Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
01/2006
01/26/2006WO2006010082A1 1,4-disubstituted naphtalenes as inhibitors of p38 map kinase
01/26/2006WO2001085170A9 Peptide deformylase inhibitors
01/26/2006US20060020039 E.g., 3-(2-(4-[(2-aminosulfonyl)phenyl]benzoylamino)phenoxy)benzamidine; 7-(2-(4-[(2-aminosulfonyl)phenyl]benzoylamino)-4-fluorophenoxy)1-aminoisoquinoline; and 3-(2-(4-[(2-aminosulfonyl)phenyl]phenylaminocarbonyl-4-chlorophenoxy)benzamidine; highly selective
01/26/2006US20060019988 Compounds, compositions, and methods
01/26/2006US20060019973 agricultural and horticultural fungal infections of plants; novel N-alkynyl-2-quinolin-(isoquinolin- and quinazolin-)oxyalkylamides; 2-(6-quinolinyloxy)-N-(4-methylpent-2-yn-4-yl) butyramide
01/26/2006DE102004031850A1 Substituirte Tetrahydroisochinoline als MMP-Inhibitoren, Verfahren zu ihrer Herstellung und ihre Verwendung als Medikament Substituirte tetrahydroisoquinolines as MMP inhibitors, to processes for their preparation and their use as a medicament
01/26/2006CA2574217A1 Diamine derivative, process of preparation thereof, and fungicide comprising diamine derivative as an active ingredient
01/25/2006EP1618087A2 Antibacterial agents
01/19/2006WO2005030130A3 Isoquinoline potassium channel inhibitors
01/19/2006US20060014954 Microporous structure of an organic metal complex
01/19/2006US20060014836 e.g. 1-(Benzofuran-2-carbonyl-3-(3-phenoxy-phenyl)-thiourea;viricides; hepatitis virus
01/19/2006US20060014830 2-amino-2-oxoethyl 1-(4'-fluoro-1,1'-biphenyl-4-yl)cyclopropylmethylcarbamate and 2-(methylamino)-2-oxoethyl 1-(4'-fluoro-1,1'-biphenyl-4-yl)cyclopropylmethylcarbamate; fatty acid amide (FAAH) hyrdrolase inhibitors; analgesics; neuropathic pain;psychological disorders; anticarcinogenic agents; AIDS
01/19/2006US20060014783 Sulfonylamino-acetic acid derivatives
01/19/2006US20060014752 Heterocyclic anti-epileptogenic agents and methods of use thereof
01/19/2006US20060014739 Androgen receptor modulators and method of treating disease using the same
01/18/2006EP1615878A2 Compounds, compositions and methods
01/18/2006CN1723194A 3,4-di-substituted cyclobutene-1,2-diones as CXC-chemokine receptor ligands
01/18/2006CN1721408A 1-benzyl tetrahydro isoquinoline compound, its preparing process and use thereof
01/17/2006CA2138930C Substituted benzenesulfonylureas and -thioureas, preparation processes and possible uses of pharmaceutical preparations based on these compounds
01/12/2006WO2006002764A1 4-trifluoromethoxyphenoxybenzol-4'-sulfonic acids, method for the production and use thereof in medicaments
01/12/2006WO2006002763A2 Substituted tetrahydroisochinolines used in the form of mmp inhibitors, method for the production and use thereof in the form of drags
01/12/2006US20060009449 Naphthaline derivatives as H3 inverse agonists
01/12/2006US20060008673 Electroluminescent efficiency
01/12/2006US20060008671 Electroluminescent efficiency
01/12/2006CA2572874A1 Urea derivative
01/12/2006CA2572126A1 4-trifluoromethoxyphenoxybenzol-4'-sulfonic acids, method for the production and use thereof in medicaments
01/12/2006CA2572125A1 Substituted tetrahydroisochinolines used in the form of mmp inhibitors, method for the production and use thereof in the form of drags
01/11/2006EP1613600A1 Substituted 4-phenyltetrahydroisoquinolines, method for the production thereof, the use of the same as medicaments, and medicament containing such compounds
01/11/2006EP1366036B1 Compounds having activity as inhibitors of cytochrome p450rai
01/10/2006US6984735 Reacting a dihalaromatic compound with sulfoxide
01/10/2006US6984647 Antiinflammatory agents; analgesics; antiarthritic agents
01/05/2006US20060004066 Method for treating ADAMTS-5-associated disease
01/05/2006US20060004041 Compounds for treatment of neurodegenerative diseases
01/05/2006DE102004028973A1 Substituierte Tetrahydro-2H-isochinolin-1-on-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Medikament Substituted tetrahydro-2H-isoquinolin-1-one derivatives, to processes for their preparation and their use as a medicament
01/05/2006CA2589565A1 Amido compounds and their use as pharmaceuticals
01/04/2006EP1611106A1 Preparation of quinapril hydrochloride
01/04/2006EP1611105A1 Isoquinoline-5-sulfonic acid amides as inhibitors of akt (protein kinase b)
01/04/2006EP1611104A1 Tetrahydroisoquinolyl acetamide derivatives for use as orexin receptor antagonists
01/04/2006EP1611102A2 Using alkylmetal reagents for directed metalation of azaaromatics
01/04/2006EP1611088A2 Hydroxamates as therapeutic agents
01/04/2006EP1363873A4 Peptide deformylase inhibitors
01/04/2006CN1717175A Quinolin-, isoquinolin-, and quinazolin-oxyalkylamides and their use as fungicides
01/03/2006US6982263 Peptidyl carbamates; treatments for osteoporosis and autoimmune diseases
12/2005
12/29/2005WO2005123743A1 Extraction of alkaloids from opium
12/29/2005WO2005123687A1 Substituted tetrahydro-2h-isoquinolin-1-one derivatives, method for the production thereof, and use of the same as medicaments
12/29/2005WO2005123089A2 Multicyclic sulfonamide compounds as inhibitors of histone deacetylase for the treatment of disease
12/29/2005US20050288304 Tetrahydronaphthylpiperazines as 5HT1B antagonists, inverse agonists and partial agonists
12/29/2005US20050288271 Arylsulfonamides and uses related thereto
12/29/2005DE19748040B4 Carbonsäurederivate, Verfahren zu ihrer Herstellung und pharmazeutische Präparate, die diese Verbindungen enthalten Carboxylic acid derivatives, processes for their preparation and pharmaceutical preparations containing these compounds
12/29/2005CA2569758A1 Extraction of alkaloids from opium
12/28/2005EP1608625A1 Acutumine and acutumine compounds, synthesis and use
12/28/2005EP1265867B1 Malonic acid derivates, processes for their preparation, their use as inhibitor of factor xa activity and pharmaceutical compositions containing them
12/28/2005EP1031563B1 Sulfonyl derivatives
12/27/2005CA2189271C Novel erythromycin derivatives, method for their preparation and their use as drugs
12/22/2005WO2005121130A2 Chemical compounds and pharmaceutical compositions containing them for the treatment of inflammatory disorders
12/22/2005WO2005121094A1 Piperazine and piperidine derivatives as anti-hiv-agents
12/22/2005WO2005121073A1 Inhibitors of histone deacetylase
12/22/2005WO2005120494A1 1-`(3r)-amino-4-(2-fluoro-phenyl)-butyl !-pyrrolidine-(2r)-carboxilic acid-benzyl amine derivatives and related compounds as dipeptidyl-peptidase iv (dpp-iv) inhibitors for the treatment of type 2 diabetes mellitus
12/22/2005WO2005053610A3 Diamine and iminodiacetic acid hydroxamic acid derivatives
12/22/2005US20050282881 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
12/22/2005US20050282858 Substituted cycloalkylcarboxamides: 1-((1-(4-Chlorophenyl)cyclopropyl)carbonyl)pyrrolidin-3-ol and 1-Acetyl-4-(4-{1-[(3-phenylpyrrolidin-1-yl)carbonyl]cyclopropyl}phenyl)piperazine; 11- beta hydroxyl steroid dehydrogenase type 1 inhibitors; mineralcorticoid receptor antagonists; antidiabetic agents
12/22/2005CA2576236A1 1-`(3r)-amino-4-(2-fluoro-phenyl)-butyl !-pyrrolidine-(2r)-carboxilic acid-benzyl amine derivatives and related compounds as dipeptidyl-peptidase iv (dpp-iv) inhibitors for the treatment of type 2 diabetes mellitus
12/22/2005CA2569111A1 Chemical compounds and pharmaceutical compositions containing them for the treatment of inflammatory disorders
12/22/2005CA2564499A1 Tetrahydropyranyl cyclopentyl tetrahy-dropyridopyridine modulators of chemokine receptor activity
12/21/2005EP1606278A1 Substituted cyclohexyl and piperidinyl derivates as melanocortin-4 receptor modulators
12/21/2005EP1605896A2 7-amino- isoindolyl compounds amd their pharmaceutical uses
12/20/2005US6977266 Pyridone derivatives having affinity for cannabinoid 2-type receptor
12/20/2005CA2302412C Aminoalkylphenol derivatives and related compounds
12/15/2005WO2005118581A1 Tetrahydro-imidazo [1,5-a] pyridin derivatives as aldosterone synthase inhibitors
12/15/2005WO2005118548A1 Substituted 1,2,3,4-tetrahydroisoquinoline derivatives
12/15/2005WO2005118547A1 Tetrahydroisoquinoline sulfonamide derivatives, the preparation thereof, and the use of the same in therapeutics
12/15/2005WO2005118540A2 Bicyclic, nitrogen-containing heterocycles as aromatase inhibitors
12/15/2005WO2005118538A2 Arylsulfonamides and uses as hydroxysteroid dehydrogenase
12/15/2005WO2005117907A2 P-chiral phospholanes and phosphocyclic compounds and their use in asymmetric catalytic reactions
12/15/2005WO2005117876A1 Dual small molecule inhibitors of cancer and angiogenesis
12/15/2005WO2005117865A1 Naphthaline derivatives useful as histamine-3-receptor ligands
12/15/2005US20050277646 N-[4-({5-(4-fluorophenyl)-4-[4-(trifluoromethyl)phenyl]pyridin-2-yl}oxy)-1,3-benzothiazol-2-yl]acetamide; vanilloid (capsaicin) receptor antagonist/agonist; antiinflammatory, analgesic, antiarthritis, antirheumatic; diseases involving sensory nerve function
12/15/2005US20050277631 Vanilloid receptor ligands and their use in treatments
12/15/2005CA2568622A1 Dual small molecule inhibitors of cancer and angiogenesis
12/15/2005CA2568163A1 Bicyclic, nitrogen-containing heterocycles as aromatase inhibitors
12/15/2005CA2568159A1 Tetrahydro-imidazo [1,5-a] pyridin derivatives as aldosterone synthase inhibitors
12/15/2005CA2561858A1 Arylsulfonamides and uses related thereto
12/14/2005EP1604983A1 Receptor antagonist
12/14/2005EP1604662A1 1-[(3R)-Amino-4-(2-fluoro-phenyl)-butyl]-pyrrolidine-(2R)-carboxylic acid benzyl amine derivatives and related compounds as dipeptidyl peptidase IV (DPP-IV) inhibitors for the treatment of type 2 diabetes mellitus
12/14/2005EP1603923A1 Metal complexes
12/14/2005EP1440052B1 Benzamide derivatives as antagonists of orexin receptors
12/14/2005EP1224165B1 Novel compounds
12/14/2005CN1231439C Novel hydronaphtalene compounds prepared by phodium catalyzed ring opening reaction in presence of phosphine ligand
12/14/2005CN1231433C Transfer hydrogenation process
12/13/2005US6974876 Method for preparing intermediates useful in synthesis of retroviral protease inhibitors
12/13/2005US6974822 Treating osteoarthritis or rheumatoid arthritis
12/08/2005WO2005115972A1 Therapeutic compounds
12/08/2005WO2005115392A2 3-(4-heteroarylcyclohexylamino) cyclopentanecarboxamides as modulators of chemokine receptors
12/08/2005WO2005115361A2 Androgen receptor modulators and method of treating disease using the same
12/08/2005WO2002057256A9 Piperazinylcarbonylquinolines and -isoquinolines
12/08/2005US20050272931 Vanilloid receptor ligands and their use in treatments
12/08/2005US20050272823 improved selectivity and pharmacokinetic properties; 6-Fluoro-1-[(1 H-indazol-4-yl)amino]-4,4-dimethyl-2-(trifluoromethyl)-1,2,3,4-tetrahydronaphthalene-2,5-diol; cyclization of imines
12/08/2005US20050272777 Vanilloid receptor ligands and their use in treatments
12/08/2005US20050272745 Novel piperidine and piperazine derivatives
12/08/2005DE102004017662B3 New 1-amino-tetrahydronaphthalene derivatives, useful for treatment of e.g. inflammation, bind with high selectivity to glucocorticoid receptors
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