Patents
Patents for C07D 235 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings (15,325)
01/2002
01/15/2002US6339082 Tricyclic compounds, preparation method and said method intermediates, application as medicines and pharmaceutical compositions containing same
01/15/2002CA2028302C Benzimidazole derivatives, their production and use
01/10/2002WO2002002533A1 Propane-1,3-dione derivatives
01/10/2002WO2002002532A1 4-alkoxy cyclohexane-1 amino carboxylic acid esters and method for the production thereof
01/10/2002DE10030664A1 Verfahren zur Herstellung von UV-Filter-Substanzen Process for the preparation of UV filter substances
01/10/2002DE10030663A1 UV-B-Filter UV-B filters
01/09/2002EP1170288A2 Diphenylureum derivatives and their use as alpha2/5-HT2c antagonists
01/09/2002EP0607439B1 Nitrogenous heterocyclic compound
01/09/2002CN1330677A Method for production of polyelectrolyte membranes and fuel cell
01/09/2002CN1330641A Crystalline forms of 3-(2,4-dichlorobenzyl)-2-methyl-N-(pentylsulfonyl)-3H-benzimidzole-5-carboxamide
01/09/2002CN1330640A Cyclic hydrazine derivatives as TNF-alpha inhibitors
01/09/2002CN1077427C Skin protecting composition containing acid hydrophilic agent for cosmetic use and application of same
01/03/2002WO2002102789A1 Antimicrobial and radioprotective compounds
01/03/2002WO2002000614A1 Aryl compounds, their preparation and their use in therapy
01/03/2002WO2001051473A8 1,2-diaryl benzimidazoles for treating illnesses associated with a microglia activation
01/03/2002US20020002169 Protein kinase inhibitors
01/03/2002DE10030375A1 Verwendung von MTP-Inhibitoren zur Senkung von ppTRL Use of MTP inhibitors to reduce ppTRL
01/02/2002EP1167360A1 Human chymase inhibitors
01/02/2002EP1167359A1 Process for the preparation of 2-arylbenzimidazole sulphonic acids and their use as UV-filters
01/02/2002EP1167358A1 2-Phenylbenzimidazole sulphonic acids as UV-B filters
01/02/2002EP1167357A1 Alpha-substituted carboxylic acid derivatives
01/02/2002EP1165557A1 ARYL AND HETEROARYL FUSED AMINOALKYL-IMIDAZOLE DERIVATIVES: SELECTIVE MODULATORS OF GABAa RECEPTORS
01/02/2002EP1165530A2 Dihetero-substituted metalloprotease inhibitors
01/02/2002EP1165519A1 Aryl and heteroaryl fused aminoalkyl-imidazole derivatives and their use as antidiabetics
01/02/2002EP1165518A2 Benzimidazole and imidazolopyridine derivatives, their preparation and their use as selective modulators of bradykinin b2 (= bk-2) receptors
01/02/2002EP1165517A1 N-benzimidazolylmethyl- and n-indolylmethyl-benzamides and their use as crf modulators
01/02/2002EP1165512A2 Method for arylating aza-heterocycles with activated aromatic compounds in the presence of cesium carbonate
01/02/2002EP1165511A2 Method of producing heterocyclic carbamates from aza-heterocyclic compounds and carbon dioxide
01/02/2002EP1165504A2 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF
01/02/2002CN1329601A New benzimidazolone-benzoxazolone-, or benzothiazolone derivatives as ion channel modulating agents
01/02/2002CN1329281A Colour photosensitive imaging element containing closed developer
01/01/2002US6335334 Hypertensive agents, anticoagulants; cardiovascular and sexual disorders, angina pectoris, and atherosclerosis
12/2001
12/27/2001WO2001097787A2 Use of microsomal triglyceride transfer protein (mtp) inhibitors for reducing the number of postprandial triglyceride-rich lipoprotein particles (pptrl)
12/27/2001WO2001064659A3 Indane derivatives and their use as cell adhesion inhibitors
12/27/2001US20010056100 Carboxylic acid or tetrazole derivatives containing carbamate groups are useful for treating the conditions associated with the urinary tract, pain, inflammation, respiratory states, edema formation of hypotensive vascular diseases
12/27/2001CA2413277A1 Use of microsomal triglyceride transfer protein (mtp) inhibitors for reducing the number of postprandial triglyceride-rich lipoprotein particles (pptrl)
12/20/2001WO2001096299A2 Indole derivatives and their use as 15-lipoxygenase inhibitors
12/20/2001WO2001096289A1 Sulfonamide derivatives
12/20/2001WO2001051456A3 Antibacterial agents
12/20/2001US20010053856 Sunscreen agents; ultraviolet radiation absorber
12/20/2001US20010053779 Antiinflammatory agents; respiratory system disorders
12/20/2001CA2411811A1 Sulfonamide derivatives
12/20/2001CA2411116A1 Indole derivatives and their use as 15-lipoxygenase inhibitors
12/19/2001EP1164418A2 Color photothermographic elements comprising blocked developing agents
12/19/2001EP1164134A1 Benzimidazole compounds and their use as modulators of the GABA A receptor complex
12/19/2001EP1164121A1 Novel carboxylic acid derivatives and process for producing the same
12/19/2001EP1163221A1 Sulfonamide derivatives as 5ht7 receptor antagonists
12/19/2001EP1094816A4 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
12/18/2001US6331640 Diaminopropionic acid derivatives
12/18/2001US6331563 N-Hydroxy-2-(Alkyl, Aryl, or Heteroaryl, Sulfanyl, Sulfinyl or Sulfonyl)-3-Substituted Alkyl, Aryl or Heteroarylamides as Matrix Metalloproteinase inhibitors
12/18/2001CA2204290C Benzimidazole derivatives, their production and use
12/18/2001CA2160725C Process for the preparation of a tetrazole derivative in two crystalline forms and novel crystalline form of said derivative
12/13/2001WO2001094341A1 Quinazoline derivatives for the treatment of tumours
12/13/2001WO2001094321A1 Bicyclic cyclohexylamines and their use as nmda receptor antagonists
12/13/2001WO2001094317A2 Method for synthesis of substituted azole libraries
12/13/2001CA2407164A1 Bicyclic cyclohexylamines and their use as nmda receptor antagonists
12/13/2001CA2345195A1 Color photothermographic elements comprising blocked developing agents
12/12/2001EP1162196A1 Fused-ring compounds and use thereof as drugs
12/12/2001EP0781126B1 Derivatives of 2-amino-1,2,3,4-tetrahydro-naphthalene active on the cardiovascular system
12/11/2001US6329360 Hetero-linked phenylglycinolamides
12/06/2001WO2001092239A1 Biciclic cyclohexylamines and their use as nmda receptor antogonists
12/06/2001US20010049447 2-(-2-(N-(3-benzoimidazol-2-yl)propyl)-N-methylamino)ethyl)-6-fluoro -1,2,3,4-tetrahydro-1-isopropyl-2-napthyl-esters; antidiabetic agents and treats microvascular or macrovascular diseases associated with diabetes.
12/06/2001US20010049446 C-C9-Heteroaryl, linked via C or N, substituted or unsubstitued by 1,3-substituents, substituted benzoylguanidine derivatives useful for treating ischemia, cardiac infarct, angina pectoris, and storke etc.
12/06/2001US20010049385 Treating obesity; suppressing appetite; treating type 2 diabetes; treatment and/or prevention of diseases and disorders related to the histamine H3 receptor.
12/06/2001CA2409006A1 Biciclic cyclohexylamines and their use as nmda receptor antogonists
12/05/2001EP1159237A1 Method of preparing surface-active alcohols and surface-active alcoholic ethers, products obtained by said method and their use
12/05/2001EP0821684B1 Benzimidazole compounds and their use as modulators of the gaba a? receptor complex
12/05/2001EP0643701B1 Benzimidazole-derived compounds, method for preparing same, and therapeutical and cosmetic uses thereof
12/05/2001CN1325397A 2-piperazino alkylatnino benzoazole derivatives: dopamine receptor subtype sepcific ligands
12/05/2001CN1325376A Novel compounds and medicinal use thereof
12/05/2001CN1325308A Use of neurotrophic factor stimulators for treatment of ophthalmic neurodegenerative diseases
12/05/2001CN1325267A Fused-benzene derivatives useful as herbicides
12/04/2001USH2007 Insecticidal N-heterocyclylalkyl-or N-[(polycyclyl)alkyl]-N′substituted piperazines
12/04/2001US6326403 Cardiovascular disorders
12/04/2001US6326395 Amidine or amide substituted furan derivatives
12/04/2001US6326384 Dry blend pharmaceutical unit dosage form
12/04/2001US6326369 Bicyclic quinone compounds, their production and use
12/04/2001US6326133 Cyanine dyes
11/2001
11/29/2001WO2001090074A2 BENZOPHENONES AS INHIBITORS OF IL-1β AND TNF-$g(a)
11/29/2001US20010047038 Treating the patient suffering for herpes viruses, and cytomegalovirus with an effective amount of sulfur or sulfoxide or sulfonyl containing heteroaromatic compounds
11/29/2001US20010047021 Tetrasubstituted benzimidazole carbamates
11/29/2001US20010047020 Benzimidazole derivatives, their production and use
11/29/2001CA2408727A1 Benzophenones as inhibitors of il-1.beta. and tnf-.alpha.
11/28/2001EP0830344B1 2-substituted benzimidazole derivatives as smooth muscle cell proliferation inhibitors
11/28/2001CN1323788A 2-pyrimidyloxy-N-amidophynylbenzyl amine, and its prepn. and use
11/27/2001US6323227 Prodrugs
11/22/2001WO2001087859A1 Naphthol derivatives
11/22/2001US20010044468 Reduced in the body to produce a benzamidine; nontoxic
11/22/2001US20010044441 And female sexual dysfunction, premature labour or dysmenorrhea
11/21/2001EP1156043A2 Drugs that enhance synaptic responses mediated by ampa receptors
11/21/2001EP1155025A1 Platinum (ii) compounds
11/21/2001EP1154771A1 Nitrosated and nitrosylated proton pump inhibitors, compositions and methods of use
11/21/2001EP0914319B1 Diarylalkyl cyclic diamine derivatives as chemokine receptor antagonists
11/21/2001EP0831910B1 Epoxy-steroidal aldosterone antagonist and angiotensin ii antagonist combination therapy for treatment of congestive heart failure
11/21/2001EP0742210B1 2-mercaptobenzimidazole derivative and antihyperlipemic or antiarteriosclerotic agent containing the same
11/21/2001CN1323291A Diaminopropionic acid derivatives
11/21/2001CN1323289A Aminoalcohol derivatives and their use as beta 3 adrenergic agonists
11/15/2001US20010041730 (1S,2S)-2-(2-(N-((3-benzoimidazol-2-yl)propyl)-N-methylamino)ethyl)-6 -fluoro-1,2,3,4-tetrahydro-1-isopropyl-2-naphthyl cyclopropanecarboxylate, for example; treating vascular disease such as gangrene, retinopathy, nephropathy
11/14/2001EP1153017A1 Bicyclic compounds and their use as integrin receptor ligands
11/13/2001US6316634 Method for preparing cycloheptimidazoles