Patents
Patents for C07D 235 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings (15,325)
07/2001
07/26/2001WO2001053272A1 Human chymase inhibitors
07/26/2001WO2001053258A1 Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
07/26/2001WO2001052847A1 Thiazole, imidazole and oxazole compounds and treatments of disorders associated with protein aging
07/26/2001US20010009919 Tris benzimidazoles; fungicides, anticarcinogenic agents, enzyme inhibitor
07/26/2001CA2398409A1 Nitrogen-containing cyclic compound and pharmaceutical composition containing the compound
07/26/2001CA2397627A1 Thiazole, imidazole and oxazole compounds and treatments of disorders associated with protein aging
07/26/2001CA2365118A1 Inhibitor against human chymase activity
07/25/2001EP1117663A2 2-piperazino alkylamino benzoazole derivatives: dopamine receptor subtype specific ligands
07/25/2001EP1117651A1 New bis-benzimidazoles
07/25/2001EP1117638A1 Biphenyl compounds substituted by camphor or hydantoin derivatives as sunscreen compositions
07/25/2001EP1117397A1 Geometrically restricted 2-indolinone derivatives as modulators of protein kinase activity
07/25/2001CN1305464A Heterocyclic compounds and methods to treat cardiac failure and other disorders
07/25/2001CN1305454A Anthranilic acid derivatives as inhibitors of CGMP phosphodiesterase
07/24/2001US6265581 Reacting specified epoxide and amine, reacting product with acid to form acid addition salt
07/24/2001US6265415 Compounds for inhibition of gastric acid secretion
07/19/2001WO2001051487A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
07/19/2001WO2001051473A1 1,2-diaryl benzimidazoles for treating illnesses associated with a microglia activation
07/19/2001WO2001051456A2 Antibacterial agents
07/19/2001WO2001044172A8 Salicylamides as serine protease and factor xa inhibitors
07/19/2001WO2000076970A3 Serine protease inhibitors
07/19/2001US20010008944 Reacting 3-alkoxy/hydroxy-2-halo-cycloheptenone derivative with alkylamidine hydrochloride to form cycloheptimidazole-8-one compound
07/19/2001CA2397575A1 Antibacterial agents
07/19/2001CA2396087A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
07/18/2001EP0850221B1 Meta-guanidine, urea, thiourea or azacyclic amino benzoic acid derivatives as integrin antagonists
07/18/2001CN1304400A Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
07/17/2001US6262295 Process for the preparation of a racemic or optically active 4-(hydroxymethyl)-2-cyclopentene derivative
07/17/2001US6262100 Nitrophenyl-sulfonyl-imidazoles and use thereof for controlling vegetable and animal pests
07/17/2001US6262095 Use of tricyclic derivatives of 1,4-dihydro-1,4-dioxo-1H-naphthalene, novel compounds obtained and their application in theraphy
07/17/2001US6262090 Aminopyridine-containing thiourea inhibitors of herpes viruses
07/17/2001US6262086 6-methoxy-2-(((4-methoxy-3, 5-dimethyl-2-pyridinyl)methyl)sulfinyl)-1h-benzimidazole; antisecretory agents
07/17/2001US6262085 Alkoxy substituted Benzimidazole compounds, pharmaceutical preparations containing the same, and methods of using the same
07/17/2001US6262066 High affinity ligands for nociceptin receptor ORL-1
07/11/2001CN1303377A Amino piperidine derivatives as integrin alpha beta 3 antagonists
07/11/2001CN1303281A Use of compounds for elevation of pyruvate dehydrogenase activity
07/10/2001CA2139653C Optically pure salts of pyridinylmethyl sulfinyl-ih- benzimidazole compounds
07/05/2001WO2001047898A2 Substituted piperazine derivatives and their use as inhibitors of the microsomal triglyceride transfer protein (mtp)
07/05/2001WO2001047896A1 Benzimidazoles, production thereof and the use thereof as antithrombotic
07/05/2001WO2001047883A1 Fused-ring compounds and use thereof as drugs
07/05/2001US20010006977 E.g., 2-(amindinophenylaminomethyl)-1-methyl-5-(1-(ethoxy-carbonyl-methylamino)-1 -(2,5-dihydropyrrolocarbonyl)-ethyl)benzimidazole; anticoagulants and antithrombolytic agents
07/05/2001CA2395249A1 Substituted piperazine derivatives, the preparation thereof and their use as medicaments
07/05/2001CA2393916A1 Benzimidazoles, the preparation thereof and their use as pharmaceutical compositions
07/05/2001CA2363274A1 Fused-ring compounds and use thereof as drugs for hepatitis c
07/04/2001EP1113332A1 Photographic element, compound, and process
07/04/2001EP1112269A2 Hiv protease inhibitors
07/04/2001EP1111993A1 Fused-benzene derivatives useful as herbicides
07/04/2001CN1302287A Bioreductive cytotoxic agents
07/04/2001CN1301702A Internmediate of anti viral medicine, their preparation and use
07/03/2001US6255494 Substituted benzimidazoles useful in treating or preventing conditions associated with excess of neuropeptide y (around arteries in heart, respiratory tract, gastrointestinal tract and genitourinary tract); etiology of psychiatric disorders
07/03/2001US6255091 Potentiating metal mediated serine protease inhibitors with cobalt or zinc ions
06/2001
06/28/2001WO2001045704A1 Inhibitors of prenyl-protein transferase
06/28/2001WO2000066104A3 Ace-2 inhibiting compounds and methods of use thereof
06/28/2001WO1999063937A9 Multivalent macrolide antibiotics
06/28/2001US20010005752 Mixing an arylsubstituted indazole compound labelled molecule with binding molecule, selectively detecting a binding event with arylsubstituted indazole labelled compound and binding molecule by fluorescence spectroscopy
06/28/2001DE19962329A1 New substituted 2-(phenylaminomethyl)-benzimidazoles, used as thrombin inhibitors, serine protease inhibitors, antithrombotic agents and intermediates
06/27/2001EP1109555A1 Novel angiogenesis inhibitors
06/27/2001EP1109552A1 Novel dna-cleaving antitumor agents
06/27/2001EP0733046B1 benzoyl guanidines, their production and their use in medicaments
06/27/2001CN1301156A Treatment of T-Helper cell tyre 2 mediated immune diseases with retinoid antagonists
06/27/2001CN1301154A Amide derivatives and nociceptin antagonists
06/26/2001US6252112 Process for the preparation of an enantiomer of a (1R, 4S) or (1S, 4R)-1-amino-4-(hydroxymethyl)-2-cyclopentene derivative
06/26/2001US6252104 3,6-disubstituted-2-oxynaphthalene derivatives; raw materials for synthesis of such materials as dyes, pigments, photosensitive materials
06/26/2001US6251689 Methods for the solid phase synthesis of combinatorial libraries of benzimidazoles benzoxazoles benzothiazoles and derivatives thereof
06/21/2001WO2001044223A1 Inhibitors of interleukin 5 gene expression
06/21/2001WO2001044172A1 Salicylamides as serine protease and factor xa inhibitors
06/21/2001US20010004669 For treatment of depression, anxiety, eating disorders, obesity, drug abuse, cluster headache, migraine, pain and chronic paroxysmal hemicrania and headache associated with vascular disorders
06/21/2001CA2394654A1 Proton pump inhibitors
06/21/2001CA2394639A1 Salicylamides as serine protease and factor xa inhibitors
06/21/2001CA2393027A1 Inhibitors of interleukin 5 gene expression
06/20/2001EP1107944A1 Aminoalcohol derivatives and their use as beta 3 adrenergic agonists
06/20/2001EP1107753A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht2 receptors
06/20/2001CN1300277A Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
06/19/2001US6248770 Cardiovascular disorders
06/14/2001WO2001042224A1 Carboxyamido derivatives
06/14/2001WO2001042199A1 Amidinophenylpyruvic acid derivative
06/14/2001WO2001002340A3 Novel aminoindanes
06/14/2001US20010003744 Therapeutic compounds
06/13/2001EP1105387A1 Prodrugs of proton pump inhibitors
06/13/2001CN1299358A Heterocyclic Topoisomerase poisons
06/13/2001CN1067060C Amino acid derivative, process for producing same, agrohorticultural fungicide, and fungicidal method
06/07/2001WO2001039773A1 Thrombopoietin mimetics
06/07/2001WO1999063940A3 INHIBITORS OF H+K+-ATPase
06/06/2001CN1298404A Inhibitors of phospholipase A2
06/06/2001CN1066729C Benzimidazole derivatives, their producing process and its therapeutic use
06/05/2001US6242644 N-(4-carbamimidoyl-phenyl)-glycine derivatives
06/05/2001US6242494 Angiogenesis inhibitors, antitumor agents, diabetic retinopathy, and antiinflammatory agents
06/05/2001US6242445 Curative effects for cardiac and nephric diseases, although having little action on blood-pressure.
06/05/2001US6242422 (Substituted)Acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
06/05/2001CA2059647C Thiocylating reagents and intermediates, thiopeptides, and methods for preparing and using same
05/2001
05/31/2001WO1999064041A9 Multibinding agents that modulate nmda receptors
05/30/2001EP1102597A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht 4 receptors
05/29/2001US6239286 Reacting 1-amino-1-cyanocyclopentane with an acyl halide; then an anhydride
05/29/2001US6239138 Vitronectin receptor antagonist
05/29/2001US6239076 Such as 3-chloro-2-(4-chloro-5-(3-phenyl-5-methylisoxazolin-5-yl)methoxy-2 -fluorophenyl)-4,5,6,7-tetrahydro-2h-indazole; herbicides for controlling rice paddy weeds
05/25/2001WO2000077027A3 Serine protease inhibitors
05/25/2001WO2000039081A3 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
05/24/2001US20010001799 Anticoagulant
05/23/2001EP1100805A1 Medicine nitrate salts
05/23/2001EP1100795A1 Disubstituted bicyclic heterocycles having, in particular, a thrombin inhibitive effect
05/23/2001EP1100781A1 High affinity ligands for nociceptin receptor orl-1
05/23/2001EP1100763A1 Diketoacid-derivatives as inhibitors of polymerases