Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005) |
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11/03/2005 | US20050245503 Therapeutic heterocycles |
11/03/2005 | US20050245500 Beta-ketoamide compounds with MCH antagonistic activity |
11/03/2005 | CA2563180A1 Non-nucleoside reverse transcriptase inhibitors |
11/02/2005 | EP1590344A2 Anti-cancer medicaments |
11/02/2005 | EP1590340A1 Inhibitors of histone deacetylase |
11/02/2005 | EP1590338A2 Modulators of melanocortin receptor |
11/02/2005 | EP1590323A2 Piperazine derivatives and their use as synthesis intermediates |
11/02/2005 | EP1590322A1 Carbonyl-amino substituted acyl phenyl urea derivatives, method for the production and use thereof |
11/02/2005 | EP1590314A2 2-aryl-acetic acids, their derivatives and pharmaceutical compositions containing them |
11/02/2005 | EP1334084A4 Phosgene-free process for preparing carbamates |
11/02/2005 | EP1309540B1 Oxidizing colorant |
11/02/2005 | EP1278719B1 Naphthamide neurokinin antagonists for use as medicaments |
11/02/2005 | EP1196371B1 Quaternary bis-ammonium salt precursors and their uses as prodrugs having an antiparasitic activity |
11/02/2005 | EP1159261B1 Antizyme modulators and their use |
11/02/2005 | CN1692109A Novel compounds as NS3-serine protease inhibitors of hepatitis c virus |
11/02/2005 | CN1692105A Cetirizine dihydrochloride polymorph and preparation method thereof |
11/02/2005 | CN1690052A Piperazine derivatives and their use in the preparation of quinolone derivatives |
11/02/2005 | CN1690041A Novel derivatives of 3, 3-diphenylpropylamines |
11/01/2005 | US6960688 Use of compounds for the elevation of pyruvate dehydrogenase activity |
11/01/2005 | US6960665 Process for arylating or vinylating or alkynating a nucleophilic compound |
11/01/2005 | US6960614 Oxygenated esters of 4-lodo phenylamino benzhydroxamic acids |
11/01/2005 | US6960612 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith |
11/01/2005 | US6960588 Tryptase inhibitors |
11/01/2005 | US6960579 administering a compound containing a biheterocylic ring with sulfonamide group: sleeping disorder, depression, anxiety, circadian rhythm disorders |
11/01/2005 | US6960355 Modified amino acid compounds useful in delivery of active agents |
10/27/2005 | WO2005100505A1 New organic luminescent element |
10/27/2005 | WO2005100345A1 Thio-substituted tricyclic and bicyclic aromatic methanesulfinyl derivatives |
10/27/2005 | WO2005100334A1 Dipeptidyl peptidase-iv inhibitors |
10/27/2005 | WO2005100325A1 Aryl glycinamide derivatives and their use as nk1 antagonists and serotonin reuptake inhibithors |
10/27/2005 | WO2005100324A1 2- ( arylalkoxy ) -1- phenylethylamine derivatives as nk1 antagonist and serotonin reuptake inhibitors |
10/27/2005 | WO2005100311A1 Bicyclic aromatic sulfinyl derivatives |
10/27/2005 | WO2005100310A1 Thio-substituted arylmethanesulfinyl derivatives |
10/27/2005 | WO2005100308A1 Thio-substituted biaryl-methanesulfinyl derivatives |
10/27/2005 | WO2005100303A1 Indene derivatives and process for the preparation thereof |
10/27/2005 | WO2005100297A1 Indene derivatives and process for the preparation thereof |
10/27/2005 | WO2005100292A1 New photoinitiators |
10/27/2005 | WO2005099353A2 A novel process for the preparation of linezolid and related compounds |
10/27/2005 | WO2005090295A3 2-phenylpropionic acid derivatives and pharmaceutical compositions containing them |
10/27/2005 | WO2005034848A3 Inhibitors of cathepsin s |
10/27/2005 | WO2004113275A3 Methods and compositions for treating amyloid-related diseases |
10/27/2005 | US20050240023 Cathepsin cysteine protease inhibitors |
10/27/2005 | US20050240018 Process for the production of n-(2,6-dimethyl-phenyl)-2-piperazin-1-yl-acetamide |
10/27/2005 | US20050240017 5-[4-(2-piperidin-1-yl-ethoxy)-phenyl]-5,11-dihydro-6-oxa-12-thia-dibenzo[a,f]azulen-2-ol; 13-[4-(2-piperidin-1-yl-ethoxy)-phenyl]-7,13-dihydro-12-oxa-benzo[4,5]cyclohepta[1,2-a]naphthalen-3-ol or derivatives or salts; for alleviating symptoms of estrogen deprivation, including bone loss |
10/27/2005 | US20050239881 viricides; polymerase inhibitors; therapy for genetic engineered virus |
10/27/2005 | US20050239870 Prevention of restenosis of blood vessels after trauma, angioplasty or stenting; aminoalkylamide, piperidine-, indole-, or pyrrole-amide derivatives; anticarcinogenic agents |
10/27/2005 | US20050239869 calcium atorvastatin (Lipitor) intermediate; from intermediate 5-(4-fluorophenyl)-2-isopropyl-1-(3-morpholin-4-yl-3-oxo-propyl)-4-phenyl-1H-pyrrole-3-carboxylic acid phenylamide; via diol esters from the 1,3,5-tricarbonyl precursors in a stereoselective ruthenium-catalyzed hydrogenation (patent indexing) |
10/27/2005 | US20050239862 Amino ceramide-like compounds and therapeutic methods of use |
10/27/2005 | US20050239849 Substituted phenoxyacetic acids |
10/27/2005 | US20050239839 Adamantylglycine-based inhibitors of dipeptidyl peptidase IV and methods |
10/27/2005 | US20050239802 E.g., 6-{2-[5-Chloro-2-(2,4-difluorobenzyloxy)- phenyl]cyclopent-1-enyl}-pyridine-2-carboxylic acid, used to treat prostaglandin mediated diseases that include inflammatory, neuropathic or visceral pain |
10/27/2005 | US20050239799 1-phenyl-4-benzylpiperazines dopamine receptor subtype |
10/27/2005 | US20050238614 Polyethylene glycol conjugates of heterocycloalkyl carboxamido propanoic acids |
10/27/2005 | CA2562554A1 Thio-substituted arylmethanesulfinyl derivatives |
10/27/2005 | CA2562401A1 Thio-substituted tricyclic and bicyclic aromatic methanesulfinyl derivatives |
10/27/2005 | CA2561555A1 Bicyclic aromatic sulfinyl derivatives |
10/26/2005 | EP1589016A1 Thio-substituted tricyclic and bicyclic aromatic methanesulfinyl derivatives |
10/26/2005 | EP1589008A1 A crystalline dibenzothiazepine derivative and its use as an antipsychotic agent |
10/26/2005 | EP1589001A1 Tricyclic aromatic and bis-phenyl sulfinyl derivatives |
10/26/2005 | EP1589000A2 (R)-Chiral halogenated 1-substitutedamino-(N+1)-alkanols useful for inhibiting cholesteryl ester transfer protein activity |
10/26/2005 | EP1588145A2 Methods, mixtures, kits and compositions pertaining to analyte determination |
10/26/2005 | EP1587518A2 Antineoplastic ether lipid compounds with modifications at the sn-3 carbon |
10/26/2005 | EP1587473A2 Thiosemicarbazones as anti-virals and immunopotentiators |
10/26/2005 | EP1183229B1 Glucagon antagonists/inverse agonists |
10/26/2005 | EP1098870B1 Nitrate salt of Cetirizine |
10/26/2005 | CN1688545A Phosphodiesterase 4 inhibitors, including n-substituted phenylamine and diphenylamine analogs |
10/26/2005 | CN1688527A Fused benzene derivative and use |
10/26/2005 | CN1688298A Composition, synthesis and therapeutic applications of polyamines |
10/26/2005 | CN1687042A Technique for producing N-formyl morpholine |
10/26/2005 | CN1687041A Method for synthesizing piperazine |
10/26/2005 | CN1224612C Acetylenic sulfonamide thiol TACE inhibitors |
10/26/2005 | CN1224598C Naphthalene derivatives |
10/25/2005 | US6958352 Compounds for inhibiting insulin secretion and methods related thereto |
10/25/2005 | US6958331 sulfonyl amine derivatives such as {2-(2,2-diphenyl-ethylamino)-5-[4-(4-isopropyl-piperazine-1-carbonyl)-piperidine-1-sulfonyl]-phenyl}-morpholin-4-yl-methanone; pain, inflammation, septic shock |
10/25/2005 | US6958243 Organic reactions with CO generating materials |
10/25/2005 | US6958205 Image forming material and ammonium compound |
10/25/2005 | CA2332461C New benzenesulfonamide derivatives, their method of preparation and the pharmaceutical compositions containing them |
10/25/2005 | CA2331053C Compositions and methods for treating conditions responsive to estrogen |
10/25/2005 | CA2331009C Compositions and methods of treatment for conditions responsive to testosterone elevation |
10/25/2005 | CA2261725C Piperidine and piperazine derivatives and their use as muscarinic antagonists |
10/25/2005 | CA2245490C 3,4-disubstituted phenylethanolaminotetralincarboxamide derivatives |
10/25/2005 | CA2147056C Novel delta-amino-gamma-hydroxy-omega-aryl-alkanoic acid amides |
10/20/2005 | WO2005097779A1 Diarylamine derivatives as calcium channel blockers |
10/20/2005 | WO2005097203A2 Serum protein conjugates of ion channel modulating compounds and uses thereof |
10/20/2005 | WO2005097092A1 Compound with vitamin k activity, particularly as additive for feeds, and preparation of the compound |
10/20/2005 | WO2005049561A3 Processes for preparing novel methylene blue derivative |
10/20/2005 | US20050234265 2-aminomethyl-5-tert-butyl-3-phenylphenol; antimalaria; used against protozoa of the genus Plasmodium, particularly emerging strains of drug-resistant Plasmodia |
10/20/2005 | US20050234125 Alpha-sulfonylamino-acetonitriles |
10/20/2005 | US20050234109 to treat Alzheimer's disease,Down syndrome and the other diseases associated with amyloid deposition; thiomethane, sulfinylmethane or sulfonylmethane compounds; 5-Chloro-4-[(4-chlorophenylsulfonyl)-(2,5-difluorophenyl)methyl]-2-(4'-hydroxypiperidin-1'-yl)pyridine |
10/20/2005 | US20050234106 1-aryl-1-heteroarylaminoalkylene-substituted, e.g., 1-[fluorophenylcyclohexylmethyl]isoquinolin-1-ylamine; antiarrhythmia agents; cardiovascular disorders |
10/20/2005 | US20050234065 Dipeptidyl peptidase-IV inhibitors |
10/20/2005 | US20050234061 N-[3-(4-chlorophenyl)-2-(3-pyridyl)-1-methylpropyl]-2-(5-trifluoromethyl-2-pyridyloxy)-2-methylpropanamide; obesity; antipsychotic agents; synergistic; cannabinoid receptor antagonists |
10/20/2005 | US20050234058 Secondary amino-and cycloamino-cycloalkanol derivatives and methods of their use |
10/20/2005 | US20050234050 Ph sensitive prodrugs of 2,6-diisopropylphenol |
10/20/2005 | US20050234046 Aryl sulfonamide and sulfonyl compounds as modulators of PPAR and methods of treating metabolic disorders |
10/20/2005 | US20050233943 Novel polyamine analog conjugates and quinone conjugates as therapies for cancers and prostate diseases |
10/20/2005 | CA2562371A1 Diarylamine derivatives as calcium channel blockers |
10/19/2005 | EP1586561A1 Bicyclic aromatic sulfinyl derivatives |
10/19/2005 | EP1586560A1 Thio-substituted arylmethanesulfinyl derivatives |
10/19/2005 | EP1586559A1 Biaryl-methanethio-, -sulphinyl- and sulphonyl derivatives |
10/19/2005 | EP1586558A2 Bis-sulfonamide hydroxyethylamino retroviral protease inhinitors |