Patents for C07D 235 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings (15,325) |
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12/25/2003 | US20030236252 Brain disorders, cardiovascular disorders, strokes, Parkinson's disease |
12/25/2003 | US20030236251 Hepatitis virus viricides |
12/24/2003 | WO2003106430A1 Benzimidazole inhibitors of poly(adp-ribosyl) polymerase |
12/24/2003 | WO2003105781A2 Ophthalmic compositions for treating ocular hypertension |
12/24/2003 | WO2003105779A2 Guanidine compounds as anesthetics and for treatment of nervous system disorders |
12/24/2003 | WO2003084916A3 Compounds that modulate ppar activity and methods for their preparation |
12/24/2003 | CA2488845A1 Opthalmic compositions containing selective m1 muscarinic agonists for treating ocular hypertension |
12/24/2003 | CA2487122A1 Guanidine compounds as anesthetics and for treatment of nervous system disorders |
12/23/2003 | US6667404 Retroviral protease inhibiting compounds |
12/23/2003 | US6667331 Non-peptidyl inhibitors of VLA-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases |
12/23/2003 | US6667324 Dry blend pharmaceutical formulations |
12/23/2003 | US6667323 Dry-blend pharmaceutical formulations |
12/23/2003 | US6667321 Alkoxy substituted benzimidazole compounds, pharmaceutical preparations containing the same, and methods of using the same |
12/23/2003 | US6667307 HIV protease |
12/23/2003 | US6667302 Heterocyclic topoisomerase poisons |
12/18/2003 | WO2003104209A1 Peptide deformylase inhibitors |
12/18/2003 | WO2003104203A1 Therapeutic molecules and methods-1 |
12/18/2003 | WO2003104195A1 4-(aryl or heteroaryl) -2-butylamine derivatives and their use as glucocorticoid ligans |
12/18/2003 | WO2003104178A1 Napththalene derivatives which inhibit the cytokine or biological activity of macrophage migration inhibitory factor (mif) |
12/18/2003 | WO2003103598A2 Amidine derivatives for treating amyloidosis |
12/18/2003 | WO2003103398A1 Insecticidal amides with nitrogen-containing benzo-fused bicyclic ring systems |
12/18/2003 | US20030232869 N3 alkylated benzimidazole derivatives as MEK inhibitors |
12/18/2003 | US20030232836 Secondary amides such as 2-(4-(2- methoxyphenyl)-1-piperazinyl )-N-(3-methylphenyl)acetamide, used for prophylaxis of impotency |
12/18/2003 | US20030232816 Benzimidazole derivatives |
12/18/2003 | US20030232810 Bicyclic cyclohexylamines and their use as nmda receptor antagonists |
12/18/2003 | US20030232808 Sulfonyl derivatives |
12/18/2003 | US20030232789 Salicylamides as serine protease and factor xa inhibitors |
12/18/2003 | US20030229950 Hair dyes |
12/18/2003 | CA2488493A1 Amidine derivatives for treating amyloidosis |
12/18/2003 | CA2487866A1 Napththalene derivatives which inhibit the cytokine or biological activity of macrophage migration inhibitory factor (mif) |
12/18/2003 | CA2487838A1 Methods and compounds for inhibiting the cytokine or biological activity of mif |
12/18/2003 | CA2486491A1 4-(aryl or heteroaryl)-2-butylamine derivatives and their use as glucocorticoid ligans |
12/17/2003 | EP1370682A2 Assay for identifying inhibitors of the rna dependent rna polymerase (ns5b) of hcv |
12/17/2003 | EP1370542A1 Bicyclic guanidine derivatives and therapeutic uses thereof |
12/17/2003 | EP1370540A1 Anti-thrombotic carboxylic acid amides, the production thereof and use of the same as medicaments |
12/17/2003 | EP1370538A1 Metalloproteinase inhibitors |
12/17/2003 | EP1370536A1 Metalloproteinase inhibitors |
12/17/2003 | EP1370535A1 Metalloproteinase inhibitors |
12/17/2003 | EP1370530A1 Acylated 1,2,3,4-tetrahydronaphthyl amines and their use as pharmaceutical |
12/17/2003 | EP1189889B1 Compositions and methods for inhibiting cell death |
12/17/2003 | CN1462303A Double-spiro organic compounds and electric-field luminescent devices |
12/17/2003 | CN1131032C Benzimidzole enteric coating preparation and preparing method thereof |
12/16/2003 | US6664353 Heterocyclic alkoxyamines as regulators in controlled radical polymerization processes |
12/11/2003 | WO2003101970A1 Imidazolium cxcr3 inhibitors |
12/11/2003 | WO2003028721A3 Substituted benzimidazole compounds and their use for the treatment of cancer |
12/11/2003 | WO2003024395A3 Linked biaryl compounds |
12/11/2003 | US20030229132 Small molecule modulators of apoptosis |
12/11/2003 | US20030229109 Vitronectin receptor antagonist bicyclic compounds, preparation method and compositions containing same |
12/11/2003 | US20030229102 Sulfonamide derivatives |
12/11/2003 | US20030229094 Acetamides and benzamides that are useful in treating sexual dysfunction |
12/11/2003 | US20030229093 Lipid diseases; metabolism diosrders; antiproliferative agents |
12/11/2003 | US20030229074 Metabolism; eating disorders; sexual disorders |
12/11/2003 | US20030229072 Cyclic and acyclic amidines and pharmaceutical compositions containing them for use as progesterone receptor binning agents |
12/11/2003 | US20030229065 Measuring drug resistance, calibration; reducing antibiotic resistance |
12/10/2003 | EP1368028A1 Benzimidazole compounds for modulating ige and inhibiting cellular proliferation |
12/10/2003 | EP0970046B1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors |
12/10/2003 | CN1461298A Compositions and methods of use thereof achiral analogues of CC-1065 and duocarmycins |
12/09/2003 | US6660870 Serotonergic compounds which possess agonist activity at 5-HT2 receptors effectively lower and control normal and elevated IOP and are useful for treating glaucoma |
12/09/2003 | US6660760 Heterocyclic aromatic compounds useful as growth hormone secretagogues |
12/09/2003 | US6660751 Sulfonamide derivatives as 5-HT7 receptor antagonists |
12/09/2003 | US6660742 Alkylation therapy; anticancer agent |
12/04/2003 | WO2003099823A2 1,3-diaza-dibenzoazulenes as inhibitors of tumour necrosis factor production and intermediates for the preparation thereof |
12/04/2003 | WO2003099814A1 Calcium receptor modulating agents |
12/04/2003 | WO2003099776A1 Calcium receptor modulating arylalkylamines |
12/04/2003 | WO2003099266A2 Acetamides and benzamides that are useful in treating sexual dysfunction |
12/04/2003 | WO2003075921A3 Mono- and bicyclic azole derivatives that inhibit the interaction of ligands with rage |
12/04/2003 | WO2003066673A8 Histogranin-like peptides and non-peptides, processes for their preparation and uses thereof |
12/04/2003 | WO2003027130A3 Transition metal complexes for preparing olefin oligomers |
12/04/2003 | US20030225285 Oxidizing a protected aminoalcohol to a chiral protected aminoaldehyde and diastereoselectively forming the aminoepoxide from said aminoaldehyde with an organometallic methylene-adding reagent in an appropriate solvent |
12/04/2003 | US20030225158 Compounds that modulate PPAR activity and methods for their preparation |
12/04/2003 | US20030225137 2-pyridinyl)-methyl)sulfinyl)-1H-benzimidazole derivatives |
12/04/2003 | US20030225136 Heterocyclic imines such as (5)6-methoxy-2-(((4-methoxy-3,5-dimethyl-2-pyridinyl)methyl)sulfinyl)-1H -benzimidazole and salts, used as antisecretory agents |
12/04/2003 | US20030225135 Dry-blend pharmaceutical formulations |
12/04/2003 | US20030225127 Heterocyclic sulfonamide derivatives |
12/04/2003 | US20030225074 E.g., 2-((4'-Methoxy(1,1'-biphenyl)-4-yl)sulfonyl)amino-4-hydroxy-5-((2 -thiazolyl)thio)-pentanoic Acid |
12/04/2003 | US20030225043 Especially for inhibiting type IV collagenase |
12/04/2003 | CA2487017A1 1,3-diaza-dibenzoazulenes as inhibitors of tumour necrosis factor production and intermediates for the preparation thereof |
12/04/2003 | CA2486564A1 Acetamides and benzamides that are useful in treating sexual dysfunction |
12/03/2003 | EP1367056A1 Drugs that enhance synaptic responses mediated by AMPA receptors |
12/03/2003 | EP1366766A1 Inhibitors of IMPDH enzyme |
12/03/2003 | CN1129583C Compound as intermediates for use in preparation of optically active 2-imidazoline-5-one or 2-imidazoline-5-thionone derivatives |
12/02/2003 | US6656956 Benzimidazole derivatives, processes for preparing them and their use as pharmaceutical compositions |
12/02/2003 | US6656954 Such as N-hydroxy-2-(((4-phenoxyphenyl)-sulfonyl)methyl) benzamide which inhibits matrix metalloprotease activity |
12/02/2003 | US6656945 6-heterocyclyl pyrazolo [3,4-d]pyrimidin-4-one cGMP-PDE inhibitors for the treatment of erectile dysfunction |
12/02/2003 | CA2246909C Method for chemical synthesis of oligonucleotides |
11/27/2003 | WO2003096980A2 Bicyclic modulators of androgen receptor function |
11/27/2003 | WO2003024899A3 CYCLIC HYDROXAMIC ACIDS AS INHIBITORS OF MATRIX METALLOPROTEINASES AND/OR TNF-α CONVERTING ENZYME (TACE) |
11/27/2003 | WO2003014064A8 Naphthylurea and naphthylacetamide derivatives as vanilloid receptor 1 (vr1) antagonists |
11/27/2003 | US20030220521 A conjugate compound comprising an antagonist of adrenergic neurotransmitter, and second residue is capable of being cleaved by a kidney enzyme; sodium channel modulators, hypotensive agents |
11/27/2003 | US20030220372 Imidazole compounds as anti-inflammatory and analgesic agents |
11/27/2003 | US20030220369 Heterocyclic sulfonamide derivatives and their use for potentiating glutamate receptor function |
11/27/2003 | US20030220367 Administering a therapeutical carbamate derivative to a patient as prostaglandin IP (12 or PGI2) antagonists |
11/27/2003 | US20030220350 For example, 3-(4-((N-(5-chlorobenzo(B)thiophen-3-carbonyl)-N-(2,2-diphenyl ethyl)amino)methyl)benzoylamino)propionic acid; for treatment or prevention of glucagon-mediated diseases such as diabetes |
11/27/2003 | US20030220341 Chemokine receptor binding heterocyclic compounds with enhanced efficacy |
11/27/2003 | US20030220326 Compounds, pharmaceutical compositions, and methods for inhibiting cyclin-dependent kinases |
11/26/2003 | EP1364945A1 Benzimidazolidinone derivatives |
11/26/2003 | EP1363890A2 Melanocortin-4 receptor binding compounds and methods of use thereof |
11/26/2003 | EP1363873A2 Peptide deformylase inhibitors |
11/26/2003 | EP0828487B1 Agents for use against parasitic protozoa |
11/26/2003 | CN1458922A Urea derivative and adhesive-molecule inhibitor containing same as ctive ingredient |