Patents for C07D 235 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings (15,325) |
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02/04/2004 | EP1385820A1 Anthranilic acid amides, method for the production thereof, their use as antiarrhythmia agents, and pharmaceutical preparations thereof |
02/04/2004 | CN1473153A Hetero-anellated ortho-aminophenols |
02/04/2004 | CN1473150A Bis-heterocyclic compounds with antitumour and chemosensitising activity |
02/03/2004 | US6686493 Antiproliferation agent; antiinflammatory agents; side effect reduction |
02/03/2004 | US6686474 Reacting benzimidazole compound with m-chloroperoxybenzoic acid in a solvent selected from the group consisting of acetone and acetone/water mixture; raising the ph of the reaction mixture; crystals are separated |
02/03/2004 | US6686384 2-anilinophenyl-substituted; inhibition of the na+/h+ exchanger |
02/03/2004 | US6686353 Diarylalkyl cyclic diamine derivatives as chemokine receptor antagonists |
02/03/2004 | US6686345 DNA-cleaving antitumor agents |
02/03/2004 | CA2092510C Crystalline forms of endo-2,3-dihydro-n-(8-methyl-8-azabicyclo-[3.2.1.]oct-3-yl)-2-oxo-1h-benzimidazole-1-carboxamide hydrochloride monohydrate and of endo-3 ethyl-2,3-dihydro-n-(8-methyl-8-azabicyclo[3.2.1.]oct-3-yl)-2-oxo-1h-benzimidazole-1-carboxamide hydrochloride monohydrate |
01/29/2004 | WO2004009017A2 Modulators of the glucocorticoid receptor and method |
01/29/2004 | WO2003066035A3 Compounds for inhibiting insulin secretion and methods related thereto |
01/29/2004 | US20040019216 Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds |
01/29/2004 | US20040019063 Nitrogen compounds such as 4-(7-Hydroxy-1,3-dioxo-tetrahydro-pyrrolo(1,2-c)imidazol-2-yl)-5,6,7,8-tetrahydronaphthalene-1-carbonitrile, used for prophylaxis of muscular disorders; aging |
01/29/2004 | US20040019058 Chemokine receptor binding heterocyclic compounds with enhanced efficacy |
01/29/2004 | US20040019041 Method for the production of imidazo-(1,2-C)(2,3)-benzodiazepines and intermediates in the production thereof |
01/28/2004 | EP1384715A1 Novel imidazolidinedione derivatives and use thereof as drugs |
01/28/2004 | EP1383757A1 Antagonists of mcp-1 function and methods of use thereof |
01/28/2004 | EP1383731A1 Biaryl compounds as serine protease inhibitors |
01/28/2004 | CN1136196C Crystalline forms of 3-(2,4-dichlorl benzyl)-2-methyl-N-(Pentylsulfonyc)-3H-benzimidzole-5-carboxamide |
01/28/2004 | CN1136193C Imide derivatives ar Salts thereof |
01/27/2004 | US6683648 Enzyme inhibitors such as 2s-(((dimethylamino)acetyl)amino)-n-(3-((((2-hydroxy-1,1 -dimethylethyl)amino)sulfonyl)(3-methyl butyl)amino)-2r-hydroxy-1s-(phenylmethyl)-propyl)-3,3-dimethyl butanamide, used for prohylaxis of viral diseases |
01/27/2004 | US6683215 N-(4-carbamimidoyl-phenyl)-glycine derivatives |
01/27/2004 | US6683191 Preparing a azole compound on a solid support resin, cleaving the compound from the solid support resin by nucleophilic substitution to further substituting by alkylation reaction |
01/27/2004 | US6683101 Such as 6-(3-(trans-4-phenylcyclohexylamino)propyl)-3h-benzoxazol-2-one; cerebral vascular disorders |
01/27/2004 | CA2292920C New spiroimidazolin derivatives, the process for preparing them and the pharmaceutical compositions that contain them |
01/27/2004 | CA2281927C Substituted benzimidazoles as non-nucleoside inhibitors of reverse transcriptase |
01/22/2004 | WO2004007500A1 Novel diketopyrrolopyrrole pigments |
01/22/2004 | WO2004007459A2 Naphthol, quinoline and isoquinoline-derivatives as modulators of vanilloid vr1 receptor |
01/22/2004 | WO2004007455A1 Heterocyclically substituted benzoylureas, method for their production and their use as medicaments |
01/22/2004 | WO2003080545A3 Substituted phenylacetic acids |
01/22/2004 | WO2003024395A8 Linked biaryl compounds |
01/22/2004 | US20040014758 Benzylcycloalkyl amines as modulators of chemokine receptor activity |
01/22/2004 | US20040014748 Cardiovascular disorders, central nervous susyem disorders |
01/22/2004 | DE10231105A1 Neue Diketopyrrolopyrrolpigmente New diketopyrrolopyrrole |
01/22/2004 | DE10210195A1 Derivate von Aza-Spiroverbindungen Derivatives of aza-spiro compounds |
01/22/2004 | CA2493374A1 Heterocyclically substituted benzoylureas, method for their production and their use as medicaments |
01/21/2004 | EP1382333A2 Use of beta 3 adrenergic receptor agonists in the treatment of dysuria |
01/21/2004 | CN1469870A A process for the preparation of bis-benzazolyl compounds |
01/21/2004 | CN1135224C Benzimidazole derivatives |
01/15/2004 | WO2004005513A2 Methods for specifically inhibiting histone deacetylase-7 and 8 |
01/15/2004 | WO2004005278A1 Bisarylsulfonamide compounds and their use in cancer therapy |
01/15/2004 | WO2004004703A1 m-PHENYLENEDIAMINE DERIVATIVE |
01/15/2004 | US20040010148 Antiinflammatory agents, antiallergens, antiproliferative agents, immunosuppressants, antidiabetic agents, cardiovascular disorders |
01/15/2004 | US20040010026 (R) 2-(4-amidinophenylaminomethyl)-1-methyl-5-[1-(carboxymethylamino)-1 (pyrrolidinocarbonyl)-ethyl]-benzimidazole, the monohydrochloride thereof, preparation thereof and the use as pharmaceutical composition |
01/15/2004 | US20040010023 Biphenyl derivatives and the use thereof as integrin inhibitors |
01/15/2004 | US20040009998 Spiro-hydantoin compounds useful as anti-inflammatory agents |
01/15/2004 | US20040009979 Use of compounds for the elevation of pyruvate dehydrogenase activity |
01/15/2004 | CA2490579A1 Methods for specifically inhibiting histone deacetylase-7 and 8 |
01/15/2004 | CA2488816A1 Bisarylsulfonamide compounds and their use in cancer therapy |
01/14/2004 | EP1380562A1 Carboxylic acid derivative and salt thereof |
01/14/2004 | EP1379527A1 Epindolidione pigments |
01/14/2004 | EP1379493A2 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses |
01/14/2004 | EP1379246A1 Nociceptin analogs |
01/14/2004 | EP1379242A1 Method for treatment of cancer and compositions for use therein |
01/14/2004 | CN1468227A Non-imidazole aryloxyalkylamines |
01/14/2004 | CN1468221A Non-imidazole aryloxypiperidines |
01/14/2004 | CN1134411C Bicyclic amino derivatives and PGD2 antagonist containing same |
01/13/2004 | US6677365 Antagonists of MCP-1 function and methods of use thereof |
01/13/2004 | US6677360 Biphenyl and biphenyl-analogous compounds as integrin antagonists |
01/13/2004 | US6676909 Method for recovery of metals from metal-containing materials using medium temperature pressure leaching |
01/08/2004 | WO2004002962A1 Novel benzimidazol-2-one derivatives and their use |
01/08/2004 | WO2004002530A1 Remedy for chronic disease |
01/08/2004 | US20040006236 Diaminopropionic acid derivatives |
01/08/2004 | US20040006162 For use as antidegradant in natural or synthetic rubber |
01/08/2004 | US20040006104 For therapy and prophylaxis of diseases and conditions associated with undesirable or abnormal inflammatory responses, such as ischemia-reperfusion injury, asthma, arthritis |
01/08/2004 | US20040006049 For therapy of prostatitis, benign prostate hyperplasia or prostate cancer |
01/08/2004 | DE10227666A1 (R)-2-(4-Amidinophenylaminomethyl)-1-methyl-5-[1-(carboxymethylamino)-1-(pyrrolidinocarbonyl)- ethyl]-benzimidazol, dessen Monohydrochlorid, Verfahren zu deren Herstellung sowie Verwendung als Arzneimittel (R) -2- (4-amidinophenylaminomethyl) -1-methyl-5- [1- (carboxymethylamino) -1- (pyrrolidinocarbonyl) - ethyl] -benzimidazole, its monohydrochloride, to processes for their preparation and use as medicaments |
01/07/2004 | EP1377549A1 Functionalized heterocycles as modulators of chemokine receptor function and methods of use therefor |
01/06/2004 | US6673257 Blends employing at least two organic compounds having known melt temperatures, exhibit improved thermal properties and performance characteristics |
01/06/2004 | US6673122 Compositions for dyeing keratin fibers containing para-aminophenols, dyeing process, novel para-aminophenols and process for their preparation |
01/02/2004 | EP1375486A1 Nitrogen-containing heteroaryl compounds having hiv integrase inhibitory activity |
01/02/2004 | EP1373283A1 Non-metallocenes, method for the production thereof and the use thereof for the polymerisation of olefins |
01/02/2004 | EP1373266A2 (diazolo-pyridinyl)-pyrimidines for use in treatment of cns disorders and diabetes |
01/02/2004 | EP1373220A1 Benzimidazoles that are useful in treating sexual dysfunction |
01/02/2004 | EP1373191A1 Acylated indanyl amines and their use as pharmaceuticals |
01/02/2004 | EP1044187B1 N-benzyl-3-indenylacetamides derivatives for treating neoplasia |
01/01/2004 | US20040002525 Obesity; osteoporosis |
01/01/2004 | US20040002524 Cardiovascular disorders; osteoporosis; central nervous system disorders |
01/01/2004 | US20040002512 Alpha-substituted carboxylic acid derivatives |
01/01/2004 | US20040002491 Melatonergic receptors |
01/01/2004 | US20040002490 Melatonergic receptors |
01/01/2004 | US20040002463 Inhibitors and methods of use thereof |
01/01/2004 | US20040001970 Organic electroluminescent materials and devices made from such materials |
12/31/2003 | WO2004000818A1 Crystalline (r)-2-(4-amidinophenylaminomethyl)-1-methyl-5-(1-(carboxymethylamino)-1(pyrrolidinocarbonyl)-ethyl)-benzimidazole, and the use thereof as antithrombotic agents |
12/31/2003 | WO2004000817A2 Benzimidazole compounds and their use as estrogen agonists/antagonists |
12/31/2003 | WO2004000256A1 Benzoxazole and benzodiazole uv-a sunscreens |
12/31/2003 | WO2003073979A3 Derivatives of azaspiro compounds for the treatment of pain |
12/31/2003 | WO2003063576A3 Arylsulfonamidobenzylic compounds |
12/31/2003 | WO2003060475A3 Melanin concentrating hormone receptor ligands: substituted 2-(4-benzyl-piperazin-1-ylmethyl)- and 2-(4-benzyl-diazepan-1-ylmethyl)-1h-benzoimidazole analogues |
12/31/2003 | CN1132832C Prepn process of 3-methyl-4 [(3-methoxy) propoxy]2-radical-methyl-thio-benzimidazole |
12/31/2003 | CN1132819C 作为TNF-α抑制剂的环状肼衍生物 Examples of the cyclic hydrazine derivative TNF-α inhibitors |
12/31/2003 | CA2487266A1 Benzimidazole compounds and their use as estrogen agonists/antagonists |
12/31/2003 | CA2485545A1 (r)-2-(4-amidinophenylaminomethyl)-1-methyl-5-(1-(carboxymethylamino)-1(pyrrolidinocarbonyl)-ethyl)-benzimidazole, the monohydrochloride thereof, preparation thereof and the use as pharmaceutical composition |
12/31/2003 | CA2445515A1 Transcription factor modulating compounds and methods of use thereof |
12/30/2003 | US6670445 Curable compounds, curable resin compositions containing the same and methods of easily disassembling cured materials |
12/30/2003 | US6668527 Non-peptidyl inhibitors of VLA-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases |
12/30/2003 | CA2052884C Angiotensin 11 antagonists in the treatment of hyperuricemia |
12/25/2003 | WO2003105853A1 1-aryl-4-substituted piperazines derivatives for use as ccr1 antagonists for the treatment of inflammation and immune disorders |
12/25/2003 | US20030236267 Benzimidazole derivatives |
12/25/2003 | US20030236260 Antiarthritic agents; autoimmune diseases; anticholesterol agents; cardiovascular disorders; antiinflammatory agents |