Patents
Patents for C07D 235 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings (15,325)
07/2002
07/11/2002WO2002024632A3 Substituted aminopropoxyaryl derivatives useful as agonists for lxr
07/11/2002WO2001024785A3 Dihydroorotate dehydrogenase inhibitors for the treatment of viral-mediated diseases
07/11/2002US20020091089 (Substituted)acyl dipeptidyl inhibitors of the ICE/ced-3 family of cysteine proteases
07/10/2002EP1221441A2 LTA4 Hydrolase inhibitors
07/10/2002EP1221314A1 New crystalline form of omeprazole
07/10/2002EP1220845A1 Aryl-sulfonamide substituted benzimidazol derivatives and use of said as tryptase inhibitors
07/10/2002EP1220844A1 Aryl sulfonamide-substituted benzimidazol derivatives thereof as tryptase inhibitors
07/10/2002EP1220836A2 Benzylcycloalkyl amines as modulators of chemokine receptor activity
07/10/2002CN1358176A Method for producing 2-heterocyclyl methyl benzoic acid derivatives
07/10/2002CN1358169A N-alkoxyalkyl-N,N-dialkylamine derivatives or salts thereof, and remedies for nerve degeneration diseases containing the same
07/10/2002CN1358094A Method for treating chronic pain using MEK inhibitors
07/10/2002CN1087285C Basic group substituted benzoyl guaniazine, its preparing process, its use as medicine or diagnostic reagent, and medicine containing the same
07/10/2002CN1087283C New LH-RH antigonists with improved effectiveness
07/09/2002CA2211444C New benzimidazol, benzoxazol and benzothiazol derivitives, the procedure for preparing them and the pharmaceutical compositions which contain them.
07/04/2002WO2002051831A1 Oxybenzamides derivatives as factor xa inhibitors
07/04/2002WO2002051810A2 Integrin receptor ligands
07/04/2002US20020086887 N-Acylsulfonamide apoptosis promoters
07/03/2002EP1219607A1 Integrase inhibitors containing aromatic heterocycle derivatives
07/03/2002EP1218352A1 Benzimidazolone derivatives having mixed serotonine and dopamine receptors affinity
07/03/2002CN1356987A Novel benzimidazole derivatives and pharmaceutical compsns. comprising these compounds
07/03/2002CN1356986A Spiroimidazolidine derivatives, their prepn. their use and pharmaceutical prepns. comprising them
07/03/2002CN1356977A Glucagon antagonists/inverse agonists
07/03/2002CN1356971A Intermediates and process for producing fluorine-contg. amino acid compound by using same
07/03/2002CN1356899A IL-8 receptor antagonists
07/02/2002US6414011 Central nervous system disorders
07/02/2002US6414008 Disubstituted bicyclic heterocycles, the preparation thereof, and their use as pharmaceutical compositions
07/02/2002US6413990 Antiinflammatory agents, antiallergens
06/2002
06/27/2002WO2002050039A1 Urea and urethane derivatives as integrin inhibitors
06/27/2002WO2002049993A2 High affinity small molecule c5a receptor modulators
06/27/2002WO2002024613A3 Resorcinol derivatives
06/27/2002US20020082429 Process for the preparation of phenylene-bis-benzimidazole-tetrasulfonic acid disodium salt
06/27/2002US20020082425 Aryl and heteroaryl fused aminoalkyl-imidazole derivatives
06/27/2002US20020082280 Method of inhibiting neoplastic cells with benzimidazole derivatives
06/27/2002DE10051318A1 New N-substituted phenyethanolamine derivatives, useful as beta-mimetics having a long duration of action, e.g. for treating asthma, chronic obstructive pulmonary disease or arrhythmia
06/26/2002EP1217000A1 Inhibitors of factor Xa and factor VIIa
06/25/2002US6410743 (1s,2s)-2-(2-(n-((3-benzoimidazol-2-yl)propyl)-n-methylamino)ethyl)-6 -fluoro-1,2,3,4-tetrahydro-1-isopropyl-2-naphthyl cyclopropanecarboxylate, for example; treating vascular disease such as gangrene, retinopathy, nephropathy
06/25/2002US6410742 Polymorphs of telmisartan
06/25/2002US6410566 Cyclic amine derivatives and their use as drugs
06/25/2002US6410561 Analgesics
06/25/2002CA2217952C A pharmaceutical composition containing benzimidazole for inhibiting the growth of cancers
06/20/2002WO2002040019A8 Benzimidazole derivatives
06/20/2002WO2002030894A3 Compositions and methods of the use thereof achiral analogues of cc-1065 and the duocarmycins
06/20/2002WO2002020495A3 Inhibitors of glycogen synthase kinase 3
06/20/2002WO2002012214A3 Non-imidazole aryloxyalkylamines as h3 receptor ligands
06/20/2002US20020077483 Preparing a azole compound on a solid support resin, cleaving the compound from the solid support resin by nucleophilic substitution to further substituting by alkylation reaction
06/20/2002US20020077329 EP4 receptor inhibitors to treat rheumatoid arthritis
06/20/2002DE10063173A1 Harnstoff- und Urethanderivate Urea and urethane
06/20/2002DE10060292A1 Verwendung substituierter Benzimidazole zur Herstellung eines Medikaments zur Behandlung von Krankheiten, welche durch Inhibierung des Na+/H+-Austauschers beeinflusst werden können und sie enthaltendes Medikament Use of substituted benzimidazoles for the manufacture of a medicament for the treatment of diseases which can be influenced by inhibiting the Na + / H + exchanger and containing medicament
06/20/2002DE10059254A1 Verfahren zur Herstellung von Phenylen-bis-benzimidazol-tetrasulfonsäure-di-natriumsalz Process for preparing phenylene-bis-benzimidazole tetrasulfonic acid disodium salt
06/19/2002EP1214318A1 Imidazo[1,2-a]pyridine and pyrazolo[2,3-a]pyridine derivatives
06/19/2002EP1214292A1 Tyrosine derivatives
06/19/2002CN1086386C Multi-drug resistance modifier
06/18/2002US6407131 5-carbonyloxy-1h-benzimidazole-2-carbamate derivatives
06/18/2002US6407130 Antiallergens, antiinflammatory and antiarthritic agents; respiratory system, gastrointestinal disorders
06/18/2002US6407105 Compounds and methods for use thereof in the treatment of cancer or viral infections
06/18/2002CA1341370C Fused polycyclic compounds, methods of manufacture, and their use as paf antagonists, antihistamines and/or antiinflammatory agents
06/13/2002WO2002046173A1 Fused heteroaromatic glucokinase activators
06/13/2002WO2002046169A1 Substituted 2-anilino-benzimidazoles and the use thereof as nhe-inhibitors
06/13/2002WO2002046168A1 Therapeutic benzimidazole compounds
06/13/2002WO2002046129A2 Inhibitors of histone deacetylase
06/13/2002WO2002015891A3 Pharmaceutical combination of angiotensin ii antagonists and ace inhibitors
06/13/2002DE10041671C1 Verfahren zur Herstellung von Imidazo[1,2-c][2,3]benzodiazepinen sowie Phenylessigsäureester und Oxazol-Derivate als Zwischenprodukte bei deren Herstellung Benzodiazepines process for the preparation of imidazo [1,2-c] [2,3] oxazole and phenylacetic acid esters and derivatives, as intermediates in the preparation thereof
06/13/2002CA2430412A1 Substituted 2-anilino-benzimidazoles and the use thereof as nhe-inhibitors
06/12/2002EP1212296A1 Phosphate mimics and methods of treatment using phosphatase inhibitors
06/12/2002EP1212269A1 Methods for preparing n- (aliphatic or aromatic)carbonyl)]-2-aminoacetamide compounds and for cyclizing such compounds
06/12/2002EP0984778B1 Neuropeptide-y ligands
06/12/2002EP0885210B1 Tricylic compounds having binding affinity for melatonin receptors, their production and use
06/12/2002CN1353695A Heterocyclically substituted benzimidazoles, production and application thereof
06/12/2002CN1353694A Alpha-substituted carboxylic acid derivatives
06/12/2002CN1353693A Substituted phenylcyclohexane carboxylic acid amides and their use as adenosine uptake inhibitors
06/12/2002CN1353605A Aryl substituted pyrazoles, imidazoles, oxazoles, thiazoles and pyrroles, and use thereof
06/11/2002US6403587 Autoimmune diseases, acute and chronic inflammatory conditions, allergic conditions, infection associated with inflammation, viral, transplantation tissue rejection, atherosclerosis, restenosis, hiv infectivity, and
06/11/2002US6403585 α-and β-amino acid hydroxyethylamino sulfonyl urea derivatives useful as retroviral protease inhibitors
06/06/2002WO2002044156A2 Benzimidazole derivatives useful as tie-2 and/or vegfr-2 inhibitors
06/06/2002WO2002044155A1 Method for producing a phenylene-bis-benzimidazole-tetrasulfonic acid disodium salt
06/06/2002WO2002014294A3 Heterocyclic sulfonamide derivatives and their use for potentiating glutamate receptor function
06/06/2002US20020068721 Purine derivatives
06/06/2002CA2430274A1 Process for the preparation of phenylene-bis-benzimidazole-tetrasulphonic acid disodium salt
06/05/2002EP1210340A1 Substituted piperazine derivatives, the production thereof and their utilization as medicaments
06/05/2002EP1210336A1 Substituted benzimidazoles as non-nucleoside inhibitors of reverse transcriptase
06/05/2002EP1210335A1 Aminocarbonyl-substituted benzimidazole derivatives, method for producing same and the use thereof as medicaments
06/05/2002EP1210327A2 New vitamin d derivatives with cyclic substructures in the side chains, method and intermediates for their production and their use in the preparation of medicaments
06/05/2002EP0971920B1 Compounds for inhibition of gastric acid secretion
06/05/2002CN1085980C Meta-guanidine, urea, thiourea or azacyclic amino benzoic and derivatives as integrin antagaonists
06/04/2002US6399643 Spiroimidazolidine derivatives, their preparation, their use and pharmaceutical preparations formed therefrom
06/04/2002US6399642 Tris benzimidazoles; fungicides, anticarcinogenic agents, enzyme inhibitor
05/2002
05/30/2002WO2002043449A1 Luminescent element material and luminescent element comprising the same
05/30/2002WO2002042278A2 Imidazole and benzimidazole caspase inhibitors and uses thereof
05/30/2002WO2002042273A2 Acid derivatives useful as serine protease inhibitors
05/30/2002WO2002042262A2 Alkylthio- and aryl(heteroyl)thio-substituted p-phenylenediamines, their manufacture and their use in rubber
05/30/2002WO2002042248A2 Naphthalene derivatives
05/30/2002WO2002041886A1 Ydroxamic acid or n-formyl hydroxylamine derivatives as inhibitors of bakterial polypeptide deformylase for treating microbial infections
05/30/2002WO2002041835A2 Estrogen receptor modulators
05/30/2002WO2002020526A3 Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binding agents
05/30/2002WO2002014275A3 Heterocyclic sulfonamide derivatives and their use for potentiating glutamate receptor function
05/30/2002WO2001021160B1 Carboxymide and aniline derivatives as selective inhibitors of pathogens
05/30/2002US20020065418 Viral polymerase inhibitors
05/30/2002US20020065278 Non-imidazole aryloxyalkylamines
05/30/2002CA2429630A1 Imidazole and benzimidazole caspase inhibitors and uses thereof
05/30/2002CA2428191A1 Acid derivatives useful as serine protease inhibitors