Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
01/2005
01/05/2005CN1183098C 3-amino-3-aryl-1-alcohol derivatives and preparation and use thereof
01/04/2005US6838584 Estrogen receptor modulators
01/04/2005US6838565 Factor x inhibitor; anticoagulants
01/04/2005US6838561 2-substituted-4-amino-phenol derivative compounds providing good oxidative coloration of hair and acceptable light fastness, fastness to shampooing and permanent wave treatment
01/04/2005US6838470 Antiischemic agents; brain disorders; cardiovascular disorders
01/04/2005US6838466 Compounds for the treatment of inflammatory disorders
01/04/2005US6838461 Psychological disorders; schizophrenia; Alzheimer's disease; Parkinson's disease; Huntington's disease; cardiovascular disorders; hypotensive agents; side effect reduction
01/04/2005US6838460 Substituted phenylamidines medicaments containing said compounds and method for production thereof
01/04/2005CA2148827C Novel 3,3-diphenylpropylamines, their use and preparation
01/04/2005CA2147155C Amide derivatives
12/2004
12/30/2004US20040266870 Inhibitors of the chemotactic activation induced by the fraction C5a of complement and from other chemotactic proteins (chemokines) that y activate a 7-transmembrane-domain receptor; psoriasis, rheumatoid arthritis, ulcerative colitis, acute respiratory distress syndrome, fibrosis; antiischemic agents
12/30/2004US20040266855 Effective against Src family; cancer, osteoporosis
12/30/2004US20040266787 Novel amorphous form of [2-[4-[(4-chlorophenyl)-phenyl methyl]-1-piperazinyl]ethoxy]acetic acid and process for the preparation thereof
12/30/2004US20040266786 1-(2 chlorophenyl-1-piperazinyl)-2-propanol-3-oxy-(2-methoxy-propenyl)-benzene; alpha 2-adrenergic/5-HT2A antagonist, 5-HT re-uptake inhibition, and anti-oxidant activities
12/30/2004US20040266785 KMST isoeugenol derivatives and pharmaceutical activity
12/30/2004US20040266784 Calcium channel inhibitors comprising benzhydril spaced from piperazine
12/30/2004US20040266782 Cyclic amine derivatives-CCR-3 receptor antagonists
12/29/2004WO2004113391A2 Improved pharmaceutical drug candidates and methods for preparation thereof
12/29/2004WO2004113312A1 Hydroxamate sulfonamides as cd23 shedding inhibitors
12/29/2004WO2004113311A1 Amorphous und crystal forms of (5-chloro-2-{2-
12/29/2004WO2004113277A2 Methods and compositions for treating amyloid-related diseases
12/29/2004WO2004113275A2 Methods and compositions for treating amyloid-related diseases
12/29/2004WO2004113270A2 Propionic acid derivatives useful in the treatment of lipid disorders
12/29/2004WO2004112787A1 Glyt1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders
12/29/2004WO2004086050A3 Labelling agents for mass spectrometry comprising tertiary amines
12/29/2004WO2004002940A8 Inhibitors of hcv ns5b polymerase
12/29/2004WO2002043648A3 Compounds active at the glucocorticoid receptor ii
12/29/2004EP1491187A1 Preventive or therapeutic agent for kidney disease
12/29/2004EP1490346A2 Stereoselective alkylation of chiral 2-methyl-4-protected piperazines
12/29/2004EP1490338A1 Use of an alfa2-adrenoreceptor antagonist for cns-related diseases
12/29/2004EP1490054A2 Hemiasterlin derivatives and uses thereof in the treatment of cancer
12/29/2004EP1265891B1 Novel lipoic acid heterocyclic or benzene derivatives, preparation and use thereof as medicines
12/29/2004EP1171419B1 Biphenyl derivatives as antagonists of the neurokinine-1 receptor
12/29/2004EP1163209A4 Compounds and compositions for delivering active agents
12/29/2004EP1102538B1 Plant growth regulator compositions
12/29/2004CN1557811A Phenoxy indenone compounds ,process for preparing same and use thereof
12/29/2004CN1182109C ((Aminoiminomethyl) amino) alkanecarboxamides and their applications in therapy
12/29/2004CN1181817C NF-KB inhibitors containing phenylmethyl benzoquinone as active ingredient
12/29/2004CA2529257A1 Methods and compositions for treating amyloid-related diseases
12/29/2004CA2529256A1 Methods and compositions for treating amyloid-related diseases
12/29/2004CA2528538A1 Dual function compounds and uses thereof
12/29/2004CA2528317A1 Hydroxamate sulfonamides as cd23 shedding inhibitors
12/29/2004CA2528234A1 Propionic acid derivatives useful in the treatment of lipid disorders
12/28/2004US6835839 Method for the production of biperiden II
12/28/2004US6835832 Catalytic hydrogenation
12/28/2004US6835831 Efficient synthesis of ceramide-like compounds by reacting an aldehyde and an amidomethylisonitrile to form a 4-amido-2-oxazoline; suppress biosynthesis of glycosphingolipids; antitumor agents; Tays-Sach, Gaucher's
12/28/2004US6835734 1,3-dioxolanes with antitussive activity
12/23/2004WO2004111025A1 Para-substituted phenyl carbamates as inhibitors of hormone sensitive lipase
12/23/2004WO2004110989A1 N-hydroxy-7-(arylamino)heptanamide derivatives useful for treating hyper-proliferative disorders
12/23/2004WO2004110986A1 Benzamide derivative or salt thereof
12/23/2004WO2004110978A2 1-aminonaphthalenes as modulators of androgen, glucocorticoid, mineralocorticoid and progesterone receptors
12/23/2004WO2004110418A2 Carbonyl compounds as inhibitors of histone deacetylase for the treatment of disease
12/23/2004WO2004110389A2 Sigma ligands for neuronal regeneration and functional recovery
12/23/2004WO2004110388A2 Sigma ligands for neuronal regeneration and functional recovery
12/23/2004WO2004110387A2 Sigma ligands for neuronal regeneration and functional recovery
12/23/2004WO2004110364A2 Thiotungstate analogues and uses thereof
12/23/2004WO2004099150A3 3-(1-naphthyl)-2-cyanopropanoic acid derivatives as estrogen receptor ligands
12/23/2004WO2003104211A3 Crystalline [2-[4-[(4-chlorophenyl)-phenyl methyl]-1-piperazinyl] ethoxy] acetic acid dihydrochloride
12/23/2004US20040260100 Sulfonylation of N-protected prolinol, hydrogenation with an alkali triethylboron hydride; N-protected-2-iodomethylpyrrolidine is formed by reacting the sulfonate with an alkali iodide salt; histamine-3 receptor modulator precursors
12/23/2004US20040260099 D-t-3',4'-ethylenedioxy-p4 derivatives; glucosyl ceramide inhibitors lower glycosphingolipid levels; anticarcinogenic, antitumor agents; angiogenesis inhibitors; tumor antigens
12/23/2004US20040260089 reacting diphosphorus pentoxide, an organic base (melamine, guanidine, piperazine), and a water releasing agent (borax, aluminum or magnesium hydroxide, or oxalic or formic acid) to form polyphosphate salts; fire retardants for thermoplastic polyamide or polyester platics
12/23/2004US20040259912 N-(4-benzhydryloxy-3-isobutyrylphenyl)-N'-(3,4-dimethoxyphenyl)urea for example; vanilloid receptor agonists; use as analgesic and or for treating urinary frequency and/or urinary incontinence
12/23/2004US20040259875 Incontinence; overactive bladder; neuropathic pain; neuralgia; analgesics; stroke; antiarthritic agents; antiinflammatory agents
12/23/2004US20040259866 Calcium channel blockers comprising two benzhydril moieties
12/23/2004US20040259861 Antiischemic agents
12/23/2004US20040259840 Using phosphoglycerides, lipid having sphingosine base, glycerides and sterol; wound healing agents; atherosclerosis
12/23/2004US20040255403 Primary intermediates for oxidative coloration of hair
12/23/2004DE10323898A1 Hydroxyamidin- und Hydroxyguanidin-Verbindungen als Urokinase-Hemmstoffe Hydroxyamidine and hydroxyguanidine compounds as inhibitors of urokinase
12/23/2004CA2528003A1 Carbonyl compounds as inhibitors of histone deacetylase for the treatment of disease
12/23/2004CA2527236A1 Thiotungstate analogues and uses thereof
12/23/2004CA2526387A1 Benzamide derivative or salt thereof
12/22/2004EP1487811A1 N-sulfonylurea apoptosis promoters
12/22/2004EP1487810A2 4-(diarylmethyl)-1-piperazinyl derivatives
12/22/2004EP1487790A1 Purified lasofoxifene and a method for purification of racemic lasofoxifene by recrystallization
12/22/2004EP1487788A1 Diaminoacid-aminoacid-polyamine based gemini surfactant compounds
12/22/2004EP1487573A2 Catalysts and method for the production of amines
12/22/2004EP1487449A1 Tyrosyl derivatives and their use as p2x7 receptor modulators
12/22/2004EP1487428A2 Amino-substituted (e)-2,6-dialkoxystyryl 4-substituted benzylsulfones for treating proliferative disorders
12/22/2004EP1080066A4 Bioreductive cytotoxic agents
12/22/2004EP0929536B1 Piperazine based cytofectins
12/22/2004CN1556703A 1H-imidazole derivatives having CB1 agonistic, CB1 partial agonistic or CB1 antagonistic activity
12/22/2004CN1181065C Aralkylformylakyl piperazine derivative and its application as brain nerve protector
12/22/2004CN1181043C Quaternary bis-ammonium salt precursors and their uses as prodrugs having antiparasitic activity
12/21/2004US6833384 Deacetylase inhibitors
12/21/2004US6833382 Streptogramins and method for preparing same by mutasynthesis
12/21/2004US6833369 Treatment of ocular neovascular diseases, neovascular glaucoma, diabetic retinopathy,
12/21/2004CA2322989C Oxidation dyeing compositions containing a cationic coupling agent, novel cationic coupling agents
12/16/2004WO2004108673A2 Inhibitors of papilloma virus
12/16/2004WO2004087685A3 Phospholipase c inhibitors for use in treating inflammatory disorders
12/16/2004WO2004052939A3 Ligands for metals and improved metal-catalyzed processes based thereon
12/16/2004WO2004050022A8 Phenylalanine derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
12/16/2004WO2003063797A8 Cycloalkyl inhibitors of potassium channel function
12/16/2004US20040254375 Process for the preparation of 2-(2-(4-(bis(4-fluorophenyl)methyl)-piperazin-1-yl)ethoxy)acetic acid derivatives or corresponding salt forms thereof and intermediates therefor
12/16/2004US20040254344 Amino acid conjugates providing for sustained systemic concentrations of gaba analogues
12/16/2004US20040254280 Blends of waxes and polymer additives
12/16/2004US20040254196 Cinnamaldehyde derivatives inhibiting growth of tumor cell and regulating cell cycle, preparations and pharmaceutical compositions thereof
12/16/2004US20040254165 Vitiligo; skin cancer; control skin coloring
12/16/2004US20040254156 opioid receptor agonists such as 2-[4-(methanesulfonylamino-methyl)-phenyl]-N-methyl-N-[1-(S)-phenyl-2-pyrrolidin-1-ylethyl]-acetamide used for preventing pain, pruritus and gastrointestinal disorders
12/16/2004US20040251452 1,3,5-Tricyano-2,4,6-tris(vinyl)benzene derivatives and method for preparing the same
12/16/2004CA2526506A1 Inhibitors of papilloma virus