| Patents for C07D 235 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings (15,325) |
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| 10/12/2000 | CA2360923A1 Process for the arylation of aza-heterocycles with activated aromatics in presence of caesium carbonate |
| 10/10/2000 | US6130235 Piperidine moieties coupled to indole, benzimidazole or benzotriazole. |
| 10/10/2000 | US6130217 Antitumor |
| 10/05/2000 | WO2000058286A2 Method of producing heterocyclic carbamates from aza-heterocyclic compounds and carbon dioxide |
| 10/05/2000 | WO2000058258A1 Novel carboxylic acid derivatives and process for producing the same |
| 10/05/2000 | WO2000057877A1 Aryl substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles, and the use thereof |
| 10/05/2000 | CA2368631A1 Aryl substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles, and the use thereof |
| 10/05/2000 | CA2361019A1 Process for the preparation of heterocyclic carbamates from aza-heterocycles and carbon dioxide |
| 10/04/2000 | EP1040098A1 Integrin receptor antagonists |
| 10/04/2000 | CN1057088C Benzimidazole, prepn. method and use thereof |
| 10/04/2000 | CN1057085C Heterocyclically substituted phenyl-cyclohexane carboxylcic acid derivatives |
| 10/03/2000 | US6127547 Halobenzimidazoles and their use as microbicides |
| 10/03/2000 | US6127415 Apoptosis inducing adamantyl derivatives and their usage as anti-cancer agents |
| 10/03/2000 | US6127380 4-aminoalkoxy-1H-benzoimidazoles |
| 10/03/2000 | US6127373 Method of treating tourette's syndrome and obsessive compulsive disorder |
| 10/03/2000 | US6127372 Sulfonamide inhibitors of aspartyl protease |
| 09/28/2000 | WO2000056918A1 Method for screening cysteine protease inhibitor |
| 09/28/2000 | WO2000056712A1 Sulfonamide derivatives as 5-ht7 receptor antagonists |
| 09/28/2000 | DE19913483A1 Verfahren zur Herstellung von Heterocyclischen Carbamaten aus Aza-Heterocyclen und Kohlendioxid Process for the preparation of heterocyclic carbamates from carbon dioxide and aza heterocycles |
| 09/28/2000 | CA2367504A1 A screening method for a cysteine protease inhibitor |
| 09/27/2000 | EP1037878A2 Metabotropic glutamate receptor antagonists for treating central nervous system diseases |
| 09/27/2000 | CN1268123A Benzimidazole derivatives |
| 09/26/2000 | US6124470 Method for working up benzimidazolone-containing reaction mixtures |
| 09/26/2000 | US6124464 Mixing a substituted sulfinyl heterocyclic compound containing an imidazole moiety with an alkylamine base or ammonia and a magnesium salt. |
| 09/26/2000 | US6124463 Treatment of affective disorder, anxiety or depression |
| 09/26/2000 | US6124321 An enzyme inhibitor for enhancing memory or treating or preventing alzheimer's disease |
| 09/26/2000 | US6124243 Method of controlling graminaceous weeds |
| 09/21/2000 | WO2000054729A2 Heterocyclic aromatic compounds useful as growth hormone secretagogues |
| 09/21/2000 | DE19912690A1 New benzimidazolyl amidine or nitrile compounds, useful as thrombin inhibitors or antithrombotic agents, for treating deep leg vein thrombosis |
| 09/21/2000 | CA2367461A1 Heterocyclic aromatic compounds useful as growth hormone secretagogues |
| 09/20/2000 | EP1036794A1 2-aryl-8-oxodihydropurine derivatives, process for producing the same, medicinal compositions containing the same, and intermediates thereof |
| 09/20/2000 | CN1056609C Benzoyl guanidines, their production and their use in medicinal compositions |
| 09/19/2000 | US6121487 Method of producing amino acids and amino-acid derivatives |
| 09/19/2000 | US6121308 Indole and benzimidazole antithrombotic compounds, such as 1-methyl-2-(n-(4-amidinophenyl)-aminomethyl)-5-(n-(hydroxycarbonylmethyl) -quinoline-8-sulphonylamino)-indole |
| 09/14/2000 | WO2000053547A1 Method of preparing surface-active alcohols and surface-active alcoholic ethers, products obtained by said method and their use |
| 09/14/2000 | WO1999063999A8 H1-histamine receptor antagonists |
| 09/14/2000 | DE19910370A1 Verfahren zur Herstellung von Tensidalkoholen und Tensidalkoholethern, die hergestellten Produkte und ihre Verwendung A process for the preparation of surfactant alcohols and surfactant alcohol ethers, the manufactured products and their use |
| 09/13/2000 | CN1056368C Preparation process for albendazole |
| 09/08/2000 | WO2000051993A2 Dihetero-substituted metalloprotease inhibitors |
| 09/08/2000 | CA2366954A1 Dihetero-substituted metalloprotease inhibitors |
| 09/06/2000 | CN1265665A Benzimidazole derivatives |
| 09/06/2000 | CN1265394A Compound as intermediates for use in preparation of optically active 2-imidazoline-5-one or 2-imidazoline-5-thionone derivatives |
| 09/06/2000 | CN1056140C Biphenyl derivatives, their preparation and theirt use for treatment of hypertension and cardiac disease |
| 09/05/2000 | US6114532 Anticoagulant |
| 09/05/2000 | US6114393 Use of inhibitors of the sodium-hydrogen exchanger for the production of a pharmaceutical for the treatment of disorders which are caused by protozoa |
| 09/05/2000 | US6114390 An argininamide or ornithinamide compound as treating memory loss, migraine, sleep disorders, pain, cardiovascular diseases, subarachnoidal bleeding, vascular-hypertrophic changes, cerebral and coronary vasospasms |
| 09/05/2000 | US6114369 N-methyl-n-(1-(4-fluorobenzyl)benzionidazol-2-yl)-n'-methyl-n-(3,5 -bis(trifluoromethyl)benzylaminocarbonyl)-1,3-propylenediamine hydrochloride, for example; substance p antagonists; antiallergic activity |
| 09/05/2000 | US6114327 Anti-viral compounds |
| 08/31/2000 | WO2000050431A1 Platinum (ii) compounds |
| 08/31/2000 | WO2000050419A1 Substituted bicyclic heterocycles and the use thereof as thrombin inhibitors |
| 08/31/2000 | WO2000050407A1 Herbicidal 2-(5-isoxazolinyl methyloxyphenyl) -4,5,6,7-tetrahydro -2h-indazole derivatives |
| 08/31/2000 | DE19907813A1 Substituierte bicyclische Heterocyclen, deren Herstellung und deren Verwendung als Arzneimittel Substituted bicyclic heterocycles, their preparation and their use as medicaments |
| 08/31/2000 | CA2364712A1 Platinum (ii) compounds |
| 08/30/2000 | EP1031563A1 Sulfonyl derivatives |
| 08/30/2000 | EP1030844A1 Compounds which inhibit tryptase activity |
| 08/30/2000 | EP1030840A1 Cyclic amine derivatives and their use as drugs |
| 08/30/2000 | EP1030662A2 Treatment of t-helper cell type 2 mediated immune diseases with retinoid antagonists |
| 08/30/2000 | CN1264704A Novel spiro imidazoline compounds, their prepn. method and medicinal compsns. containing same |
| 08/29/2000 | US6110944 LTA4, hydrolase inhibitors |
| 08/29/2000 | US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds |
| 08/29/2000 | US6110906 Androgen derivatives for use in the inhibition of sex steroid activity |
| 08/24/2000 | WO2000049005A1 Bicyclic compounds and their use as integrin receptor ligands |
| 08/24/2000 | CA2362862A1 Bicyclic compounds and their use as integrin receptor ligands |
| 08/23/2000 | EP1029861A1 Benzisothiazol-piperazinyl derivative and its use as neuroleptic |
| 08/23/2000 | EP1028953A1 Aromatic heterocyclic compounds as anti-inflammatory agents |
| 08/23/2000 | EP0820447B1 Process for making 2-aryl benz(ox, thi, imid)azoles and 2-aminoaryl aminobenz(ox, thi, imid)azoles |
| 08/23/2000 | CN1264385A Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and compositions containing same |
| 08/23/2000 | CN1264367A Nitrophenyl-sulfonyl-imidazoles and use thereof for controlling vegetable and animal pests |
| 08/23/2000 | CN1263887A Benzimidazole derivative and hair maintaining agent, skin external use agent |
| 08/22/2000 | US6107329 Hypotensive agents; cardiovascular disorders |
| 08/16/2000 | EP1028112A1 Phenylglycinolamides linked by a hetero-atom with antiatherosclerotic agents |
| 08/16/2000 | EP1028111A1 Amide derivatives or salts thereof |
| 08/16/2000 | EP1026950A1 Treatment of schizophrenia with ampakines and neuroleptics |
| 08/16/2000 | CN1055469C Optically pure salts of pyridinylmethyl sulfinyl-1H-benzimidazole compounds, its preparing method and use |
| 08/16/2000 | CN1055465C Optical active 2-imidazoline-5-thione derivatives and preparating method and use thereof |
| 08/15/2000 | US6103747 Substituted imidazole derivative used as antagonists against muscarinic acetylcholine receptor on smooth muscles, treats dysuria |
| 08/15/2000 | US6103745 Useful for high fungicidal, insecticidal and acaricidal activity |
| 08/15/2000 | US6103744 Administering to the patient a dopamine autoreceptor agonists for the treatment of schizophrenia, parkinson,s disease, tourette,s syndrom, alcoholism and drug addiction |
| 08/15/2000 | US6103736 Showing an inhibitory action on gastric acid secretion and a protective action of gastric mucosa; 2-(hetero)aryl-3-aminoimidazo-(2,1-a)isoquinolines; antiulcer agents; |
| 08/10/2000 | WO1999063936A9 Novel therapeutic agents that modulate endothelin receptors |
| 08/08/2000 | US6100404 Erythromycin compounds |
| 08/08/2000 | US6100283 Prodrug phosphate derivative for poly (adp-ribose) polymerase enzyme inhibitor for administering in conjunction with antitumor drug or radiotherapy |
| 08/08/2000 | US6100264 5H, 10H-imidazo [1,2-A] indeno [1,2-E] pyrazin-4-one derivatives, their preparation, their intermediates and medicaments containing them |
| 08/03/2000 | WO2000044709A2 ACETYLENIC α-AMINO ACID-BASED SULFONAMIDE HYDROXAMIC ACID TACE INHIBITORS |
| 08/03/2000 | DE19903126A1 New sulphur substituted sulphonylaminocarboxylic acid N-arylamide derivatives used for treating e.g. cardiovascular diseases and atherosclerosis |
| 08/03/2000 | DE19901921A1 Polymorphe von Telmisartan, Verfahren zu deren Herstellung und deren Verwendung zur Herstellung eines Arzneimittels Polymorphs of telmisartan, to processes for their preparation and their use for the preparation of a medicament |
| 08/03/2000 | CA2356299A1 Acetylenic .alpha.-amino acid-based sulfonamide hydroxamic acid tace inhibitors |
| 07/27/2000 | WO2000043371A2 Fused ring heteroaryl and heterocyclic compounds which inhibit leukocyte adhesion mediated by vla-4 |
| 07/27/2000 | WO2000043370A1 Telmisartan polymorphs, methods for producing same and their use in the preparation of a medicament |
| 07/27/2000 | WO2000018767A3 2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands |
| 07/27/2000 | WO1999066944A9 Methods for identifying novel multimeric agents that modulate receptors |
| 07/27/2000 | WO1999064033A9 Phosphodiesterase-v modulator drugs and their uses |
| 07/27/2000 | WO1999063994A9 MULTIBINDING INHIBITORS OF HMG-CoA REDUCTASE |
| 07/27/2000 | WO1999057098A3 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2 |
| 07/27/2000 | CA2359112A1 Fused ring heteroaryl and heterocyclic compounds which inhibit leukocyte adhesion mediated by vla-4 |
| 07/26/2000 | EP1022272A1 Substituted fused heterocyclic compounds |
| 07/26/2000 | EP1021199A1 PEPTIDE-CONTAINING $g(a)-KETOAMIDE CYSTEINE AND SERINE PROTEASE INHIBITORS |
| 07/26/2000 | EP1021188A1 Inhibitors of prenyl-protein transferase |
| 07/25/2000 | US6093735 Selective β-3 adrenergic agonists |
| 07/25/2000 | US6093734 Pyridyl methyl sulfinyl benzimidazole type proton pump inhibitor drugs having a hydrolyzable sulfinyl or arylsulfonyl group attached to the benzimidazole nitrogen; gastrointestinal disorders |