Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
05/1999
05/12/1999EP0915087A2 Sulfonamide substituted fused five-membered ring compounds, their use as medicaments as well as pharmaceutical compositions containing them
05/12/1999EP0915086A1 Phenylsulfonamide derivatives
05/12/1999EP0914605A1 Molecular model for vla-4 inhibitors
05/12/1999EP0914321A1 Indole derivatives for the treatment of osteoporosis
05/12/1999EP0914319A1 Diarylalkyl cyclic diamine derivatives as chemokine receptor antagonists
05/12/1999EP0808162B1 Use of carbazole compounds for the manufacture of a medicament for the treatment of congestive heart failure
05/12/1999EP0729470B1 Herbicidal pyrrolopyridine compounds
05/12/1999CN1216531A Indole derivatives useful as endothelin receptor antagonists
05/11/1999US5902884 Reacting carbazole or alkyl, alkoxy, nitro or halogen substitued derivative with an alkyl halide in an inert solvent with an inorganic base and di- or tri-, alkylamine catalyst; no aftertreatment required to remove catalyst
05/11/1999US5902791 Metalloproteinase inhibitors
05/06/1999WO1999021854A1 Bis-quaternary ammonium derivatives as neuromuscular relaxants
05/06/1999WO1999021849A1 Processes for producing 7-isoindolinequinolonecarboxylic derivatives and intermediates therefor, salts of 7-isoindolinequinolonecarboxylic acids, hydrates thereof, and composition containing the same as active ingredient
05/06/1999WO1999021848A2 Novel 1-(n'-(arylalkylaminoalkyl))aminoisoindoles; a new class of dopamine receptor subtype specific ligands
05/06/1999WO1999021837A1 Substituted benzene compounds, process for their preparation, and herbicidal and defoliant compositions containing them
05/06/1999WO1999021831A1 Tricyclic compounds as cgmp-pde inhibitors
05/06/1999WO1999021824A1 Cyclic amino acids and derivatives thereof useful as pharmaceutical agents
05/06/1999WO1999021811A1 Method of separating optical isomers
05/06/1999WO1999021559A1 MORPHOLINO-N-ETHYL ESTER PRODRUGS OF INDOLE sPLA2 INHIBITORS
05/06/1999WO1999021557A1 Antagonists of gonadotropin releasing hormone
05/06/1999WO1999021553A1 Antagonists of gonadotropin releasing hormone
05/06/1999WO1999021546A1 N,N-DIETHYLGLYCOLAMIDO ESTER PRODRUGS OF INDOLE sPLA2 INHIBITORS
05/06/1999WO1999021545A1 ISOPROPYL ESTER PRODRUGS OF INDOLE sPLA2 INHIBITORS
05/06/1999WO1999015493A8 9,10-dihydro-9,10-ethanoanthracene derivatives as phospholipase inhibitors
05/06/1999EP0913430A1 Condensed azo compound and process for producing the same
05/06/1999EP0912573A1 Camptothecin-skeleton compounds isolated from mappia foetida and the use thereof as syntones for novel medicaments as well as therapeutical agents
05/06/1999EP0912570A1 Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors
05/06/1999EP0912567A1 Carboline derivatives
05/06/1999EP0912513A1 Fibrinogen receptor antagonist prodrugs
05/06/1999EP0912511A1 5-indolyl-2,4-pentadienoic acid derivatives useful as inhibitors of bone resorption
05/06/1999EP0912510A1 Nickel catalyzed addition of -nh- containing compounds to vinyl and aryl halides
05/06/1999EP0912496A1 Inhibition of matrix metalloproteases by acetylene containing compounds
05/06/1999EP0912487A1 Substituted oxobutyric acids as matrix metalloprotease inhibitors
05/06/1999EP0912175A1 Fibrinogen receptor antagonists
05/06/1999DE19748763A1 Verwendung von Vasopressin-Antagonisten Use of vasopressin antagonists
05/06/1999CA2568251A1 Process for preparing substituted 7-bromoquinolone-carboxylic acid derivatives
05/06/1999CA2309135A1 N,n-diethylglycolamido ester prodrugs of indole spla2 inhibitors
05/06/1999CA2308454A1 Antagonists of gonadotropin releasing hormone
05/06/1999CA2308443A1 Morpholino-n-ethyl ester prodrugs of indole spla2 inhibitors
05/06/1999CA2308069A1 Antagonists of gonadotropin releasing hormone
05/06/1999CA2307815A1 Substituted benzene compounds, process for their preparation, and herbicidal and defoliant compositions containing them
05/06/1999CA2306878A1 Bis-quaternary ammonium derivatives as neuromuscular relaxants
05/04/1999US5900430 Cytokine inhibitors
05/04/1999US5900227 Multicyclic nitrone spin trapping compositions
05/04/1999CA2184604C Bicyclic carbamates
04/1999
04/29/1999WO1999020599A1 Pharmaceutically active compounds and methods of use
04/29/1999WO1998057931A3 Quinoline-indole antimicrobial agents, uses and compositions related thereto
04/29/1999CA2307597A1 Pharmaceutically active compounds and methods of use
04/28/1999EP0910572A1 Inhibitors of picornavirus 3c proteases and methods for their use and preparation
04/28/1999EP0910565A1 Amide derivatives as selective neuropeptide y receptor antagonists
04/28/1999EP0910564A1 D-amino acid derived inhibitors of cysteine and serine proteases
04/28/1999EP0910373A1 Use of substituted azaspirane in the treatment of asthma
04/28/1999EP0910372A1 Pharmaceutical compositions containing mesembrine and related compounds
04/28/1999EP0784629B1 Peptidyl compounds and their therapeutic use as inhibitors of metalloproteases
04/28/1999EP0559738B1 Methods for detection and quantitation of cell subsets within subpopulations of a mixed cell population
04/28/1999CN1215400A Piperazine and piperidine compounds
04/28/1999CN1215390A Substituted phenyl keto enols as pesticides and herbicides
04/28/1999CN1215056A Process for preparation of N-tertiary butyl amide
04/28/1999CN1215049A (3-oxioisoindolin-1-ylidine) propandinitrile derivatives and method for preparing the same
04/28/1999CN1043142C Quinolone and naphthyridone-carboxylic acid derivatives and preparation process
04/27/1999US5898075 Process for the separation of the enantiomers of a bicyclic lactam
04/22/1999WO1999019298A1 iso-CBI AND iso-CI ANALOGS OF CC-1065 AND THE DUOCARMYCINS
04/22/1999WO1999019296A1 Aminobutanoic acid derivatives
04/22/1999WO1999019293A1 Novel aryloxy-alkyl-dialkylamines
04/22/1999WO1999018794A1 Method for treating alzheimer's disease
04/22/1999WO1999006361A3 N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases
04/22/1999CA2306420A1 Iso-cbi and iso-ci analogs of cc-1065 and the duocarmycins
04/22/1999CA2305262A1 Method for treating alzheimer's disease
04/21/1999EP0909762A2 Binuclear Iridium(I) phosphine complexes and their use as catalysts for the asymmetric hydroamination of olefins
04/21/1999EP0909174A1 TREATMENT OF CYSTIC DISEASE WITH TNF-$g(a)
04/21/1999CN1214690A Specific immunophilin ligands as antiasthmatics and immunosuppressants
04/21/1999CN1214683A 1,3,4-oxadiazine derivatives and their use as pesticides
04/20/1999CA2188798C Tryptamine derivatives as 5-ht-1d receptor ligands
04/15/1999WO1999018074A1 Novel lactam metalloprotease inhibitors
04/15/1999WO1999018066A1 Amidocarboxylic acid derivatives
04/15/1999WO1999017778A1 α-KETOAMIDE MULTICATALYTIC PROTEASE INHIBITORS
04/15/1999WO1999009025A3 2-(4-aryl or heteroaryl-piperazin-1-ylmethyl)-1h-indole derivatives interacting with the dopamine d4 receptor
04/15/1999CA2305808A1 Amidocarboxylic acid derivatives
04/15/1999CA2305679A1 Novel lactam metalloprotease inhibitors
04/14/1999EP0908448A1 Thermally stable aminosulfur trifluorides
04/14/1999EP0908445A1 Oxidation dyeing composition for keratin fibres containing an amino acid derivative as oxidation base and aminoacid derivatives
04/14/1999EP0907639A1 Polymorphic compounds
04/14/1999EP0907318A1 Antioxidant compound
04/14/1999EP0810991B1 1-aryl-2-acylamino-ethane compounds and their use as neurokinin especially neurokinin 1 antagonists
04/14/1999EP0510068B1 NEW CENTRALLY ACTING 6,7,8,9-TETRAHYDRO-3H-BENZ(e)INDOLE HETEROCYCLICS
04/14/1999CN1214043A Benzyl(idene)-lactam derivatives, their prepn. and their use as selective (ant) agaonists of 5-ht1A-and/or 5-ht1D receptors
04/14/1999CN1214041A Sulfonated amino acid derivatives and metalloproteinase inhibitors contg. same
04/14/1999CN1214039A Carbamoyloxy derivatives of mutiline and their use as antibacterials
04/13/1999CA2044491C Novel process for industrial preparation of 4-chloro-3-sulfamoyl n-(2,3-dihydro 2-methyl 1h-indol -1-yl) benzamide
04/13/1999CA2044186C Novel process for industrial preparation of 4-chloro 3-sulfamoyl n-(2,3-dihydro 2-methyl 1h-indol-1-yl) benzamide from 2,3-dihydro 2-methyl 1h-indole and hydroxylamine-0-sulfonic acid
04/13/1999CA2001988C Hydroxylamine derivatives
04/08/1999WO1999016748A1 Utilizing spirocyclic phenyl keto-enols as pesticides and herbicides
04/08/1999WO1999016707A1 Synthesis method for solution with high grade chloramine
04/08/1999WO1999016453A1 Method for the treatment of cystic fibrosis
04/08/1999WO1999003823A3 Novel polyamine analogues as therapeutic and diagnostic agents
04/08/1999CA2304482A1 Method for the treatment of cystic fibrosis
04/08/1999CA2303135A1 High grade chloramine synthesis
04/07/1999EP0906284A1 Tricyclic amine derivatives
04/07/1999EP0906283A1 Substituted benzamide derivatives and their use as anticonvulsants
04/07/1999EP0906094A1 Substituted n- (aminoiminomethyl or aminomethyl)phenyl]propyl amides
04/07/1999EP0659181B1 Sulfonamide inhibitors of hiv-aspartyl protease