Patents
Patents for C07D 235 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings (15,325)
02/2003
02/20/2003WO2003014079A1 Stable polymorph of flibanserin, technical process for its preparation and the use thereof for preparing medicaments
02/20/2003WO2003014064A1 Naphthylurea and naphthylacetamide derivatives as vanilloid receptor 1 (vr1) antagonists
02/20/2003WO2003013539A1 Neuroprotective drug
02/20/2003WO2002068399B1 Aryl carbamate derivatives, preparation and use thereof
02/20/2003WO2002065979A3 (diazolo-pyridinyl)-pyrimidines for use in treatment of cns disorders and diabetes
02/20/2003WO2002049993A3 High affinity small molecule c5a receptor modulators
02/20/2003WO2002024635A3 Aminoalcohol derivatives
02/20/2003CA2455754A1 Amine derivatives
02/19/2003CN1398252A Dehydroamino acids compounds
02/18/2003US6521623 N,N'-disubstituted benzimidazolone derivatives with affinity at the serotonin and dopamine receptors
02/13/2003WO2003011835A1 Benzimidazolylalkyl-aryl(alkan) oic acid derivatives and their use as antihyperglycaemics
02/13/2003WO2003011812A1 NOVEL AMINE DERIVATIVE HAVING HUMAN β-TRYPTASE INHIBITORY ACTIVITY AND DRUGS CONTAINING THE SAME
02/13/2003WO2003011219A2 Mediators of hedgehog signaling pathways, compositions and uses related thereto
02/13/2003WO2002036580A9 Benzoxazole lpaat- beta inhibitors and uses thereof
02/13/2003US20030032663 Inhibition of the interaction of RAGE with its ligands; treatment acute and chronic inflammation, the development of diabetic late complications, Alzheimer's disease, erectile dysfunction, and tumor invasion and metastasis.
02/13/2003CA2456096A1 Novel amine derivative having human .beta.-tryptase inhibitory activity and medecine containing the same
02/13/2003CA2455100A1 Mediators of hedgehog signaling pathways,compositions and uses related thereto
02/12/2003EP1283205A1 Naphthol derivatives
02/12/2003EP1283202A1 Method for preparing heterocyclic-carboxylic acids
02/12/2003EP0944601B1 Guanidinylamino heterocycle compounds useful as alpha-2 adrenoceptor agonists
02/12/2003CN1397148A Luminescent element material and luminescent element comprising the same
02/12/2003CN1101385C Substituted benzimidazole derivatives and its preparation method and medicine use
02/11/2003US6518292 Heterocyclic aromatic compounds usefuls as growth hormone secretagogues
02/11/2003US6518291 Inosine-5'-monophosphate dehydrogenase inhibitors
02/06/2003WO2003009807A2 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods
02/06/2003US20030027842 Halogenobenzimidazoles
02/06/2003US20030027823 N,N'-disubstituted benzimidazolone derivatives with affinity at the serotonin and dopamine receptors
02/06/2003US20030027807 Vitronectin receptor antagonists, their preparation and their use
02/06/2003US20030027714 Late transition metal complexes, their use as catalysts and polymers therefrom
02/06/2003CA2452159A1 Cytoprotective compounds, pharmaceutical and cosmetic formulations, and methods
02/05/2003CN1395568A 1,2-diaryl benzimidazole derivative for treating illnesses associated with microglia activation
02/05/2003CN1395562A Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
02/05/2003CN1395467A Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents
02/05/2003CN1100776C Process for preparing magnesium salt of substituted sulphinyl heterocycle
02/05/2003CN1100748C Inhibition of matrix metalloproteases by 2-substituted-4-(4-substituted phenyl)-4-oxobutyric acids
02/04/2003US6515124 Dehydroamino acids
02/04/2003US6515023 Thrombin receptor antagonists
01/2003
01/30/2003WO2003007945A1 Viral polymerase inhibitors
01/30/2003WO2003007931A1 Sulfonamide derivatives
01/30/2003WO2002092088A3 Novel use of 2h-benzimidazol-2-one, 1,3-dihadro-1-(2{4-{3-(trifluoromethyl}phenyl]-1-piperazinyl}ethyl)- and its physiologically acceptable acid addition salts
01/30/2003WO2002012247A1 Method for the production of imidazo-(1,2-c)(2,3)-benzodiazepines and intermediates in the production thereof
01/30/2003US20030022935 Acylated 1,2,3,4-tetrahydronaphthyl amines and their use as pharmaceutical agents
01/30/2003CA2417804A1 Method for the production of imidazo-(1,2-c)(2,3)-benzodiazepines and intermediates in the production thereof
01/29/2003EP1105387B1 Prodrugs of proton pump inhibitors
01/29/2003CN1100056C Compound for inhibition of gastric acid secretion
01/29/2003CN1100042C Method for reducing amount of by-products in carbendazim by adding diazotization agents
01/28/2003US6512000 Aminocarbonyl-substituted benzimidazoles having tryptase-inhibitory activity
01/28/2003CA2254905C Tricyclic functional dyes for contrast enhancement in optical imaging
01/23/2003WO2003006670A2 2-[5-(5-carbamimidoyl-1h-heteroaryl)-6-hydroxybiphenyl-3-yl]-succinic acid derivatives as factor viia inhibitors
01/23/2003WO2003006438A1 Benzimidazole derivatives for treating microglia-activation associated diseases such as inflammatory, allergic, infectious or autoimmune diseases
01/23/2003WO2003006423A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003WO2003006011A1 2-[5-(5-carbamimidoyl-1h-heteroaryl)-6-hydroxybiphenyl-3-yl]-succinic acid derivatives as factor viia inhibitors
01/23/2003WO2002041835A3 Estrogen receptor modulators
01/23/2003WO2002036562A3 1-aryl- or 1-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-6 ligands
01/23/2003US20030018059 Antiinflammatory agents; antihistamines; antiallergens
01/23/2003US20030018025 Psychological disorders, antidepressants, Parkinson's disease
01/23/2003CA2453503A1 N-(3-amino-2-hydroxy-propyl) substituted alkylamide compounds
01/23/2003CA2452391A1 2-[5-(5-carbamimidoyl-1h-heteroaryl)-6-hydroxybiphenyl-3-yl]-succinic acid derivatives as factor viia inhibitors
01/22/2003EP1277752A1 Process for producing optically active sulfoxide derivative
01/22/2003EP1277742A1 Method for preparing halomethyl heterocyclic compounds
01/22/2003EP1277739A1 Method for preparing heterocyclic-carboxylic acids
01/22/2003EP1277729A1 Ppar (gamma) modulators
01/22/2003EP1071660B1 N-sulphonyl and n-sulphinyl phenylglycinamide
01/22/2003CN1099416C Integrin receptor antagonisis
01/21/2003US6509365 Useful as inhibitors of poly(ADP-ribose)polymerase and for the production of drugs.
01/16/2003WO2003004479A1 4-aryl quinols and analogs thereof as therapeutic agents
01/16/2003WO2003004464A2 Heterocyclic amide derivatives and the use thereof as pesticides
01/16/2003WO2003004023A1 1-alkyl-2-aryl-benzimidazole derivatives, their use for producing medicaments and pharmaceutical preparations containing said derivatives
01/16/2003WO2002046129A3 Inhibitors of histone deacetylase
01/16/2003US20030013891 Process for the preparation of N,N'-carbonyldiazoles and azolide salts
01/16/2003US20030013847 Pyruvate derivatives
01/16/2003US20030013846 Cytoprotective agents
01/16/2003US20030013751 Viricides; enzyme inhibitors
01/16/2003US20030013677 Anticancer agents
01/16/2003US20030013657 Reducing oxidation stresses; central nervous system disorders; antiinflammatory agents
01/16/2003US20030013656 Reducing oxidation stresses; central nervous system disorders; antiinflammatory agents
01/16/2003CA2452592A1 4-aryl quinols and analogs thereof as therapeutic agents
01/15/2003CN1391565A Benzophenones as inhibitors of reverse transcriptase
01/15/2003CN1098841C Novel amide derivatives and medicinal compositions thereof
01/15/2003CN1098838C Substituted N-(indole-2-carbonyl)-beta-alanimamides and derivatives as antidiabetic agents
01/14/2003US6506876 LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use
01/14/2003US6506783 A pharmaceutical composition that inhibits the growth of tumors and cancers in mammals and can be used to treat viral infections that comprises a fungicide is disclosed. The particular fungicide used is a benzimidazole derivative
01/14/2003US6506769 Heterocyclic compounds useful as inhibitors of tyrosine kinases
01/14/2003US6506738 Treatment of viral infections. More particularly, the invention provides benzimidazolone derivatives for the treatment of respiratory syncytial virus infection.
01/09/2003WO2003002532A1 Cyclic diamine compounds having fused-ring groups
01/09/2003WO2003002122A1 Beta-hydroxyamine derivatives useful in treatment of alzheimer's disease
01/09/2003US20030009033 Substituted condensation products of N-benzyl-3-indenylacent amides with heterocyclic aldehydes for neoplasia
01/09/2003US20030008915 Acylated 6,7,8,9-tetrahydro-5H-benzocycloheptenyl amines and their use as pharmaceutical agents
01/09/2003US20030008907 Intermediates for the synthesis of benzimidazole derivatives and a process for the preparation thereof
01/09/2003US20030008906 Administering benzothiazole compound for therapy, prophylaxis of disease
01/09/2003US20030008884 Fungicidal phenyl (thio) urea and phenyl (thio) carbamate derivatives
01/09/2003US20030008878 Administering benzimidazole compound for therapy of sexual dysfunction in a human
01/09/2003US20030008796 Composition and method for bleaching a substrate
01/09/2003CA2452039A1 Beta-hydroxyamine derivatives useful in treatment of alzheimer's disease
01/08/2003EP1273571A1 Nitrogenous compounds and antiviral drugs containing the same
01/08/2003EP1272473A1 Process for preparing substituted benzimidazole compounds
01/08/2003EP1272176A1 Adamantyl derivatives as anti-cancer agents
01/08/2003EP0946175B1 USE OF A COMBINATION OF H+, K+ -ATPase INHIBITORS AND GLUCOCORTICOIDS IN THE TREATMENT OF NASAL POLYPS
01/08/2003EP0859768B1 Amine acid salt compounds and process for the production thereof
01/08/2003CN1098261C Process for optical purification of enantiomerically enriched benzimidazole derivatives
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