for preparing same
08/17/2005CN1654461A Process for preparing bis-phenyl fluorozine and its use as medicine in treatment of cardiovascular and cerebrovascular diseases
08/17/2005CN1215055C Arylsulfonamido-substituted hydroxamic acid derivatives
08/16/2005US6930189 Chiral ligand
08/16/2005US6930185 Anorectic agents; obesity; such as 4'-chloro-N-(6-((N,N-dimethylamino)methyl)-2-naphthyl)(1,1'-biphenyl)-4 -carbox-amide
08/16/2005US6930106 Inhibitors of HCV NS5B polymerase
08/16/2005CA2280985C Compound containing urea and use of the compound in the field of cosmetics and/or dermatology
08/16/2005CA2166059C Novel intermediates for the preparation of antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives
08/11/2005WO2005073208A1 Piperazino sensitisers
08/11/2005WO2005073207A1 Process for preparing optically active cetirizine or its salt
08/11/2005WO2005073206A1 Selective estrogen receptor modulators
08/11/2005WO2005073205A1 Selective estrogen receptor modulators
08/11/2005WO2005073204A1 Selective estrogen receptor modulators for the treatment of vasomotor symptoms
08/11/2005WO2005073190A1 Selective estrogen receptor modulators
08/11/2005WO2005056510A3 Novel ligands that are activators of the rar receptors, use in human medicine and in cosmetics
08/11/2005WO2005051914A8 Benzylether and benzylamino beta-secretase inhibitors for the treatment of alzheimer's disease
08/11/2005WO2005020897A3 Compositions and methods for the treatment of disease associated with trp-p8 expression
08/11/2005US20050176987 Method for producing vinyl, aryl and heteroaryl acetic acids and derivatives thereof
08/11/2005US20050176963 Reacting 1-(bicyclo(2.2.1)hept-5-en-2-yl)-3-piperidine-1-propanone withdiphenylmagnesium
08/11/2005US20050176962 Aminating a -cyanophenylalanine derivative with hydroxylamine hydrochloride in the presence of sodium carbonate in alcoholic-aqueous solution at reflux temperature to a 3-amidino derivative; chemical intermediates as highly efficient urokinase inhibitors
08/11/2005US20050176821 Meta-substituted phenylene sulphonamide derivatives
08/11/2005US20050176820 Oxygenated esters of 4-iodo phenylamino benzhydroxamic acids
08/11/2005US20050176766 2,3-Oxidosqualene-lanosterol cyclase inhibitors
08/11/2005US20050176764 Medicine for treating cancer
08/11/2005US20050176732 Enantiomers of 1-(4-chlorophenyl)phenylmethyl]-4-[(4-methylphenyl)sulfonyl]piperazine
08/11/2005US20050176731 N-[5-({(2S)-3-[(4-{4-[(4-benzylpiperidin-1-yl)carbonyl]phenyl}cyclohexyl)amino]-2-hydroxypropyl}oxy)-2-hydroxyphenyl]methanesulfonamide; beta 3 receptors agonist; gastrointestinal diseases; antiobesity, antidiabetic, cicatrizing agents, tocolytics, dysmenorrhea, antiglaucomatous; amidation
08/11/2005US20050176727 Male erectile dysfunction; 1-(3-chlorophenyl)-3-(4-pyridin-2-yl-piperazin-1-yl)propan-1-one O-methyloxime
08/11/2005US20050173683 Materials, methods, and uses for photochemical generation of acids and/or radical species
08/11/2005DE19728335B4 Piperazin-Derivate und diese enthaltenden Oxidationsfärbemittel sowie deren Verwendung Piperazine derivatives and containing oxidation dyes and their use
08/10/2005EP1561744A2 Amine derivatives, process for producing the same and their use as antimycotic agent
08/10/2005EP1560810A1 Bifunctional phenyliso(thio)cyanates; method and intermediate products for the production thereof
08/10/2005EP1560574A2 Antileishmanial dinitroaniline sulfonamides with activity against parasite tubulin
08/10/2005EP1395265A4 Combretastatin a-3 prodrug
08/10/2005EP1333795A4 Novel coupler for use in oxidative hair dyeing
08/10/2005EP1157002B1 1,2,3,4-tetrahydro-1-naphthalenamine compounds useful in therapy
08/10/2005CN1653043A Method for the production of sulphamic acid halogenides
08/10/2005CN1653042A Aminoalcohol derivatives as beta-3 adrenergic receptor agonists
08/10/2005CN1653037A Substituted tetracycline compounds
08/10/2005CN1653033A Method of purifying quaternary alkylammonium salt and quaternary alkylammonium salt
08/10/2005CN1653025A NK1 antagonists
08/10/2005CN1652788A Method of treating diabetes
08/10/2005CN1652779A Treatment of chemokine mediated diseases
08/10/2005CN1652761A Preventive or therapeutic agent for kidney disease
08/10/2005CN1652759A Small molecule entry inhibitors
08/09/2005US6927224 Anticancer agents; osteoporosis
08/09/2005US6927222 Compounds
08/09/2005US6927218 Aryl N-cyanoguanidines and methods related thereto
08/09/2005CA2310627C Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance p antagonists
08/09/2005CA2258217C Substituted cyclopentane compounds useful as neuraminidase inhibitors
08/04/2005WO2005070921A1 Polyethylene glycol conjugates of heterocycloalkyl carboxamido propanoic acids
08/04/2005WO2005070910A2 Derivatives of 1-piperazine- and 1-homopiperazine-carboxylates, preparation method thereof and use of same as inhibitors of the faah enzyme
08/04/2005WO2005070909A1 An improved process for the preparation of gefitinib