Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
08/1998
08/20/1998WO1998035951A2 New aminopiperazine derivatives
08/20/1998WO1998035939A1 Malonic diamide derivatives and use thereof
08/20/1998WO1998035701A1 Drug targeting
08/20/1998CA2280874A1 Bioreductive conjugate for targeting a therapeutic agent
08/20/1998CA2251368A1 Amide derivatives as selective neuropeptide y receptor antagonists
08/19/1998EP0859004A1 Piperidine derivatives having anxiolytic effect
08/19/1998EP0858996A1 Nerve cell protective agents
08/19/1998EP0858995A1 Process for the preparation of N-alkyl carbazoles
08/19/1998EP0858444A1 Cyclopentyl tachykinin receptor antagonists
08/19/1998EP0767783B1 Substituted alkyldiamine derivatives and their use as tachykinin antagonists
08/19/1998EP0667860B1 Aza spiro alkanes derivatives as therapeutic agents
08/19/1998EP0663825B1 USE OF MELATONIN in low oral doses TO INDUCE SLEEP
08/19/1998CN1190890A Cyclo-oxygenase inhibitor and amidine derivative salts, preparation method thereof, use thereof as drugs, and pharmaceutical compositions containing said salts
08/19/1998CN1190650A Substituted phenyl acetanides, process for their preparation and intermediates thereof
08/18/1998US5795914 Phenylalkan(en)oic acid
08/18/1998US5795907 Gastin and CCK receptor ligands
08/18/1998US5795890 Sulfonamide derivatives
08/18/1998CA2161768C 3-(indol-3-yl) propenoic acid derivatives and as nmda antagonists
08/18/1998CA2036876C Derivatives having a naphthalenic structure; process for preparing the same and pharmaceutical compositions containing them
08/18/1998CA1340005C Pharmaceutical composition for the treatment of psoriasis
08/13/1998WO1998034935A1 Fibrinogen receptor antagonist prodrugs
08/13/1998WO1998034632A1 Compounds and compositions for delivering active agents
08/13/1998WO1998018466A3 Anti-neurogenic inflammatory compounds and compositions and methods of use thereof
08/13/1998CA2279927A1 Fibrinogen receptor antagonist prodrugs
08/12/1998CN1190389A Farnesyl transferase inhibitors, its preparation and medicine composition thereof
08/12/1998CN1039491C Tetrahydro-carbazole compound and its preparation and application
08/11/1998US5792786 Sustained and prolonged wound healing agents
08/11/1998US5792783 Capable of modulating tyrosine kinase signal transduction in order to regulate, modulate and/or inhibit abnormal cell proliferation
08/11/1998US5792771 For treating tumors, vascular system disorders, diabetes, diabetic retinopathy, rheumatoid arthritis and hemangioma
08/06/1998WO1998033878A2 Activators for per compounds
08/06/1998WO1998033795A1 Nanomolar, non-peptide inhibitors of cathepsin d
08/06/1998WO1998033758A1 Bicyclic quinone compounds, their production and use
08/06/1998WO1998024763A3 Immunotherapeutic imides/amides as pde iv and tnf inhibitors
08/06/1998DE19704143A1 Aktivatoren für anorganische Perverbindungen Activators for inorganic per
08/06/1998CA2280096A1 Nanomolar, non-peptide inhibitors of cathepsin d
08/06/1998CA2276171A1 Bicyclic quinone compounds, their production and use
08/05/1998EP0856511A1 Calcium salt of indomethacin pentahydrate and its preparation
08/05/1998EP0480006B1 Process for producing gramine derivates
08/05/1998CN1189820A N-substituted 4-hydroxyindole derivatives and keratin fibre dyeing compsns. containing same
08/05/1998CN1189494A Substituted isoazalene compound
08/05/1998CN1189493A New Substituted biphenyl or phenylpyridine compounds, process for their preparation and pharmaceutical compositions containing them
08/04/1998US5789491 Fluorinated imides for imparting repellency of low surface tension fluids to thermoplastic polymers
08/04/1998US5789434 Derivatives of substituted 4-biarylbutyric acid as matrix metalloprotease inhibitors
08/04/1998US5789404 Central nervous system disorders and antiserotonin agents
08/04/1998US5789402 Compounds having effects on serotonin-related systems
07/1998
07/30/1998WO1998032802A1 Soluble chromophores having improved solubilising groups
07/30/1998WO1998032759A1 Method of making (1s, 4r)-1-azabicyclo[2.2.1]heptan-3-one and (1r, 4s), 1-azabicyclo[2.2.1]heptan-3-one
07/30/1998WO1998032736A1 Process for producing benzylsuccinic acid derivatives
07/30/1998WO1998032734A1 SUBSTITUTED β-THIOCARBOXYLIC ACIDS
07/30/1998WO1998032733A1 Sulfonyl urea derivatives and their use in the control of interleukin-1 activity
07/30/1998WO1998032727A1 Process for producing optically active benzylsuccinic acid and intermediate therefor
07/30/1998WO1998032438A1 Il-8 receptor antagonists
07/30/1998WO1998023565A3 Aminoguanidines and alkoxyguanidines as protease inhibitors
07/30/1998CA2278427A1 Il-8 receptor antagonists
07/30/1998CA2275965A1 Soluble chromophores having improved solubilising groups
07/30/1998CA2269683A1 Method of making (1s, 4r)-1-azabicyclo¬2.2.1|heptan-3-one and (1r, 4s), 1-azabicyclo¬2.2.1|heptan-3-one
07/29/1998EP0854874A1 Macrocyclic lactone compounds and their production process
07/29/1998EP0854865A1 Combinatorial solid phase synthesis of a library of indole derivatives
07/29/1998EP0854863A1 Esters and amides as pla2 inhibitors
07/29/1998EP0740668B1 Tetracyclic derivatives, process of preparation and use
07/29/1998EP0722434B1 Nitric esters having anti-inflammatory and/or analgesic activity and process for their preparation
07/29/1998EP0717732B1 Polyamidic acid derivatives with antigastrin activity, a method for their preparation, and their pharmaceutical use
07/29/1998CN1189153A Alkyl dihalogenated phenyl-substituted ketoenols useful as pesticides and herbicides
07/28/1998US5786523 Naphthol derivatives and process for producing the same
07/28/1998US5786488 Dehydrobromination of a dibromobenzoquinones with at least one indoles in a polar solvent and a metal carbonate to form an antitumor agent
07/28/1998US5786483 α-and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
07/28/1998US5786356 Selective β3 adrenergic agonists
07/28/1998CA2127561C 3-azabicyclohexane compound intermediates for producing antibacterial compounds
07/23/1998WO1998031667A1 Amino-iminoisoindolenine benzene sulfonate, and process for the preparation of nitrate and benzene sulfonate salts of amino-aminoisoindolenine derivatives
07/23/1998WO1998031661A1 Benzamidine derivatives
07/23/1998CA2278180A1 Benzamidine derivatives
07/22/1998EP0854382A1 Heat development image forming process and heptamethine cyanine compound
07/22/1998EP0853614A1 Substituted tetralylmethylen-oxindole analogues as tyrosine kinase inhibitors
07/22/1998EP0853612A1 Alpha-hydrazino acid derivatives and method for making same
07/22/1998EP0748312B1 Bicyclic carbamates as leukotriene d4 antagonists
07/22/1998EP0725775B1 Certain fused pyrrolecarboxanilides; a new class of gaba brain receptor ligands
07/22/1998EP0677042B1 Selective ligands of 5ht1d-5ht1b receptors derived from indole-piperazine useful as medicaments
07/22/1998EP0635002B1 Novel perhydroisoindole derivatives and preparation thereof
07/22/1998CN1188475A Process for producing guanidine derivatives, intermediates therefor and their production
07/21/1998US5783738 Optically active diphosphines, preparation thereof according to a process for the resolution of the racemic mixture and use thereof
07/21/1998US5783708 Hexahydroisoindole derivatives
07/21/1998US5783701 Anti-hiv viricides
07/21/1998US5783682 Oligonucleotide mimics having nitrogen-containing linkages
07/21/1998US5783594 Administering to treat glioma, colon cancer and immunological disordaers
07/21/1998US5783593 Inhibitors of squalene synthetase and protein farnesyltransferase
07/21/1998US5783590 6-heterocyclic-4-amino-1,2,2A,3,4,5-hexahydrobenz CD!indoles
07/21/1998US5783575 Antagonists, their preparation and use
07/16/1998WO1998030992A2 Fluorescent cyanine dyes
07/16/1998WO1998030569A1 Asymmetric synthesis and catalysis with chiral heterocyclic compounds
07/16/1998WO1998030546A1 TRICYCLIC BENZO[e]ISOINDOLES AND BENZO[h]ISOQUINOLINES
07/16/1998WO1998030541A1 C-terminal ketone hydroxamic acid inhibitors of matrix metalloproteinases and tnfa secretion
07/16/1998WO1998030540A1 Efficient synthesis of a chiral mediator
07/16/1998CA2277105A1 C-terminal ketone hydroxamic acid inhibitors of matrix metalloproteinases and tnfa secretion
07/16/1998CA2276074A1 Efficient synthesis of a chiral mediator
07/15/1998EP0853085A1 Piperidine derivatives having anxiolytic effect
07/15/1998CN1187813A Fatty acid esters as bioactive compounds
07/15/1998CN1187812A Indole derivatives as CGMP-PDE inhibitors
07/15/1998CN1039119C Condensed heterocyclic ketone derivatives, their production and use
07/14/1998US5780645 Procedure for alkylation of imides
07/14/1998US5780632 Imide derivatives and their production and use