Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780) |
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03/04/1999 | CA2295017A1 Process for preparing enantiomerically enriched n-derivatised lactams |
03/03/1999 | EP0899270A1 Indolylmethyl-N,N'-bisacylpiperazines as neurokinine receptor antagonists |
03/03/1999 | EP0899259A1 Process for the preparation of cis-hexahydroisoindolines |
03/03/1999 | EP0724570B1 Amidino derivatives useful as nitric oxide synthase inhibitors |
03/03/1999 | EP0674641B1 Pyrrolopyrimidines as crf antagonists |
03/03/1999 | EP0605697B1 Indol derivatives for the treatment of migraine |
03/03/1999 | CN1209818A Method of producing press-moulding materials with polyisocyanate binders and using latent, heat-activable catalyst |
03/03/1999 | CN1209805A Noval fused pyrrolecarboxamides and new class of GABA brain receptor ligands |
03/03/1999 | CN1209803A Conformationally restricted aromatic inhibitors of microsomal triglyceride transfer protein and method therefor |
03/03/1999 | CN1042331C 4,6-dichloro-3-substituted-2-carboxy indole derivative |
03/03/1999 | CN1042328C Substituted cyclohexane derivative and medicine containing same |
03/02/1999 | US5877329 Coupling/ring closure of a 2-halo or 2-trifluoromethylsulfonyloxy aniline and an alkyl ketone, indomethacin precursors |
03/02/1999 | US5877202 Indole derivatives useful to treat estrogen-related neoplasms and disorders |
03/02/1999 | US5877200 Cyclic amides |
03/02/1999 | US5877199 Heterocyclic compounds, their preparation and their therapeutic use |
03/02/1999 | US5877190 Substituted biphenyl compounds |
03/02/1999 | US5876710 Drug delivery; using a brominated benzamide compound |
03/02/1999 | US5876465 Compositions for dyeing keratin fibres containing 2-iminoindoline derivatives and dyeing process |
02/28/1999 | CA2246407A1 Use of inhibitors of the sodium-hydrogen exchanger for the production of a pharmaceutical for the treatment of disorders which are caused by protozoa |
02/25/1999 | WO1999009025A2 2-(4-aryl or heteroaryl-piperazin-1-ylmethyl)-1h-indole derivatives interacting with the dopamine d4 receptor |
02/25/1999 | WO1999009007A1 Solid phase synthesis of 2,3-disubstituted indole compounds |
02/25/1999 | DE19837386A1 New CCR-3 antagonist piperazine derivatives and analogues |
02/24/1999 | EP0897912A1 Amidino derivatives useful as nitric oxide synthase inhibitors |
02/24/1999 | CN1209129A Antagonists of gonadotropin releasing hormone |
02/24/1999 | CN1209119A Novel tricyclic compounds and drug compositions contg. same |
02/23/1999 | US5874473 Substituted cycloalkanecarboxylic acid derivatives as matrix metalloprotease inhibitors |
02/18/1999 | WO1999007681A1 2-acylaminopropanamines as tachykinin receptor antagonists |
02/18/1999 | WO1999007679A1 Peptidyl compounds having mmp and tnf inhibitory activity |
02/18/1999 | WO1999007678A1 Indole derivatives as mcp-1 receptor antagonists |
02/18/1999 | WO1999007677A1 2-acylaminopropanamines as tachykinin receptor antagonists |
02/18/1999 | WO1999007667A1 Novel ethylamine derivatives |
02/18/1999 | WO1999007378A1 Nicotine antagonists for nicotine-responsive neuropsychiatric disorders |
02/18/1999 | WO1999007351A2 Indole derivatives and their use as mcp-1 antagonists |
02/18/1999 | CA2298702A1 2-acylaminopropanamines as tachykinin receptor antagonists |
02/18/1999 | CA2298701A1 2-acylaminopropanamines as tachykinin receptor antagonists |
02/18/1999 | CA2297290A1 Chemical compounds |
02/18/1999 | CA2295535A1 Indole derivatives as mcp-1 receptor antagonists |
02/18/1999 | CA2245043A1 Ccr-3 receptor antagonists |
02/17/1999 | EP0896580A1 Specific immunophilin ligands as antiasthmatics and immunosuppressants |
02/17/1999 | EP0896533A2 Pentafluorobenzenesulfonamides and analogs |
02/17/1999 | CN1208413A Antagonists of gonadotropin releasing hormone |
02/17/1999 | CN1208347A Substituted N-[(aminoiminomethyl or aminomethyl) phenyl] propyl amides |
02/17/1999 | CN1042133C N-substituted azabicycloheptane derivatives, the preparation and use thereof |
02/17/1999 | CN1042131C Novel N-cinnamoyl-2-methyl-5-methoxy-3-indol acetate, preparation of same and pharmaceutical containing same |
02/16/1999 | US5872253 1-(3-heterocyclyphenyl)-s-triazine-2,4,6-oxo or thiotrione herbicidal agents |
02/16/1999 | US5872145 Formulation of 5-HT agonist and NSAID for treatment of migraine |
02/16/1999 | US5872117 Treating cerebrovascular dementia, senile dementia, alzheimer's dementia, sequelae of ischemic encephalopathy and cerebral apoplexy |
02/16/1999 | US5872100 Peptides containing D-2-Alkyl-Tryptophan |
02/11/1999 | WO1999006433A1 Compounds which inhibit leukocyte adhesion mediated by vla-4 |
02/11/1999 | WO1999006406A1 4-OXO-3,5-DIHYDRO-4H-PYRIDAZINO[4,5-b]-INDOLE-1-ACETAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION IN THERAPY |
02/11/1999 | WO1999006384A1 1-(n-phenylaminoalkyl)-piperazine derivatives substituted at position 2 of the phenyl ring |
02/11/1999 | WO1999006368A1 Special 3-azabicyclo[3.1.0]hexanes, method for producing and modifying the same, and their use |
02/11/1999 | WO1999006367A1 Caspases and apoptosis |
02/11/1999 | WO1999006361A2 N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases |
02/11/1999 | WO1999006340A2 Sulfonylamino substituted hydroxamic acid derivatives as metalloprotease inhibitors |
02/11/1999 | WO1999006042A1 Caspases and apoptosis |
02/11/1999 | WO1999006041A1 SUBSTITUTED ALKANOHYDROXAMIC ACIDS AND METHOD OF REDUCING TNFα LEVELS |
02/11/1999 | CA2298668A1 Caspases and apoptosis |
02/11/1999 | CA2298617A1 Acyclic metalloprotease inhibitors |
02/11/1999 | CA2298509A1 Special 3-azabicyclo[3.1.0]hexanes, method for producing and modifying the same, and their use |
02/11/1999 | CA2297757A1 Caspases and apoptosis |
02/11/1999 | CA2297095A1 1-(n-phenylaminoalkyl)-piperazine derivatives substituted at position 2 of the phenyl ring |
02/11/1999 | CA2295295A1 Substituted alkanohydroxamic acids and method of reducing tnf.alpha. levels |
02/11/1999 | CA2290746A1 Compounds which inhibit leukocyte adhesion mediated by vla-4 |
02/09/1999 | US5869692 Compositions for dyeing keratinous fibers containing n-substituted derivatives of 4-hydroxyindole, new derivatives, process for preparing them, their use for dyeing, and dyeing processes |
02/09/1999 | US5869663 Intermediates for neurokinin receptor antagonists |
02/09/1999 | US5869518 Azacycloalkane derivatives, their preparation and their application in therapy |
02/09/1999 | US5869489 Trypthophan ureas as neurokinnin antagonists |
02/09/1999 | CA1340382C Process for the preparation of 2-arylpropionic acids |
02/04/1999 | WO1999005105A1 Thermodynamically stable modification of 1-(4-carbazolyloxy)-3-[2-(2-methoxyphenoxy)ethylamino]-2-propanole, process for its preparation and pharmaceutical compositions containing it |
02/04/1999 | WO1999005104A1 Indole compounds as cox-2 inhibitors |
02/04/1999 | WO1999005096A2 Urokinase inhibitors |
02/04/1999 | WO1999004780A1 Therapeutic or prophylactic agent for glomerulopathy |
02/04/1999 | DE19733439A1 Neue 6-endo-Amino-3-azabicyclo(3.1.0)hexande, Verfahren zu deren Herstellung und deren Verwendung zur Herstellung von Chinolon- und Naphthyridincarbonsäure-Derviaten mit verbesserten Eigenschaften New 6-endo-amino-3-azabicyclo (3.1.0) hexande, processes for their preparation and their use for the preparation of quinolone and naphthyridine-Derviaten with improved properties |
02/04/1999 | CA2294300A1 Urokinase inhibitors |
02/03/1999 | EP0894789A1 Substituted indole-2-carboxylic acids as glucosyl transferase inhibitors |
02/03/1999 | EP0894089A1 Novel heterocyclic compounds having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions containing them |
02/03/1999 | EP0894085A1 Benzyl(idene)-lactam derivatives, their preparation and their use as selective (ant)agonists of 5-ht1a- and/or 5-ht1d receptors |
02/03/1999 | EP0862553A4 Cbi analogs of cc-1065 and the duocarmycins |
02/03/1999 | EP0623619B1 PREPARATION METHOD OF ARENO[e]INDOLS |
02/03/1999 | CN1207100A Novel indole-2,3-done-3-oxime derivatives |
02/02/1999 | US5866611 Phenoxypropylamine inhibitors of squalene synthese, useful in treating diseases in which a lowering of cholesterol is desirable. |
02/02/1999 | US5866594 Indole-2-carboxylate derivatives and fungicidal compositions for agricultural or horticultural use containing the derivatives as active component |
02/02/1999 | US5866587 Hydroxamide derivatives of fused piperidine derivatives |
02/02/1999 | US5866577 Aromatic amidine derivatives and salts thereof |
02/02/1999 | US5866545 Antiinflammatory agents; nervous system disorders; gastrointestinal disorders; urogenital disorders |
02/02/1999 | US5866318 Administering to nerve cells apopototic stimulant; calibration |
01/29/1999 | CA2243882A1 Substituted indole-2-carboxylic acids as glucosyl transferase inhibitors |
01/28/1999 | WO1999003831A1 3-benzoylindole derivatives and drugs containing the same |
01/28/1999 | WO1999003823A2 Novel polyamine analogues as therapeutic and diagnostic agents |
01/28/1999 | WO1999003468A1 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith |
01/28/1999 | WO1999003467A1 Pharmaceutical compositions and methods for treating compulsive disorders using pyrrolidine derivatives |
01/28/1999 | WO1999003465A1 Antibiotics containing indole derivatives |
01/28/1999 | WO1998038984A3 Formulations for hydrophobic pharmaceutical agents |
01/28/1999 | CA2297413A1 Novel polyamine analogues as therapeutic and diagnostic agents |
01/28/1999 | CA2294772A1 3-benzoylindole derivatives and drugs containing the same |
01/28/1999 | CA2289055A1 Kappa agonist compounds, pharmaceutical formulations and method of prevention and treatment of pruritus therewith |
01/27/1999 | EP0893440A1 Thermodynamically stable modification of 1-(4-carbazolyloxy)-3-[2-(2-methoxyphenoxy)ethylamino]-2-propanole, process for its preparation and pharmaceutical compositions containing it |
01/27/1999 | EP0892780A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS |
01/27/1999 | CN1206405A Imides as PDE III, PDE IV and TNF inhibitors |