Patents
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
02/2001
02/01/2001WO2001007402A1 Antiviral agents
02/01/2001WO2001007400A1 Carboxylic acid derivatives and adhesion molecule inhibitors containing the same as the active ingredient
02/01/2001WO2001007029A2 Substituted guanidines and the use thereof
02/01/2001WO2001007020A2 Carboxylic acid amides, medicaments containing these compounds and the use and production thereof
02/01/2001DE19935693A1 Verfahren zur Herstellung geschützter Acylguanidine durch Mukaiyama Reaktion Process for the preparation of protected acylguanidines by Mukaiyama reaction
02/01/2001DE19935219A1 Carbonsäureamide, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Herstellung Carboxamides, medicaments containing these compounds, their use and production
02/01/2001CA2382757A1 Carboxylic acid derivatives and adhesion molecule inhibitors which contain the same as effective ingredients
01/2001
01/31/2001EP1072576A1 Fluorinating agent, process for producing the same, and use thereof
01/31/2001EP1071670A1 Novel diphenyl-substituted 5-ring-heterocycles, method for producing them and their use as medicaments
01/31/2001EP1071666A1 Azacycloalkane derivatives, preparation and therapeutic application
01/31/2001EP0842152B1 N-(4-substituted-benzyl)-2-aminolactam derivatives
01/31/2001CN1282319A Aminobutanoic acid derivatives
01/31/2001CN1282318A Optically active intermediates for preparation of optically active substituted oximex, hydrazones and olefins useful as neurokinin antagonists
01/31/2001CN1061339C Novel sulfonamide inhibitors of aspartyl protease
01/30/2001US6180796 Sulfonamide derivatives
01/30/2001US6180646 Retroviral protease inhibitors
01/30/2001US6180623 Used as analgesics and anti-pruritic agents
01/25/2001WO2001005783A1 Bradykinin b1 receptor antagonists
01/25/2001WO2001005767A1 Organic compounds
01/25/2001WO2001005765A1 Cyclic amides and imides having selective antagonist activity at alpha-1d adrenergic receptor
01/25/2001WO2001005742A1 Quaternary bis-ammonium salt precursors and their uses as prodrugs having an antiparasitic activity
01/25/2001WO2001005399A1 Anti-ischemic agent
01/25/2001WO2001005354A2 Improved process for the preparation of benzenesulfonylureas as oral hypoglycemic agents of the second generation
01/25/2001WO2001005230A1 Alpha-hydroxy-gamma-[[(carbocyclic-or heterocyclic-substituted)amino]carbonyl]alkanamide derivatives and uses thereof
01/25/2001WO2000071515A3 INHIBITORS OF FACTOR Xa
01/25/2001WO2000066587A3 Polyamines and their use in therapy
01/25/2001DE19934394A1 New N-phenylnaphthalenesulfonamide derivatives useful for treatment and prevention of viral infection, especially cytomegalovirus
01/25/2001DE19934321A1 New N-phenyl-naphthalenesulfonamide derivatives are antiviral agents especially useful for treating cytomegalovirus infections
01/25/2001CA2379891A1 Quaternary bis-ammonium salt precursors and their uses as prodrugs having an antiparasitic activity
01/25/2001CA2379064A1 Bradykinin b1 receptor antagonists
01/25/2001CA2375954A1 Alpha-hydroxy-gamma-¬¬(carbocyclic-or heterocyclic-substituted)amino|carbonyl|alkanamide derivatives and uses thereof
01/24/2001EP0837852B1 Pesticidal sulfur compounds
01/24/2001EP0610377B1 Tri-substituted tetrahydrofuran antifungals
01/23/2001USRE37029 Antipsychotic and analgesic agents
01/23/2001US6177464 Bactericides
01/23/2001US6177446 Synergistic
01/23/2001US6177428 Treatment of sexual dysfunction; stimulation of endogenous nitrogen monoxide synthesis
01/23/2001US6177427 Treatment of glaucoma and ocular hypertension
01/23/2001US6177408 Compounds such as 3-(1-methyl-4(1-methyl-4(1-methyl-4(4-n,n-bis(2 -chloroethyl)aminocinnamoylamido)pyrrole-2-carboxamido)pyrrole-2 -carboxamido)pyrrole-2-carboxamido)propionamidine
01/23/2001CA2296884C Targeted liposomes and methods for liposome-protein coupling
01/23/2001CA2197451C Neuroprotective 3-(piperidinyl-1)-chroman-4,7-diol and 1-(4-hydrophenyl)-2-(piperidinyl-1)-alkanol derivatives
01/23/2001CA2196885C Carboxamide compounds (changed to n-(2-(pyrrolidinyl-1)-1-phenylethyl) acetamides as kappa receptor antagonists)
01/23/2001CA2021340C Cyclic vinylogous n-hydroxy-n-methylureas useful as 5-lipoxygenase inhibitors
01/18/2001WO2001004116A2 Neurotrophic pyrrolidines and piperidines, and related compositions containing them
01/18/2001WO2000071516A3 INHIBITORS OF FACTOR Xa
01/18/2001WO2000059285A3 NOVEL LACTAM INHIBITORS OF MATRIX METALLOPROTEINASES, TNF-α, AND AGGRECANASE
01/18/2001WO1999064049A9 Novel antibacterial agents
01/18/2001CA2379149A1 Neurotrophic pyrrolidines and piperidines, and related compositions and methods
01/17/2001EP1069125A2 Carbamate derivatives of 4-amino-3-isoxazolidinones, 3-amino-1-hydroxypyrrolidin-2-ones and 1-amino-1-cyclopropanecarboxylic acid analogs, a process for their preparation and their use as medicaments
01/17/2001EP1068304A1 Treatment of parasitic diseases by inhibition of cysteine proteases of the papain superfamily
01/17/2001EP1068185A1 Compounds with activity on muscarinic receptors
01/17/2001EP1068183A2 Process for the preparation of a 2-oxopyrrolidine compound
01/17/2001EP1068182A1 Process for preparing a protected 4-aminomethyl-pyrrolidin-3-one
01/17/2001EP1068178A1 NON-PEPTIDE GnRH AGENTS
01/17/2001EP0983258A4 N-hydroxy 4-sulfonyl butanamide compounds
01/17/2001EP0490919B1 Cytoprotective compounds bearing unsaturated hydrocarbon groups having 16 to 20 carbon atoms
01/17/2001CN1280565A Heterocyclic compounds having NOS inhibitory activities
01/17/2001CN1280564A Method for producing salts of cyclic amidines
01/17/2001CN1280128A Process for preparing cis-1-{2-[4-(6-methoxy-2-phenyl-1,2,3,4-tetralin-1-group)phenoxy]ethyl} pyrrolidine
01/16/2001US6174989 Synthetic rubbers and vulcanization for tires
01/16/2001US6174975 Addition polymerization, catalysts and coordination compounds
01/16/2001US6174915 Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses
01/16/2001US6174905 As carcinostatic agent to a hematologic malignancy and a solid carcinoma
01/16/2001US6174898 Method of treating filariae
01/16/2001US6174839 As herbicide
01/16/2001CA2200192C Amidino and guanidino substituted inhibitors of trypsin-like enzymes
01/16/2001CA2010800C Protein labelling
01/11/2001WO2001002381A1 Piperazine derivatives as modulators of chemokine receptor activity
01/11/2001WO2001002376A1 Amino-alkyl derivatives
01/11/2001WO2001002368A1 N-heterocyclic derivatives with neuronal activity
01/11/2001WO2001002358A2 Cyclized amide derivatives for treating or preventing neuronal damage
01/11/2001WO2001002354A1 Phthalamide derivatives, intermediates in the production thereof, and agricultural/horticultural insecticides and method of using the same
01/11/2001WO2001002353A1 Method for producing a 4-(pyrrole-1-yl)-benzoylguanidine derivative
01/10/2001EP1067138A1 Hydroxyproline derivatives
01/10/2001EP1067136A1 New peptide derivatives
01/10/2001EP1066295A2 Synthesis of compounds and libraries of compounds
01/10/2001EP1066258A1 Aryl phenyl substituted cyclic ketoenols
01/10/2001EP1066256A1 The use of derivatives of 2-oxopyrrole as crop protection agents and novel 2-oxopyrroles
01/10/2001CN1279686A Inhibitors of nucleoside metabolism
01/10/2001CN1279680A Imidazole derivatives with inhabiting activity to transterasa and preparing method thereof
01/10/2001CN1060472C Hydroxamic acid derivatives with tricylic substitution, their preparing methods, medicines containing them and uses thereof
01/09/2001US6172261 Biosynthesis using chain extension
01/09/2001US6172255 Alkoxy-alkyl-substituted 1-H-3-aryl-pyrrolidine-2,4-diones used as herbicides and pesticides
01/09/2001US6172234 Optically active cyclic amino acid ester derivatives and processes for producing the same
01/09/2001US6172113 Bicyclic amino derivatives and PGD2 antagonist containing the same
01/09/2001US6172108 Hydrazide compounds
01/09/2001US6172102 Pyrrole derivatives and medicinal composition
01/09/2001US6172083 Applying 4-phenoxyquinoline and 3-(halophenyl)-4-cyanopyrrole derivatives as synergistic mixture
01/09/2001US6172068 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
01/09/2001US6172060 Therapy for sexual disorders
01/09/2001US6172057 Antiinflammatory agents; antiarthritic agents; antitumor agents
01/09/2001US6171595 Skin external preparation
01/09/2001US6171522 Heterocyclic aromatic anion salts, and their uses as ionic conducting materials
01/04/2001WO2001000575A1 Heterocyclic dicarboxylic acid diamide derivatives, agricultural/horticultural insecticides and method of using the same
01/04/2001WO2001000574A1 Pyrrole derivatives
01/04/2001WO2001000229A1 Combination of tumors necrocis factor (tnf) antagonists and cox-2 inhibitors for the treatment of inflammation
01/04/2001WO2001000206A1 Vla-4 inhibitor compounds
01/04/2001DE19929857A1 Verfahren zur Herstellung eines 4-(Pyrrol-1-yl)-benzoylguanidinderivates A method for producing a 4- (pyrrol-1-yl) -benzoylguanidinderivates
01/04/2001CA2369308A1 Vla-4 inhibitor compounds
01/04/2001CA2369145A1 Combination of tumors necrocis factor (tnf) antagonists and cox-2 inhibitors for the treatment of inflammation