Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
10/2006
10/19/2006US20060234349 Fungal cell wall synthesis gene
10/19/2006US20060234283 reporter system reflecting the transport process that transports GPI-anchored proteins to the cell wall was constructed and compounds inhibiting this process were discovered; antifungal agents; inhibiting expression of cell wall glycoproteins and preventing pathogens from showing pathogenicity
10/18/2006CN1849117A Entry inhibitors of the HIV virus
10/17/2006US7122673 Cyclization of imines to form compounds such as 4-Phenyl-6H-(1)Benzopyrano(4',3':4,5)pyrrolo(2,1-a)isoquinolin-6-one, used as nontoxic modulators of multidrug resistant cells; antitumor agents
10/17/2006US7122672 N-alkynyl-2-quinolin-(isoquinolin- and quinazolin-)oxyalkylamides; treating agricultural and horticultural fungal infections of plants
10/17/2006US7122580 management, treatment and/or control of diseases caused in intrinsic clotting pathway utilizing factor IX such as stroke, myocardial infarction, aneurysm surgery, and deep vein thrombosis associated with surgical procedures etc
10/17/2006US7122559 Useful as anticoagulants in therapy and prophylaxis of cardiovascular diseases, as anti-inflammatory agents, and as metastasis inhibitors in therapy of cancer
10/17/2006CA2275686C Isoquinolinamine and phthalazinamine derivatives which interact with crf receptors
10/17/2006CA2197207C Hiv protease inhibitor combination
10/12/2006WO2006108107A1 Diarylamine-containing compounds and compositions, and their use as modulators of steroid hormone nuclear receptors
10/12/2006WO2006061217A3 Saquinavir derivatives useful in immunoassay
10/12/2006WO2006060225A3 Process for asymmetric synthesis of hexahydropyrimido[1,2-a] azepine-2-carboxamides and related compounds
10/12/2006WO2006020049A3 Aryl-and heteroaryl-substituted tetrahydroisoquinolines and use thereof to block reuptake of norepinephrine, dopamine, and serotonin
10/12/2006US20060229333 Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors
10/12/2006CA2603250A1 Diarylamine-containing compounds and compositions, and their use as modulators of steroid hormone nuclear receptors
10/11/2006EP1710238A1 Benzophenones as inhibitors of reverse transcriptase
10/11/2006EP1708999A1 Bronchorelaxing compounds
10/11/2006EP1708994A1 Aryloxyalkylcarbamate-type derivatives, preparation method thereof and use of same in therapeutics
10/11/2006EP1708698A1 3-(4-piperidine-1ylmethyl-phenyl)-propion acid-phenylamide-derivatives and related compounds used in the form of mch antagonists (melanine concentrating hormone) for treating eating disorders
10/11/2006EP1469851B1 Melanocortin receptor agonists
10/11/2006EP1216232B1 Heterocyclic compounds and methods for modulating cxcr3 function
10/11/2006CN1845740A Piperazine derivatives for the treatment of HIV infections
10/10/2006US7119103 β3-Adrenoreceptor agonists, agonist compositions and methods of using
10/10/2006CA2253407C Inorganic ion receptor-active compounds
10/05/2006WO2006105127A2 Hydroxysteroid dehydrogenase inhibitors
10/05/2006WO2006104141A1 3-propenylcephem derivative
10/05/2006WO2006102998A1 Substituted tetrahydroisochinolines as mmp inhibitors, related production method and use as medicine
10/05/2006WO2006102760A1 Inhibitors of histone deacetylase
10/05/2006WO2005115392A8 3-(4-heteroarylcyclohexylamino) cyclopentanecarboxamides as modulators of chemokine receptors
10/05/2006WO2004060308A3 Thiosemicarbazones as anti-virals and immunopotentiators
10/05/2006US20060223847 Anti-coronavirus drug
10/05/2006US20060220004 with Tris(2-bromo-6-pyridyl)phosphine oxide ligands; organic light-emitting diodes, integrated circuits, organic field-effect transistors, thin-film transistors, organic solar cells, and/or laser diodes
10/05/2006DE102005015040A1 Substituierte Tetrahydroisochinoline als MMP-Inhibitoren, Verfahren zu ihrer Herstellung und ihre Verwendung als Medikament Substituted tetrahydroisoquinolines as MMP inhibitors, to processes for their preparation and their use as a medicament
10/05/2006CA2603589A1 Inhibitors of histone deacetylase
10/05/2006CA2603345A1 New heterocyclic compounds, their preparation and their use as medicaments, in particular as anti-alzheimer agents
10/04/2006EP1372653B1 Acylated piperidine derivatives as melanocortin-4 receptor agonists
10/04/2006EP0906091B1 Amidinohydrazones as protease inhibitors
10/03/2006US7115743 For treatment of leukemia, carcinomas, adenocarcinomas, and melanoma; assaying metabolism via cytochromes
10/03/2006US7115664 Peptidomimetic ligands for cellular receptors and ion channels
10/03/2006US7115652 Aspartyl protease inhibitors
10/03/2006US7115646 Cyclic diamines and derivatives as factor Xa inhibitors
10/03/2006US7115607 Substituted piperazinyl amides and methods of use
10/03/2006US7115605 Peptide deformylase inhibitors
10/03/2006US7115600 Histamine-3 receptor modulators
09/2006
09/28/2006WO2006100100A1 Tetrahydronaphthalene derivatives, method for their production and their use as anti-inflammatory agents
09/28/2006US20060217416 Antihypoxic agents; adjust concentration of erythropoietin concentration in blood; strokes; antiepileptic agents; neurodegenerative disease ; liver disorders; antiischemic agents
09/28/2006US20060217384 e.g. 1-((3-Phenyl-1,2,4-triazolo(3,4-a)phthalazines-6-yl)carbonyl)piperidine; high affinity to the benzodiazepine site of GABAA receptors; central nervous system (CNS) diseases such as depression, anxiety, and attention deficit disorder
09/28/2006US20060217372 Diaryl ethers as opioid receptor antagonist
09/28/2006CA2598205A1 Tetrahydronaphthalene derivatives, process for their production and their use as anti-inflammatory agents
09/27/2006EP1704856A1 Hsp90 family protein inhibitor
09/27/2006EP1286967B1 Cyclohexane derivatives and their use as therapeutic agents
09/26/2006US7112586 Substituted diamine derivatives useful as motilin antagonists
09/21/2006WO2006099060A2 Process for the preparation of opioid modulators
09/21/2006WO2006098982A1 Process for the preparation of opioid modulators
09/21/2006WO2006098855A2 Processes for preparing morphinans and intermediates thereof
09/21/2006WO2006098308A1 Novel anthranilic acid derivative or salt thereof
09/21/2006WO2006097323A1 TETRAHYDRO-ISOQUINOLIN-l-ONES FOR THE TREATMENT OF CANCER
09/21/2006WO2006067587A3 Nonnucleoside inhibitors of hiv-1 reverse transcriptase
09/21/2006WO2006063294A3 Novel inhibitors of histone deacetylase for the treatment of disease
09/21/2006US20060211863 Process for the preparation of opioid modulators
09/21/2006US20060211675 Preventives/remedies for urinary disturbance
09/21/2006US20060211590 Organic catalyst with enhanced solubility
09/21/2006US20060211107 Protease inhibitor conjugates and antibodies useful in immunoassay
09/21/2006CA2602609A1 Novel anthranilic acid derivative or salt thereof
09/21/2006CA2601674A1 Process for the preparation of opioid modulators
09/21/2006CA2601481A1 Process for the preparation of opioid modulators
09/21/2006CA2600687A1 Processes for preparing morphinans and intermediates thereof
09/20/2006EP1701724A2 Alkylamino, arylamino, and sulfonamido cyclopentyl amide modulators of chemokine receptor activity
09/20/2006EP1611106B1 Preparation of quinapril hydrochloride
09/20/2006EP1392363B1 Use of mGLuR5 antagonists in the manufacture of a medicament in the treatment of Fragile X syndrome, Autism and Mental Retardation
09/20/2006CN1835924A Fused compounds that inhibit vanilloid receptor subtype 1(vr1) receptor
09/20/2006CN1275944C Process for preparing (s)-6,7-dimethoxy-1,2,3,4-tetrahydro isoquinoline-3-carboxylic acid
09/19/2006US7109224 Acyl guanidine compounds and use thereof
09/19/2006US7109212 Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors
09/14/2006WO2006095922A1 Tetrahydroisoquinoline compound and medicinal use thereof
09/14/2006US20060205772 Amide derivatives and their use as inhibitors of 11-beta-hydroxysteroid dehydrogenase type I
09/13/2006EP0917462B1 Cell adhesion inhibitors
09/13/2006CN1832925A New p2x7 receptor avtagonists and their use
09/13/2006CN1274670C Diaminopropionic acid derivatives
09/12/2006US7105702 For use as catalysts in asymmetric reactions, such as, hydrogenation, hydride transfer, allylic alkylation, hydrosilylation, hydroboration, hydrovinylation, hydroformylation, olefin metathesis, hydrocarboxylation
09/12/2006US7105701 Multibinding compounds for agonists for phenolic derivatives for adrenergic receptors with carriers
09/12/2006US7105538 4-oxo-4-[2-(5-pyridin-4-yl-[1,3,4]oxadiazol-2-yl)-pyrrolidin-1-yl]-butyric acid ethyl ester; inhibition of serotonin re-uptake; analgesic effect
09/12/2006US7105536 Compounds
09/12/2006US7105507 Cyclohexane derivatives and their use as therapeutic agents
09/12/2006CA2241788C Novel n-(arylsulphonyl)amino acid derivatives, their preparation process and pharmaceutical compositions containing them
09/08/2006WO2006093823A1 2- [ isoquinolin-s - carbonyl ) amino] -propionic acid derivatives as inhibitors of factors xi and ix for the treatment of thrombosis
09/08/2006WO2005117907A3 P-chiral phospholanes and phosphocyclic compounds and their use in asymmetric catalytic reactions
09/08/2006CA2599808A1 2- [ isoquinolin-s - carbonyl ) amino] -propionic acid derivatives as inhibitors of factors xi and ix for the treatment of thrombosis
09/07/2006US20060199826 Cyclopropane compounds and pharmaceutical use thereof
09/06/2006EP1697304A1 Peroxisome proliferator activated receptor modulators
09/05/2006US7101892 2-(4-benzenesulfonyl-4-methyl-pentyl)-5-phenyl-2-aza-bicyclo[2.2.1]heptane; useful for treating sleep disorder, depression, anxiety
09/05/2006US7101881 N-(4-Chlorophenylacetyl)-8-(4-methylpiperazinyl)-tetrahydroisoquinoline; treating anxiety, depression, dysthymia, major depressive disorder, migraine, post-traumatic stress disorder, avoidant personality disorder, borderline personality disorder, phobias
08/2006
08/31/2006WO2006090783A1 Process for production of 4-fluoroisoquinoline-5-sulfonyl halide or salt thereof
08/31/2006WO2006074223A3 Pharmaceutical compounds as activators of caspases and inducers of apoptosis and the use thereof
08/31/2006WO2005080313A9 Sulfonamide derivatives for the treatment of diseases
08/31/2006US20060194798 Bicyclic-substituted amines as histamine-3 receptor ligands
08/30/2006EP1694410A2 Cyclopropane compounds and pharmaceutical use thereof
08/30/2006EP1694329A2 Diamine and iminodiacetic acid hydroxamic acid derivates
08/30/2006EP1318811B1 Cyclopentyl modulators of chemokine receptor activity
08/30/2006CN1826115A Substituted piperidine compounds and methods of their use
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