Patents
Patents for C07D 235 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings (15,325)
09/2001
09/20/2001WO2001068591A1 Carboxylic acid derivatives as ip antagonists
09/20/2001WO2001068585A1 Novel amide compounds
09/19/2001EP1134213A2 Process for the preparation of substituted N-(indole-2-carbonyl)- glycinamides
09/19/2001EP1133477A1 Substituted benzimidazoles and their use as parp inhibitors
09/19/2001EP0880522B1 5H,10H-IMIDAZO[1,2-a]INDENO[1,2-e]PYRAZINE-4-ONE DERIVATIVES AMPA AND NMDA RECEPTORS ANTAGONISTS, PREPARATION THEREOF, INTERMEDIATES THEREOF AND DRUGS CONTAINING SAME
09/19/2001EP0538297B1 Antiviral tetrahydroimidazo 1,4]benzodiazepin-2-(thio)ones
09/19/2001CN1313846A C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cystenine proteases
09/19/2001CN1313766A DNA-cleaving antitumor agents
09/18/2001US6291678 Process for the preparation of chiral keto-heterocycles of basic amino acids
09/18/2001US6291503 β-phenylalanine derivatives as integrin antagonists
09/18/2001US6291499 2-cyclohexyl benzimidazole NMDA/NR2B antagonists
09/13/2001WO2001066526A1 Ester derivatives of dimethylpropionic acid and pharmacetuical compositions containing them
09/13/2001WO2000059886A3 Benzimidazole abd imidazolophyridine derivaties, their preparation and their use as selective modulators of bradykinin b2 (=bk-2) receptors
09/13/2001WO2000059883A3 Method for producing n-aryl-aza-heterocycles in the presence of cesium carbonate
09/13/2001US20010021775 Benzimidazolinones, benzoxazolinones, benzopiperazinones, indanones, and derivatives thereof as inhibitors of factor Xa
09/12/2001EP1132381A1 Ester derivatives of dimethylpropionic acid and pharmaceutical compositions containing them
09/12/2001EP1132087A1 Remedies for polycystic ovary syndrome
09/12/2001EP1131308A1 New piperazine and piperidine compounds
09/12/2001EP1131301A1 2-phenylbenzimidazoles and 2-phenylindoles, and production and use thereof
09/12/2001EP0888317B1 Substituted 4-hydroxy-phenylalcanoic acid derivatives with agonist activity to ppar-gamma
09/12/2001CN1312806A Prodrugs of proton pump inhibitors
09/11/2001US6288236 Benzimidazole compounds containing a benzoxazole or benzothiazole ring, and compositions and methods of use containing the same
09/11/2001US6288234 Fluorinated heterocyclic amido amine compounds as drugs
09/11/2001US6288231 Peptide-containing α-ketoamide cysteine and serine protease inhibitors
09/11/2001US6288100 Benzimidazole derivatives
09/11/2001US6288086 N-hydroxy-2-(alkyl, aryl, or heteroaryl, sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
09/11/2001US6288055 Analgesic agents
09/07/2001WO2001064676A2 INHIBITORS OF p38-α KINASE
09/07/2001WO2001064659A2 Indane derivatives and their use as cell adhesion inhibitors
09/07/2001WO2001010841A3 Fluorene derivatives as integrin inhibitors
09/06/2001US20010020021 Metalloprotease inhibitor
09/05/2001EP1130017A2 Azole derivatives and their use as superoxide radical inhibitors
09/05/2001EP0830345B1 Styryl benzimidazole derivatives as inhibitors of smooth muscle cell proliferation
09/05/2001CN1311777A High affinity ligands for nociceptin receptor ORL-1
09/05/2001CN1311679A Benzimidazole derivatives as modulators of IgE
09/05/2001CN1311675A Compounds having IgE affecting properties
09/05/2001CN1070489C Process for synthesis of substituted sulphoxides
09/05/2001CN1070368C Method for prepn. of pharmaceutical composition contg. imidazo [2,1-6] [3] benzoazepine derivatives
09/04/2001US6284759 2-piperazinoalkylaminobenzo-azole derivatives: dopamine receptor subtype specific ligands
09/04/2001CA2224062C Substituted n-(indole-2-carbonyl)-glycinamides and derivatives as glycogen phosphorylase inhibitors
08/2001
08/30/2001WO2001062741A1 Tetrahydronaphtalene derivatives and their use
08/30/2001WO2001062740A1 Mibefradil analogues and their use
08/29/2001EP1127880A2 Phenylacetic acid derivatives substituted by a heterocycle and their use as A-II antagonists and as inhibitors of smooth muscle cell proliferation
08/29/2001EP1127869A1 Novel compounds and medicinal use thereof
08/29/2001EP1127052A1 Substituted 2-phenylbenzimidazoles, the production thereof and their use
08/29/2001EP0889877B1 META-SUBSTITUTED PHENYLENE DERIVATIVES AND THEIR USE AS ALPHAvBETA3 INTEGRIN ANTAGONISTS OR INHIBITORS
08/29/2001CN1310721A Medicine nitrate salts
08/29/2001CN1310629A Coadministration of ACAT and MMP inhibitors for the treatment of atherosclerotic lesions
08/28/2001US6281363 Antiinflammatory agents; antiarthritic agents; autoimmune disorders
08/28/2001US6281237 N-phenyl benzimidazolecarboxamide and N-phenyl indolecarboxamide derivatives
08/28/2001US6281218 Benzimidazolone derivatives having mixed serotonin and dopamine receptors affinity
08/23/2001WO2001060803A1 Fused imidazolium derivatives
08/22/2001EP1124528A1 Multivalent macrolide antibiotics
08/22/2001CN1309633A Diacylhydrazine derivs. as integrain inhibitors
08/22/2001CN1309325A Photographic element, compound and method
08/21/2001US6278027 3-Substituted-2-halocycloheptenone compounds and a method for manufacturing same
08/21/2001US6277877 Substituted n-(indole-2-carbonyl)glycinamides and derivates as glycogen phosphorylase inhibitors
08/21/2001US6277849 N-sulphonyl and N-sulphinyl amino acid amides as microbiocides
08/21/2001US6277845 Hydrazono-benzazulene derivatives, pharmaceutical compositions and intermediates
08/21/2001CA2207348C Benzimidazole derivatives
08/21/2001CA2083606C Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use
08/16/2001WO2001058879A1 2-phenylcarbamoyl-benzimidazoles
08/16/2001WO2001058878A1 2-carboxamide-benzimidazoles useful in the treatment and prevention of ischemic reperfusion injury
08/16/2001WO2001058877A1 Interferon ω production potentiators
08/16/2001WO2001058853A1 Dehydroamino acids
08/16/2001WO2001010842A3 Melanocortin-4 receptor binding compounds and methods of use thereof
08/16/2001WO2001009096A3 Potassium channel openers
08/16/2001WO2000015212A3 Antifungal activity of dicationic molecules
08/16/2001EP1123272A1 (substituted)acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
08/16/2001EP0558677B1 Biologically active amines
08/16/2001CA2399799A1 2-phenylcarbamoyl-benzimidazoles
08/16/2001CA2399795A1 2-carboxamide-benzimidazoles useful in the treatment and prevention of ischemic reperfusion injury
08/16/2001CA2397993A1 Dehydroamino acids
08/15/2001CN1308622A Biphenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia
08/15/2001CN1308614A Benzimidazoles, production thereof and use thereof medicaments
08/15/2001CN1308608A Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
08/15/2001CN1308606A Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use pharmaceutical preparations comprising them
08/15/2001CN1308542A Sucoinamide inhibitors of interleukin-1& beta, converting enzyme
08/15/2001CN1308536A Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
08/15/2001CN1308534A Angiogenesis inhibitors
08/14/2001US6274600 Heteroatom substituted benzoyl derivatives that enhance synaptic responses mediated by AMPA receptors
08/09/2001WO2001056563A1 Adamantyl derivatives as anti-cancer agents
08/09/2001WO2000059878A3 INHIBITORS OF LFA-1 BINDING TO ICAMs AND USES THEREOF
08/08/2001EP1121342A1 Diaminopropionic acid derivatives
08/08/2001EP0965342B1 Preparation for percutaneous administration containing 6-amino-5-chloro-1-isopropyl-2-(4-methyl-1-piperazinyl)benzimidazole
08/07/2001US6271390 Suppression of the IgE-dependent allergic response by benzimidazole analogs
08/07/2001US6271340 Living free radical polymerization initiated by an alkoxyamine initiator or nitroxide
08/07/2001US6271249 Diphenyl imidazoles as potassium channel modulators
08/07/2001US6271241 Cycloalkyl and aryl fused aminoalkyl-imidazole derivatives: modulators and GLP-1 receptors
08/07/2001CA2213197C Certain bridged 4-phenyl-2-aminomethylimidazoles; new dopamine receptor subtype specific ligands
08/02/2001WO2000076971A3 Serine protease inhibitors
08/02/2001WO2000066564A8 Benzimidazolones and analogues and their use as progesterone receptor ligands
08/02/2001WO2000066175A3 Conjugates as therapies for cancer and prostate diseases
08/02/2001US20010011092 High affinity ligands for nociceptin receptor ORL-1
08/01/2001CN1069098C Novel imidazole derivative and process for producing same
07/2001
07/31/2001US6268508 For crop protection
07/31/2001US6268507 Hydantoin derivatives
07/31/2001US6268502 Process of synthesis of 5-methoxy- 2-[(4-methoxy-3,5-dimethy-2-pyridyl)methyl]sulfiny-1h-benzimidazole
07/31/2001US6268385 Dry blend pharmaceutical formulations
07/31/2001US6268313 Dihalopropene compounds, insecticidal/acaricidal agents containing same, and intermediates for their production