Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
07/2005
07/20/2005CN1642535A Tuberculosis treatment using pleuromutilin derivatives
07/20/2005CN1642531A Palatable chewable tablet
07/20/2005CN1211353C Unsaturated hydroximic acid derivatives as PARP inhibitors
07/19/2005US6919482 A 1,4-bis(N-(2-(4-hydroxy-3-hydroxymethylphenyl) -2-hydroxyethyl)amino)-cyclohexane or alkyl-cyclohexane or -pyrazine derivatives; treating respiratory diseases disorders, asthma, bronchitis, nervous system injury
07/19/2005US6919481 Alkoxyamines containing a vinyl group, their applications and methods of their production
07/19/2005US6919367 Substituted thioacetamides
07/19/2005US6919350 Compositions and methods for reducing respiratory depression and attendant side effects of mu opioid compounds
07/19/2005US6919336 Hallogenated aminobenzophenones and aminobenzoylpyridines as inhibitors of IL-1 and TNF
07/14/2005WO2005063773A1 Ionic liquid, method for producing same, double layer capacitor comprising same, and lithium battery
07/14/2005WO2005063729A1 3-(4-benzyloxyphenyl)propanoic acid derivatives
07/14/2005WO2005063705A1 Benzene compounds disubstituted with cyclic groups at the 1- and 2-positions
07/14/2005WO2005063697A2 Substituted n-aryl amidines as selective d1 dopamine receptor antagonists for the treatment of obesity and cns disorders
07/14/2005WO2005063689A1 Benzamide derivative
07/14/2005WO2005063680A1 Process for the preparation of arylamines
07/14/2005WO2005063247A1 Aryl sulfonamide compounds and uses related thereto
07/14/2005WO2005063239A1 3-(4-piperidine-1ylmethyl-phenyl)-propion acid-phenylamide-derivatives and related compounds used in the form of mch antagonists (melanine concentrating hormone) for treating eating disorders
07/14/2005WO2005063222A1 Hsp90 FAMILY PROTEIN INHIBITOR
07/14/2005WO2005040142B1 Novel keto-oxadiazole derivatives as cathepsin inhibitors
07/14/2005WO2004113277A8 Methods and compositions for treating amyloid-related diseases
07/14/2005US20050154233 Disproportionation of a N-oxy-2,2,6,6-tetramethylpiperidine or N-oxy-2,2,5,5-tetramethylpyrrolidine; separation of the protonated hydroxylamine from the nitrosonium compound using a hydrophobic resin; recyclable oxidation catalysts for carbohydrate oxidation
07/14/2005US20050154232 Nitrosation of the diphenylamine with an alkali metal nitrite in an acidic medium; the nitrosodiphenylamines increase the bioavailability of endothelial nitrogen monoxide; the diphenylamines are used as antioxidants and free radical scavengers; insulin resistance
07/14/2005US20050154230 Urea derivatives
07/14/2005US20050154202 Substituted aryl amides
07/14/2005US20050154015 Substituted 4H-chromene and analogs as activators of caspases and inducers of apoptosis and the use thereof
07/14/2005US20050154011 such as S)-3-Methylcarbamoyl-7-sulfoamino-3,4-dihydro-1H-isoquinoline-2-carboxylic acid tert-butyl ester, used in the treatment of protein tyrosine phosphatase (PTPase) mediated disorder such as diabetes
07/14/2005US20050153996 Compounds that modulate ppar activity and methods for their preparation
07/14/2005US20050153981 N1-phenacyl-N4-[2-(benzylamino)-2-oxo-ethyl] piperazine; as neuroprotective agents, in the treatment of ischemic cerebral apoplexy, human cerebral infraction; antiischemic agents for brain disorders; side effect reduction
07/14/2005US20050153371 Conjugated small molecules
07/14/2005US20050153366 Protein-protein interaction antagonist screening libraries based upon 1,4-disubstituted naphthalenes and related scaffolds
07/14/2005DE10360151A1 New 3-oxo-1-propenyl azo compounds useful as 5-HT receptor antagonists e.g. for treating psychoses, neurological disorders, amyotrophic lateral sclerosis and eating disorders
07/14/2005CA2551610A1 3-(4-benzyloxyphenyl)propanoic acid derivatives
07/14/2005CA2551602A1 Methods for controlling sr protein phosphorylation, and antiviral agents whose active ingredients comprise agents that control sr protein activity
07/14/2005CA2550679A1 Substituted n-aryl amidines as selective d1 dopamine receptor antagonists for the treatment of obesity and cns disorders
07/14/2005CA2550649A1 3-(4-piperidine-1ylmethyl-phenyl)-propion acid-phenylamide-derivatives and related compounds used in the form of mch antagonists (melanine concentrating hormone) for treating eating disorders
07/14/2005CA2548309A1 Aryl sulfonamide compounds and uses related thereto
07/13/2005EP1553092A1 Aralkyl formyl-alkyl piperazine derivatives and their uses as cerebral nerve protective agent
07/13/2005EP1553074A1 Fused benzene derivative and use
07/13/2005EP1552836A1 Anti-neurodegenerative agents
07/13/2005EP1551822A2 Pentacyclic oxepines and derivatives thereof, process for their preparation and pharmaceutical compositions containing them
07/13/2005EP1551799A1 Cyclohexyl sulphones as gamma-secretase inhibitors
07/13/2005EP1551797A1 Cyclohexyl sulphone derivatives as gamma-secretase inhibitors
07/13/2005EP1551795A1 Inhibitors of histone deacetylase
07/13/2005EP1161415B1 N-cyanomethylamides as protease inhibitors
07/13/2005EP1144364B1 Multicyclic compounds which inhibit leukocyte adhesion mediated by vla-4
07/13/2005EP1020426B1 Amine derivatives and process for producing the same
07/13/2005CN1639142A Method for producing 3-amidinophenylalanine derivatives
07/13/2005CN1639133A Novel antibacterial compounds, process for their preparation and pharmaceutical compositions containing them
07/13/2005CN1639126A Nitrosodiphenylamine derivatives and their pharmaceutical use against oxidative stress pathologies
07/13/2005CN1639125A New inhibitors of histone deacetylase
07/13/2005CN1639096A Process for producing trans-4-amino-1-cyclohexanecarboxylic acid derivative
07/13/2005CN1638773A Pharmaceutical preparations containing aminobenzene- sulfonic acid derivatives as the active ingredient
07/13/2005CN1638757A 组织蛋白酶半胱氨酸蛋白酶抑制剂 Cathepsin cystatin
07/13/2005CN1637018A Novel effectors of dipeptidyl peptidase IV
07/13/2005CN1636986A Benzophenones as inhibitors of reverse transcriptase
07/13/2005CN1636985A Benzophenones as inhibitors of reverse transcriptase
07/13/2005CN1636984A Benzophenones as inhibitors of reverse transcriptase
07/13/2005CN1636980A 二肽腈组织蛋白酶k抑制剂 Dipeptide nitrile cathepsin inhibitors k
07/13/2005CN1636597A Compounds for the treatment of female sexual dysfunction
07/13/2005CN1636593A Novel effectors of dipeptidyl peptidase IV
07/13/2005CN1210270C Novel use of phenylheteroalkylamine derivatives
07/13/2005CN1210263C N-hydroxy-2-(alkyl, aryl or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
07/12/2005US6916957 Antiinflammatory agents; antihistamines; antiallergens
07/12/2005US6916927 Pyrazolopyrimidinones which inhibit type 5 cyclic guanosine 3′,5′-monophosphate phosphodiesterase (cGMP-PDE5) for the treatment of sexual dysfunction
07/12/2005US6916926 Process for the preparation of (±) 1-3-dioxolanes and the optical resolution thereof
07/12/2005US6916850 Pyruvate derivatives
07/12/2005US6916812 Dietetic agents
07/12/2005US6916802 Synthase inhibitors for lowering glycosphingolipid levels; anticancer agents; for treatment of Gaucher's disease
07/12/2005US6916797 α-arylethylpiperazine derivatives as neurokinin antagonists
07/12/2005US6916461 Metal complexes that contain perfluoroalkyl, process for their production and their use in NMR diagnosis
07/12/2005US6916347 Making 2-amino-5-substituted-amino-phenol derivatives by reduction, hydrogenation, amination, hydroxylation; oxidation color dyes, hair dye mixture including coupler and developer oxidizers, yellow color shades, colorfastness
07/07/2005WO2005061459A1 Biaryl sulfonamides and methods for using same
07/07/2005WO2005060456A2 Method for treating adamts-5-associate disease
07/07/2005WO2005049593A3 N-acylsulfonamide apoptosis promoters
07/07/2005WO2005037810A3 Cyclopropyl methanone derivatives, the preparation and the therapeutic use thereof
07/07/2005WO2005032471A3 Benzylether and benzylamino beta-secretase inhibitors for the treatment of alzheimer's disease
07/07/2005US20050148774 Isotopically enriched N-substituted piperazine acetic acids and methods for the preparation thereof
07/07/2005US20050148773 labeling reagents; powerful tools for analyte analysis, including but not limited to multiplex proteomic analysis; comprises one or more heavy atom isotopes; intermediates in the synthesis of active esters of N-substituted piperazine acetic acid
07/07/2005US20050148771 Active esters of N-substituted piperazine acetic acids, including isotopically enriched versions thereof
07/07/2005US20050148672 reacting methyl bromide and 2-[(1R)-3-(diisopropylamino)-1-phenylpropyl]-4-(trifluoromethyl) phenol; formation of (3R)-3-[2-hydroxy-5-(trifluoromethyl)phenyl]-N,N-diisopropyl-N-methyl-3-phenylpropan-1-aminium bromide; asthma, chronic obstructive pulmonary disorder, allergic and infectious rhinitis
07/07/2005US20050148656 Carboxylic derivates
07/07/2005US20050148625 Use of estrogen antagonists and estrogen agonists inhibiting pathological conditions
07/07/2005US20050148613 Carbonylamino-derivatives as novel inhibitors of histone deacetylase
07/07/2005US20050148595 heterocylcyclic amines used for treating or preventing conditions ameliorated by monoamine reuptake such as vasomotor symptoms, sexual dysfunction, gastrointestinal and genitourinary disorders, chronic fatigue syndrome, fibromylagia syndrome, nervous system disorders
07/07/2005US20050148584 N-(3-(2-(4-morpholino)ethyloxy)phenyl)-N-{(cis3-(benzylamino)cyclohexyl)methyl}-N'-phenylurea; useful for the treatment of gastrointestinal reflux disorders, eating disorders leading to obesity and irritable bowel syndrome
07/07/2005US20050147563 Imaging lymph nodes with a Gadolinium complex of 10-[2-hydroxy-4-aza-5-oxo-7-aza-7-(perfluorooctylsulfonyl)-nonyl]-1,4,7-tris (carboxymethyl)-1,4,7,10-tetraazacyclododecane; in vivo contrast media in nuclear spin tomography; blood-pool agents, lymphographic agents
07/07/2005DE10358539A1 Carbonsäureamidderivate Carboxamide
07/07/2005DE10354327A1 New perfluorocarboxylates, conductive perfluorocarboxylates with organic cation and electrolytes, e.g. for electrochemical double layer capacitor, are prepared from perfluorocarboxylic ester and tertiary amine or heterocyclic phosphine
07/07/2005CA2548513A1 Biaryl sulfonamides and methods for using same
07/07/2005CA2547575A1 Method for treating adamts-5-associated disease
07/06/2005EP1549627A1 1-phenylalkyl-piperazines
07/06/2005EP1549600A1 Ketones
07/06/2005EP1549283A1 Merocyanine derivatives for cosmetic use
07/06/2005EP1233961B1 Method for producing 5-(1-piperazinyl)-benzofuran-2-carboxamide by transition metal-catalyzed amination
07/06/2005EP1216225B1 Novel derivatives of dicarboxylic acid having pharmaceutical properties
07/06/2005CN1634901A Process for preparing N-benzyl piperazine
07/06/2005CN1209354C Salt of phenylacetyl-(N-methyl)leucine-aspartic acid- phenylalanine-(N-methyl)piperazine
07/06/2005CN1209353C Estrogen agonist/antagonist metabolites
07/06/2005CN1209352C Hydrazine derivatives
07/05/2005US6914137 Adjustment of pH
07/05/2005US6914058 1-(p-(thiomorpholino)phenyl)-1,2,3-triazole derivatives