Patents for C07D 235 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings (15,325) |
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05/22/2003 | US20030096852 Inhibiting binding interaction between hGH (human growth hormone) or a mutant thereof and an hGH binding protein or receptor in mammal administering benzimidazole compound |
05/22/2003 | US20030096845 Alkoxy substituted benzimidazole compounds, pharmaceutical preparations containing the same, and methods of using the same |
05/22/2003 | US20030096826 Inhibitors of interleukin-1 beta converting enzyme and other cysteine proteases in the ICE family |
05/22/2003 | CA2466971A1 Benzimidazol- or indol-aminoacetonitrile derivatives for parasite control |
05/22/2003 | CA2464419A1 Benzimidazoles useful as protein kinase inhibitors |
05/21/2003 | EP1311512A1 Late transition metal complexes, their use as catalysts and polymers therefrom |
05/21/2003 | EP1311499A2 Bicyclic compounds as h3 receptor ligands |
05/21/2003 | EP1311489A1 Biphenyl derivatives and the use thereof as integrin inhibitors |
05/21/2003 | EP1311482A2 Non-imidazole aryloxypiperidines as h3 receptor ligands |
05/21/2003 | EP1311478A1 Novel thiourea compounds and the pharmaceutical compositions containing the same |
05/21/2003 | CN1418870A 3,4-dibidro-1H-anphthalene derivatives used as high selectivity inhibitor of cyclooxygenase-2 |
05/20/2003 | US6566566 Dimerization of a C6-12 olefin mixture in which the hexene isomer fraction has less than 30% by weight of linear isomers in the presence of a nickel catalyst; derivatization to give primary alcohols, and optional subsequent alkoxylation |
05/20/2003 | US6566533 Reacting aza-heterocyclic compounds (indoles and carbazoles) with alkyl- or aryl-halides in the presence of carbon dioxide and alkali carbonate |
05/20/2003 | US6566509 Compound for use as bactericide |
05/20/2003 | US6566381 For therapy of arthritis, cancer, cardiovascular disorder, skin disorder, ocular disorder, inflammation and gum disease |
05/20/2003 | CA2144962C 1-(2-oxo-acetyl)-piperidine-2-carboxylic acid derivatives as multi-drug-resistant cancer cell sensitizers |
05/20/2003 | CA2110693C Amino acid derivative anticonvulsant |
05/15/2003 | US20030092912 Brain disorders, anticonvulsants, antidepressants, drug abruse |
05/15/2003 | US20030092728 Antagonists of MCP-1 function and methods of use thereof |
05/14/2003 | EP1309577A2 Heterocyclic sulfonamide derivatives and their use for potentiating glutamate receptor function |
05/14/2003 | EP1309563A1 Heterocyclic-hydroxyimino-fluorenes and their use for inhibiting protein kinases |
05/14/2003 | EP1309562A1 4-alkoxy cyclohexane-1 amino carboxylic acid esters and method for the production thereof |
05/14/2003 | CN1418210A Carbocyclik side chain containing, N-substituted Metalloprotease inhibitors |
05/14/2003 | CN1418209A Carbocyclic side chain containing metalloprotease inhibitors |
05/14/2003 | CN1418191A Novel thiourea derivatives and the pharmaceutical compositions containing thd same |
05/14/2003 | CN1418187A Carboxylic acid derivatives as IP antagonists |
05/13/2003 | US6562972 Method for preparing quinoxaline-5- and 6-carboxylic acids (I) which comprises contacting an aqueous alkaline suspension of a 5- or 6-halomethyl quinoxaline (II) with oxygen in the presence of a transition metal catalyst, to form the |
05/13/2003 | US6562854 Compositions comprising a substituted benzimidazole useful for treating immunomediated inflammatory disorders |
05/13/2003 | US6562851 Antiinflammatory and antiasthmatic agents; inhibitors of alpha4 beta1 mediated cell adhesion |
05/08/2003 | WO2003037876A1 Crystalline sodium salt of telmisartan and the use of the same as an angiotensin antagonist |
05/08/2003 | US20030087945 Sulfonylaminocarboxylic acids |
05/08/2003 | US20030087943 2-phencycarbamoyl-benzimidazoles |
05/08/2003 | US20030087928 Novel anilide compounds and drugs containing the same |
05/08/2003 | US20030087306 Methods for identifying novel multimeric agents that modulate receptors |
05/07/2003 | EP1307460A1 Method for the production of imidazo-(1,2-c)(2,3)-benzodiazepines and intermediates in the production thereof |
05/07/2003 | EP0966454B1 Disubstituted bicyclic heterocycles, their production and use as medicaments |
05/07/2003 | EP0940387B1 Phenylethanolamine compounds useful as beta3 agonist, process for producing the same, and intermediates in the production of the same |
05/07/2003 | CN1107503C Optically pure compoun as medicinal use |
05/06/2003 | US6559308 The present invention relates to a method for preparing quinoxaline-5- and 6-carboxylic acids. The method comprises contacting an aqueous suspension of a 5- or 6-hydroxymethyl quinoxaline with oxygen in the presence of a transition metal |
05/06/2003 | US6559167 Prodrugs of the pyridyl methyl sulfinyl benzimidazole type proton pump inhibitor drugs have a hydrolyzable arylsulfonyl or heteroarylsulfonyl group attached to the benzimidazole nitrogen. The prodrugs of the invention hydrolyze under |
05/02/2003 | EP1306368A2 3,4-dihydro-1H-naphtalene derivatives as a highly selective cyclooxygenase-2 inhibitor |
05/02/2003 | EP1305300A1 Novel, slow-acting betamimetics, a method for their production and their use as medicaments |
05/02/2003 | EP1185516B1 Substituted phenylcyclohexane carboxylic acid amides that have an adenosine uptake inhibiting effect |
05/02/2003 | EP0963371B1 Substituted benzimidazoles as non-nucleoside inhibitors of reverse transcriptase |
05/02/2003 | EP0910563B1 Integrin receptor antagonists |
05/02/2003 | EP0724387B1 Angiotension ii receptor antagonists for the treatment of chronic anti-inflammatory diseases |
05/01/2003 | WO2003035602A1 Lipid modulators |
05/01/2003 | WO2003035072A1 Use of flibanserin in the treatment of sexual disorders |
05/01/2003 | US20030083518 Substituted alcohols useful in treatment of Alzheimer's disease |
05/01/2003 | US20030083517 Methods of preparing sulfinamides and sulfoxides |
05/01/2003 | US20030083504 N- (4-carbamimidoyl-phenyl) -glycine derivatives |
05/01/2003 | US20030083361 Naphtho(1,2-d)imidazole derivatives; treating thrombocytopenia |
05/01/2003 | US20030083315 Benzimidazole derivatives for treating an inflammatory disease, an allergy disease, a respiratory disease, a cardiovascular disorder or a bone disorder |
04/30/2003 | CN1414849A Carboxylic acid amides, medicaments containing these compounds and the use and preparation thereof |
04/24/2003 | WO2003033484A1 Substituted piperazine cyclohexane carboxilic acid amides and the use thereof |
04/24/2003 | WO2003032984A1 2-phenyl benzimidazoles and imidazo-[4,5]-pyridines as cdsi/chk2-inhibitors and adjuvants to chemotherapy or radiation therapy in the treatment of cancer |
04/24/2003 | US20030078431 Biheterocyclic compounds having high anticoagulant activity, used as inhibitors of factor Xa |
04/24/2003 | US20030078425 N-oxyl compound contained in an easily polymerizable material can be sufficiently decreased and loss of easily polymerizable material (acrylic or methacrylic acids or their esters) is little |
04/24/2003 | CA2463426A1 Substituted piperazine cyclohexane carboxilic acid amides and the use thereof |
04/23/2003 | EP1304110A2 Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors |
04/23/2003 | EP1303641A2 Method for recovery of copper from sulfidic ore materials using super-fine grinding and medium temperature pressure leaching |
04/23/2003 | EP1303493A1 Method for the production of n,n'-carbonyldiazoles and azolide salts |
04/23/2003 | EP1303483A1 Novel thiourea derivatives and the pharmaceutical compositions containing the same |
04/23/2003 | EP0844998B1 Halobenzimidazoles and their use as microbicides |
04/23/2003 | CN1413210A Non-peptidyl inhibitors of VLA-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases |
04/23/2003 | CN1413204A Method for producing therapeutic agents for ulcers |
04/23/2003 | CN1412183A New preparation method of timixatan |
04/22/2003 | US6552216 Molecular model for VLA-4 inhibitors |
04/22/2003 | US6552042 Anticoagulants |
04/22/2003 | CA2287054C 1,3,8-triazaspiro¬4,5|decanone compounds as orl1-receptor agonists |
04/17/2003 | WO2003031418A1 3,4-dihydro-1h-naphthalene derivatives as a highly selective cyclooxygenase-2 inhibitor |
04/17/2003 | WO2003031415A1 Mibefradil-based compounds as calcium channel blockers useful in the treatment of hypertension and angina |
04/17/2003 | WO2003030902A1 Imidazole derivates as anti-inflammatory agents |
04/17/2003 | WO2001094341A9 Quinazoline derivatives for the treatment of tumours |
04/17/2003 | WO1999064401A3 Imidazolyl derivatives and their use as somatostatin receptor ligands |
04/17/2003 | WO1999043212A3 Wood preservatives |
04/17/2003 | US20030073848 Accelerated process for preparing O-methyl phenols, N-methyl heteroaromatic compounds, and methylated aminophenols |
04/17/2003 | US20030073847 Dihalopropene compounds, insecticidal/acaricidal agents containing same, and intermediates for their production |
04/17/2003 | US20030073745 Apoptosis inducing adamantyl derivatives and their usage as anti-cancer agents, especially for cervical cancers and dysplasias |
04/17/2003 | US20030073731 Alkylation therapy; anticancer agent |
04/17/2003 | US20030073712 Antiinflamamtory agents; antiischemic agents |
04/17/2003 | US20030073699 Compounds and methods to treat cardiac failure and other disorders |
04/17/2003 | US20030073690 Controlling pain in mammals |
04/17/2003 | CA2462913A1 Mibefradil-based compounds as calcium channel blockers useful in the treatment of hypertension and angina |
04/16/2003 | EP1302468A1 Processes and intermediates for manufacturing retroviral protease inhibiting compounds |
04/16/2003 | EP1301488A1 Squaric acid derivatives containing a bicyclic heteroaromatic ring as integrin antagonists |
04/16/2003 | EP1301487A2 Viral polymerase inhibitors |
04/16/2003 | EP1301464A1 Biphenylcarboxylic acid amides, production thereof and use thereof as medicaments |
04/16/2003 | EP1094812A4 Angiogenesis inhibitors |
04/16/2003 | EP0972769B1 Novel amide derivatives and medicinal compositions thereof |
04/16/2003 | CN1411444A Vitronectin receptor antagonist bicyclic compounds, preparation method and compositions containing same |
04/16/2003 | CN1410047A Composition containing specific single cation monoazo dye for dyeing human cutin fiber |
04/16/2003 | CN1105716C Benzimidazole derivatives with antihistaminic activity |
04/15/2003 | US6548547 Sulfonylamino carboxylic acid N-arylamides as guanylate cyclase activators |
04/15/2003 | US6548505 Radioprotectors |
04/15/2003 | US6548502 Preventing disorder selected from pathological gambling, attention deficit disorder with hyperactivity disorder, substance addiction such as drug and alcohol and sex in a mammals by administering pyrido(1,2-a) pyrazine derivatives |
04/15/2003 | CA2097715C Indan derivatives |
04/10/2003 | WO2003029245A1 Spiro-hydantoin compounds useful as anti-inflammatory agents |
04/10/2003 | WO2003029211A1 Difluoroalkene derivative, pest control agent containing the same, and intermediate therefor |
04/10/2003 | WO2003029199A1 Benzene derivatives, process for preparing the same and use thereof |