Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
01/2002
01/02/2002CN1329589A N-aralkylaminotetralins as ligands for neuroptide YY5 receptor
01/02/2002CN1328998A Preparation method of 3-oxyindole derivative for synthesizing indigo
01/02/2002CN1328997A Method for synthesizing indigo by using N-substituted glycine or glycine ester
01/02/2002CN1328824A Compound for curing female sexual disorder
01/02/2002CN1077109C S type 2-substituted hydroxy 2-indolidinylbutyric ester compounds and process for preparation thereof
01/01/2002US6335463 Copper catalyzed arylation of 2,5-dichlorobenzoic acid with n-(4-fluorophenyl)glycine in which alkali metal salts are employed in aqueous alkaline environment
01/01/2002US6335460 Treating retroviral infections, including human immunodeficiency virus, and aids
01/01/2002US6335450 Efficient cyclic-bridged cyanine dyes
01/01/2002US6335360 Indoline-2-carboxylic amide derivatives; obesity, eating and psychological disorders
01/01/2002US6335359 Topically applying to skin or scalp to treat dermatitis or acne; side effect reduction
01/01/2002US6335334 Hypertensive agents, anticoagulants; cardiovascular and sexual disorders, angina pectoris, and atherosclerosis
01/01/2002US6335333 Matrix metalloproteinase inhibitors
01/01/2002CA2215333C Heterocyclic substituted piperazinone derivatives as tachykinin receptor antagonists
12/2001
12/27/2001WO2001098267A1 3-azabicyclo (3.1.0) hexane derivatives having opioid receptor affinity
12/27/2001WO2001098256A1 Thyroid receptor ligands, pharmaceutical compositions comprising them and their use in the treatment of disorders influenced by thyroid hormones
12/27/2001WO2001097810A2 Use of therapeutic benzamide derivatives
12/27/2001WO2001097787A2 Use of microsomal triglyceride transfer protein (mtp) inhibitors for reducing the number of postprandial triglyceride-rich lipoprotein particles (pptrl)
12/27/2001WO2001097782A1 Stable gabapentin having ph within a controlled range
12/27/2001WO2001097751A2 New formulation comprising a betablocker and optionally a cholesterol-lowering agent
12/27/2001WO2001063345A9 Photochemically controlled photonic crystal diffraction
12/27/2001WO2000064864A9 N-protected amines and their use as prodrugs
12/27/2001US20010056113 Methods for the inhibition of angiogenesis with 6-amino EM-12
12/27/2001US20010056112 Synthetic compounds for treatment of inflammation
12/27/2001US20010056100 Carboxylic acid or tetrazole derivatives containing carbamate groups are useful for treating the conditions associated with the urinary tract, pain, inflammation, respiratory states, edema formation of hypotensive vascular diseases
12/27/2001US20010056099 Method of reducing morbidity and the risk of mortality
12/27/2001US20010056096 Administering to a patient suffering from hypercholesterolemia, hyperlipedimea and other metabolic disorders an effective amount of hydrozone, oxime or imine derivatives
12/27/2001US20010056094 3-(Cycloalkanoheteroarylidenyl)-2-Indolinone Protein Tyrosine Kinase Inhibitors
12/27/2001US20010055567 Uses water-soluble dyes and their biomolecule adducts, each having specific photophysical and pharmaco-chemical properties, as contrast media for fluorescence and transillumination diagnostics
12/27/2001CA2413277A1 Use of microsomal triglyceride transfer protein (mtp) inhibitors for reducing the number of postprandial triglyceride-rich lipoprotein particles (pptrl)
12/27/2001CA2412188A1 3-azabicyclo¬3.1.0|hexane derivatives useful in therapy
12/27/2001CA2411100A1 New formulation comprising a betablocker and optionally a cholesterol-lowering agent
12/26/2001CN1328554A Eletriptan hydrobromide monohydrate
12/26/2001CN1328471A Near infrared fluorescent contrast agent and fluorescence imaging
12/26/2001CN1328455A Use of N-substituted azabicycloalkane derivatives for treating diseases of central nervous system
12/25/2001US6333339 3-Benzylpiperidine
12/25/2001US6333323 Indole derivatives with antiviral activity
12/25/2001CA2052424C 2-(4-piperidinyl)-1h-pyrido¬4,3-b|indol-1-ones and related compounds, intermediates and a process for their preparation
12/20/2001WO2001096336A2 6,5-fused bicyclic heterocycles
12/20/2001WO2001096305A1 Serine protease inhibitors
12/20/2001WO2001096300A1 Growth hormone secretagogues
12/20/2001WO2001096299A2 Indole derivatives and their use as 15-lipoxygenase inhibitors
12/20/2001WO2001096298A2 1,2,4-trisubstituted benzenes as inhibitors of 15-lipoxygenase
12/20/2001WO2001096297A2 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
12/20/2001WO2001051456A3 Antibacterial agents
12/20/2001WO2001046121A3 Exciplexes
12/20/2001WO2001016108A3 Bicyclic androgen and progesterone receptor modulator compounds and methods
12/20/2001US20010053778 Pharmaceutical compositions of glycogen phosphorylase inhibitors
12/20/2001DE10029285A1 New 3-(anilino-methylidene)-2-indolinone derivatives, are kinase inhibitors and cell proliferation inhibitors, useful e.g. for treating tumors, metastasis, rheumatoid arthritis or psoriasis
12/20/2001CA2412618A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
12/20/2001CA2412462A1 6,5-fused bicyclic heterocycles
12/20/2001CA2411495A1 1,2,4-trisubstituted benzenes as inhibitors of 15-lipoxygenase
12/20/2001CA2411116A1 Indole derivatives and their use as 15-lipoxygenase inhibitors
12/19/2001EP1163225A1 Compounds and methods for modulation of estrogen receptors
12/19/2001EP1163220A1 Tricyclic indole-2-carboxylic acid compound used as nmda receptor antagonist
12/19/2001EP1163219A1 Substituted 1-oxo- and 1,3-dioxoisoindolines and their use in pharmaceutical compositions for reducing inflammatory cytokine levels
12/19/2001EP1163208A2 Caspase inhibitors and uses thereof
12/19/2001EP0912573B1 Camptothecin-skeleton compounds isolated from mappia foetida and the use thereof as syntones for novel medicaments as well as therapeutical agents
12/19/2001CN1327469A Organic electroluminescent element
12/19/2001CN1327444A Alpha 1 beta-adrenergic receptor antagonists
12/19/2001CN1327383A Pharmaceutical for treatment of neurological and neuropsychiatric disorders
12/19/2001CN1326930A Method for producing cyclic compounds
12/19/2001CN1076348C 3-bustituted oxindole derivatives as patassium path regulating agent
12/18/2001US6331636 Treatment of central nervous system disorders, diabetes, hypertension, impotency, appetite control
12/18/2001US6331632 Cyanine dye phosphoramidites
12/18/2001US6331563 N-Hydroxy-2-(Alkyl, Aryl, or Heteroaryl, Sulfanyl, Sulfinyl or Sulfonyl)-3-Substituted Alkyl, Aryl or Heteroarylamides as Matrix Metalloproteinase inhibitors
12/18/2001US6331554 Antipicornaviral compounds, compositions containing them, and methods for their use
12/18/2001US6331507 Substituted aromatic thiocarboxylic acid amides and their use as herbicides
12/18/2001CA2031897C Carbamoyl derivatives
12/13/2001WO2001094359A1 Chiral ligands for asymmetric catalysis
12/13/2001WO2001094312A2 Indolinone derivatives as protein kinase/phosphatase inhibitors
12/13/2001WO2001094311A1 Cytoprotectors
12/13/2001WO2001094310A1 Methods for making bis-heterocyclic alkaloids
12/13/2001WO2001068599A3 Dosing form for reagents, use of said dosing form in organic chemical synthesis and production of said dosing form
12/13/2001WO2001049275A3 Methods and compositions for mitigating pain using nitrate esters
12/13/2001WO2001032647A3 Benz`f!indoles for use in the treatment of 5ht receptor related disorders
12/13/2001US20010051657 Malonamic acids and derivatives thereof as thyroid receptor ligands
12/13/2001DE10032134C1 Compositions for oxidative dyeing of keratinic fibers, especially human hair, comprise new or known 2-hydroxy-5-amino-biphenyl derivatives as developers
12/13/2001CA2410509A1 Indolinone derivatives as protein kinase/phosphatase inhibitors
12/13/2001CA2410410A1 Chiral ligands for asymmetric catalysis
12/12/2001EP1161948A2 Pharmaceutical or food composition for treatment of brain edema
12/12/2001EP1161434A1 Pyridopyranoazepine derivatives, preparation and therapeutic use
12/12/2001EP1161422A1 Amine derivatives as protease inhibitors
12/12/2001EP1161418A1 1-acyl-7-nitroindoline derivatives, their preparation and their use as photocleavable precursors
12/12/2001EP1161415A2 N-cyanomethylamides as protease inhibitors
12/12/2001EP1161233A2 Lxr modulators
12/12/2001EP1119546A4 Process for preparing toluenesulfinates
12/12/2001EP0968175B1 Spiro compounds and the use thereof
12/12/2001EP0781126B1 Derivatives of 2-amino-1,2,3,4-tetrahydro-naphthalene active on the cardiovascular system
12/12/2001CN1326347A 2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indole in combination with estrogens
12/11/2001US6329550 For therapy of emphysema, osteoporosis, rheumatoid arthritis and neoplastic diseases
12/11/2001US6329531 For therapy of alzheimer's disease
12/11/2001US6329443 Acrylates and actinic radiation-curable compositions containing them
12/11/2001US6329421 Diaryl bicyclic heterocycles as inhibitors of cyclooxygenase-2
12/11/2001US6329416 Administering to female of child bearing age for 28 consecutive days: first phase dosage of progestational agent; second phase of antiprogesin compound, and third phase of placebo for contraception
12/11/2001US6329405 As ileal bile acid transporter inhibitor, for therapy of hyperlipemia
12/11/2001US6329402 Heterocycle-containing carboxylic acid derivative and drug containing the same
12/11/2001US6329394 Medical use for tachykinin antagonists
12/11/2001US6329372 Phenylalanine derivatives
12/11/2001US6329366 Heterocyclic, piperidine, indole derivitives for treatment of nervous system disorders and serotonin antagonist
12/11/2001US6328855 Method for producing (+)-exo-6-phenyl-3-azabicyclo-[3.2.0]heptanes