Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
04/2000
04/26/2000EP0994862A2 Sulphonamide derivatives being 5-ht6 receptor antagonists and process for their preparation
04/26/2000EP0810998B1 Phenyl diketone derivatives as herbicides
04/26/2000CN1251569A Noval compounds, their use and preparation
04/26/2000CN1251523A Sulphonamide derivatives
04/26/2000CN1051765C Stereoselective synthesizing process for enantiomorph pure 3-amino-1,2-twice substituted pyrrolidine
04/26/2000CN1051764C Stereoselective synthesizing process for enantiomorph pure 3-amino-1,2-twice substituted pyrrolidine
04/25/2000US6054579 Reacting a difunctional component containing an activated carbon, an amine capable of forming an imine with the activated carbon, and an isocyanide in a nucleophilic polar protic solvent
04/25/2000US6054482 Hydrolysis of gabapentin or the lactam to form acid addition salt, conversion to pure compound by ion exchanging; antiepileptic agents
04/25/2000US6054445 Kappa opioid agonist activity; analgesics and anti-pruritic agents
04/20/2000WO2000021928A1 Substituted pyrrolidinone, thiazolidinone or oxazolidinone as herbicides
04/20/2000WO2000021927A2 Pyrrole-2,5-diones as gsk-3 inhibitors
04/20/2000WO2000021920A1 Diaminopropionic acid derivatives
04/20/2000WO2000021530A1 Peripherally acting anti-pruritic opiates
04/20/2000WO2000003737A3 Water-soluble drugs and methods for their production
04/20/2000WO1999064000A9 Novel therapeutic agents that modulate neurokinin receptors
04/20/2000CA2346464A1 Peripherally acting anti-pruritic opiates
04/19/2000EP0994110A1 Sulphonamide derivatives
04/19/2000EP0993458A1 3-benzylpiperidine
04/19/2000EP0993445A1 New oxime sulfonates and the use thereof as latent sulfonic acids
04/19/2000EP0993442A1 Hydrazine derivatives
04/19/2000EP0738262B1 Novel heterocyclic compounds
04/19/2000CN1251119A Polymeric amines
04/19/2000CN1251037A Triaryl methane compounds for sickle cell disease
04/18/2000US6051720 Removal of contaminants from N-methyl-2-pyrrolidone
04/18/2000US6051610 Compounds useful as neuroprotectants, anticonvulsants, anxiolytics, analgesics, muscle relaxants or adjuvants to general anesthetics
04/18/2000US6051573 Treatment of GLC1A glaucoma with non-steroidal glucocorticoid antagonists
04/18/2000US6051568 Thrombin inhibitors, their preparation and use
04/18/2000US6051243 Polyaromatic amide compounds and pharmaceutical/cosmetic compositions comprised thereof
04/13/2000WO2000020382A1 Energetic nitramine-linked azoles and hydroxylammonium salts as oxidizers, initiators and gas generators
04/13/2000WO2000002850A3 Sulfonylamino carboxylic acid n-arylamides as guanylate cyclase activators
04/13/2000DE19844787A1 Disubstituierte Pyrrolidinone, diese Verbindung enthaltende Arzneimittel und deren Verwendung sowie ihre Herstellung Disubstituted pyrrolidinone, comprising this compound medicines and their use, and their preparation
04/12/2000EP0992492A1 Small molecule inhibitors of rotamase enzyme activity
04/12/2000EP0991753A1 Protease inhibitors
04/12/2000EP0991654A1 Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and compositions containing same
04/12/2000EP0991627A1 Pyrimidinone compounds, pharmaceutical compositions containing the compounds and the process for preparing the same
04/12/2000EP0991620A1 Pyrrolidine carboxylic acid derivatives as endothelin antagonists
04/12/2000EP0991619A1 INHIBITORS OF $g(a) 4?$g(b) 1?MEDIATED CELL ADHESION
04/12/2000EP0991417A1 Complex formation between dsdna and oligomer of heterocycles
04/12/2000EP0807265B1 Crosslinked polymers
04/12/2000EP0759917B1 Novel selective inhibitors of viral or bacterial neuraminidases
04/11/2000US6048860 Kappa agonist anti-pruritic pharmaceutical formulations and method of treating pruritus therewith
04/11/2000US6048637 Nonaqueous secondary battery
04/11/2000CA1340955C Stilbene derivatives
04/11/2000CA1340952C Chemiluminescent 1,2-dioxetane compounds
04/06/2000WO2000018735A1 2-substituted heterocyclic sulfonamides
04/06/2000WO2000018733A1 Heterocyclic 2-substituted ketoamides useful for treating hair loss in mammals
04/06/2000WO2000018732A2 Disubstituted pyrrolidinones, medicaments containing these compounds, their use and the production thereof
04/06/2000WO2000018724A1 (R)-CHIRAL HALOGENATED 1-SUBSTITUTEDAMINO-(n+1)-ALKANOLS USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY
04/06/2000WO2000018721A1 Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity
04/06/2000WO2000018361A2 Method of treating hair loss using sulfonamides
04/06/2000WO2000018358A2 Method of treating hair loss using ketoamides
04/05/2000EP0990646A1 Process for preparing 3-(7-amidino-2-naphthyl)-2-phenylpropionic acid derivatives
04/05/2000EP0990645A1 Novel sulfonamide derivatives
04/05/2000EP0990439A1 Bisaryl compounds and cancer remedies containing the same
04/05/2000EP0989857A1 Novel therapeutic agents that modulate enzymatic processes
04/05/2000CN1249748A Small molecules useful in treatment of inflamatory disease
04/05/2000CN1249682A Use of angiotension II antagonists to treat symptomatic heart failure
04/04/2000US6046213 Neuroprotective 3-(piperidinyl-1)-chroman-4,7-diol and 1-(4-hydroxyphenyl)-2-(piperidinyl-1)-alkanol derivatives
04/04/2000US6046211 Amidino derivatives useful as nitric oxide synthase inhibitors
03/2000
03/30/2000WO2000017228A2 Stereoselective process for enalapril
03/30/2000WO2000017182A1 PROCESS FOR OBTAINING HMG-CoA REDUCTASE INHIBITORS OF HIGH PURITY
03/30/2000WO2000017176A2 Benzoylguanidine derivatives with advantageous properties, method for producing them and their use in the production of medicaments
03/30/2000WO2000017162A1 Novel thiol derivatives, process for producing the same and utilization thereof
03/30/2000WO2000017161A1 Cyclic ester or amide derivatives
03/30/2000WO2000016765A1 Method and composition for treatment of inflammatory bowel disease
03/30/2000WO2000016763A2 Antimalarial agents
03/30/2000WO2000016603A2 Bridged heterocyclic derivatives
03/30/2000CA2344913A1 Antimalarial agents
03/30/2000CA2344438A1 Method and composition for treatment of inflammatory bowel disease
03/30/2000CA2344412A1 Thiol compound, their production and use
03/30/2000CA2344376A1 Bridged heterocyclic derivatives
03/30/2000CA2343645A1 Process for obtaining hmg-coa reductase inhibitors of high purity
03/30/2000CA2343193A1 Improved stereoselective process for enalapril
03/30/2000CA2341036A1 Cyclic ester or amide derivatives
03/29/2000EP0988284A1 A process for the production of n-methyl pyrrolidone
03/29/2000EP0988263A1 Process for the production of radioiodinated neuroreceptor agents
03/29/2000CN1248434A Keratin fibre dyeing composition using cation direct dye and thickening polymer
03/29/2000CN1050841C Indole derivatives and medicinal composition having same
03/28/2000US6043366 Useful in treating disorders involving the orphanin fq(a seventeen amino acid long peptide) receptor.
03/28/2000US6043261 Pyrrolodino imidines useful as nitric oxide synthase inhibitors
03/28/2000US6043243 Pyrrolidine derivative, anti-ulcer drug, and antibacterial drug
03/28/2000US6043240 Useful as antipsychotic and analgesic agents
03/28/2000US6043239 Heterocyclic compounds
03/28/2000US6042620 p-diaminobenzene derivative compounds and dye compositions containing same
03/28/2000CA2180978C Pyrrolidine-containing monomers and oligomers
03/28/2000CA2177821C Prolyl endopeptidase inhibitors
03/28/2000CA2160270C 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
03/23/2000WO2000015634A2 Hiv protease inhibitors
03/23/2000WO2000015614A1 Novel compounds
03/23/2000WO2000015611A1 Branched alkyl pyrrolidine-3-carboxylic acids
03/23/2000WO2000015610A1 The preparation of n-substituted-hydroxycycloalkylamine derivatives
03/23/2000WO2000015603A1 Benzene derivatives and medicinal use thereof
03/23/2000WO1999063983A9 MULTIBINDING AGENTS THAT MODULATE PPARη AND RXR RECEPTORS
03/23/2000DE19843489A1 New benzoylguanidine derivatives are Na+/H+ exchange inhibitors, useful for treatment of ischemia and other circulation disorders, tumors, prostatic hypertrophy and diabetic complications
03/23/2000DE19841895A1 Neues Verfahren zur Herstellung von 3-Amino-2-oxo-pyrrolidinen, neue Zwischenprodukte und deren Verwendung New process for the preparation of 3-amino-2-oxo-pyrrolidines, to novel intermediates and their use
03/23/2000CA2343837A1 The preparation of n-substituted-hydroxycycloalkylamine derivatives
03/23/2000CA2343101A1 Benzene derivatives and medicinal use thereof
03/23/2000CA2341440A1 Novel compounds
03/23/2000CA2339275A1 5,6-dihydro-4-hydroxy-2-pyranones as hiv aspartyl protease inhibitors
03/22/2000EP0987267A1 Carbapenem compounds, use thereof, and intermediate compounds of the same